
Recettore dell'adenosina
I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.
Trovati 242 prodotti di "Recettore dell'adenosina"
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Adenosine receptor inhibitor 1
CAS:<p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>Formula:C17H19ClFN5O3Colore e forma:SolidPeso molecolare:395.82A1/A3 AR antagonist 2
CAS:<p>The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.</p>Formula:C22H16N2O3SColore e forma:SolidPeso molecolare:388.44AB-MECA
CAS:<p>AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.</p>Formula:C18H21N7O4Purezza:98%Colore e forma:SolidPeso molecolare:399.4A2AAR/HDAC-IN-1
CAS:<p>A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.</p>Formula:C24H21N7O2Colore e forma:SolidPeso molecolare:439.47LASSBio-1359
CAS:LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.Formula:C17H18N2O3Purezza:98%Colore e forma:SolidPeso molecolare:298.34PSB 11 hydrochloride
CAS:<p>PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.</p>Formula:C16H18ClN5OPurezza:98%Colore e forma:SolidPeso molecolare:331.8Adenosine receptor antagonist 3
CAS:<p>Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].</p>Formula:C16H14N6SColore e forma:SolidPeso molecolare:322.39Adentri
CAS:Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.Formula:C18H24N4O3Purezza:98%Colore e forma:SolidPeso molecolare:344.41A2A receptor antagonist 3
CAS:<p>A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).</p>Formula:C26H26N6O2Colore e forma:SolidPeso molecolare:454.52MRS1186
CAS:<p>MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).</p>Formula:C16H12ClN5O2Purezza:98%Colore e forma:SolidPeso molecolare:341.75Adenosine receptor A1 antagonist 5
CAS:<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Formula:C17H20N4O2Purezza:99.97%Colore e forma:SolidPeso molecolare:312.37MRS1177
CAS:<p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>Formula:C20H12ClN5O2Purezza:98%Colore e forma:SolidPeso molecolare:389.79XU1
CAS:<p>XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or</p>Formula:C12H8N2OPurezza:98.58% - 99.59%Colore e forma:SolidPeso molecolare:196.2HEMADO
CAS:<p>HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).</p>Formula:C17H23N5O4Purezza:98%Colore e forma:SolidPeso molecolare:361.4A1AR antagonist 6
CAS:<p>A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].</p>Formula:C17H15N3O2Colore e forma:SolidPeso molecolare:293.32Lu AA41063
CAS:<p>Lu AA41063 is a potent and selective antagonist of the hA2A receptor.</p>Formula:C16H17F2N3O2SColore e forma:SolidPeso molecolare:353.39Neladenoson dalanate HCl
CAS:<p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>Formula:C35H35Cl2N7O4S2Purezza:98%Colore e forma:SolidPeso molecolare:752.73A3AR antagonist 1
CAS:<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Formula:C32H24N4O4SColore e forma:SolidPeso molecolare:560.62Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Formula:C23H21FN8OColore e forma:SolidPeso molecolare:444.46CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Formula:C18H20N6Colore e forma:SolidPeso molecolare:320.39
