Recettore dell'adenosina
I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.
Trovati 242 prodotti di "Recettore dell'adenosina"
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FR-194921
CAS:<p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>Formula:C23H23N5OColore e forma:SolidPeso molecolare:385.46CVT-2759
CAS:<p>CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.</p>Formula:C17H24N6O6Colore e forma:SolidPeso molecolare:408.41Adenosine receptor inhibitor 2
CAS:<p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>Formula:C17H20BrN5O2Colore e forma:SolidPeso molecolare:406.28Acefylline piperazine
CAS:<p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>Formula:C9H10N4O4·xC4H10N2Colore e forma:SolidPeso molecolare:562.54JNJ-40255293
CAS:<p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>Formula:C23H22N4O3Purezza:98%Colore e forma:SolidPeso molecolare:402.45AK-IN-1
CAS:<p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>Formula:C22H21N3O4Colore e forma:SolidPeso molecolare:391.42ATL-801
CAS:<p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>Formula:C24H25N7O3Colore e forma:SolidPeso molecolare:459.5Kira8 Hydrochloride
CAS:<p>Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.</p>Formula:C31H30Cl2N6O3SPurezza:98%Colore e forma:SolidPeso molecolare:637.58A2AAR/HDAC-IN-2
CAS:<p>A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.</p>Formula:C23H26N6O4Colore e forma:SolidPeso molecolare:450.49Theophylline sodium glycinate
CAS:<p>Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.</p>Formula:C9H12N5NaO4Colore e forma:SolidPeso molecolare:277.216hA2AAR antagonist 1
CAS:<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Formula:C15H15N5OColore e forma:SolidPeso molecolare:281.31LUF5831
CAS:<p>LUF5831 is an agonist of adenosine A1 receptor.</p>Formula:C15H12N4O2SColore e forma:SolidPeso molecolare:312.35Draflazine
CAS:<p>Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.</p>Formula:C30H33Cl2F2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:604.52LUF5981
CAS:<p>LUF5981 is a selective agonist of human adenosine A1 receptor.</p>Formula:C24H23N3Colore e forma:SolidPeso molecolare:353.46Cirazoline hydrochloride
CAS:<p>Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.</p>Formula:C13H17ClN2OPurezza:99.863%Colore e forma:SolidPeso molecolare:252.74Bamifylline Hydrochloride
CAS:<p>Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.</p>Formula:C20H28ClN5O3Colore e forma:SolidPeso molecolare:421.92MRS1067
CAS:<p>MRS1067 is an antagonist of A3 adenosine receptor.</p>Formula:C19H16Cl2O3Colore e forma:SolidPeso molecolare:363.23MRE3008F20
CAS:<p>MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.</p>Formula:C21H20N8O3Purezza:97.29%Colore e forma:SolidPeso molecolare:432.44A2AR-antagonist-1
CAS:<p>Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.</p>Formula:C27H25N5O2Purezza:98%Colore e forma:SolidPeso molecolare:451.52VUF 5574
CAS:<p>VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.</p>Formula:C21H17N5O2Purezza:99.53%Colore e forma:SolidPeso molecolare:371.39ST3932
CAS:<p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>Formula:C12H16N8OPurezza:98%Colore e forma:SolidPeso molecolare:288.31APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formula:C18H22N6O4Purezza:99.88%Colore e forma:SolidPeso molecolare:386.41N6-Cyclopentyladenosine
CAS:<p>N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of</p>Formula:C15H21N5O4Purezza:99.84%Colore e forma:SolidPeso molecolare:335.36Sonedenoson
CAS:<p>Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.</p>Formula:C18H20ClN5O5Purezza:99.79%Colore e forma:SolidPeso molecolare:421.84Evodenoson
CAS:<p>Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.</p>Formula:C23H29N7O6Purezza:99.75% - 99.83%Colore e forma:SolidPeso molecolare:499.52N-[(4-Aminophenyl)methyl]adenosine
CAS:<p>N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).</p>Formula:C17H20N6O4Purezza:98.75%Colore e forma:SolidPeso molecolare:372.38BAY 60-6583
CAS:<p>BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3</p>Formula:C19H17N5O2SPurezza:98.46% - 99.8%Colore e forma:SolidPeso molecolare:379.44ANR 94
CAS:<p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>Formula:C9H13N5OPurezza:98.9%Colore e forma:SolidPeso molecolare:207.23Adenosine antagonist-1
CAS:<p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>Formula:C18H13N7SPurezza:99.28% - 99.95%Colore e forma:SolidPeso molecolare:359.41ST-1535
CAS:<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Formula:C12H16N8Purezza:99.64% - 99.69%Colore e forma:SolidPeso molecolare:272.31MRS1220
CAS:<p>MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic</p>Formula:C21H14ClN5O2Purezza:98.43%Colore e forma:SolidPeso molecolare:403.82N 0861
CAS:<p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>Formula:C13H17N5Purezza:98.78%Colore e forma:SolidPeso molecolare:243.31Selodenoson
CAS:<p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>Formula:C17H24N6O4Purezza:99.52%Colore e forma:SolidPeso molecolare:376.41ISAM-140
CAS:<p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>Formula:C19H19N3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:337.37GW-493838
CAS:<p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>Formula:C21H21ClFN7O4Purezza:99.11% - 99.58%Colore e forma:SolidPeso molecolare:489.89GS-9667
CAS:<p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>Formula:C21H24FN5O4SPurezza:99.76% - 99.77%Colore e forma:SolidPeso molecolare:461.51A2A receptor antagonist 1
CAS:<p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>Formula:C16H12FN5OPurezza:99.52% - 99.93%Colore e forma:SolidPeso molecolare:309.3LAS38096
CAS:<p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>Formula:C17H12N6OPurezza:99.18% - 99.95%Colore e forma:SolidPeso molecolare:316.32N6-(2-Phenylethyl)adenosine
CAS:<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Formula:C18H21N5O4Purezza:99.83%Colore e forma:SolidPeso molecolare:371.392'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formula:C16H22ClN5O4Purezza:99.93%Colore e forma:SolidPeso molecolare:383.83KI-7
CAS:<p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>Formula:C23H18N2O2Purezza:98.33%Colore e forma:SolidPeso molecolare:354.4FK-453
CAS:<p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>Formula:C23H25N3O2Purezza:99.44%Colore e forma:SolidPeso molecolare:375.46GP3269
CAS:<p>GP3269 is a selective, potent, orally active human adenosine kinase (AK) inhibitor (IC50: 11 nM) with anticonvulsant effects in rats.</p>Formula:C23H21FN4O3Colore e forma:SolidPeso molecolare:420.44PSB-1115 potassium salt
CAS:<p>PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1].</p>Formula:C14H13KN4O5SColore e forma:SolidPeso molecolare:388.44MRS3558
CAS:<p>MRS3558 is an agonist of A3 adenosine receptors.</p>Formula:C20H20Cl2N6O3Colore e forma:SolidPeso molecolare:463.32ABT-702 hydrochloride
CAS:<p>ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].</p>Formula:C22H20BrClN6OColore e forma:SolidPeso molecolare:499.79KFM19
CAS:<p>KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.</p>Formula:C16H22N4O3Purezza:98.62%Colore e forma:SolidPeso molecolare:318.37Neladenoson dalanate
CAS:<p>Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.</p>Formula:C35H34ClN7O4S2Colore e forma:SolidPeso molecolare:716.27Sulmazole
CAS:<p>Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.</p>Formula:C14H13N3O2SPurezza:99.94%Colore e forma:SolidPeso molecolare:287.34Xanthine amine congener
CAS:<p>Xanthine amine congener is an Adenosine receptor antagonist.</p>Formula:C21H28N6O4Purezza:99.7%Colore e forma:SolidPeso molecolare:428.48
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