
Recettore dei cannabinoidi
I recettori dei cannabinoidi sono GPCR che mediano gli effetti dei cannabinoidi endogeni (endocannabinoidi) e fitocannabinoidi, come quelli presenti nella cannabis. I due principali tipi di recettori dei cannabinoidi, CB1 e CB2, sono coinvolti nella regolazione di una vasta gamma di processi fisiologici, tra cui la percezione del dolore, l'appetito, l'umore e la funzione immunitaria. I modulatori dei recettori dei cannabinoidi hanno un potenziale terapeutico nel trattamento di condizioni come il dolore cronico, l'epilessia e la sclerosi multipla. Presso CymitQuimica, offriamo una vasta gamma di modulatori di recettori dei cannabinoidi di alta qualità per supportare la tua ricerca in neurofarmacologia, gestione del dolore e immunologia.
Trovati 217 prodotti di "Recettore dei cannabinoidi"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurezza:99.28% - 99.83%Colore e forma:SolidPeso molecolare:487.4GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormula:C23H24Cl2N2O3Purezza:99.82% - 99.93%Colore e forma:SolidPeso molecolare:447.35Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Formula:C20H37NO2Purezza:99.97%Colore e forma:SolidPeso molecolare:323.51Ref: TM-T8425
1mg34,00€5mg64,00€1mL*10mM (DMSO)80,00€10mg95,00€25mg156,00€50mg225,00€100mg329,00€200mg495,00€AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Formula:C21H19Cl2IN4O2Purezza:98.6% - >99.99%Colore e forma:White To Off-White SolidPeso molecolare:557.21Ref: TM-T2264
1mg80,00€5mg169,00€1mL*10mM (DMSO)233,00€10mg259,00€25mg523,00€50mg750,00€100mg1.035,00€500mg2.062,00€AM-2232
CAS:AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Formula:C24H20N2OPurezza:99.37%Colore e forma:SolidPeso molecolare:352.43LY2828360
CAS:LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Formula:C22H27ClN6OPurezza:98.45% - 99.51%Colore e forma:SolidPeso molecolare:426.94CID 16020046
CAS:CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.Formula:C25H19N3O4Purezza:99.03%Colore e forma:SolidPeso molecolare:425.44Otenabant
CAS:Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formula:C25H25Cl2N7OPurezza:99.43%Colore e forma:SolidPeso molecolare:510.42CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formula:C33H31Cl2F3N6O3S2Purezza:99.08% - 99.76%Colore e forma:SolidPeso molecolare:751.67Ref: TM-T5996
1mg82,00€2mg110,00€5mg180,00€1mL*10mM (DMSO)215,00€10mg258,00€25mg423,00€50mg588,00€100mg793,00€500mg1.594,00€Tetrahydromagnolol
CAS:Tetrahydromagnolol can activate cannabinoid (CB) receptors.Formula:C18H22O2Purezza:99.86% - >99.99%Colore e forma:SolidPeso molecolare:270.37BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体,其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formula:C23H23ClN2O4Purezza:97.70%Colore e forma:SolidPeso molecolare:426.89CB1/2 agonist 3
CAS:CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formula:C25H41NO2Purezza:98.78%Colore e forma:SolidPeso molecolare:387.6S-Methoprene
CAS:S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Formula:C19H34O3Purezza:97.05% - 98.55%Colore e forma:SolidPeso molecolare:310.47Dehydroabiethylamine
CAS:Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Formula:C20H31NPurezza:98.79%Colore e forma:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidPeso molecolare:285.47PSB-KK1445
CAS:PSB-KK1445 is a potent and selective agonist of GPR18, exhibiting EC50 values of 45.4 nM for humans and 124 nM for mice. The selectivity of PSB-KK1445 for GPR18 over the CB receptor subtypes GPR55 and GPR183 exceeds 200-fold.Formula:C24H23FN6O2Peso molecolare:446.48GPR55 agonist 3
CAS:Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Formula:C19H16F4N4Colore e forma:SolidPeso molecolare:376.35PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Formula:C22H31NO3Colore e forma:SolidPeso molecolare:357.49CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Formula:C24H23N3O4S2Purezza:98%Colore e forma:SolidPeso molecolare:481.59VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formula:C18H26N2O3Colore e forma:SolidPeso molecolare:318.41GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Formula:C22H18N2O2Colore e forma:SolidPeso molecolare:342.39

