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Recettore dei cannabinoidi

Recettore dei cannabinoidi

I recettori dei cannabinoidi sono GPCR che mediano gli effetti dei cannabinoidi endogeni (endocannabinoidi) e fitocannabinoidi, come quelli presenti nella cannabis. I due principali tipi di recettori dei cannabinoidi, CB1 e CB2, sono coinvolti nella regolazione di una vasta gamma di processi fisiologici, tra cui la percezione del dolore, l'appetito, l'umore e la funzione immunitaria. I modulatori dei recettori dei cannabinoidi hanno un potenziale terapeutico nel trattamento di condizioni come il dolore cronico, l'epilessia e la sclerosi multipla. Presso CymitQuimica, offriamo una vasta gamma di modulatori di recettori dei cannabinoidi di alta qualità per supportare la tua ricerca in neurofarmacologia, gestione del dolore e immunologia.

Trovati 217 prodotti di "Recettore dei cannabinoidi"

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  • O-2093

    CAS:
    anandamide uptake inhibitor
    Formula:C34H43Cl2NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:584.62

    Ref: TM-T23100

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • CID1172084

    CAS:
    CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.
    Formula:C23H18FN5O2S2
    Colore e forma:Solid
    Peso molecolare:479.55

    Ref: TM-T27016

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • CB2 receptor agonist 3

    CAS:
    GP 2A is a selective agonist of CB2 receptor.
    Formula:C24H23Cl2N3O
    Colore e forma:Solid
    Peso molecolare:440.36

    Ref: TM-T24097

    25mg
    690,00€
    50mg
    898,00€
    100mg
    1.566,00€
  • TC-C 14G

    CAS:
    CB1 receptor inverse agonist
    Formula:C24H17Cl2F2NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:492.3

    Ref: TM-T23427

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • (R)-SLV 319

    CAS:
    (R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.
    Formula:C23H20Cl2N4O2S
    Colore e forma:Solid
    Peso molecolare:487.4

    Ref: TM-T22140

    5mg
    1.018,00€
    10mg
    1.513,00€
  • Olorinab

    CAS:
    Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.
    Formula:C18H23N5O3
    Purezza:97.67% - 98.47%
    Colore e forma:Solid
    Peso molecolare:357.41

    Ref: TM-T14302

    1mg
    56,00€
    5mg
    119,00€
    10mg
    187,00€
    25mg
    378,00€
    50mg
    560,00€
  • AM-1235

    CAS:
    AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.
    Formula:C24H21FN2O3
    Purezza:99.92%
    Colore e forma:Solid
    Peso molecolare:404.43

    Ref: TM-T29930

    1mg
    315,00€
    5mg
    745,00€
    10mg
    1.018,00€
    25mg
    1.431,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • CB1 agonist 1

    CAS:
    CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.
    Formula:C24H24N2O5S
    Purezza:98.56%
    Colore e forma:Solid
    Peso molecolare:452.52

    Ref: TM-T62761

    5mg
    74,00€
    10mg
    107,00€
    25mg
    216,00€
    50mg
    354,00€
    100mg
    567,00€
  • SR144528

    CAS:
    SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).
    Formula:C29H34ClN3O
    Purezza:99.63%
    Colore e forma:Solid
    Peso molecolare:476.05

    Ref: TM-T16928

    1mg
    43,00€
    5mg
    95,00€
    10mg
    155,00€
    25mg
    339,00€
    50mg
    507,00€
    100mg
    730,00€
    1mL*10mM (DMSO)
    95,00€
  • Nonabine

    CAS:
    Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.
    Formula:C25H33NO2
    Purezza:99.82% - 99.94%
    Colore e forma:Solid
    Peso molecolare:379.54

    Ref: TM-T28187

    1mg
    139,00€
    5mg
    333,00€
    10mg
    504,00€
    25mg
    817,00€
    50mg
    1.121,00€
    100mg
    1.510,00€
  • CB1R antagonist 1

    CAS:
    CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.
    Formula:C18H23F3N2O3S
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:404.45

    Ref: TM-T61989

    5mg
    74,00€
    10mg
    116,00€
    25mg
    188,00€
    50mg
    279,00€
    100mg
    416,00€
  • CB2R PAM

    CAS:
    CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in neuropathic pain relief.
    Formula:C21H24BrFN2O2
    Purezza:99.09%
    Colore e forma:Solid
    Peso molecolare:435.33

    Ref: TM-T37075

    1mg
    52,00€
    5mg
    113,00€
    10mg
    167,00€
    25mg
    265,00€
    50mg
    404,00€
    100mg
    593,00€
    500mg
    1.243,00€
  • SCH-336

    CAS:

    SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.

    Formula:C23H25NO8S3
    Purezza:95.01%
    Colore e forma:Solid
    Peso molecolare:539.64

    Ref: TM-T24771

    5mg
    52,00€
    10mg
    78,00€
    25mg
    160,00€
    50mg
    225,00€
    100mg
    325,00€
    200mg
    469,00€
  • PSB-CB5

    CAS:
    PSB-CB5 (GPR18-IN-32)2 is a GRP18 antagonist with anti-inflammatory activity and can be used to study obesity and metabolic disorders.
    Formula:C20H17ClN2O2S
    Purezza:99.26%
    Colore e forma:Solid
    Peso molecolare:384.88

    Ref: TM-T27019

    1mg
    84,00€
    5mg
    173,00€
    10mg
    294,00€
    25mg
    492,00€
  • AZD1940

    CAS:
    AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.
    Formula:C20H29F2N3O2S
    Purezza:98.68%
    Colore e forma:Solid
    Peso molecolare:413.52

    Ref: TM-T30252

    1mg
    130,00€
    5mg
    311,00€
    10mg
    535,00€
    25mg
    847,00€
    50mg
    1.169,00€
    100mg
    1.586,00€
    1mL*10mM (DMSO)
    344,00€
  • JTE-907

    CAS:
    JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。
    Formula:C24H26N2O6
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:438.47

    Ref: TM-T19705

    1mg
    56,00€
    5mg
    126,00€
    10mg
    187,00€
    25mg
    329,00€
    50mg
    490,00€
    100mg
    700,00€
    1mL*10mM (DMSO)
    150,00€
  • O-2050

    CAS:
    O-2050: strong CB1 antagonist (Ki 2.5 nM), CB2 inhibitor (Ki 0.2 nM); reduces mouse food intake, increases activity.
    Formula:C23H31NO4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:417.56

    Ref: TM-T23099

    25mg
    2.033,00€
    50mg
    2.645,00€
    100mg
    3.345,00€
  • Heptadecanoyl ethanolamide

    CAS:
    Heptadecanoyl ethanolamide, an endogenous cannabinoid, serves as a synthetic analog of PEA, featuring an odd-numbered (17-carbon) fatty acid chain [1].
    Formula:C19H39NO2
    Colore e forma:Solid
    Peso molecolare:313.52

    Ref: TM-T84594

    10mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
  • COR659

    CAS:
    COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
    Formula:C16H16ClNO3S
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:337.82

    Ref: TM-T36520

    1mg
    38,00€
    5mg
    86,00€
    10mg
    123,00€
    25mg
    215,00€
    50mg
    299,00€
    100mg
    411,00€
    200mg
    560,00€
    1mL*10mM (DMSO)
    94,00€
  • PF-03550096

    CAS:
    PF-03550096, an orally active synthetic cannabinoid (CB), selectively binds to peripheral CB2 receptors with a Ki value of 7.9 nM, demonstrating analgesic activity [1].
    Formula:C19H28N4O4
    Colore e forma:Solid
    Peso molecolare:376.45

    Ref: TM-T84412

    10mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta