
Recettore dei cannabinoidi
I recettori dei cannabinoidi sono GPCR che mediano gli effetti dei cannabinoidi endogeni (endocannabinoidi) e fitocannabinoidi, come quelli presenti nella cannabis. I due principali tipi di recettori dei cannabinoidi, CB1 e CB2, sono coinvolti nella regolazione di una vasta gamma di processi fisiologici, tra cui la percezione del dolore, l'appetito, l'umore e la funzione immunitaria. I modulatori dei recettori dei cannabinoidi hanno un potenziale terapeutico nel trattamento di condizioni come il dolore cronico, l'epilessia e la sclerosi multipla. Presso CymitQuimica, offriamo una vasta gamma di modulatori di recettori dei cannabinoidi di alta qualità per supportare la tua ricerca in neurofarmacologia, gestione del dolore e immunologia.
Trovati 217 prodotti di "Recettore dei cannabinoidi"
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Δ9-THCH
CAS:Δ9-THCH, a phytocannabinoid analytical reference standard, is present in a Cannabis variety cultivated for medicinal use. In the United States, it is classified as a Schedule I compound. This product is designated for research and forensic applications.Formula:C22H32O2Colore e forma:SolidPeso molecolare:328.49CB1-IN-3
CB1-IN-3 (Compound 6i) is a potent inhibitor of the cannabinoid receptor type 1 (CB1). It holds potential for research in obesity, inflammation, and neurological disorders.Colore e forma:Odour SolidCannabidivarinic acid
CAS:Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.Formula:C20H26O4Colore e forma:SolidPeso molecolare:330.42Taranabant racemate
CAS:Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.Formula:C27H25ClF3N3O2Purezza:98%Colore e forma:SolidPeso molecolare:515.95Virodhamine
CAS:Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formula:C22H37NO2Purezza:98%Colore e forma:SoildPeso molecolare:347.53WIN 55,212-2 Mesylate
CAS:WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) is a potent aminoalkylindole cannabinoid (CB) receptor agonist with Kis of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively. Cannabinoid analogue WIN 55,212-2 Mesylate exhibited a novel anticancer effect against human tumors.Formula:C28H30N2O6SPurezza:98% - 99.71%Colore e forma:White To Off-White SolidPeso molecolare:522.61AM251
CAS:AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).Formula:C22H21Cl2IN4OPurezza:97.43% - 98.79%Colore e forma:A Crystalline SolidPeso molecolare:555.24Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.Formula:C52H83N13O14Purezza:99.86%Colore e forma:SolidPeso molecolare:1114.29Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFormula:C21H32O2Purezza:99.59% - 99.92%Colore e forma:SolidPeso molecolare:316.48Ref: TM-TN1465
1mg145,00€2mg215,00€5mg314,00€10mg474,00€25mg808,00€50mg1.111,00€100mg1.501,00€1mL*10mM (DMSO)324,00€PSB-SB-487
CAS:PSB-SB-487 is antagonist of GPR55.Formula:C26H32O4Purezza:98.53%Colore e forma:SolidPeso molecolare:408.53Ref: TM-T8975
1mg38,00€5mg85,00€10mg126,00€25mg245,00€50mg364,00€100mg507,00€200mg697,00€1mL*10mM (DMSO)93,00€ML-191
CAS:ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formula:C24H25N3O3Purezza:99.58%Colore e forma:SolidPeso molecolare:403.47ML-184
CAS:ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.Formula:C25H34N4O3SPurezza:99.45%Colore e forma:SolidPeso molecolare:470.63JD-5037
CAS:JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Formula:C27H27Cl2N5O3SPurezza:99.54% - 99.84%Colore e forma:SolidPeso molecolare:572.51Ref: TM-T4453
1mg44,00€2mg58,00€5mg95,00€10mg140,00€25mg246,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)106,00€ML-193
CAS:ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formula:C28H25N5O4SPurezza:97.74%Colore e forma:SolidPeso molecolare:527.59Ref: TM-T22103
5mg47,00€10mg73,00€25mg110,00€50mg166,00€100mgPrezzo su richiesta1mL*10mM (DMSO)63,00€Otenabant hydrochloride
CAS:Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).Formula:C25H26Cl3N7OPurezza:99.79% - ≥95%Colore e forma:SolidPeso molecolare:546.88Olivetol
CAS:Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.Formula:C11H16O2Purezza:99.98%Colore e forma:(Melting Point 102-106°F) (Ntp 1992)Peso molecolare:180.24CB1 antagonist 4
CAS:TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Formula:C30H25Cl2F3N4OSPurezza:98.97%Colore e forma:SolidPeso molecolare:617.51Ref: TM-T8511
2mg48,00€5mg97,00€10mg160,00€25mg273,00€50mg427,00€100mg630,00€200mg895,00€1mL*10mM (DMSO)163,00€Bay 59-3074
CAS:<p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>Formula:C18H13F6NO4SPurezza:97.68% - 99.69%Colore e forma:SolidPeso molecolare:453.36AM1241
CAS:AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Formula:C22H22IN3O3Purezza:98.937% - 99.1%Colore e forma:SolidPeso molecolare:503.33Ref: TM-T6755
2mg38,00€5mg51,00€10mg88,00€25mg172,00€50mg290,00€100mg523,00€500mg1.130,00€1mL*10mM (DMSO)93,00€Org 27569
CAS:Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity andFormula:C24H28ClN3OPurezza:>99.99% - ≥95%Colore e forma:SolidPeso molecolare:409.95A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurezza:99.94%Colore e forma:SolidPeso molecolare:310.45Ref: TM-T7375
2mg35,00€5mg71,00€10mg115,00€25mg187,00€50mg274,00€100mg390,00€200mg527,00€1mL*10mM (DMSO)66,00€RTICBM-189
CAS:RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formula:C15H14Cl2N2OPurezza:99.96%Colore e forma:SolidPeso molecolare:309.19Ref: TM-T9466
2mg37,00€5mg50,00€10mg88,00€25mg170,00€50mg264,00€100mg389,00€200mg550,00€1mL*10mM (DMSO)71,00€GW842166X
CAS:GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formula:C18H17Cl2F3N4O2Purezza:99.47%Colore e forma:SolidPeso molecolare:449.25β-Caryophyllene
CAS:β-Caryophyllene ((-)-(E)-Caryophyllene) acts as an CB2 receptor agonist.Formula:C15H24Purezza:95.43% - 99.11%Colore e forma:Turpentine (Ntp 1992)Peso molecolare:204.35N-Oleoyl glycine
CAS:N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated AktFormula:C20H37NO3Purezza:97.43%Colore e forma:SolidPeso molecolare:339.51RVD-Hpα acetate(1193362-76-3 free base)
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formula:C67H109N19O19Purezza:99.87%Colore e forma:SolidPeso molecolare:1484.71Ref: TM-TP1939L1
1mg213,00€5mg464,00€10mg677,00€25mg1.035,00€50mg1.406,00€100mg1.882,00€500mg3.771,00€yangonin
CAS:Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.Formula:C15H14O4Purezza:98.82% - 99.55%Colore e forma:Pale Yellow PowderPeso molecolare:258.27Ref: TM-T3S0738
1mg70,00€5mg135,00€10mg207,00€25mg349,00€50mg515,00€100mg735,00€1mL*10mM (DMSO)177,00€ARN272
CAS:ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Formula:C27H20N4O2Purezza:98.23%Colore e forma:SolidPeso molecolare:432.47Voacamine
CAS:<p>Voacamine: an indole alkaloid, CB1 antagonist, inhibits P-gp, may affect rhythm.</p>Formula:C43H52N4O5Purezza:98.54% - 99.82%Colore e forma:SolidPeso molecolare:704.9Hemopressin (rat) acetate(568588-77-2 free base)
Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.Formula:C5H81N13O14Purezza:99.37%Colore e forma:SolidPeso molecolare:1148.31AM-2232
CAS:AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Formula:C24H20N2OPurezza:99.37%Colore e forma:SolidPeso molecolare:352.43(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurezza:99.28% - 99.83%Colore e forma:SolidPeso molecolare:487.4AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Formula:C21H19Cl2IN4O2Purezza:98.6% - >99.99%Colore e forma:White To Off-White SolidPeso molecolare:557.21Ref: TM-T2264
1mg85,00€5mg172,00€10mg274,00€25mg552,00€50mg792,00€100mg1.093,00€500mg2.175,00€1mL*10mM (DMSO)245,00€GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormula:C23H24Cl2N2O3Purezza:99.82% - 99.93%Colore e forma:SolidPeso molecolare:447.35Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Formula:C20H37NO2Purezza:99.97%Colore e forma:SolidPeso molecolare:323.51Ref: TM-T8425
1mg35,00€5mg67,00€10mg90,00€25mg164,00€50mg239,00€100mg348,00€200mg522,00€1mL*10mM (DMSO)85,00€LY2828360
CAS:LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Formula:C22H27ClN6OPurezza:98.45% - 99.51%Colore e forma:SolidPeso molecolare:426.94CID 16020046
CAS:<p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>Formula:C25H19N3O4Purezza:99.03%Colore e forma:SolidPeso molecolare:425.44Otenabant
CAS:Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formula:C25H25Cl2N7OPurezza:99.43%Colore e forma:SolidPeso molecolare:510.42CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formula:C33H31Cl2F3N6O3S2Purezza:99.08% - 99.76%Colore e forma:SolidPeso molecolare:751.67Ref: TM-T5996
1mg87,00€2mg116,00€5mg190,00€10mg271,00€25mg445,00€50mg622,00€100mg837,00€500mg1.681,00€1mL*10mM (DMSO)226,00€Tetrahydromagnolol
CAS:Tetrahydromagnolol can activate cannabinoid (CB) receptors.Formula:C18H22O2Purezza:99.86% - >99.99%Colore e forma:SolidPeso molecolare:270.37BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体,其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formula:C23H23ClN2O4Purezza:97.70%Colore e forma:SolidPeso molecolare:426.89CB1/2 agonist 3
CAS:CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formula:C25H41NO2Purezza:98.78%Colore e forma:SolidPeso molecolare:387.6S-Methoprene
CAS:<p>S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.</p>Formula:C19H34O3Purezza:97.05% - 98.55%Colore e forma:SolidPeso molecolare:310.47Dehydroabiethylamine
CAS:Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Formula:C20H31NPurezza:98.79%Colore e forma:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidPeso molecolare:285.47PSB-KK1445
CAS:PSB-KK1445 is a potent and selective agonist of GPR18, exhibiting EC50 values of 45.4 nM for humans and 124 nM for mice. The selectivity of PSB-KK1445 for GPR18 over the CB receptor subtypes GPR55 and GPR183 exceeds 200-fold.Formula:C24H23FN6O2Peso molecolare:446.48GPR55 agonist 3
CAS:Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Formula:C19H16F4N4Colore e forma:SolidPeso molecolare:376.35PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Formula:C22H31NO3Colore e forma:SolidPeso molecolare:357.49CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Formula:C24H23N3O4S2Purezza:98%Colore e forma:SolidPeso molecolare:481.59VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formula:C18H26N2O3Colore e forma:SolidPeso molecolare:318.41GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Formula:C22H18N2O2Colore e forma:SolidPeso molecolare:342.39

