Recettore dei cannabinoidi

I recettori dei cannabinoidi sono GPCR che mediano gli effetti dei cannabinoidi endogeni (endocannabinoidi) e fitocannabinoidi, come quelli presenti nella cannabis. I due principali tipi di recettori dei cannabinoidi, CB1 e CB2, sono coinvolti nella regolazione di una vasta gamma di processi fisiologici, tra cui la percezione del dolore, l'appetito, l'umore e la funzione immunitaria. I modulatori dei recettori dei cannabinoidi hanno un potenziale terapeutico nel trattamento di condizioni come il dolore cronico, l'epilessia e la sclerosi multipla. Presso CymitQuimica, offriamo una vasta gamma di modulatori di recettori dei cannabinoidi di alta qualità per supportare la tua ricerca in neurofarmacologia, gestione del dolore e immunologia.

Trovati 215 prodotti di "Recettore dei cannabinoidi"

Purezza (%)

100

prodotti per pagina.

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CB2 receptor agonist 2
CAS:
- 1314230-75-5
CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.
Formula:C₃₀H₃₆N₂O₄
Purezza:99.75%
Colore e forma:Solid
Peso molecolare:488.62
Ref: TM-T22009
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APP-FUBINACA
CAS:
- 1185282-03-4
APP-FUBINACA is a cannabinoid receptor agonist, classified as a phenylalanine amide-based indazole-3-carboxamide derivative. It exhibits neurostimulatory effects.
Formula:C₂₄H₂₁FN₄O₂
Colore e forma:Solid
Peso molecolare:416.45
Ref: TM-T203471
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TRPV1/CB2 agonist 1
TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.
Colore e forma:Odour Solid
Ref: TM-T200749
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CB1R agonist 1
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.
Formula:C₂₀H₁₈F₃N₃O₃S
Colore e forma:Solid
Peso molecolare:437.435
Ref: TM-T206337
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N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide
CAS:
- 1258011-97-0
N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide: binds CB1 (Ki=365 nM), activates PPARα (EC50=698 nM), reduces rat food intake, no FAAH inhibition.
Formula:C₂₇H₄₅NO₃
Colore e forma:Solid
Peso molecolare:431.661
Ref: TM-T38223
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VIP36
VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.
Formula:C₂₇H₃₅FN₆O₄
Colore e forma:Solid
Peso molecolare:526.603
Ref: TM-T206705
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CB2 receptor antagonist 2
Compound 39, also known as CB2 receptor antagonist 2, is a potent CB2 antagonist exhibiting an IC50 of 0.33 μM.
Colore e forma:Odour Solid
Ref: TM-T82772
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(−)-6α-hydroxy Cannabidiol
CAS:
- 58940-28-6
(−)-6α-Hydroxy Cannabidiol, an analytical reference standard and a phytocannabinoid metabolite, serves primarily as a metabolite of cannabidiol (CBD). This product is designed for use in research and forensic applications.
Formula:C₂₁H₃₀O₃
Colore e forma:Solid
Peso molecolare:330.46
Ref: TM-TN7529
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CB1-IN-3
CB1-IN-3 (Compound 6i) is a potent inhibitor of the cannabinoid receptor type 1 (CB1). It holds potential for research in obesity, inflammation, and neurological disorders.
Colore e forma:Odour Solid
Ref: TM-T210564
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Δ9-THCH
CAS:
- 36482-24-3
Δ9-THCH, a phytocannabinoid analytical reference standard, is present in a Cannabis variety cultivated for medicinal use. In the United States, it is classified as a Schedule I compound. This product is designated for research and forensic applications.
Formula:C₂₂H₃₂O₂
Colore e forma:Solid
Peso molecolare:328.49
Ref: TM-TN7523
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Cannabigerorcinic Acid
CAS:
- 69734-83-4
Cannabigerorcinic acid, structurally akin to recognized phytocannabinoids, serves as an analytical reference standard designed for research and forensic purposes.
Formula:C₁₈H₂₄O₄
Colore e forma:Solid
Peso molecolare:304.386
Ref: TM-TN7556
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Tocrifluor T1117
CAS:
- 1186195-59-4
Fluorescent form of AM 251, CB1 receptor antagonist
Formula:C₅₆H₅₃Cl₂N₇O₅
Purezza:98%
Colore e forma:Solid
Peso molecolare:974.97
Ref: TM-T23464
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Taranabant racemate
CAS:
- 701977-00-6
Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.
Formula:C₂₇H₂₅ClF₃N₃O₂
Purezza:98%
Colore e forma:Solid
Peso molecolare:515.95
Ref: TM-T13081
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Virodhamine
CAS:
- 287937-12-6
Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.
Formula:C₂₂H₃₇NO₂
Purezza:98%
Colore e forma:Soild
Peso molecolare:347.53
Ref: TM-T64371
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LY2828360
CAS:
- 1231220-79-3
LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.
Formula:C₂₂H₂₇ClN₆O
Purezza:98.45% - 99.51%
Colore e forma:Solid
Peso molecolare:426.94
Ref: TM-T7316
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Otenabant
CAS:
- 686344-29-6
Otenabant (CP-945598) has been investigated for the treatment of Obesity.
Formula:C₂₅H₂₅Cl₂N₇O
Purezza:99.43%
Colore e forma:Solid
Peso molecolare:510.42
Ref: TM-T3530
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CB1-IN-1
CAS:
- 1429239-98-4
CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.
Formula:C₃₃H₃₁Cl₂F₃N₆O₃S₂
Purezza:99.08% - 99.76%
Colore e forma:Solid
Peso molecolare:751.67
Ref: TM-T5996
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A-836339
CAS:
- 959746-77-1
A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.
Formula:C₁₆H₂₆N₂O₂S
Purezza:99.94%
Colore e forma:Solid
Peso molecolare:310.45
Ref: TM-T7375
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AM251
CAS:
- 183232-66-8
AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).
Formula:C₂₂H₂₁Cl₂IN₄O
Purezza:97.43% - 98.79%
Colore e forma:A Crystalline Solid
Peso molecolare:555.24
Ref: TM-T1915
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PSB-SB-487
CAS:
- 1399049-81-0
PSB-SB-487 is antagonist of GPR55.
Formula:C₂₆H₃₂O₄
Purezza:98.53%
Colore e forma:Solid
Peso molecolare:408.53
Ref: TM-T8975