Recettore GNRH
I recettori dell'ormone di rilascio delle gonadotropine (GnRH) sono GPCR che si legano al GnRH, un ormone responsabile della regolazione del rilascio dell'ormone luteinizzante (LH) e dell'ormone follicolo-stimolante (FSH) dalla ghiandola pituitaria. Questi recettori sono cruciali per la funzione riproduttiva e sono bersagliati nelle terapie per condizioni come il cancro alla prostata, l'endometriosi e l'infertilità. Gli agonisti e gli antagonisti dei recettori del GnRH sono anche utilizzati nelle tecnologie di riproduzione assistita. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori del GnRH di alta qualità per supportare la tua ricerca in salute riproduttiva, endocrinologia e terapia ormonale.
Trovati 83 prodotti di "Recettore GNRH"
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Alarelin Acetate
CAS:Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.Formula:C56H78N16O12Purezza:99.81% - >99.99%Colore e forma:White PowderPeso molecolare:1167.34Degarelix acetate(214766-78-6 free base)
CAS:Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Formula:C84H107ClN18O18Purezza:98.66%Colore e forma:SolidPeso molecolare:1692.34(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Formula:C32H30F5N3O5Purezza:99.08%Colore e forma:SolidPeso molecolare:631.59Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Formula:C72H95ClN14O14Purezza:>99.99%Colore e forma:SolidPeso molecolare:1416.06[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide is a LHRH peptide analogue.Formula:C58H82N16O12Peso molecolare:1195.37Onvitrelin ucalontide
CAS:Onvitrelin ucalontide is a LHRH analogue with anticancer effect; halts breast, ovarian, and prostate tumors in mice.Formula:C163H243N43O32Peso molecolare:3316.94Kisspeptin-54(human)
CAS:Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.Formula:C258H401N79O78Purezza:98%Colore e forma:SolidPeso molecolare:5857.49AG 045572
CAS:AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 isFormula:C30H37NO5Purezza:99.96%Colore e forma:SolidPeso molecolare:491.62LHRH
CAS:Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and hasFormula:C55H74N16O14Purezza:98%Colore e forma:SolidPeso molecolare:1183.27LGnRH-III, lamprey
CAS:GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.Formula:C59H74N18O14Purezza:98%Colore e forma:SolidPeso molecolare:1259.33MI 1544
CAS:MI 1544 is a LHRH antagonist.Formula:C71H94ClN17O13Colore e forma:SolidPeso molecolare:1429.09Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS:LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.Formula:C60H73N15O13Purezza:98%Colore e forma:SolidPeso molecolare:1212.31Phoenixin-14
CAS:<p>Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/</p>Formula:C75H110N18O20Purezza:98%Colore e forma:SolidPeso molecolare:1583.78RS 18286
CAS:RS 18286 is a LHRH antagonist.Formula:C74H101Cl2N17O14Colore e forma:SolidPeso molecolare:1523.6LHRH, Ala(6)-
CAS:LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formula:C56H77N17O13Colore e forma:SolidPeso molecolare:1196.32Avorelin
CAS:Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.Formula:C65H85N17O12Purezza:98%Colore e forma:SolidPeso molecolare:1296.48(D-Trp6)-LHRH free acid
CAS:(D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .Formula:C64H81N17O14Peso molecolare:1312.43APTAA-LHRH
CAS:APTAA-LHRH is a gonadorelin antagonist.Formula:C69H91Cl2N17O14Purezza:98%Colore e forma:SolidPeso molecolare:1453.47Azaline
CAS:Azaline is a gonadorelin antagonist.Formula:C74H106ClN23O12Purezza:98%Colore e forma:SolidPeso molecolare:1545.26Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Formula:C27H28F3N3O8SPurezza:99.64%Colore e forma:SolidPeso molecolare:611.59LH-RH (4-10)
CAS:LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Formula:C33H53N11O9Peso molecolare:747.84Lamprey LH-RH I
CAS:Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Formula:C58H79N15O15Peso molecolare:1226.34(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS:(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Formula:C53H62N12O11Peso molecolare:1043.13Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).Formula:C44H80N14O15Peso molecolare:1044.59276Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Formula:C74H92ClN17O13Purezza:98%Colore e forma:SolidPeso molecolare:1463.08[D-Phe2,6, Pro3]-LH-RH
CAS:[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).Formula:C59H80N14O13Peso molecolare:1193.35Human follicular gonadotropin releasing peptide
CAS:Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH)Formula:C68H94N22O27Peso molecolare:1651.61Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Formula:C162H26N56O44SPeso molecolare:3724.17Prolactin Releasing Peptide (1-31), human
CAS:Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).Formula:C160H252N56O42SPurezza:98%Colore e forma:SolidPeso molecolare:3664.15Surfagon
CAS:Surfagon is an effective LHRH agonist.Formula:C56H78N16O12Purezza:98%Colore e forma:SolidPeso molecolare:1167.34[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:<p>[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.</p>Formula:C67H84N16O13Colore e forma:SolidPeso molecolare:1321.48[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Formula:C54H71N15O14Purezza:98%Colore e forma:SolidPeso molecolare:1154.23Fsh receptor-binding inhibitor fragment(bi-10)
CAS:<p>FSH antagonist bi-10 suppresses ovulation, induces follicular atresia, and may help in ovarian cancer by downregulating FSHR/ERβ.</p>Formula:C42H67N13O19Colore e forma:SolidPeso molecolare:1058.06Zebrafish Kisspeptin-1
CAS:<p>Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.</p>Formula:C58H84N16O15Colore e forma:SolidPeso molecolare:1245.39GnRH Associated Peptide (1-24), human
CAS:<p>GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.</p>Formula:C117H190N32O43Colore e forma:SolidPeso molecolare:2732.95LH-RH (7-10)
CAS:LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.Formula:C19H36N8O4Colore e forma:SolidPeso molecolare:440.54(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:<p>Analog of LHRH, stimulates LH and FSH release, controls reproduction.</p>Formula:C59H84N18O14Colore e forma:SolidPeso molecolare:1269.41Kisspeptin-54(human) TFA
Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.Formula:C258H401N79O78·C2HF3O2Colore e forma:SolidPeso molecolare:5971.45sGnRH-A
CAS:sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Formula:C64H83N17O12Colore e forma:SolidPeso molecolare:1282.45Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Formula:C75H110N18O20·xC2HF3O2Purezza:99.11%Colore e forma:SolidPeso molecolare:1583.78 (free base)Kisspeptin 13
CAS:<p>Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.</p>Formula:C78H107N21O18Colore e forma:SolidPeso molecolare:1626.81Azaline B
CAS:Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.Formula:C80H102ClN23O12Colore e forma:SolidPeso molecolare:1613.27A 76154
CAS:A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).Formula:C70H93FN12O12Colore e forma:SolidPeso molecolare:1313.584Wy 43657
CAS:Wy 43657 is a gonadorelin antagonist.Formula:C71H86N14O13Purezza:98%Colore e forma:SolidPeso molecolare:1343.554LUF5771
CAS:LUF5771: potent allosteric recLH & Org 43553 inhibitor, partial LH receptor activator with low efficacy.Formula:C24H23NO2Colore e forma:SolidPeso molecolare:357.44Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Formula:C59H84N16O12Colore e forma:SolidPeso molecolare:1209.4Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormula:C61H88N16O14Purezza:98.1%Colore e forma:SolidPeso molecolare:1269.45Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurezza:98.64% - 99.97%Colore e forma:SolidPeso molecolare:623.63Sufugolix
CAS:Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.Formula:C36H31F2N5O4SPurezza:97.78%Colore e forma:SolidPeso molecolare:667.72Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formula:C23H31FO5Purezza:99.47%Colore e forma:CoaPeso molecolare:406.49Fertirelin
CAS:Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).Formula:C55H76N16O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:1153.29Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formula:C74H100ClN17O18Purezza:98.38%Colore e forma:SolidPeso molecolare:1551.17Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormula:C82H117ClN18O15Purezza:96.05%Colore e forma:SolidPeso molecolare:1630.4LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretionFormula:C61H78N18O16Purezza:99.66%Colore e forma:SolidPeso molecolare:1319.38Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formula:C68H90N18O14Purezza:99.92%Colore e forma:SolidPeso molecolare:1383.55Deslorelin acetate(57773-65-6 free base)
<p>Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)</p>Formula:C66H87N17O14Purezza:99.84%Colore e forma:SolidPeso molecolare:1342.5Buserelin Acetate (57982-77-1 free base)
CAS:<p>Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).</p>Formula:C62H90N16O15Purezza:99.31% - 99.78%Colore e forma:SolidPeso molecolare:1299.48Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formula:C66H86N18O15Purezza:99.90%Colore e forma:White PowderPeso molecolare:1371.53Elagolix sodium
CAS:<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Formula:C32H29F5N3NaO5Purezza:99.71%Colore e forma:SolidPeso molecolare:653.57Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purezza:99.98%Colore e forma:SolidPeso molecolare:1382.55Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurezza:99.33%Colore e forma:SolidPeso molecolare:508.42Goserelin acetate
CAS:<p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>Formula:C61H88N18O16Purezza:99.77% - >99.99%Colore e forma:White Crystalline PowderPeso molecolare:1329.46Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Formula:C55H74N16O13Colore e forma:SolidPeso molecolare:1167.29Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Formula:C80H104ClN21O14Colore e forma:SolidPeso molecolare:1619.27NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Formula:C27H24F3N3O3Colore e forma:SolidPeso molecolare:495.49BAY 1214784
CAS:BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.Formula:C29H26ClF4N3O5S2Colore e forma:SolidPeso molecolare:672.11Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Formula:C70H92ClN17O14·xC2H4O2Purezza:97.96%Colore e forma:SolidPeso molecolare:1491.11Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurezza:98.60% - 98.97%Colore e forma:SolidPeso molecolare:544.5[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Formula:C56H77N17O13Colore e forma:SolidPeso molecolare:1196.325α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFormula:C21H36O2Colore e forma:SolidPeso molecolare:320.51BAY-784
CAS:<p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>Formula:C29H26ClF4N3O5S2Purezza:98%Colore e forma:SolidPeso molecolare:672.11T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFormula:C37H37F2N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:657.77BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Formula:C27H21ClFN3O2Purezza:98%Colore e forma:SolidPeso molecolare:473.93DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Formula:C11H17Cl2NOSColore e forma:SolidPeso molecolare:282.22Abarelix acetate
CAS:Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formula:C72H95ClN14O14·xC2H4O2Colore e forma:SolidPeso molecolare:1476.14BAY-899
CAS:BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.Formula:C25H19F2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:459.45(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Formula:C25H19F2N5O2Colore e forma:SolidPeso molecolare:459.45GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Formula:C31H28F5N7O6SPurezza:98%Colore e forma:SolidPeso molecolare:721.65GnRH antagonist 2
CAS:<p>GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.</p>Formula:C28H27F2N9O5Purezza:98.08%Colore e forma:SolidPeso molecolare:607.57Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Formula:C80H102ClN15O14Colore e forma:SolidPeso molecolare:1533.21Merigolix
CAS:Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Formula:C36H35F7N4O6Colore e forma:SolidPeso molecolare:752.68Goserelin acetate(65807-02-5 Free base)
<p>Goserelin acetate （ICI-118630 acetate） is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.</p>Purezza:99.77%Colore e forma:Odour SolidDimethandrolone Undecanoate
CAS:Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.Formula:C31H50O3Purezza:99.65% - >99.99%Colore e forma:SolidPeso molecolare:470.73Ref: TM-T27176
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