Recettore GNRH
I recettori dell'ormone di rilascio delle gonadotropine (GnRH) sono GPCR che si legano al GnRH, un ormone responsabile della regolazione del rilascio dell'ormone luteinizzante (LH) e dell'ormone follicolo-stimolante (FSH) dalla ghiandola pituitaria. Questi recettori sono cruciali per la funzione riproduttiva e sono bersagliati nelle terapie per condizioni come il cancro alla prostata, l'endometriosi e l'infertilità. Gli agonisti e gli antagonisti dei recettori del GnRH sono anche utilizzati nelle tecnologie di riproduzione assistita. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori del GnRH di alta qualità per supportare la tua ricerca in salute riproduttiva, endocrinologia e terapia ormonale.
Trovati 86 prodotti per "Recettore GNRH".
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Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormula:C61H88N16O14Purezza:99.74%Colore e forma:SolidPeso molecolare:1269.45Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurezza:98.64% - 99.97%Colore e forma:White SolidPeso molecolare:623.63Ref: TM-T3630
2mg39,00€5mg58,00€1mL*10mM (DMSO)81,00€10mg93,00€25mg167,00€50mg250,00€100mg408,00€200mg585,00€Sufugolix
CAS:Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.Formula:C36H31F2N5O4SPurezza:97.78%Colore e forma:SolidPeso molecolare:667.72Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formula:C23H31FO5Purezza:99.47%Colore e forma:SolidPeso molecolare:406.49Fertirelin
CAS:Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).Formula:C55H76N16O12Purezza:>99.99%Colore e forma:White SolidPeso molecolare:1153.29Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formula:C74H100ClN17O18Purezza:98.38%Colore e forma:White SolidPeso molecolare:1551.17Ref: TM-T5520L
1mg50,00€5mg95,00€10mg142,00€1mL*10mM (DMSO)239,00€25mg276,00€50mg414,00€100mg608,00€500mg1.288,00€Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormula:C82H117ClN18O15Purezza:96.05%Colore e forma:SolidPeso molecolare:1630.4LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretionFormula:C61H78N18O16Purezza:96.65%Colore e forma:SolidPeso molecolare:1319.38Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formula:C68H90N18O14Purezza:99.92%Colore e forma:SolidPeso molecolare:1383.55Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)Formula:C66H87N17O14Purezza:99.96%Colore e forma:White SolidPeso molecolare:1342.5Buserelin Acetate (57982-77-1 free base)
CAS:Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).Formula:C62H90N16O15Purezza:98.37% - 99.78%Colore e forma:White SolidPeso molecolare:1299.48Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formula:C66H86N18O15Purezza:99.59% - 99.90%Colore e forma:White SolidPeso molecolare:1371.53Ref: TM-T21410
5mg52,00€10mg78,00€1mL*10mM (DMSO)116,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formula:C32H29F5N3NaO5Purezza:99.71%Colore e forma:White SolidPeso molecolare:653.57Ref: TM-T5031
2mg34,00€5mg50,00€1mL*10mM (DMSO)71,00€10mg75,00€25mg137,00€50mg215,00€100mg340,00€200mg504,00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purezza:99.98%Colore e forma:SolidPeso molecolare:1382.55Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurezza:99.33% - 99.95%Colore e forma:White SolidPeso molecolare:508.42Goserelin acetate
CAS:Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.Formula:C61H88N18O16Purezza:99.77% - >99.99%Colore e forma:SolidPeso molecolare:1329.46EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Formula:C15H27N5O6Colore e forma:SolidPeso molecolare:373.4Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Formula:C55H74N16O13Colore e forma:SolidPeso molecolare:1167.29Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Formula:C70H92ClN17O14·xC2H4O2Purezza:99.97%Colore e forma:SolidPeso molecolare:1491.11Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Formula:C80H104ClN21O14Colore e forma:SolidPeso molecolare:1619.27BAY 1214784
CAS:BAY 1214784 is a selective and orally active human GnRH-R antagonist, which can effectively reduce plasma luteinizing hormone levels by up to 49%.Formula:C29H26ClF4N3O5S2Purezza:100% - 99.77%Colore e forma:White SolidPeso molecolare:672.11NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Formula:C27H24F3N3O3Colore e forma:SolidPeso molecolare:495.49Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurezza:98.60% - 99.77%Colore e forma:SolidPeso molecolare:544.55α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFormula:C21H36O2Colore e forma:SolidPeso molecolare:320.51DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Formula:C11H17Cl2NOSColore e forma:SolidPeso molecolare:282.22BAY-784
CAS:BAY-784 is a potent GnRH receptor antagonist with nanomolar activity in human and rat receptors, widely used in endocrine and reproductive research.Formula:C29H26ClF4N3O5S2Purezza:99.22% - 99.75%Colore e forma:White SolidPeso molecolare:672.11BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Formula:C27H21ClFN3O2Purezza:98%Colore e forma:SolidPeso molecolare:473.93T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFormula:C37H37F2N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:657.77[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Formula:C56H77N17O13Colore e forma:SolidPeso molecolare:1196.32Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Formula:C80H102ClN15O14Colore e forma:SolidPeso molecolare:1533.21Merigolix
CAS:Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Formula:C36H35F7N4O6Colore e forma:SolidPeso molecolare:752.68(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Formula:C25H19F2N5O2Colore e forma:SolidPeso molecolare:459.45BAY-899
CAS:BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.Formula:C25H19F2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:459.45Abarelix acetate
CAS:Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formula:C72H95ClN14O14·xC2H4O2Colore e forma:SolidPeso molecolare:1476.14GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Formula:C28H27F2N9O5Purezza:98.08%Colore e forma:SolidPeso molecolare:607.57GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Formula:C31H28F5N7O6SPurezza:98%Colore e forma:SolidPeso molecolare:721.65
