Proteasi HIV
Gli inibitori della proteasi dell'HIV sono una classe di farmaci antiretrovirali che bersagliano specificamente l'enzima proteasi del virus dell'immunodeficienza umana (HIV). Inibendo questo enzima, questi composti impediscono al virus di elaborare le sue poliproteine in proteine mature e funzionali, bloccando così la produzione di nuovi virioni infettivi. Gli inibitori della proteasi dell'HIV sono una pietra miliare della terapia antiretrovirale altamente attiva (HAART) utilizzata per gestire l'HIV/AIDS. Presso CymitQuimica, offriamo una varietà di inibitori della proteasi dell'HIV per supportare la vostra ricerca nel trattamento dell'HIV, nella resistenza ai farmaci e nella virologia.
Trovati 506 prodotti di "Proteasi HIV"
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Temsavir
CAS:Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.Formula:C24H23N7O4Purezza:99.14%Colore e forma:SolidPeso molecolare:473.48Ref: TM-T4665
2mg42,00€5mg64,00€10mg97,00€25mg170,00€50mg293,00€100mg434,00€200mg610,00€1mL*10mM (DMSO)64,00€Doravirine
CAS:Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.Formula:C17H11ClF3N5O3Purezza:99.65% - 99.79%Colore e forma:SolidPeso molecolare:425.75Ref: TM-T3632
1mg49,00€2mg69,00€5mg97,00€10mg170,00€25mg335,00€50mg520,00€100mg750,00€500mg1.549,00€1mL*10mM (DMSO)131,00€Delavirdine mesylate
CAS:Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI).Formula:C23H32N6O6S2Purezza:99.99%Colore e forma:Light Brown SolidPeso molecolare:552.67Fostemsavir
CAS:Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.Formula:C25H26N7O8PPurezza:98.95%Colore e forma:SolidPeso molecolare:583.49Ref: TM-T3523
1mg59,00€5mg120,00€10mg170,00€25mg283,00€50mg432,00€100mg622,00€200mg873,00€1mL*10mM (DMSO)156,00€Raltegravir
CAS:<p>Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIV</p>Formula:C20H21FN6O5Purezza:99.86% - >99.99%Colore e forma:SolidPeso molecolare:444.42Bictegravir
CAS:Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).Formula:C21H18F3N3O5Purezza:97.6% - 99.51%Colore e forma:SolidPeso molecolare:449.38Ref: TM-T4493
1mg35,00€5mg66,00€10mg96,00€25mg185,00€50mg311,00€100mg469,00€200mg682,00€1mL*10mM (DMSO)66,00€Dolutegravir sodium
CAS:<p>Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature</p>Formula:C20H18F2N3NaO5Purezza:98% - 99.46%Colore e forma:SolidPeso molecolare:441.36I-XW-053 sodium
CAS:I-XW-053 sodium inhibits the replication of a diverse panel of primary HIV-1 isolates in Peripheral blood mononuclear cell with no appreciable cytotoxicity.Formula:C22H16N2NaO2Colore e forma:SolidPeso molecolare:363.372PTACH
CAS:PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).Formula:C20H26N2O2S2Purezza:87.44% - 99.74%Colore e forma:SolidPeso molecolare:390.56Darunavir Ethanolate
CAS:Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Formula:C29H43N3O8SPurezza:99.84% - 99.86%Colore e forma:SolidPeso molecolare:593.74Ref: TM-T3335
5mg37,00€10mg52,00€25mg80,00€50mg111,00€100mg165,00€200mg236,00€500mg399,00€1mL*10mM (DMSO)48,00€Thiamine disulfide
CAS:Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.Formula:C24H34N8O4S2Purezza:99.81% - 99.81%Colore e forma:CoaPeso molecolare:562.71Inosine pranobex
CAS:Inosine pranobex (Delimmun) has a lot of immunomodulatory effects, including inducing T-lymphocyte differentiation, augmenting macrophage and NK cell functions.Formula:C52H78N10O17Purezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:1115.23Peptide T acetate(106362-32-7 free base)
Peptide T acetate is an octapeptide from the V2 region of HIV-1 gp120.Formula:C37H59N9O18Purezza:99.47%Colore e forma:SolidPeso molecolare:917.91Indinavir sulfate
CAS:<p>Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.</p>Formula:C36H49N5O8SPurezza:99.75% - >99.99%Colore e forma:White PowderPeso molecolare:711.87Darunavir
CAS:Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Formula:C27H37N3O7SPurezza:99.67% - 99.76%Colore e forma:White Amorphous SolidPeso molecolare:547.66Peldesine dihydrochloride
CAS:Peldesine (BCX 34) dihydrochloride is an inhibitor of PNP in humans, rats, and mice, also hindering T-cell proliferation, used in lymphoma and HIV research.Formula:C12H13Cl2N5OColore e forma:SolidPeso molecolare:314.17HIV-1 Nef-IN-1
CAS:HIV-1 Nef-IN-1 is an inhibitor of HIV-1 Nef protein. It efficiently competes for Nef-SH3Hck interactions(Kd : 6.7 μM).Formula:C18H16O2Purezza:99.90%Colore e forma:SolidPeso molecolare:264.32Fosamprenavir sodium
CAS:Fosamprenavir sodium is an HIV protease inhibitor that is the water soluble prodrug of amprenavir.Formula:C25H34N3Na2O9PSColore e forma:SolidPeso molecolare:629.57HODHBt
CAS:HODHBt is a STAT5-SUMO protein-protein interaction inhibitor.Formula:C7H5N3O2Purezza:99.45% - 99.95%Colore e forma:Off-White To Yellow SolidPeso molecolare:163.13BMS-707035
CAS:BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.Formula:C17H19FN4O5SPurezza:99.78%Colore e forma:SolidPeso molecolare:410.42Cobicistat
CAS:Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.Formula:C40H53N7O5S2Purezza:97.36% - 99.62%Colore e forma:SolidPeso molecolare:776.02Ref: TM-T6246
1mg46,00€2mg59,00€5mg93,00€10mg124,00€25mg212,00€50mg350,00€100mg505,00€1mL*10mM (DMSO)111,00€Dolutegravir
CAS:<p>Dolutegravir (GSK1349572), HIV integrase inhibitor with IC50 of 2.7 nM, partly effective against some raltegravir-resistant HIV strains.</p>Formula:C20H19F2N3O5Purezza:98.97% - 99.75%Colore e forma:White To Pale Yellow SolidPeso molecolare:419.38Saquinavir
CAS:<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Formula:C38H50N6O5Purezza:99.50% - >99.99%Colore e forma:SolidPeso molecolare:670.84TAT
CAS:<p>TAT peptide (YGRKKRRQRRR), originating from the human immunodeficiency virus-1 (HIV-1) transactivator of transcription (TAT), enhances the solubility and</p>Formula:C64H118N32O14Purezza:>99.99%Colore e forma:SolidPeso molecolare:1559.83HIV-1 Inhibitor 18A
CAS:HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.Formula:C14H11N5O2SPurezza:99.79%Colore e forma:SolidPeso molecolare:313.33Ref: TM-T24141
1mg115,00€5mg227,00€10mg313,00€25mg535,00€50mg752,00€100mg1.064,00€1mL*10mM (DMSO)217,00€Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Formula:C20H20FN6O5·KPurezza:98% - 99.55%Colore e forma:Off-White SolidPeso molecolare:482.51Dexelvucitabine
CAS:Dexelvucitabine (RVT), a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.Formula:C9H10FN3O3Purezza:98.25%Colore e forma:SolidPeso molecolare:227.19Nelfinavir Mesylate
CAS:Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM).Formula:C33H49N3O7S2Purezza:95.81% - 99.97%Colore e forma:A White Or Almost White PowderPeso molecolare:663.89LDC4297 hydrochloride
CAS:LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Formula:C23H29ClN8OColore e forma:SolidPeso molecolare:468.982,4-Dihydroxypyridine
CAS:2,4-Dihydroxypyridine: a pyridine derivative, chelates metals, assesses ion levels, measures enzymatic reactions, and quantifies biomolecules.Formula:C5H5NO2Purezza:97.79%Colore e forma:White To Yellow-Beige Crystals OrPeso molecolare:111.1lavendustin B
CAS:Lavendustin B inhibits Tyrosine Kinase and HIV-1 integrase-LEDGF/p75 interaction.Formula:C21H19NO5Purezza:95.72%Colore e forma:Off-White SolidPeso molecolare:365.38Ref: TM-T4182
1mg42,00€5mg88,00€10mg134,00€25mg283,00€50mg419,00€100mg607,00€200mg1.206,00€1mL*10mM (DMSO)87,00€Rolipram
CAS:Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.Formula:C16H21NO3Purezza:99.22% - >99.99%Colore e forma:SolidPeso molecolare:275.34PMEDAP
CAS:PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiencyFormula:C8H13N6O4PPurezza:99.77%Colore e forma:SolidPeso molecolare:288.2RN-18
CAS:RN-18 is an inhibitor of HIV-1 viral infectivity factor (IC50: 6 μM in nonpermissive H9 cells).Formula:C20H16N2O4SPurezza:97.21% - 98.39%Colore e forma:SolidPeso molecolare:380.42Tenofovir alafenamide
CAS:Tenofovir alafenamide (GS-7340) is a nucleotide reverse transcriptase inhibitor (NRTI) and a novel ester prodrug of the antiretroviral tenofovir.Formula:C21H29N6O5PPurezza:99.68% - 99.81%Colore e forma:SolidPeso molecolare:476.47Obefazimod
CAS:<p>Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).</p>Formula:C16H10ClF3N2OPurezza:99.86%Colore e forma:SolidPeso molecolare:338.71Ref: TM-T8311
2mg39,00€5mg62,00€10mg87,00€25mg187,00€50mg301,00€100mg437,00€200mg617,00€1mL*10mM (DMSO)65,00€IMB-301
CAS:IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.Formula:C19H17Cl2FN2OPurezza:99.72%Colore e forma:SolidPeso molecolare:379.26Ref: TM-T9212
1mg48,00€5mg97,00€10mg156,00€25mg259,00€50mg369,00€100mg530,00€200mg720,00€1mL*10mM (DMSO)105,00€Filgotinib
CAS:Filgotinib (GLPG0634) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and TYK2 are 10 nM, 28 nM, 810 nM, and 116 nM, respectively.Formula:C21H23N5O3SPurezza:98.03% - ≥95%Colore e forma:SolidPeso molecolare:425.5Filgotinib maleate
CAS:Filgotinib maleate, a selective oral JAK1 inhibitor, treats RA and Crohn's. IC50s: JAK1-10nM, JAK2-28nM, JAK3-810nM, TYK2-116nM.Formula:C25H27N5O7SColore e forma:SolidPeso molecolare:541.58Dimercaprol
CAS:Dimercaprol (Dicaptol) is an anti-gas warfare agent that is effective against Lewisite (dichloro(2-chlorovinyl)arsine) and formerly known as British Anti-Formula:C3H8OS2Purezza:98.91% - 99.64%Colore e forma:Viscous Oily LiquidPeso molecolare:124.22Etravirine
CAS:Etravirine (R165335) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.Formula:C20H15BrN6OPurezza:97.61% - 99.74%Colore e forma:White To Off-White SolidPeso molecolare:435.28Ref: TM-T2551
2mg35,00€5mg52,00€10mg80,00€25mg149,00€50mg216,00€100mg329,00€200mg485,00€1mL*10mM (DMSO)52,00€Lamivudine 13C,15N2
CAS:Lamivudine 13C,15N2, a BCH-189 impurity, blocks HIV/HBV reverse transcriptase as an NRTI.Formula:C8H9N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:246.22Nelfinavir
CAS:Nelfinavir (AG1341), with Ki=2 nM, is an HIV treatment and broad-spectrum anticancer drug.Formula:C32H45N3O4SPurezza:98.16% - 99.5%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:567.78Suvizumab
CAS:Suvizumab (KD-247) is a neutralizing anti-HIV-1 antibody with IC50 values of 0.1-1.0 µg/mL; it lowers viral load and prevents infection.Colore e forma:LiquidElipovimab
CAS:Elipovimab, a potent and broadly neutralizing antibody against HIV-1, targets and eliminates HIV-infected cells [1].Colore e forma:LiquidSemzuvolimab
CAS:Semzuvolimab, a murine IgG1κ antibody, targets the p55 T-cell surface antigen T4/Leu-3 (CD4).Colore e forma:LiquidNevirapine-d3
CAS:Nevirapine-d3 is a deuterated compound of Nevirapine. Nevirapine has a CAS number of 129618-40-2. Nevirapine is a benzodiazepine non-nucleoside reverse transcriptase inhibitor. In combination with other antiretroviral drugs, nevirapine reduces HIV viral loads and increases CD4 counts, thereby retarding or preventing the damage to the immune system and reducing the risk of developing AIDS.Formula:C15H11D3N4OPeso molecolare:269.32Benzalphthalide
CAS:Benzalphthalide (NSC-2824) is a chemical compound with anti-HIV activity.Formula:C15H10O2Purezza:99.94%Colore e forma:Pale Yellow To Yellow Crystalline PowderPeso molecolare:222.24Nipamovir
CAS:<p>Nipamovir is a nitroimidazole prodrug that exhibits antiviral activity comparable to SAMT-247 and NS-1040 in cellular assays and a human ex vivo model of HIV infection, with low toxicity. Nipamovir has EC50 values of 3.64±3.28 and 3.23±2.81 μM for CEM-SS/HIV-1RF and hPBMC/HIV-192HT599, respectively [1].</p>Formula:C14H15N5O4SColore e forma:SolidPeso molecolare:349.37Antiviral agent 55
CAS:Antiviralagent 55 (Compound 95) is an inhibitor of human immunodeficiency viruses 1 and 2 (HIV1 and HIV2), demonstrating antiviral activity.Formula:C21H20N2O4Colore e forma:SolidPeso molecolare:364.39
