Proteasi HIV
Gli inibitori della proteasi dell'HIV sono una classe di farmaci antiretrovirali che bersagliano specificamente l'enzima proteasi del virus dell'immunodeficienza umana (HIV). Inibendo questo enzima, questi composti impediscono al virus di elaborare le sue poliproteine in proteine mature e funzionali, bloccando così la produzione di nuovi virioni infettivi. Gli inibitori della proteasi dell'HIV sono una pietra miliare della terapia antiretrovirale altamente attiva (HAART) utilizzata per gestire l'HIV/AIDS. Presso CymitQuimica, offriamo una varietà di inibitori della proteasi dell'HIV per supportare la vostra ricerca nel trattamento dell'HIV, nella resistenza ai farmaci e nella virologia.
Trovati 506 prodotti di "Proteasi HIV"
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Benzalphthalide
CAS:Benzalphthalide (NSC-2824) is a chemical compound with anti-HIV activity.Formula:C15H10O2Purezza:99.94%Colore e forma:Pale Yellow To Yellow Crystalline PowderPeso molecolare:222.24Nipamovir
CAS:<p>Nipamovir is a nitroimidazole prodrug that exhibits antiviral activity comparable to SAMT-247 and NS-1040 in cellular assays and a human ex vivo model of HIV infection, with low toxicity. Nipamovir has EC50 values of 3.64±3.28 and 3.23±2.81 μM for CEM-SS/HIV-1RF and hPBMC/HIV-192HT599, respectively [1].</p>Formula:C14H15N5O4SColore e forma:SolidPeso molecolare:349.37Antiviral agent 55
CAS:Antiviralagent 55 (Compound 95) is an inhibitor of human immunodeficiency viruses 1 and 2 (HIV1 and HIV2), demonstrating antiviral activity.Formula:C21H20N2O4Colore e forma:SolidPeso molecolare:364.39A3N19
CAS:A3N19 is a potent inhibitor of HIV-1 non-nucleoside reverse transcriptase and is able to act on HIV-1 IIIB (EC50: 3.28 nM).Formula:C31H31N9O2SColore e forma:SolidPeso molecolare:593.7HIV-1 inhibitor-23
CAS:HIV-1 inhibitor-23 suppresses HIV reverse transcriptase, effective on wild-type (EC50: 24.9 nM) and K103N mutant (EC50: 10.4 nM), with in vitro stability.Formula:C30H26N6O4SColore e forma:SolidPeso molecolare:566.63R 82150
CAS:R 82150 is an antiviral and a member of the tetrahydroimidazo[4,5,1-jk]-[1,4]-benzodiazepin-2(1H)-thione family.Formula:C16H21N3SPurezza:98%Colore e forma:SolidPeso molecolare:287.42Fostemsavir disodium
CAS:Fostemsavir disodium is an HIV-1 attachment inhibitor and prodrug of the small-molecule inhibitor BMS-626529.Formula:C25H24N7Na2O8PColore e forma:SolidPeso molecolare:627.45Docosylferulate
CAS:Docosylferulate is a biochemical that has been studied for its inhibition on Hep G2 cells and anti-tumor activities.Formula:C32H54O4Colore e forma:SolidPeso molecolare:502.77DLC27-14
CAS:DLC27-14 is an HIV-1 Nef specific protein disorder catalyzer.Formula:C25H25NO4Colore e forma:SolidPeso molecolare:403.47BMS-509744
CAS:BMS-509744 is a selective, ATP-competitive Itk inhibitor, IC50 of 19 nM. It inhibits IL-8 expression and HIV infection, ameliorates pulmonary inflammation.Formula:C32H41N5O4S2Purezza:99.70%Colore e forma:SolidPeso molecolare:623.83Ref: TM-T14674
1mg48,00€2mg63,00€5mg92,00€10mgPrezzo su richiesta25mg354,00€50mg628,00€100mg1.008,00€200mg1.359,00€1mL*10mM (DMSO)127,00€HIV-1 inhibitor-32
CAS:HIV-1 inhibitor-32 is a potent inhibitor of HIV-1 that acts on wild-type HIV (IC50: 34 nM) and can be used in AIDS research.Formula:C26H29N5O3SColore e forma:SolidPeso molecolare:491.61HIV-1 protease-IN-2
CAS:HIV-1 protease-IN-2: strong HIV-1 protease blocker, IC50 2.53 nM, fights DRV-sensitive/resistant HIV-1.Formula:C27H34N4O7SColore e forma:SolidPeso molecolare:558.65HIV-1 inhibitor-46
CAS:HIV-1 inhibitor-46, compound 13d, is a potent non-nucleoside reverse transcriptase inhibitor with an EC50 of 1.425 μM, useful in AIDS research.Formula:C24H21ClN4OSColore e forma:SolidPeso molecolare:448.97HIV-1 inhibitor-37
CAS:HIV-1 inhibitor-37, a potent HIV-1 suppressant, shows promise as a novel latent reactivator.Formula:C14H11Cl3N4OColore e forma:SolidPeso molecolare:357.62Complestatin
CAS:"Complestatin, from Streptomyces lavendulae, yields hydroxyphenylglycines & a chromophore; blocks HIV-1 gp120-CD4 binding; antimicrobial."Formula:C61H45Cl6N7O15Colore e forma:SolidPeso molecolare:1328.77Tenofovir maleate
CAS:Tenofovir Disoproxil Fumarate is a nucleotide reverse transcriptase inhibitor used in the treatment of HIV and chronic Hepatitis B.Formula:C13H18N5O8PColore e forma:SolidPeso molecolare:403.28Nevirapine quinone methide
CAS:Nevirapine quinone methide is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used to treat HIV-1 infection and AIDS.Formula:C15H12N4OColore e forma:SolidPeso molecolare:264.28Stampidine
CAS:Stampidine prevents HIV-1, effective against resistant strains at subnanomolar levels.Formula:C20H23BrN3O8PPurezza:98%Colore e forma:SolidPeso molecolare:544.29HIV-1 inhibitor-30
CAS:HIV-1 inhibitor-30 (10i) targets RT enzyme, EC50=40nM, IC50=80nM. Effective against seven NNRTI-resistant HIV-1 strains.Formula:C19H20ClN3O2Colore e forma:SolidPeso molecolare:357.83Edelfosine
CAS:inhibits phosphatidylinositol phospholipase CFormula:C27H58NO6PPurezza:98%Colore e forma:SolidPeso molecolare:523.73(+)-Dihydrocalanolide A
CAS:DHCal A (NSC 678323) is an oral nonnucleoside Reverse Transcriptase inhibitor for HIV research.Formula:C22H28O5Colore e forma:SolidPeso molecolare:372.45HIV-IN-5
CAS:HIV-IN-5 (5r) inhibits HIV-1 with 0.16 μM IC50, targeting NNIBP as a NNRTI.Formula:C30H24N2O8SColore e forma:SolidPeso molecolare:572.59HIV-1 inhibitor-47
CAS:HIV-1 Inhibitor-47 blocks Vif-APOBEC3G interaction, has 14.33 μM IC50, and may yield antianxiety and antipsychotic derivatives.Formula:C12H14N6Colore e forma:SolidPeso molecolare:242.28L 870810
CAS:L 870810 is a small-molecule inhibitor of HIV-1 integrase with potent antiviral activity in cell culture and good pharmacokinetic properties.Formula:C20H19FN4O4SColore e forma:SolidPeso molecolare:430.45Isoescin IA
CAS:Isoescin IA is a triterpenoid saponin isolated from the seeds of Aesculus chinensis. It has anti-HIV-1 protease activity.Formula:C55H86O24Purezza:96.00%Colore e forma:SolidPeso molecolare:1131.26HIV-1 protease-IN-5
CAS:HIV-1 protease-IN-5 is an HIV-1 protease inhibitor (IC50: 1.64 nM). HIV-1 protease-IN-5 exhibits significant effects on wild-type and DRV-resistant HIV-1.Formula:C27H29F3N2O7SColore e forma:SolidPeso molecolare:582.59DPC-963
CAS:DPC-963 is a RNA-directed DNA polymerase inhibitor.Formula:C14H9F5N2OColore e forma:SolidPeso molecolare:316.23Brecanavir
CAS:Brecanavir is a tyrosyl-based arylsulfonamide, high affinity, protease inhibitor (PI) for the treatment of human immunodeficiency virus type 1.Formula:C33H41N3O10S2Colore e forma:SolidPeso molecolare:703.82ZINC04177596
CAS:ZINC04177596 is a novel Nef Protein Inhibitor with anti-HIV activity.Formula:C22H16N6O4Colore e forma:SolidPeso molecolare:428.4APA-H-MPO
CAS:APA-H-MPO is a PCAF bromodomain/Tat-AcK50 association inhibitor.Formula:C9H16ClN3O2Colore e forma:SolidPeso molecolare:233.7HIV-1 inhibitor-42
CAS:HIV-1 inhibitor-42 (5b) strongly blocks HIV-1 (IC50: 0.06μM) and its RT RNA/DNA polymerases (IC50: 0.518/0.072μM).Formula:C22H20N2O5SColore e forma:SolidPeso molecolare:424.47EP39
EP39 is a potent HIV-1 inhibitor, stabilizing the SP1 domain's helix and blocking virus maturation.Formula:C38H62N2O5Colore e forma:SolidPeso molecolare:626.91SJ-3366
CAS:SJ3366 is a unique and highly potent nonnucleoside reverse transcriptase human immunodeficiency virus type 1 and HIV-2 inhibitor.Formula:C21H24N2O3Colore e forma:SolidPeso molecolare:352.43HIV-1 protease-IN-1
CAS:HIV-1 protease-IN-1, potent HIV inhibitor; IC50=90pM, fights B/C-HIV strains with EC50=89-13.59/8.23nM.Formula:C25H35N3O6SColore e forma:SolidPeso molecolare:505.63VEC-5
CAS:VEC-5: an HIV-1 inhibitor, outperforms RN18 by better binding with Vif in studies.Formula:C29H21NO4Purezza:98%Colore e forma:SolidPeso molecolare:447.48HIV-1 inhibitor-38
CAS:HIV-1 inhibitor-38, or Compound 91, shows promise as a strong latency reversing agent against HIV-1.Formula:C15H13Cl3N6Colore e forma:SolidPeso molecolare:383.66ZINC36617540
CAS:ZINC36617540 is a novel Nef Protein Inhibitor with anti-HIV activity.Formula:C21H17N5OColore e forma:SolidPeso molecolare:355.39GSK-364735 sodium
CAS:GSK-364735 sodium is an HIV-1 IN inhibitor.Formula:C19H17FN3NaO4Colore e forma:SolidPeso molecolare:393.34DMJ-I-228
CAS:DMJ-I-228 is a specific inhibitor of HIV-1 entry through interaction with the Env spike by virtue of the incorporation of a guandinium group.Formula:C19H19ClFN5O4Colore e forma:SolidPeso molecolare:435.84BMS 378806
CAS:BMS-378806 is an orally bioavailable HIV-1 inhibitor that interferes with gp120-CD4 interaction.Formula:C22H22N4O4Colore e forma:SolidPeso molecolare:406.43gp120-IN-2
CAS:gp120-IN-2 is a potent HIV-1 inhibitor (IC50 = 7.5 μM) with low cytotoxicity (CC50 = 112.93 μM).Formula:C15H18N2O5Colore e forma:SolidPeso molecolare:306.31A 80987
CAS:A 80987 is an inhibitor of HIV-1 protease.Formula:C37H43N5O6Colore e forma:SolidPeso molecolare:653.77GW-695634
CAS:<p>GW-695634, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Formula:C26H21Cl2N3O6SColore e forma:SolidPeso molecolare:574.43HIV-1 inhibitor-31
CAS:HIV-1 inhibitor-31 (compound 4) is a potent inhibitor of HIV-1. HIV-1 inhibitor-31 can be used in the study of AIDS.Formula:C21H13Cl2N3O2Colore e forma:SolidPeso molecolare:410.25Deaminase inhibitor-1
CAS:Deaminase inhibitor-1 is an APOBEC3G DNA Deaminase inhibitor with an IC 50 value of 18.9 μM [1].Formula:C11H12BrN3OSColore e forma:SolidPeso molecolare:314.2HIV-1 inhibitor-50
CAS:HIV-1 inhibitor-50 is a non-nucleoside reverse transcriptase inhibitor (NNRTI) that targets HIV-1 reverse transcriptase (IC50 = 50 nM).Formula:C24H18FN5O2Colore e forma:SolidPeso molecolare:427.43S-1360
CAS:S-1360 is an inhibitor of HIV-1 integrase.Formula:C16H12FN3O3Purezza:98%Colore e forma:SolidPeso molecolare:313.28PF-46396
CAS:PF-46396 is a HIV maturation inhibitor and can be used against HIV-1 clade B and C.Formula:C27H29F3N2OColore e forma:SolidPeso molecolare:454.53Tenofovir diphosphate
CAS:TFV-DP inhibits DNA polymerases, mimics dATP, and is used by HIV-1's reverse transcriptase.Formula:C9H16N5O10P3Colore e forma:SolidPeso molecolare:447.17HIV-1 inhibitor-39
CAS:HIV-1 inhibitor-39: blocks HIV-1, anti-RT (IC50=15.75 μM), toxic to MT-4 cells (CC50=112.9 μM).Formula:C20H17ClN4O4S4Colore e forma:SolidPeso molecolare:541.09
