
Proteasi HIV
Gli inibitori della proteasi dell'HIV sono una classe di farmaci antiretrovirali che bersagliano specificamente l'enzima proteasi del virus dell'immunodeficienza umana (HIV). Inibendo questo enzima, questi composti impediscono al virus di elaborare le sue poliproteine in proteine mature e funzionali, bloccando così la produzione di nuovi virioni infettivi. Gli inibitori della proteasi dell'HIV sono una pietra miliare della terapia antiretrovirale altamente attiva (HAART) utilizzata per gestire l'HIV/AIDS. Presso CymitQuimica, offriamo una varietà di inibitori della proteasi dell'HIV per supportare la vostra ricerca nel trattamento dell'HIV, nella resistenza ai farmaci e nella virologia.
Trovati 502 prodotti di "Proteasi HIV"
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Thiamine disulfide
CAS:Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.Formula:C24H34N8O4S2Purezza:99.81% - 99.81%Colore e forma:CoaPeso molecolare:562.71Inosine pranobex
CAS:Inosine pranobex (Delimmun) has a lot of immunomodulatory effects, including inducing T-lymphocyte differentiation, augmenting macrophage and NK cell functions.Formula:C52H78N10O17Purezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:1115.23Indinavir sulfate
CAS:<p>Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.</p>Formula:C36H49N5O8SPurezza:99.75% - >99.99%Colore e forma:White PowderPeso molecolare:711.87Ganoderic acid B
CAS:Ganoderic acid B: quality marker for G. lucidum products, inhibits telomerase & EBV activation, moderates HIV-1 protease.Formula:C30H44O7Purezza:99.09% - 99.97%Colore e forma:SolidPeso molecolare:516.67Amprenavir
CAS:<p>Amprenavir (KVX-478) is a synthetic derivative of hydroxyethylamine sulfonamide that selectively binds to and inhibits human immunodeficiency virus (HIV)</p>Formula:C25H35N3O6SPurezza:99.60% - 99.87%Colore e forma:Off-White To Pale YellowPeso molecolare:505.63LDC4297 hydrochloride
CAS:LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Formula:C23H29ClN8OColore e forma:SolidPeso molecolare:468.98Peldesine dihydrochloride
CAS:Peldesine (BCX 34) dihydrochloride is an inhibitor of PNP in humans, rats, and mice, also hindering T-cell proliferation, used in lymphoma and HIV research.Formula:C12H13Cl2N5OColore e forma:SolidPeso molecolare:314.17Rolipram
CAS:Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.Formula:C16H21NO3Purezza:99.22% - >99.99%Colore e forma:SolidPeso molecolare:275.34HODHBt
CAS:HODHBt is a STAT5-SUMO protein-protein interaction inhibitor.Formula:C7H5N3O2Purezza:99.45% - 99.95%Colore e forma:Off-White To Yellow SolidPeso molecolare:163.13Dimercaprol
CAS:Dimercaprol (Dicaptol) is an anti-gas warfare agent that is effective against Lewisite (dichloro(2-chlorovinyl)arsine) and formerly known as British Anti-Formula:C3H8OS2Purezza:98.91% - 99.64%Colore e forma:Viscous Oily LiquidPeso molecolare:124.22Saquinavir
CAS:<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Formula:C38H50N6O5Purezza:99.50% - >99.99%Colore e forma:SolidPeso molecolare:670.84Bictegravir
CAS:Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).Formula:C21H18F3N3O5Purezza:97.6% - 99.51%Colore e forma:SolidPeso molecolare:449.38Rilpivirine
CAS:Rilpivirine (R278474) is a diarylpyrimidine derivative and reverse transcriptase inhibitor with antiviral activity against HIV-1 that is used in the treatmentFormula:C22H18N6Purezza:97.22% - 98.83%Colore e forma:SolidPeso molecolare:366.42Fostemsavir
CAS:Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.Formula:C25H26N7O8PPurezza:98.95%Colore e forma:SolidPeso molecolare:583.49IMB-301
CAS:IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.Formula:C19H17Cl2FN2OPurezza:99.72%Colore e forma:SolidPeso molecolare:379.26Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Formula:C20H20FN6O5·KPurezza:98% - 99.55%Colore e forma:Off-White SolidPeso molecolare:482.51Dexelvucitabine
CAS:Dexelvucitabine (RVT), a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.Formula:C9H10FN3O3Purezza:98.25%Colore e forma:SolidPeso molecolare:227.19Des(benzylpyridyl) Atazanavi
CAS:The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.Formula:C26H43N5O7Purezza:98% - 99.75%Colore e forma:SolidPeso molecolare:537.65PMEDAP
CAS:PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiencyFormula:C8H13N6O4PPurezza:99.77%Colore e forma:SolidPeso molecolare:288.2Cobicistat
CAS:Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.Formula:C40H53N7O5S2Purezza:97.36% - 99.62%Colore e forma:SolidPeso molecolare:776.02
