Proteasi HIV
Gli inibitori della proteasi dell'HIV sono una classe di farmaci antiretrovirali che bersagliano specificamente l'enzima proteasi del virus dell'immunodeficienza umana (HIV). Inibendo questo enzima, questi composti impediscono al virus di elaborare le sue poliproteine in proteine mature e funzionali, bloccando così la produzione di nuovi virioni infettivi. Gli inibitori della proteasi dell'HIV sono una pietra miliare della terapia antiretrovirale altamente attiva (HAART) utilizzata per gestire l'HIV/AIDS. Presso CymitQuimica, offriamo una varietà di inibitori della proteasi dell'HIV per supportare la vostra ricerca nel trattamento dell'HIV, nella resistenza ai farmaci e nella virologia.
Trovati 506 prodotti di "Proteasi HIV"
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(S)-BI-1001
CAS:(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).Formula:C19H15BrClNO3Purezza:98%Colore e forma:SolidPeso molecolare:420.68HIV-IN-4
CAS:HIV-IN-4 (Compound 12) is a potent HIV inhibitor that exhibits promising anti-HIV activities [1].Formula:C14H18N2O3Colore e forma:SolidPeso molecolare:262.3HIV-1 inhibitor-16
CAS:HIV-1 inhibitor-16: potent with EC50 1.3 nM for wild-type; inhibits K103N, E138K, Y181C, L100I strains; good solubility; stable; low CYP impact; non-toxic.Formula:C23H16F2N6Colore e forma:SolidPeso molecolare:414.41HIV-1 inhibitor-57
CAS:<p>HIV-1 Inhibitor-57 (Compound 12g) is an antiviral agent that potently inhibits both wild-type and five common NNRTI-resistant strains of HIV-1, exhibiting EC50</p>Formula:C25H24FN5O3SColore e forma:SolidPeso molecolare:493.55SARS-CoV-IN-3
CAS:SARS-CoV-IN-3 is an effective SARS-CoV replication inhibitor.Formula:C25H28ClFeN3OPurezza:98%Colore e forma:SolidPeso molecolare:477.81Mesoxalic acid
CAS:Mesoxalic acid is a dicarboxylic acid and a ketonic acid which blocks RT translocation.Formula:C3H2O5Purezza:98%Colore e forma:SolidPeso molecolare:118.04SAMT-247
CAS:SAMT-247 is an HIV inhibitor that acts by modifying the nucleocapsid NCp7 region of Gag in infected cells and blocking Gag processing and reducing infectivity.Formula:C12H14N2O3SColore e forma:SolidPeso molecolare:266.32TMC310911
CAS:TMC310911 is an oral HIV-1 protease inhibitor with an EC50 of 2.2-14.2 nM, effective against various HIV-1 strains.Formula:C38H53N5O7S2Purezza:98%Colore e forma:SolidPeso molecolare:755.99Reverse transcriptase-IN-3
Reverse transcriptase-IN-3, a pyrimidine carboxamide, inhibits HIV-1 including mutant strains.Formula:C28H31N7O4SColore e forma:SolidPeso molecolare:561.66DQBS
CAS:DQBS is an HIV-1 Nef function antagonist.Formula:C22H17ClN4O4SPurezza:98%Colore e forma:SolidPeso molecolare:468.91HIV-1 integrase inhibitor 7
CAS:HIV-1 integrase inhibitor 7 is a potent HIV-1 integrase inhibitor (IC50: 33.3 nM).Formula:C30H26O16Purezza:98%Colore e forma:SolidPeso molecolare:642.52β-L-D4A
CAS:beta-L-D4A inhibits HIV-1 reverse transcriptase, stopping DNA synthesis.Formula:C10H11N5O2Purezza:99.45%Colore e forma:SolidPeso molecolare:233.23MK-4965
CAS:MK-4965 is a new type of non-nucleoside reverse transcriptase inhibitor with antiviral activity.Formula:C20H13Cl2N5O2Colore e forma:SolidPeso molecolare:426.26gp120-IN-1
CAS:gp120-IN-1 (4e) is a potent HIV-1 inhibitor, IC50 2.2 μM, CC50 100.90 μM, and blocks HIV entry.Formula:C15H18N2O4SColore e forma:SolidPeso molecolare:322.38HIV-1 inhibitor-25
CAS:Compound R-12a is a potent HIV-1 reverse transcriptase inhibitor (IC50: 0.1061 nM), with low cytotoxicity and effective against multiple mutants.Formula:C26H19N5O2Colore e forma:SolidPeso molecolare:433.46LEDGIN6
CAS:HIV-1 integrase inhibitor 2 is used for the treatment of human immunodeficiency virus (HIV) infection.Formula:C21H20ClNO2Colore e forma:SolidPeso molecolare:353.84NIT
CAS:NIT is an HIV-1 protease inhibitor.Formula:C15H7N3O4S2Purezza:98%Colore e forma:SolidPeso molecolare:357.36HIV-1 inhibitor-36
CAS:HIV-1 inhibitor-36 (Compound 2) is a potent HIV-1 inhibitor with significant potential as a novel latency reversing agent [1].Formula:C14H14Cl2N2O2SColore e forma:SolidPeso molecolare:345.24HIV-1 inhibitor-24
CAS:HIV-1 inhibitor-24 (S-12a) blocks HIV reverse transcription effectively (IC50: 9.5 nM), low toxicity, well-tolerated in mice, good heart safety.Formula:C26H19N5O2Colore e forma:SolidPeso molecolare:433.46DPC-681
CAS:DPC-681 is a potent and selective HIV protease inhibitor (IC90s: 4 to 40 nM for wild-type HIV-1).Formula:C35H48FN5O5SColore e forma:SolidPeso molecolare:669.85
