
Proteasi HIV
Gli inibitori della proteasi dell'HIV sono una classe di farmaci antiretrovirali che bersagliano specificamente l'enzima proteasi del virus dell'immunodeficienza umana (HIV). Inibendo questo enzima, questi composti impediscono al virus di elaborare le sue poliproteine in proteine mature e funzionali, bloccando così la produzione di nuovi virioni infettivi. Gli inibitori della proteasi dell'HIV sono una pietra miliare della terapia antiretrovirale altamente attiva (HAART) utilizzata per gestire l'HIV/AIDS. Presso CymitQuimica, offriamo una varietà di inibitori della proteasi dell'HIV per supportare la vostra ricerca nel trattamento dell'HIV, nella resistenza ai farmaci e nella virologia.
Trovati 502 prodotti di "Proteasi HIV"
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HIV protease-IN-1
CAS:HIV protease-IN-1 (compound 1·succinate), a potent non-peptidic inhibitor of HIV protease, is utilized for AIDS research [1].Formula:C39H40ClF7N10O7Colore e forma:SolidPeso molecolare:929.24Pegaldesleukin
CAS:Pegaldesleukin, a PEG-IL2 conjugate, exhibits antiviral properties, potentially slowing HIV progression, preserving immune function.Colore e forma:Liquid(Iso)-Fosdevirine
CAS:(Iso)-Fosdevirine ( (Iso)-GSK2248761), a reverse transcriptase (NNRTI) inhibitor with anti-HIV activity, is used in the study of neurological diseases.Formula:C20H17ClN3O3PPurezza:99.93%Colore e forma:SoildPeso molecolare:413.79TAT peptide
TAT peptide, a CPP, delivers molecules into cells by traversing membrane barriers using aa49-57 of TAT protein.Formula:C65H124N34O15Purezza:98%Colore e forma:SolidPeso molecolare:1621.91GLR-19
CAS:GLR-19 is an anti-HIV peptide with demonstrated antiviral activity against HSV-2 [1] [2].Formula:C102H194N40O20Purezza:98%Colore e forma:SolidPeso molecolare:2300.89Lopinavir Metabolite M-1
CAS:Lopinavir Metabolite M-1, derived from Lopinavir, inhibits HIV protease (Ki=0.7 pM) and shows antiviral activity in vitro.Formula:C37H46N4O6Colore e forma:SolidPeso molecolare:642.78Peritassine A
CAS:Peritassine A, an alkaloid derived from Tripterygium wilfordii Hook. f., exhibits anti-HIV properties.Formula:C38H47NO18Colore e forma:SolidPeso molecolare:805.783Hinnuliquinone
CAS:Hinnuliquinone is an anti-HIV agent.Formula:C32H30N2O4Purezza:98%Colore e forma:SolidPeso molecolare:506.59Hypoglaunine D
CAS:Hypoglaunine D, an anti-HIV analogue of Triptonine B, inhibits HIV in H9 cells with an EC50 of 22 μg/ml.Formula:C41H47NO19Colore e forma:SolidPeso molecolare:857.81QYL-685
CAS:QYL-685 is a methylenecyclopropane nucleoside analog.Formula:C20H24N7O5PColore e forma:SolidPeso molecolare:473.42Carbovir triphosphate
CAS:Carbovir triphosphate (CBV-TP), a phosphorylated metabolite, serves as a research tool for studying human immunodeficiency virus (HIV) [1].Formula:C11H16N5O11P3Colore e forma:SolidPeso molecolare:487.19Amdoxovir
CAS:Amdoxovir is a reverse transcriptase inhibitor.Formula:C9H12N6O3Colore e forma:SolidPeso molecolare:252.23HIV-1 inhibitor-12
HIV-1 inhibitor-12: potent at inhibiting HIV-1 capsid protein polymerization with 9 nM IC50.Formula:C42H36ClF10N7O5S2Colore e forma:SolidPeso molecolare:1008.35SDZ 283-910
CAS:SDZ 283-910 is used as a statine-derived inhibitor.Formula:C46H59N5O9Purezza:98%Colore e forma:SolidPeso molecolare:826.004CA inhibitor 1
CAS:CA inhibitor 1 (GS-6207 analog) is a potent inhibitor of the HIV capsid.Formula:C41H36ClF8N7O5S2Purezza:98%Colore e forma:SolidPeso molecolare:958.34Delavirdine
CAS:<p>Delavirdine, an NNRTI for HIV-1, is used in HAART.</p>Formula:C22H28N6O3SColore e forma:SolidPeso molecolare:456.56(±)-BI-D
CAS:(±)-BI-D is an effective ALLINI(An allosteric IN inhibitor) that binds integrase at the LEDGF/p75 binding site (IC50: 2.4–2.9 μM).Formula:C25H27NO4Colore e forma:SolidPeso molecolare:405.492-Hydroxyisoquinoline-1,3(2H,4H)-dione
CAS:Hydroxyisoquinoline-1,3(2H,4H)-dione (compound 6a) acts as an inhibitor of both HIV-1 integrase (IN) and HIV-1 reverse transcriptase ribonuclease H (RT RNase H), exhibiting IC50 values of 6.32 µM and 5.9 µM, respectively.Formula:C9H7NO3Peso molecolare:177.16Isoquinoline
CAS:Compound PDK0035, with CAS No. 119-65-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0035 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C9H7NPeso molecolare:129.15

