Antibatterico
Gli inibitori antibatterici sono composti che prendono di mira le cellule batteriche, inibendo la loro crescita o uccidendole direttamente. Questi inibitori sono essenziali nello sviluppo di trattamenti per le infezioni batteriche e sono ampiamente utilizzati nella ricerca per studiare la fisiologia batterica, i meccanismi di resistenza e l'efficacia di nuovi agenti antibatterici. Presso CymitQuimica offriamo una gamma di inibitori antibatterici per supportare la vostra ricerca in microbiologia, malattie infettive e sviluppo di farmaci.
Trovati 3423 prodotti di "Antibatterico"
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Aquayamycin
CAS:Aquayamycin is an anthraquinone derivative and inhibitor of the enzyme tyrosine hydroxylase..Formula:C25H26O10Colore e forma:SolidPeso molecolare:486.47Keto lovastatin
CAS:Keto lovastatin is an impurity of lovastatin with antibacterial properties. Lovastatin is a cell-permeable HMG-CoA reductase (HMG-CoA reductase) inhibitor used to reduce cholesterol levels.Formula:C24H34O6Colore e forma:SolidPeso molecolare:418.523Alpibectir
CAS:Alpibectir has antibacterial activity [1].Formula:C12H14F6N2O2Colore e forma:SolidPeso molecolare:332.24DNA Gyrase-IN-13
CAS:DNA Gyrase-IN-13 (compound 1b) is an inhibitor of DNA gyrase with bacteriostatic properties. It exhibits an IC50 of 1.81 μM against Staphylococcus aureus DNA gyrase.Formula:C15H21N3O3SColore e forma:SolidPeso molecolare:323.41Kikumycin A
CAS:Kikumycin A, an antibiotic produced by Streptomyces, exhibits antimicrobial activity against both Gram-positive and Gram-negative bacteria. Additionally, it demonstrates antitrichomonal activity with a minimum inhibitory concentration (MIC) of 25 μg/mL against Trichomonas foetus.Formula:C13H17N7O2Colore e forma:SolidPeso molecolare:303.32MT0703
CAS:MT0703 is a cephalosporin antibiotic featuring an aminothiazolylglycyl moiety with a 1,5-dihydroxy-4-pyridinone-2-carbonyl group, displaying potent activity against Pseudomonas species.Formula:C26H25N7O9S3Colore e forma:SolidPeso molecolare:675.71Cephalosporin C
CAS:Cephalosporin C exhibits relatively weak resistance to Gram-positive and Gram-negative bacteria. It is stable against penicillinase, but can be decomposed by cephalosporinase. When hydrolyzed to remove its side chain, it yields 7-amino-cefenoic acid (7-ACA), which is an essential raw material for the production of semisynthetic cephalosporins.Formula:C16H21N3O8SColore e forma:SolidPeso molecolare:415.418AAA-10 formic
AAA-10 formic is an orally active inhibitor of intestinal bacterial bile salt hydrolase (BSH) against B.Formula:C26H43FO7SColore e forma:SolidPeso molecolare:518.68CM-728
CAS:CM-728 is an oxazanonaphthoquinone that exhibits cytotoxic and antibacterial properties. It acts as a human peroxidase-1 inhibitor and serves as a source of oxidative stress affecting mitochondrial function.Formula:C22H14N2O5Colore e forma:SolidPeso molecolare:386.357Bilanafos
CAS:Bilanafos is an agent of Anti-Bacterial.Formula:C11H22N3O6PPurezza:98%Colore e forma:SolidPeso molecolare:323.28Antitubercular agent-29
Compound 6xa inhibits drug-resistant tuberculosis with MICs 0.03 μg/mL for DS-Mtb and 0.03-0.06 for DR-Mtb, SI>40 for Vero cells.Formula:C20H12ClN3O5Colore e forma:SolidPeso molecolare:409.78Benzisothiazolone
CAS:Benzisothiazolone is an isothiazolinone fungicide that demonstrates growth inhibitory activity against Escherichia coli ATCC 8739 and yeast NCYC 1354. It is utilized in studies investigating growth inhibition models.Formula:C7H5NOSColore e forma:SolidPeso molecolare:151.197-Hydroxytropolone
CAS:7-Hydroxytropolone (3-Hydroxytropolone) is an antibiotic that exhibits activity against Gram-positive and Gram-negative bacteria, as well as yeasts and fungi. It also functions as an inhibitor of 2''-O-adenylate transferase.Formula:C7H6O3Colore e forma:SolidPeso molecolare:138.12Avibactam sodium dihydrate
Avibactam sodium dihydrate (NXL-104) is a reversible covalent inhibitor for CTX-M-15 and TEM-1 β-lactamases with IC50s of 5 nM and 8 nM.Formula:C7H14N3NaO8SColore e forma:SolidPeso molecolare:323.26Metallo-β-lactamase-IN-16
CAS:Metallo-β-lactamase-IN-16 (compound 18), a sulfone-containing metallo-β-lactamase inhibitor, exhibits antimicrobial activity. It effectively inhibits various metallo-β-lactamases, including NDM-1 (New Delhi metallo-β-lactamase-1), IMP-1 (imipenemase-1), VIM-1 (Verona Integron-encoded Metallo-β-lactamase), and VIM-2. The IC50 values for these enzymes are 0.16 nM, 0.23 nM, 0.31 nM, and 1.0 nM respectively.Formula:C16H16N8O4S3Colore e forma:SolidPeso molecolare:480.54NBTI 5463
CAS:NBTI 5463 is a bacterial type II topoisomerase (topoisomerase II) inhibitor with antimicrobial properties. It effectively inhibits GyrA and TopoIV in Pseudomonas aeruginosa and Escherichia coli. By binding to topoisomerase II, NBTI 5463 prevents DNA cleavage and re-ligation, thereby impeding bacterial DNA replication and transcription. This compound shows potential for research into Gram-negative bacterial infections.Formula:C25H30N6O4Colore e forma:SolidPeso molecolare:478.54PF 03709270
CAS:PF 03709270 is an oral prodrug of sulopenem with broad-spectrum antibacterial effects on gram-positive and gram-negative bacteria.Formula:C19H27NO7S3Purezza:98%Colore e forma:SolidPeso molecolare:477.61(4-Aminobenzoyl)-D-glutamic acid
CAS:(4-Aminobenzoyl)-D-glutamic acid (Compound 17) exhibits competitive inhibitory activity against the H2-pterin synthesis system, affecting folic acid synthesis and subsequently inhibiting bacterial growth.Formula:C12H14N2O5Colore e forma:SolidPeso molecolare:266.25VEGFR-2/DHFR-IN-1
Compound 8b inhibits VEGFR-2/DHFR, combats various bacteria, and fights cancer cells.Formula:C20H18ClNO4Colore e forma:SolidPeso molecolare:371.81Antibacterial agent 236
CAS:Anti bacterial agent 236 (Compound 4l), an orally effective inhibitor of DNA gyrase and topoisomerase IV (with IC50 values of 3.2 and 300 nM in Staphylococcus aureus, respectively), exhibits broad-spectrum antibacterial activity. It also demonstrates favorable pharmacokinetic properties in mice.Formula:C26H27N5O2SColore e forma:SolidPeso molecolare:473.59Colistin adjuvant-2
Colistin adjuvant-2 is a compound that acts as a potentiation agent for colistin, effectively enhancing its activity against Gram-negative bacteria [1].Formula:C14H7Cl2F3N2OColore e forma:SolidPeso molecolare:347.12MtTMPK-IN-9
MtTMPK-IN-9 moderately inhibits MtbTMPK (IC50: 48 μM), has submicromolar Mycobacterium activity, and is non-toxic, aiding tuberculosis research.Formula:C25H26N6O7Colore e forma:SolidPeso molecolare:522.51Antibacterial agent 81
CAS:Antibacterial agent 81 blocks DNA transcription, targets S. aureus (MIC 12.5μM) & M. smegmatis (MIC 7.8μM). Used in infection research.Formula:C33H28N2O8Colore e forma:SolidPeso molecolare:580.58MurA-IN-6
CAS:MurA-IN-6 (Compound L16) is a selective MurA inhibitor with an IC50 of 26.63 μM. It exhibits antibacterial activity by inhibiting the function of MurA, a key protein essential for bacterial cell wall synthesis.Formula:C22H17N3O3SColore e forma:SolidPeso molecolare:403.454BM635 mesylate
BM635 mesylate inhibits MmpL3; kills Divergent bacterium with 0.6 µM MIC50; boosts bioavailability.Formula:C26H33FN2O4SColore e forma:SolidPeso molecolare:488.6114α-Demethylase/DNA Gyrase-IN-1
14α-Demethylase/DNA Gyrase-IN-1 (Compound 7c) is a potent inhibitor of 14α-Demethylase/DNA Gyrase with antibacterial activity.Formula:C26H22N4O4Colore e forma:SolidPeso molecolare:454.48Deprodone
CAS:Deprodone is an active compound that inhibits key processes such as bacterial cell wall synthesis by interacting with hydrolase and transferase proteins of methicillin-resistant Staphylococcus aureus (MRSA). It is applied in the research of MRSA infections, inflammatory skin diseases, intestinal disorders, and fatty acid metabolism disorders.Formula:C21H28O4Colore e forma:SolidPeso molecolare:344.44PqsR-IN-1
PqsR-IN-1, potent PqsR inhibitor, curbs pyocyanin in Pseudomonas aeruginosa with low cytotoxicity.Formula:C17H18ClN3OSColore e forma:SolidPeso molecolare:347.86DNA Gyrase-IN-1
DNA Gyrase-IN-1: potent, selective promoter inhibitor. IC50: 2.6 μM, inhibits Mtb, MIC: 0.49 μM. Useful for tuberculosis research.Formula:C24H24FN7O6Colore e forma:SolidPeso molecolare:525.49GT-055
GT-055 (LCB18-055) is a novel inhibitor of broad-spectrum β-lactamase.Formula:C13H20F3N5O8SColore e forma:SolidPeso molecolare:463.39PCTR1
CAS:PCTR1, derived from DHA, hastens inflammation resolution and boosts macrophage function, reducing PGE2, PGD2, and TXB2 in mice.Formula:C32H47N3O9SColore e forma:SolidPeso molecolare:649.8Antibacterial synergist 1
Compound 20P is a potent antibacterial, inhibits biofilms with IC50 4.5 μM, and reduces pyocyanin at IC50 8.6 μM.Formula:C19H24N2O4Colore e forma:SolidPeso molecolare:344.4DNA Gyrase-IN-16
CAS:DNA Gyrase-IN-16 (Compound 9) is an inhibitor of DNA gyrase, with an IC50 of 1.609 μM. It exhibits antibacterial properties, effectively inhibiting S. aureus and MRSA, with a MIC of 3.125 μM for both.Formula:C17H15N3O3Colore e forma:SolidPeso molecolare:309.319MtMetAP1-IN-1
MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.Formula:C15H10BrN5O2SColore e forma:SolidPeso molecolare:404.24Thiolactomycin
CAS:Thiolactomycin is a novel reversible dual inhibitor of D-amino acid oxidase (DAO) and D-Aspartate oxidase (DDO).Formula:C11H14O2SPurezza:98%Colore e forma:SolidPeso molecolare:210.29HldA/E-IN-1
CAS:HldA/E-IN-1 (compound 8) is a dual inhibitor of HldA/E, exhibiting IC50 values of 17.2 μM and 67.8 μM, respectively. This compound is utilized in research on antibacterial infections.Formula:C8H17FO13P2Colore e forma:SolidPeso molecolare:402.16Penethamate hydriodide
CAS:Penethamate hydriodide is a diethylaminoethyl ester prodrug of penicillin, utilized via intramuscular injection to treat mastitis in cattle.Formula:C22H32IN3O4SColore e forma:SolidPeso molecolare:561.477MBX-1162
CAS:MBX-1162, a bis-indole compound, has demonstrated unique substrate specificity related to MepA and MepR in studies investigating its resistance mechanisms in Staphylococcus aureus. It has not shown cross-resistance with related compounds.Formula:C30H28N6Colore e forma:SolidPeso molecolare:472.58MtTMPK-IN-3
CAS:MtTMPK-IN-3 inhibits Mycobacterium tuberculosis kinase with IC50 0.12μM, MIC 12.5μM on Mtb, cytotoxic EC50 12.5μM on MRC-5 cells.Formula:C23H23Cl2N3O3Colore e forma:SolidPeso molecolare:460.35Antibacterial agent 113
Antibacterial agent 113 targets multiple bacteria including P. aeruginosa and E. coli, showing efficacy at MIC 15625 μM.Formula:C29H18ClN5OColore e forma:SolidPeso molecolare:487.944-Bromo A23187
CAS:4-Bromo A23187 is a halogenated analog of the calcium ionophore A-23187. 4-Bromo A23187 is a calcium modulator and induces apoptosis in different cells.Formula:C29H36BrN3O6Purezza:98%Colore e forma:SolidPeso molecolare:602.52BWC0977
CAS:BWC0977 is an effective topoisomerase inhibitor that disrupts bacterial DNA replication by targeting both DNA gyrase and topoisomerase IV. The minimum inhibitory concentration (MIC90) of BWC0977 against MDR (multi-drug resistant) Gram-negative bacteria ranges from 0.03 to 2 µg/mL.Formula:C22H21FN6O5Colore e forma:SolidPeso molecolare:468.44Ro 24-4383
CAS:Ro 24-4383 is a carbamate-linked dual-action antibacterial agent.Formula:C32H31FN8O10S2Purezza:98%Colore e forma:SolidPeso molecolare:770.76NBTIs-IN-5
CAS:NBTIs-IN-5 inhibits Mycobacterium abscessus DNA with IC50 1.5μM, halts growth at MIC90 0.4μM.Formula:C24H25F3N4O2Colore e forma:SolidPeso molecolare:458.48Diclosulam
CAS:Diclosulam (XDE 564) is an herbicide with a Ki value of less than 32 nM. It exhibits a MIC of 6.25 and 12.5 μM, and a MIC50 of 1.40 and 3.01 μM against the CBS10913 and CBS12373 strains, respectively.Formula:C13H10Cl2FN5O3SColore e forma:SolidPeso molecolare:406.22L-threo-β-Hydroxyaspartic acid
CAS:L-threo-β-Hydroxyaspartic acid is an amino acid antibiotic with activity against Bacillus subtilis, Xanthomonas oryzae, Mycobacterium phlei, and Botrytis cinerea.Formula:C4H7NO5Colore e forma:SolidPeso molecolare:149.102BAS-118
CAS:BAS-118 is a benzamide derivative exhibiting antibacterial activity. For 100 randomly selected strains of Helicobacter pylori, its MIC50, MIC90, and MIC range were ≤0.003, 0.013, and ≤0.003-0.025 mg/L, respectively. BAS-118 shows potential for research as an anti-H. pylori agent.Formula:C20H18N2O2Colore e forma:SolidPeso molecolare:318.369BRL-42715
CAS:BRL-42715 is an effective inhibitor of bacterial beta-lactamases.Formula:C10H7N4NaO3SPurezza:98%Colore e forma:SolidPeso molecolare:286.24Cefoxazole
CAS:Cefoxazole is a β-lactam antibiotic featuring an isoxazole structure, known for its antibacterial activity. It can be utilized in the study of infectious diseases.Formula:C21H18ClN3O7SColore e forma:SolidPeso molecolare:491.902MRL-494
MRL-494, a small-molecule BamA inhibitor, resists efflux and outer membrane permeability, with antibacterial properties.Formula:C26H35FN16O2Purezza:98%Colore e forma:SolidPeso molecolare:622.66
