
Altri inibitori
Questa categoria comprende una vasta gamma di inibitori che non rientrano nelle classificazioni standard ma sono comunque fondamentali per varie ricerche biochimiche e farmacologiche. Questi inibitori possono bersagliare vie, enzimi e interazioni molecolari uniche o meno studiate, fornendo strumenti preziosi per aree di ricerca specializzate. Presso CymitQuimica, offriamo una selezione diversificata di inibitori di alta qualità che coprono molteplici bersagli biologici e discipline di ricerca, permettendoti di esplorare nuove strade terapeutiche e approfondire la tua comprensione dei processi biologici complessi.
Trovati 37827 prodotti di "Altri inibitori"
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Erizepine
CAS:<p>Erizepine, an octopamine receptor 3 (OAR3) antagonist, exhibits a Ki value of 474 nM. This compound is utilized in insect research.</p>Formula:C20H22N2Colore e forma:SolidPeso molecolare:290.4Naltalimide
CAS:<p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>Formula:C28H28N2O5Purezza:98%Colore e forma:SolidPeso molecolare:472.53Pamiparib maleate
CAS:<p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>Formula:C44H42F2N8O14Purezza:98%Colore e forma:SolidPeso molecolare:944.859LK-732
CAS:<p>LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.</p>Formula:C25H29N5O3SColore e forma:SolidPeso molecolare:479.59Ambelline
CAS:<p>Ambelline has antitumor activity.</p>Formula:C18H21NO5Purezza:98%Colore e forma:SolidPeso molecolare:331.36Ro-51
CAS:<p>dual P2X3 and P2X2/3 antagonist</p>Formula:C17H23IN4O4Purezza:98%Colore e forma:SolidPeso molecolare:474.29G-9791
CAS:<p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>Formula:C26H26ClFN6O2Purezza:98%Colore e forma:SolidPeso molecolare:508.98Hymenidin
CAS:Hymenidin, isolated from the Okinawan sponge Hymeniacidon sp., is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor.Formula:C11H12BrN5OPurezza:96.85% - 99.52%Colore e forma:SolidPeso molecolare:310.15Acetoxycycloheximide
CAS:<p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>Formula:C17H25NO6Colore e forma:SolidPeso molecolare:339.38Moflomycin
CAS:<p>Moflomycin is an anthracycline derivative. It exhibits a higher antileukemic activity compared to other anthracyclines.</p>Formula:C25H25IO10Purezza:98%Colore e forma:SolidPeso molecolare:612.36GSK 932121
CAS:<p>GSK 932121: potent antimalarial, targets P. falciparum by inhibiting cytochrome bc1 in the electron transport chain.</p>Formula:C20H15ClF3NO4Purezza:98%Colore e forma:SolidPeso molecolare:425.79Pillaromycin A
CAS:<p>Pillaromycin A exhibits activity against mycobacteria, Gram-positive bacteria, and Gram-negative bacteria, although it is less effective against Gram-negative bacteria. Additionally, it possesses antitumor properties.</p>Formula:C28H30O11Colore e forma:SolidPeso molecolare:542.531Fomecin A
CAS:<p>Fomecin A exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, and weak activity against fungi. It also possesses antiviral activity against the influenza virus PR-8.</p>Formula:C8H8O5Colore e forma:SolidPeso molecolare:184.146L2H2-6OTD
CAS:<p>L2H2-6OTD is a telomerase inhibitor with G-quadruplex loops; IC50: 15 nM.</p>Formula:C30H30N10O8Colore e forma:SolidPeso molecolare:658.62CH5447240
CAS:<p>CH5447240: potent hPTHR1 agonist, treats Hypoparathyroidism, EC50 12 nM, 55% oral bioavailability, raises rat serum calcium.</p>Formula:C26H39N5O4SPurezza:98%Colore e forma:SolidPeso molecolare:517.68Detoxin D1
CAS:<p>Detoxin D1 is a selective blasticidin S antagonist.</p>Formula:C28H41N3O8Purezza:98%Colore e forma:SolidPeso molecolare:547.64Foroxymithine
CAS:<p>Foroxymithine is an inhibitor of angiotensin-converting enzyme.</p>Formula:C22H37N7O11Purezza:98%Colore e forma:SolidPeso molecolare:575.57Flurdihydroergotamine
CAS:<p>Flurdihydroergotamine, a serotonin 5HT1 receptor agonist, is used as an antimigraine drug.</p>Formula:C34H36F3N5O5Purezza:98%Colore e forma:SolidPeso molecolare:651.68MRS2279
CAS:<p>Selective, high affinity competitive antagonist of the P2Y1 receptor</p>Formula:C13H18ClN5O8P2Purezza:98%Colore e forma:SolidPeso molecolare:469.71SMP-797 HCl
CAS:<p>SMP-797 HCl, an ACAT (acyl-CoA-cholesterol acyltransferase) inhibitor, is used potentially for the treatment of Hyperlipidemia.</p>Formula:C34H44ClN5O4Purezza:98%Colore e forma:SolidPeso molecolare:622.20FR 901537
CAS:<p>FR 901537 is a new aromatase inhibitor with antitumor effects.</p>Formula:C23H29N3O6S2Purezza:98%Colore e forma:SolidPeso molecolare:507.62Lorajmine
CAS:Lorajmine, a monochloroacetyl derivative of ajmaline, is a class Ia antiarrhythmic agent that is rapidly hydrolyzed to ajmaline by plasma and tissue esterases.Formula:C22H27ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:402.91Dinordrin I diacetate
CAS:<p>Dinordrin I diacetate is an implantation inhibitor and hormone.</p>Formula:C25H32O4Purezza:98%Colore e forma:SolidPeso molecolare:396.52Esorubicin
CAS:<p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>Formula:C27H29NO10Colore e forma:SolidPeso molecolare:527.52Alentemol hydrobromide
CAS:<p>Alentemol hydrobromide is a Dopamine agonist.</p>Formula:C19H26BrNOPurezza:98%Colore e forma:SolidPeso molecolare:364.32Juvenimicin A2
CAS:<p>Juvenimicin A2 is effective against Gram-positive bacteria and certain Gram-negative bacteria.</p>Formula:C30H51NO8Colore e forma:SolidPeso molecolare:553.728Seldomycin factor 3
CAS:<p>Seldomycin factor 3 (XK 88-3) is an aminoglycoside antibiotic with broad-spectrum antibacterial activity.</p>Formula:C17H35N5O9Colore e forma:SolidPeso molecolare:453.488Quadrilineatin
CAS:<p>Quadrilineatin exhibits antifungal and antibacterial properties.</p>Formula:C10H10O4Colore e forma:SolidPeso molecolare:194.184Sannamycin F
CAS:<p>Sannamycin F is an aminoglycoside antibiotic that exhibits mild antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C18H35N5O6Colore e forma:SolidPeso molecolare:417.5Enteromycin
CAS:<p>Enteromycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C6H8N2O5Colore e forma:SolidPeso molecolare:188.138Polyoxin A
CAS:<p>Polyoxin A is a nucleoside-based antifungal antibiotic.</p>Formula:C23H32N6O14Colore e forma:SolidPeso molecolare:616.532FMK-MEA
CAS:<p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>Formula:C21H26FN5O2Purezza:98%Colore e forma:SolidPeso molecolare:399.46Cryptosporiopsin
CAS:<p>Cryptosporiopsin can be isolated from strains of Cryptosporiopsis sp. and Sporormia affinis. It exhibits antimicrobial activity against various basidiomycetes, alga fungi, ascomycetes, and glaucomycetes responsible for wood decay. Additionally, it inhibits the germination of Phytophthora potatoes spores. Cryptosporiopsin also shows some activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C10H10Cl2O4Colore e forma:SolidPeso molecolare:265.09Chlorflavonin
CAS:<p>Chlorflavonin exhibits antifungal activity against several fungi, including Aspergillus, yeast, and Botrytis cinerea, with exceptionally strong activity against Aspergillus nidulans, where the minimum inhibitory concentration is as low as 0.08 μg/mL.</p>Formula:C18H15ClO7Colore e forma:SolidPeso molecolare:378.761Piperazinomycin
CAS:<p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>Formula:C18H20N2O2Colore e forma:SolidPeso molecolare:296.362-Hydroxybutirosin
CAS:<p>2-Hydroxybutirosin is an antibiotic that can be found in Bacillus circulans.</p>Formula:C21H41N5O13Colore e forma:SolidPeso molecolare:571.576Roselipin 1A
CAS:<p>Roselipin 1A inhibits diacylglycerol acyltransferase (DGAT) in rats.</p>Formula:C40H72O14Colore e forma:SolidPeso molecolare:776.991Dihydrocompactin
CAS:<p>Dihydrocompactin is an antifungal metabolite derived from Penicillium citrinum and acts as an inhibitor of 3-hydroxy-3-methylglutaryl coenzyme-A reductase (HMG-CoA reductase).</p>Formula:C23H36O5Colore e forma:SolidPeso molecolare:392.529Pilatin
CAS:<p>Pilatin exhibits inhibitory effects on both bacteria and fungi, and it strongly suppresses the incorporation of thymidine and uridine into DNA and RNA in Ehrlich ascites tumor cells.</p>Formula:C21H26O7Colore e forma:SolidPeso molecolare:390.427Pacidamycin 5T
CAS:<p>Pacidamycin 5T is found in the bacterium Streptomyces coeruleorubidus [NRRL 18370].</p>Formula:C36H44N8O12Colore e forma:SolidPeso molecolare:780.78Parimycin
CAS:<p>Parimycin exhibits activity against Gram-positive and Gram-negative bacteria, as well as tumors, but shows no efficacy against fungi. It inhibits tumor cells such as GXF 251L, H640, LXFA 629L, MCF-7, and MEXF 514L, with an IC70 range of 0.9-6.7 μg/mL.</p>Formula:C22H20O7Colore e forma:SolidPeso molecolare:396.3916-Hydroxyroridin L-2
CAS:<p>16-Hydroxyroridin L-2 is a member of the verrucarin subclass of antibiotics with antitumor properties.</p>Formula:C29H38O10Colore e forma:SolidPeso molecolare:546.6061-Hydroxyoxaunomycin
CAS:<p>1-Hydroxyoxaunomycin is an antibiotic that inhibits the growth of U210 cells as well as the synthesis of DNA and RNA, with IC50 values of 0.0005 μg/mL, 1.00 μg/mL, and 0.76 μg/mL, respectively.</p>Formula:C26H29NO11Colore e forma:SolidPeso molecolare:531.509Gentamicin C2
CAS:<p>Gentamicin C2 is an aminoglycoside antibiotic.</p>Formula:C20H41N5O7Colore e forma:SolidPeso molecolare:463.569Monamycin H1
CAS:<p>Monamycin H1 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.</p>Formula:C34H56ClN7O8Colore e forma:SolidPeso molecolare:726.30Bacithrocin B
CAS:<p>Bacithrocin B is a thrombin inhibitor that suppresses the activity of thrombin, Factor Xa, trypsin, and papain, with IC50 values of 84 μM, 17 μM, 1.7 μM, and 0.02 μM, respectively.</p>Formula:C19H29N5O3Colore e forma:SolidPeso molecolare:375.465Glidobactin G
CAS:<p>Glidobactin G is an antitumor antibiotic with activity against pathogenic fungi and yeasts. Additionally, Glidobactin G prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Formula:C27H44N4O7Colore e forma:SolidPeso molecolare:536.6619-cis-13,14-Dihydroretinoic acid
CAS:<p>9-cis-13,14-Dihydroretinoic acid (9CDHRA) is a selective retinoid X receptor (RXR) agonist with a Kd of 90 nM. It can ameliorate memory deficits caused by impaired RXR signaling in vivo. This compound shows potential for research in the fields of neuroscience and metabolic diseases.</p>Formula:C20H30O2Colore e forma:SolidPeso molecolare:302.451Curvulic acid
CAS:<p>Curvulic acid exhibits relatively weak activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C11H12O6Colore e forma:SolidPeso molecolare:240.209Carzinophillin A
CAS:<p>Carzinophillin A exhibits inhibitory effects on both ascites carcinoma and Yoshida sarcoma.</p>Formula:C31H33N3O11Colore e forma:SolidPeso molecolare:623.607Haliangicin D
CAS:<p>Haliangicin D exhibits antifungal activity against filamentous fungi and is also effective against oomycetes, though it lacks antibacterial properties.</p>Formula:C22H32O5Colore e forma:SolidPeso molecolare:376.49L-2,5-Dihydrophenylalanine
CAS:<p>L-2,5-Dihydrophenylalanine can induce apoptosis in human medulloblastoma leukemia cells [HL-60].</p>Formula:C9H13NO2Colore e forma:SolidPeso molecolare:167.21Oximidine Ⅲ
CAS:<p>Oximidine III is an antitumor antibiotic that selectively inhibits the growth of rat fibroblast 3Y1 cells and induces mutations in various tumor genes. The inhibitory effects of Oximidine III on vH-ras-3Y1, v-src-3Y1 cells, and normal 3Y1 cells have IC50 values of 14 nM, 4.5 nM, and 140 nM, respectively. Additionally, Oximidine III arrests cells with RAS or SRC mutations in the G1 phase of the cell cycle and increases the expression of p21WAF1.</p>Formula:C23H24N2O6Colore e forma:SolidPeso molecolare:424.45NB-533
CAS:<p>NB-533 is a macrocyclic peptidic BACE-1 inhibitor.</p>Formula:C33H55N3O4Colore e forma:SolidPeso molecolare:557.81Megovalicin G
CAS:<p>Megovalicin G is effective against Bacillus subtilis and Escherichia coli, and it also acts on Pseudomonas aeruginosa.</p>Formula:C35H61NO7Colore e forma:SolidPeso molecolare:607.86Monamycin B
CAS:<p>Monamycin B is an ester peptide antibiotic with activity against Gram-positive bacteria.</p>Formula:C33H55N7O8Colore e forma:SolidPeso molecolare:677.8320S Proteasome-IN-4
CAS:<p>20S Proteasome-IN-4: brain-penetrant, parasite-specific, oral, inhibits T.b. brucei proteasome (IC50: 6.3nM), for HAT research.</p>Formula:C20H18ClF2N3O3Colore e forma:SolidPeso molecolare:421.839-Hydroxycrisamicin
CAS:9-Hydroxycrisamicin exhibits moderate activity against Gram-positive bacteria with a minimum inhibitory concentration (MIC) ranging from 6.25 to 25 μg/mL. Additionally, 9-Hydroxycrisamicin demonstrates significant growth inhibition towards various human tumor cell lines.Formula:C32H22O13Colore e forma:SolidPeso molecolare:614.51Monamycin I
CAS:Monamycin I is an ester peptide antibiotic with activity against Gram-positive bacteria.Formula:C35H58ClN7O8Colore e forma:SolidPeso molecolare:740.33GC 14
CAS:<p>GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 200 nM and 35 nM for hTRα and hTRβ, respectively.</p>Formula:C26H27NO6Purezza:98%Colore e forma:SolidPeso molecolare:449.5RIP1 kinase inhibitor 1
CAS:<p>RIP1 kinase inhibitor 1 is an orally available and brain-penetrating inhibitor of RIP1 kinase with pKi of 9.04.</p>Formula:C24H20ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:461.9CI-1029
CAS:<p>CI-1029: HIV protease inhibitor, combats mutant strains, high efficacy, good bioavailability in animals.</p>Formula:C28H37NO4SColore e forma:SolidPeso molecolare:483.6613-Hydroxyglucopiericidin A
CAS:<p>13-Hydroxyglucopiericidin A is an antibiotic with potent antitumor cell activity.</p>Formula:C31H47NO10Colore e forma:SolidPeso molecolare:593.706Hypercalin B
CAS:<p>Hypercalin B is an antibacterial agent isolated from the hexane and chloroform extracts of Hypericum acmosepalum. It demonstrates activity against multidrug-resistant strains of Staphylococcus aureus, with a minimum inhibitory concentration (MIC) ranging from 0.5 to 128 mg/L.</p>Formula:C33H42O5Colore e forma:SolidPeso molecolare:518.684Fleephilone
CAS:<p>Fleephilone is a fungal metabolite isolated from Trichoderma harzianum. It acts as an HIV REV/RRE binding inhibitor, hindering the interaction between REV protein and RRE RNA with an IC50 of 7.6 μM.</p>Formula:C24H27NO7Colore e forma:SolidPeso molecolare:441.474Pradimicin Q
CAS:<p>Pradimicin Q is an antibiotic exhibiting cytotoxicity against human colon HCT-116 cells and mouse melanoma B16-F10 cells, with IC50 values of 75 μg/mL and 100 μg/mL, respectively.</p>Formula:C24H16O10Colore e forma:SolidPeso molecolare:464.378Saframycin Mx2
CAS:<p>Saframycin Mx2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C29H38N4O8Colore e forma:SolidPeso molecolare:570.634BMS-986120
CAS:BMS-986120: Oral, reversible PAR4 antagonist. IC50: 9.5 nM (human), 2.1 nM (monkey). Potent, selective antiplatelet.Formula:C23H23N5O5S2Colore e forma:SolidPeso molecolare:513.59Pelagiomicin C
CAS:Pelagiomicin C exhibits activity against both Gram-positive and Gram-negative bacteria.Formula:C17H15N3O5Colore e forma:SolidPeso molecolare:341.318AZ14145845
<p>AZ14145845 is an in vivo potent and highly selective type I1/2 Mer/Axl bispecific kinase inhibitor.</p>Formula:C32H35N9OColore e forma:SolidPeso molecolare:561.68G-4120
CAS:<p>G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.</p>Formula:C26H36N8O11SColore e forma:SolidPeso molecolare:668.68ZK824859 hydrochloride (2271122-53-1 free base)
ZK824859 hydrochloride: oral, selective uPA inhibitor, IC50s: 79 nM (uPA), 1580 nM (tPA), 1330 nM (plasmin).Formula:C23H23ClF2N2O4Purezza:98%Colore e forma:SolidPeso molecolare:464.896-Hydroxytetrangulol
CAS:<p>6-Hydroxytetrangulol is an inducer of CPP32 protease found in Streptomyces.</p>Formula:C19H12O5Colore e forma:SolidPeso molecolare:320.30Cepacin A
CAS:<p>Cepacin A is an alkyne antibiotic with antibacterial properties, exhibiting a minimum inhibitory concentration (MIC) of 0.2 μg/mL against Staphylococcus. Additionally, Cepacin A displays a degree of toxicity in mice, with an LD50 of 30 mg/kg when administered intraperitoneally.</p>Formula:C16H14O4Colore e forma:SolidPeso molecolare:270.28COTC
CAS:<p>COTC is an anticancer bacterial metabolite; inhibits glyoxalase with GSH, halts HeLa cell growth, and fights tumor in Ehrlich murine model.</p>Formula:C11H14O6Colore e forma:SolidPeso molecolare:242.23EBOV-GP-IN-1
<p>EBOV-GP-IN-1 (Compound 28) is a potent inhibitor of Ebola entry, acting on the Ebola virus envelope glycoprotein (EBOV-GP) (IC50: 0.05 μM).</p>Formula:C25H40ClN3O2Colore e forma:SolidPeso molecolare:450.06Lp-PLA2-IN-5
CAS:<p>Lp-PLA2-IN-5 inhibits Lp-PLA2 and PAF-AH, potentially useful in Alzheimer's and atherosclerosis studies.</p>Formula:C23H18F5N3O4Colore e forma:SolidPeso molecolare:495.4MDL-27788
CAS:<p>MDL-27788 is a tricyclic inhibitor.</p>Formula:C24H26N2O5SColore e forma:SolidPeso molecolare:454.5417β-HSD1-IN-1
<p>17β-HSD1-IN-1 (Compound 1) can be used in the non-small cell lung cancer (NSCLC) research.</p>Formula:C21H21NO3Colore e forma:SolidPeso molecolare:335.4Amidinomycin
CAS:<p>Amidinomycin primarily acts against Gram-positive bacteria.</p>Formula:C9H18N4OPeso molecolare:198.27Norplicacetin
CAS:<p>Norplicacetin exhibits activity against Gram-positive bacteria and mycobacteria.</p>Formula:C24H33N5O7Peso molecolare:503.55BAY-693
CAS:<p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>Formula:C26H30F3N7O2Colore e forma:SolidPeso molecolare:529.56Melanoxazal
CAS:<p>Melanoxazal is an inhibitor of melanin biosynthesis, effectively suppressing melanin formation in silkworm larva hemolymph with an IC50 of 30.1 μg/mL, and it also exhibits strong inhibitory effects on mushroom tyrosinase (IC50 of 4.2 μg/mL), while lacking antibacterial activity.</p>Formula:C8H9NO3Peso molecolare:167.16Papyracon D
CAS:<p>Papyracon D exhibits moderate inhibitory effects on L1210 and HL60 cells and shows mild inhibition against nematodes. It also has a slight inhibitory effect on Gram-positive bacteria.</p>Formula:C14H18O5Peso molecolare:266.29Oryzoxymycin
CAS:<p>Oryzoxymycin is an aromatic derivative antibiotic with activity against Gram-negative bacteria.</p>Formula:C10H13NO5Peso molecolare:227.21Polvitolimod
CAS:<p>Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.</p>Formula:C13H14FN5O4Colore e forma:SolidPeso molecolare:323.28Cinnatriacetin A
CAS:<p>Cinnatriacetin A exhibits activity against Gram-positive bacteria.</p>Formula:C23H20O5Colore e forma:SolidPeso molecolare:376.402Coriolin B
CAS:<p>Coriolin B exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, yeast, and Trichomonas vaginalis. At a concentration of 5 μg/mL, Coriolin B inhibits 61.6% of Yoshida sarcoma growth but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>Formula:C23H36O6Colore e forma:SolidPeso molecolare:408.528Azicemicin A
CAS:<p>Azicemicin A exhibits mild antibacterial activity and shows no acute toxicity when administered via intraperitoneal injection to mice at a dosage of 150 mg/kg.</p>Formula:C23H25NO9Colore e forma:SolidPeso molecolare:459.446Polyozellin
CAS:<p>Polyozellin is a prolyl endopeptidase inhibitor with properties effective against inflammation, cancer, and diseases related to oxidative stress.</p>Formula:C22H14O10Colore e forma:SolidPeso molecolare:438.341Purine phosphoribosyltransferase-IN-1
<p>Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.</p>Formula:C11H15N5Na4O10P2Colore e forma:SolidPeso molecolare:531.17Phencomycin
CAS:<p>Phencomycin exhibits mild activity against Gram-positive bacteria and inhibits physiologically important enzymes such as renin, with an IC50 of 440 μg/mL.</p>Formula:C15H10N2O4Colore e forma:SolidPeso molecolare:282.251Polyoxin J
CAS:<p>Polyoxin J is a nucleoside antifungal antibiotic, notably effective against sheath blight in rice.</p>Formula:C17H25N5O12Peso molecolare:491.41Diatretyne Ⅰ
CAS:Diatretyne I (Diatretyne amide) exhibits mild activity against Gram-positive bacteria.Formula:C8H5NO3Colore e forma:SolidPeso molecolare:163.13Maltophilin
CAS:<p>Maltophilin is a broad-spectrum antifungal antibiotic that exhibits no antibacterial activity against either Gram-positive or Gram-negative bacteria.</p>Formula:C29H38N2O6Peso molecolare:510.62Combretastatin A1 phosphate
CAS:<p>Combretastatin A1 phosphate: potent anti-angiogenic and tumor vascular disruptor, with research potential in pancreatic neuroendocrine tumors.</p>Formula:C18H22O12P2Colore e forma:SolidPeso molecolare:492.31Enactin Ia
CAS:<p>Enactin Ia is found in Streptomyces roseoviridis and exhibits mild antibacterial activity.</p>Formula:C20H38N2O6Colore e forma:SolidPeso molecolare:402.526Methyl 5-thia-6,8,11,14-eicosatetraenoate
CAS:<p>Methyl 5-thia-6,8,11,14-eicosatetraenoate is a bioactive chemical.</p>Formula:C20H32O2SColore e forma:SolidPeso molecolare:336.53Azirinomycin
CAS:<p>Azirinomycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C4H5NO2Colore e forma:SolidPeso molecolare:99.088Anti-inflammatory agent 18
<p>Anti-inflammatory agent 18: NO activity blocker (IC50: 15.94 μM), hampers HMGB1-induced inflammation, potential for COVID-19, sepsis study.</p>Formula:C30H50O6Colore e forma:SolidPeso molecolare:506.71Griseorhodin G
CAS:<p>Griseorhodin G is a quinone antibiotic with antitumor activity.</p>Formula:C25H18O12Peso molecolare:510.40Formadicin C
CAS:<p>Formadicin C exhibits the strongest activity among all components against certain strains of Pseudomonas, Proteus, and Alcaligenes.</p>Formula:C24H26N4O10Peso molecolare:530.48BI-207524
CAS:<p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>Formula:C35H36ClN5O5Colore e forma:SolidPeso molecolare:642.14Antileishmanial agent-5
<p>Antileishmanial agent-4, a ribonucleoside analogue, targets L.infantum and T.cruzi with EC50s of 0.68 μM and 0.83 μM.</p>Formula:C17H17ClN4O4Colore e forma:SolidPeso molecolare:376.79MK-2748
CAS:<p>MK-2748 is an inhibitor of NS3 protease, hepatitis C virus.</p>Formula:C42H56N6O10SColore e forma:SolidPeso molecolare:836.99NA 0346
CAS:<p>NA 0346 is a derivative of SF 2370 that shows long lasting antihypertensive action as well as potent protein kinases inhibitory activity.</p>Formula:C26H22N4O3Colore e forma:SolidPeso molecolare:438.48O-GlcNAcase-IN-1
<p>O-GlcNAcase-IN-1 is a potent and novel inhibitor of O-GlcNAcase(OGA) with an IC 50 value of 46 nM.</p>Formula:C15H22N6Colore e forma:SolidPeso molecolare:286.38Tezampanel hydrate
CAS:<p>Tezampanel is used for the treatment of migraine, neuropathic pain.</p>Formula:C13H23N5O3Colore e forma:SolidPeso molecolare:297.35SARS-CoV-2-IN-24
<p>SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.</p>Formula:C27H30N4O5Colore e forma:SolidPeso molecolare:490.55ODN 2088
CAS:<p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>Colore e forma:SolidP-gp modulator 2
<p>P-gp modulator 2 (Compound 27) is a potent competitive and metabotropic P-glycoprotein (P-gp) modulator.</p>Formula:C22H20BrN3O4Colore e forma:SolidPeso molecolare:470.32Fulvoferruginin
CAS:<p>Fulvoferruginin exhibits cytotoxicity and antifungal properties, particularly against Paecilomyces.</p>Formula:C15H18O3Colore e forma:SolidPeso molecolare:246.30Sulprostone
CAS:<p>EP3 and EP1 receptor agonist</p>Formula:C23H31NO7SPurezza:98%Colore e forma:White To Off-White SolidPeso molecolare:465.562-Hydroxy-5-iminoazacyclopent-3-ene
CAS:<p>2-Hydroxy-5-iminoazacyclopent-3-ene is a pyrroline-class antibiotic with mild activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C4H6N2OColore e forma:SolidPeso molecolare:98.103UNC9426
CAS:<p>UNC9426 is an orally active, potent and selective TYRO3 inhibitor with an IC50 of 2.1 nM. UNC9426 reduces platelet aggregation without prolonging bleeding time.</p>Formula:C32H34F6N6OPurezza:98.051%Colore e forma:SolidPeso molecolare:632.642Mimocine
CAS:<p>Mimosine, a plant amino acid, is known to act as a normoxic inducer of hypoxia-inducible factor (HIF).</p>Formula:C15H14N2O5Colore e forma:SolidPeso molecolare:302.28CGC 11144
CAS:<p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>Formula:C40H100Cl10N10Colore e forma:SolidPeso molecolare:1075.82SphK2-IN-2
<p>SphK2-IN-2 (21g) is a potent and selective inhibitor of SphK2 (IC50: 0.23 μM).</p>Formula:C21H25ClN10OColore e forma:SolidPeso molecolare:468.945-cis Carbaprostacyclin
CAS:<p>5-cis Carbaprostacyclin: a PGI2 stable analog; poor human platelet aggregation inhibitor (IC50: 2.8 μM); weakens rabbit artery relaxation (EC50: 104 μM).</p>Formula:C21H34O4Colore e forma:SolidPeso molecolare:350.49Menoxymycin A
CAS:<p>Menoxymycin A is an antibiotic with cytotoxic properties. It inhibits the growth of KB and N18-RE-105 cells, with IC50 values of 0.86 μM and 0.14 μM, respectively.</p>Formula:C24H27NO9Colore e forma:SolidPeso molecolare:473.4732-Hydroxygentamicin C2
CAS:<p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H41N5O8Colore e forma:SolidPeso molecolare:479.568Istamycin Y0
CAS:<p>Istamycin Y0 is an aminoglycoside antibiotic found in *Streptomyces tenjimariensis* [ATCC 31603]. This compound exhibits weak antibacterial activity against only a limited range of bacteria.</p>Formula:C14H30N4O4Colore e forma:SolidPeso molecolare:318.41Cystothiazole A
CAS:<p>Cystothiazole A exhibits antifungal properties, effectively inhibiting Candida albicans, Saccharomyces cerevisiae, and Aspergillus fumigatus with minimum inhibitory concentrations (MIC) of 0.4 μg/mL, 0.1 μg/mL, and 1.6 μg/mL, respectively. It also demonstrates inhibitory activity against human tumor cells such as HPT-116 and K562, with MIC values of 130 ng/mL and 110 ng/mL. However, it shows no antibacterial activity.</p>Formula:C20H26N2O4S2Colore e forma:SolidPeso molecolare:422.561Sannamycin J
CAS:<p>Sannamycin J is an aminoglycoside antibiotic found in *Streptomyces sannanensis* sp. KC-7038. This compound exhibits relatively weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C14H30N4O4Colore e forma:SolidPeso molecolare:318.41Bacithrocin C
CAS:<p>Bacithrocin C is a thrombin inhibitor that suppresses the activity of thrombin, factor Xa, trypsin, and papain, with IC50 values of 80 μM, 15 μM, 1.3 μM, and 0.02 μM, respectively.</p>Formula:C18H27N5O3Colore e forma:SolidPeso molecolare:361.439Endophenazine A
CAS:<p>Endophenazine A exhibits activity against Gram-positive bacteria and filamentous fungi such as Mucor and Penicillium, but demonstrates limited herbicidal effect on Lemna.</p>Formula:C18H16N2O2Colore e forma:SolidPeso molecolare:292.332Rosiptor acetate
CAS:<p>Rosiptor (AQX-1125) activates SHIP1, inhibits Akt, and reduces inflammation and allergy in rodents.</p>Formula:C22H39NO4Purezza:98%Colore e forma:Solid PowderPeso molecolare:381.55PKCiota-IN-1
CAS:<p>PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).</p>Formula:C25H22FN5OColore e forma:SolidPeso molecolare:427.47MPro N3
CAS:<p>Mpro inhibitor blocks MHV-A29, HCoV-229E, FOPV (IC50: 2.7–8.8 μM), and SARS-CoV-2 (IC50: 16.8 μM) in plaque assays.</p>Formula:C35H48N6O8Colore e forma:SolidPeso molecolare:680.79Rhamnitol
CAS:<p>Rhamnitol, the reduction product of L-rhamnose, can be observed during the metabolism of rhamnose in the body. Rhamnitol is promising for use in assessing intestinal permeability and studying carbohydrate metabolism.</p>Formula:C6H14O5Colore e forma:SolidPeso molecolare:166.17NRX-2663
CAS:<p>NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).</p>Formula:C20H13F3N2O5Colore e forma:SolidPeso molecolare:418.32PD-1-IN-17 TFA
<p>PD-1-IN-17 TFA is a potent PD-1 inhibitor, blocking 92% of splenocyte growth at 100 nM.</p>Formula:C15H23F3N6O9Colore e forma:SolidPeso molecolare:488.375(S),6(S)-DiHETE
CAS:<p>5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.</p>Formula:C20H32O4Colore e forma:SolidPeso molecolare:336.47Chicamycin B
CAS:<p>Chicamycin B exhibits antitumor properties and has mild activity against gram-positive bacteria.</p>Formula:C13H14N2O4Colore e forma:SolidPeso molecolare:262.261Glisoprenin E
CAS:<p>Glisoprenin E is an inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT) that can prevent the formation of hydrophobic surface adhesion cells in Pyricularia oryzae.</p>Formula:C45H86O9Colore e forma:SolidPeso molecolare:771.16Feudomycin B
CAS:<p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>Formula:C28H31NO10Colore e forma:SolidPeso molecolare:541.546Dihydroabikoviromycin
CAS:<p>Dihydroabikoviromycin is a secondary metabolite of Streptomyces anulatus and acts as a polyketide synthase inhibitor.</p>Formula:C10H13NOColore e forma:SolidPeso molecolare:163.216Narbomycin
CAS:<p>Narbomycin exhibits activity against Gram-positive bacteria.</p>Formula:C28H47NO7Colore e forma:SolidPeso molecolare:509.675Formadicin A
CAS:<p>Formadicin A exhibits strong activity against various Pseudomonas, Proteus, and Alcaligenes bacteria.</p>Formula:C30H34N4O16Colore e forma:SolidPeso molecolare:706.608Feigrisolide C
CAS:<p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>Formula:C21H36O7Colore e forma:SolidPeso molecolare:400.506Deoxyfrenolicin
CAS:<p>Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.</p>Formula:C18H18O6Colore e forma:SolidPeso molecolare:330.332PD-1/PD-L1-IN-16
<p>PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.</p>Formula:C34H30N4O4Colore e forma:SolidPeso molecolare:558.634"-Demethylgentamicin C2
CAS:<p>4"-Demethylgentamicin C2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C19H39N5O7Colore e forma:SolidPeso molecolare:449.54Dermostatin B
CAS:<p>Dermostatin B is a polyene antibiotic with antifungal properties, suitable for research on fungal infections.</p>Formula:C41H66O11Colore e forma:SolidPeso molecolare:734.956CXCR4 probe 1
CAS:<p>CXCR4 probe 1, a specific PET tracer, targets CXCR4 with antagonist TN14003 (IC50: 6.9 nM), aiding in imaging CXCR4-related diseases and tumors.</p>Formula:C24H30FN5O4SColore e forma:SolidPeso molecolare:502.59Haloquinone
CAS:<p>Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.</p>Formula:C17H12O5Colore e forma:SolidPeso molecolare:296.274Vulolisib
CAS:<p>Vulolisib inhibits PI3K (α: IC50 0.2nM, β: 168nM, γ: 90nM, δ: 49nM), taken orally with anti-cancer properties.</p>Formula:C18H19F2N5O3SColore e forma:SolidPeso molecolare:423.444-Nitrochalcone
CAS:<p>4-Nitrochalcone (2-(4-Nitrobenzylidene)acetophenone) inhibits proteasomes and suppresses TNFα-induced NF-κB activity.</p>Formula:C15H11NO3Colore e forma:SolidPeso molecolare:253.257(Z),11(Z)-Nonacosadiene
CAS:<p>7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.</p>Formula:C29H56Colore e forma:SolidPeso molecolare:404.75Pyloricidin A2
CAS:<p>Pyloricidin A2 is an antibiotic effective against Helicobacter pylori, produced by Bacillus species HC-70. It exhibits strong anti-Helicobacter pylori activity but shows no activity against other bacteria and yeast.</p>Formula:C32H53N5O10Colore e forma:SolidPeso molecolare:667.79Fudecalone
CAS:<p>Fudecalone is produced by the Penicillium strain FO-2030. It completely inhibits the coccidian parasite Eimeria Tenella that is resistant to Monensin.</p>Formula:C15H22O3Colore e forma:SolidPeso molecolare:250.33BW A868C
CAS:BW A868C is a potent, selective PGD2 antagonist and a BW245C analogue, inert to other prostaglandin receptors.Formula:C25H37N3O5Colore e forma:SolidPeso molecolare:459.5811-Hydroxynovobiocin
CAS:<p>11-Hydroxynovobiocin exhibits activity against Gram-negative bacteria.</p>Formula:C31H36N2O12Colore e forma:SolidPeso molecolare:628.62Ophiobolin D
CAS:<p>Ophiobolin D is a terpene antibiotic with mild inhibitory effects on Staphylococcus aureus.</p>Formula:C25H36O4Colore e forma:SolidPeso molecolare:400.55Heme Oxygenase-2-IN-1
<p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>Formula:C19H17N3O2Colore e forma:SolidPeso molecolare:319.36CGP 22979
CAS:<p>CGP 22979 is a renal selective vasodilator prodrug.</p>Formula:C16H24N4O4Colore e forma:SolidPeso molecolare:336.39PD-L1-IN-1
<p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>Formula:C21H23N5O2Colore e forma:SolidPeso molecolare:377.44Pyrisulfoxin A
CAS:<p>Pyrisulfoxin A is an antibiotic that can be found in Streptomyces callfornicus [BS-75].</p>Formula:C13H13N3O3SColore e forma:SolidPeso molecolare:291.326Seldomycin factor 1
CAS:<p>Seldomycin factor 1 (XK 88-1) is an aminoglycoside antibiotic known for its broad-spectrum antibacterial activity.</p>Formula:C17H34N4O10Colore e forma:SolidPeso molecolare:454.473Kigamicin A
CAS:<p>Kigamicin A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) ranging from 0.025 to 0.78 μg/mL.</p>Formula:C34H35NO13Colore e forma:SolidPeso molecolare:665.64Matlystatin F
CAS:<p>Matlystatin F is an inhibitor of metalloproteinases (MMP).</p>Formula:C27H44N6O6Colore e forma:SolidPeso molecolare:548.675LY3325656
CAS:<p>LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.</p>Formula:C21H23F3N6O2Colore e forma:SolidPeso molecolare:448.44Thiazolo[5,4-c]pyridin-4(5H)-one
CAS:<p>Thiazolo[5,4-c]pyridin-4(5H)-one is a compound used for diagnostic imaging of TDP-43, in PET imaging of neurodegenerative diseases ALS、AD、FTD、LATE.</p>Formula:C22H22FN5O2SPurezza:98.75%Colore e forma:SolidPeso molecolare:439.51Plumbemycin A
CAS:<p>Plumbemycin A is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Formula:C12H20N3O9PColore e forma:SolidPeso molecolare:381.28Chandrananimycin C
CAS:<p>Chandrananimycin C exhibits activity against Mucor fungi and demonstrates anti-tumor properties against cancer cell lines such as CCL HT29, MFXF 529L, and MACL McF-7.</p>Formula:C17H16N2O3Colore e forma:SolidPeso molecolare:296.32Quorum Sensing-IN-1
<p>Quorum Sensing-IN-1 is a small-molecule inhibitor of quorum sensing.</p>Formula:C13H10N2O2S2Colore e forma:SolidPeso molecolare:290.36Exatecan-amide-cyclopropanol
CAS:<p>Exatecan-amide-cyclopropanol potently inhibits SK-BR-3 and U87 cancer cells (IC50 0.12 and 0.23 nM)</p>Formula:C28H26FN3O6Purezza:98.308%Colore e forma:SolidPeso molecolare:519.52Hydroxynybomycin
CAS:<p>Hydroxynybomycin is an antibiotic with activity against Gram-negative bacteria.</p>Formula:C16H14N2O5Colore e forma:SolidPeso molecolare:314.293C20 Sphingomyelin (d18:1/20:1)
CAS:<p>C20 Sphingomyelin (d18:1/20:1) (Compound SM:20:1) is a type of sphingolipid. This compound shows potential for research related to motor neuron diseases, such as amyotrophic lateral sclerosis (ALS) and primary lateral sclerosis (PLS).</p>Formula:C43H85N2O6PColore e forma:SolidPeso molecolare:757.119Melithiazole B
CAS:<p>Melithiazol B is an antibiotic and a potent inhibitor of β-methoxyacrylate (MOA), with both antifungal and cytotoxic properties.</p>Formula:C20H24N2O4S2Colore e forma:SolidPeso molecolare:420.546Hypnophilin
CAS:<p>Hypnophilin exhibits multiple activities, including effectiveness against Gram-positive bacteria, Gram-negative bacteria, yeasts, molds, and tumors.</p>Formula:C15H20O3Colore e forma:SolidPeso molecolare:248.318Phosmidosine
CAS:<p>Phosmidosine inhibits cell cycle progression and morphological recovery in srcts-NRK cells. Additionally, Phosmidosine exhibits antifungal properties.</p>Formula:C16H24N7O8PColore e forma:SolidPeso molecolare:473.38Belatacept
CAS:<p>Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.</p>Colore e forma:LiquidB-3852
CAS:<p>B-3852 is a Bradykinin inhibitor.</p>Formula:C55H74F3N15O11Colore e forma:SolidPeso molecolare:1178.27Calphostin A
CAS:<p>Calphostins, from Cladosporium fungus, inhibit PKC; calphostin C is most potent, used as a biochemical tool.</p>Formula:C44H38O12Colore e forma:SolidPeso molecolare:758.77Glidobactin B
CAS:<p>Glidobactin B is an antitumor antibiotic. It is active against pathogenic fungi and yeasts and can prolong the survival time of mice inoculated with leukemia P388 cells.</p>Formula:C29H46N4O6Colore e forma:SolidPeso molecolare:546.699Echinocandin B nucleus
CAS:<p>Echinocandin B nucleus (A-30912 A nucleus) is the reaction product catalyzed by Echinocandin B decarboxylase. It serves as an intermediate in the semisynthetic production of antifungal agents.</p>Formula:C34H51N7O15Colore e forma:SolidPeso molecolare:797.807Carnostatine
<p>Carnostatine (SAN9812), a potent CN1 inhibitor with 11 nM K i, may boost renal carnosine to treat DN.</p>Formula:C10H16N4O4Purezza:98%Colore e forma:SolidPeso molecolare:256.26Ayapin
CAS:<p>Ayapin, found in sunflowers, is a primary plant phytoalexin. It inhibits the growth of S. scerorotiorum, with an IC50 of 0.16 mM indicating 50% inhibition. Ayapin is utilized in studies on controlling sclerotinia stem rot.</p>Formula:C10H6O4Colore e forma:SolidPeso molecolare:190.15OUN58101
CAS:<p>OUN58101, also MDK-8101/BI-D, is an RSV L-protein inhibitor with no formal name, first reported in patent WO 2005042530.</p>Formula:C32H36N6O6Colore e forma:SolidPeso molecolare:600.66Melithiazole A
CAS:<p>Melithiazol A is an antibiotic and a potent β-methoxyacrylate (MOA) inhibitor with antifungal and cytotoxic properties.</p>Formula:C20H26N2O4S2Colore e forma:SolidPeso molecolare:422.5615-Hydroxymethylblasticidin S
CAS:<p>5-Hydroxymethylblasticidin S is a broad-spectrum antibiotic found in Streptomyces setonii.</p>Formula:C18H28N8O6Colore e forma:SolidPeso molecolare:452.465Acetylstachyflin
CAS:<p>Acetylstachyflin is an antibiotic effective against the influenza A virus.</p>Formula:C25H33NO5Colore e forma:SolidPeso molecolare:427.53Salvinorin A Propionate
CAS:<p>Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.</p>Formula:C24H30O8Colore e forma:SolidPeso molecolare:446.49Cinatrin C2
CAS:<p>Cinatrin C2, a phospholipase A2 (PLA2) inhibitor, has an IC50 value of 800 μM and can be extracted from the Circinotrichum falcatisporum strain RF-641.</p>Formula:C18H30O8Colore e forma:SolidPeso molecolare:374.426Purine phosphoribosyltransferase-IN-2
<p>Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.</p>Formula:C11H15N5Na4O10P2Colore e forma:SolidPeso molecolare:531.17Exfoliazone
CAS:<p>Exfoliazone is a phenazinic antibiotic with activity against Trichoderma viride, exhibiting an ED50 for inhibiting mycelial growth of 70 μg/mL.</p>Formula:C15H12N2O4Colore e forma:SolidPeso molecolare:284.267PI3K-IN-23
<p>PI3K-IN-23 is a (E)-9-oxooctadec-10-en-12-ynoic acid analogue that promotes glucose uptake (EC50: 7.00 μM).</p>Formula:C24H33NO4SColore e forma:SolidPeso molecolare:431.59Fluoropolyoxin L
CAS:<p>Fluoropolyoxin L exhibits inhibitory activity against Escherichia coli and Enterococcus faecalis.</p>Formula:C16H22FN5O12Colore e forma:SolidPeso molecolare:495.371Miyakamide A2
CAS:<p>Miyakamide A2 is an antibiotic with insecticidal properties. It inhibits the growth of brine shrimp and exhibits weak activity against Xanthomonas species. The IC50 for inhibiting P388 cells is 12.2 μg/mL.</p>Formula:C31H32N4O3Colore e forma:SolidPeso molecolare:508.611TP-030-1
CAS:<p>TP-030-1, RIPK1 inhibitor: K(i) hRIPK1 at 3.9nM, IC50 mRIPK1 at 4.2μM; targets inflammation, neurodegeneration research.</p>Formula:C23H22N4O3Colore e forma:SolidPeso molecolare:402.45NSC 357754
CAS:NSC 357754 is an inhibitor of Claudin. It can enhance transepithelial electrical resistance and reduce specific cation permeability. NSC 357754 is useful for research involving Claudin-2 and/or Claudin-15 mediated intestinal disorders.Formula:C26H20N4O2Colore e forma:SolidPeso molecolare:420.463Kigamicin B
CAS:<p>Kigamicin B exhibits activity against gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) ranging from 0.025 to 0.78 μg/mL.</p>Formula:C40H45NO15Colore e forma:SolidPeso molecolare:779.78TCMDC-125431
<p>TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.</p>Formula:C25H27N3O2SColore e forma:SolidPeso molecolare:433.57HS-731
CAS:<p>HS-731 is a μ-Opioid Receptor Agonist.</p>Formula:C20H26N2O5Colore e forma:SolidPeso molecolare:374.43Glutaminyl cyclases-IN-1
<p>Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.</p>Formula:C25H30N6O2SColore e forma:SolidPeso molecolare:478.61Z57346765
CAS:<p>Z57346765 is a specific PGK1 inhibitor that inhibits PGK1-dependent cell proliferation by decreasing the metabolic enzyme activity of PGK1 during glycolysis.</p>Formula:C17H18N4OPurezza:99.85%Colore e forma:SolidPeso molecolare:294.35Antiplatelet agent 3
CAS:<p>Antiplatelet agent 3 (Compound K-10) is a compound with antiplatelet aggregation activity, exhibiting IC50 values of 2.55, 3.22, and 2.09 mg/mL for platelet aggregation induced by ADP, AA, and COL, respectively. It holds potential for research in cardiovascular diseases.</p>Formula:C38H32N2O5Colore e forma:SolidPeso molecolare:596.671GSK3527497 HCl
CAS:<p>GSK3527497: potent TRPV4 inhibitor, IC50=12 nM, targets heart/respiratory issues, for oral/IV use, low-dose effective.</p>Formula:C17H17Cl2FN4O4SColore e forma:SolidPeso molecolare:463.3054Cuevaene A
CAS:<p>Cuevaene A can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. It exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and demonstrates moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>Formula:C21H22O5Colore e forma:SolidPeso molecolare:354.396

