Altri inibitori
Questa categoria comprende una vasta gamma di inibitori che non rientrano nelle classificazioni standard ma sono comunque fondamentali per varie ricerche biochimiche e farmacologiche. Questi inibitori possono bersagliare vie, enzimi e interazioni molecolari uniche o meno studiate, fornendo strumenti preziosi per aree di ricerca specializzate. Presso CymitQuimica, offriamo una selezione diversificata di inibitori di alta qualità che coprono molteplici bersagli biologici e discipline di ricerca, permettendoti di esplorare nuove strade terapeutiche e approfondire la tua comprensione dei processi biologici complessi.
Trovati 37827 prodotti di "Altri inibitori"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Phosmidosine
CAS:<p>Phosmidosine inhibits cell cycle progression and morphological recovery in srcts-NRK cells. Additionally, Phosmidosine exhibits antifungal properties.</p>Formula:C16H24N7O8PColore e forma:SolidPeso molecolare:473.38Clavicoronic acid
CAS:<p>Clavicoronic acid, a β-lactamase inhibitor, boosts penicillin antibiotics against resistant bacteria.</p>Formula:C15H18O4Colore e forma:SolidPeso molecolare:262.3Eprociclovir Na
CAS:<p>Eprociclovir Na (A-5021) is 15x stronger than acyclovir at inhibiting herpesviruses, showing promise for EHV1 and herpetic keratitis treatment.</p>Formula:C11H14N5NaO3Colore e forma:SolidPeso molecolare:287.25PDE-I2
CAS:<p>PDE-I2 is a parasite schizogony inhibitor.</p>Formula:C25H23N5O8Colore e forma:SolidPeso molecolare:521.48Oleuroside
CAS:<p>Oleuroside can protect against mitochondrial dysfunction in models of early Alzheimer's disease and brain ageing.</p>Formula:C25H32O13Purezza:98%Colore e forma:SolidPeso molecolare:540.51Melithiazole A
CAS:<p>Melithiazol A is an antibiotic and a potent β-methoxyacrylate (MOA) inhibitor with antifungal and cytotoxic properties.</p>Formula:C20H26N2O4S2Colore e forma:SolidPeso molecolare:422.561Scorodonin
CAS:<p>SScorodonin exhibits antibacterial, antistreptomycete, and antifungal properties. It inhibits DNA-dependent RNA polymerase with an IC50 of 25 μg/mL.</p>Formula:C7H7ClOColore e forma:SolidPeso molecolare:142.583Damavaricin D
CAS:<p>Damavaricin D exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>Formula:C38H49NO12Colore e forma:SolidPeso molecolare:711.795ABCA1 inducer 1
CAS:<p>ABCA1 inducer 1, a non-lipid inducer of ABCA1, enhances ABCA1 expression in E3/4FAD mice expressing human APOE 3/4, augments the lipidation of apolipoprotein (APOE), and reverses various Alzheimer's disease (AD) phenotypes without increasing triglycerides.</p>Formula:C24H24Cl2N2O7S2Colore e forma:SolidPeso molecolare:587.49UTPγS trisodium salt
CAS:<p>P2Y2 and P2Y4 receptor agonist</p>Formula:C9H12N2Na3O14P3SPurezza:98%Colore e forma:SolidPeso molecolare:566.15Bagremycin B
CAS:<p>Bagremycin B is produced by the bacterium Streptomyces strain Tu 4128. It exhibits weak activity against Gram-positive bacteria, Saccharomyces cerevisiae, and Candida albicans.</p>Formula:C17H15NO4Colore e forma:SolidPeso molecolare:297.305Ezomycin A1
CAS:<p>Ezomycin A1 is an antifungal antibiotic effective primarily against plant pathogens such as Sclerotinia and Botrytis. It is used to prevent and control diseases like Sclerotinia rot, gray mold, and candidiasis in crops.</p>Formula:C26H38N8O15SColore e forma:SolidPeso molecolare:734.69Acetylstachyflin
CAS:<p>Acetylstachyflin is an antibiotic effective against the influenza A virus.</p>Formula:C25H33NO5Colore e forma:SolidPeso molecolare:427.53AVE-1330A sodium
CAS:<p>AVE-1330A sodium is a beta-Lactamase inhibitor.</p>Formula:C7H10N3NaO6SColore e forma:SolidPeso molecolare:287.23Luffariellolide
CAS:<p>Luffariellolide is a terpene compound obtained from the marine sponge Hyrtios communis that is an HSF-PLA2 inhibitor and a RAR agonist.</p>Formula:C25H38O3Purezza:98%Colore e forma:SolidPeso molecolare:386.57Heparastatin
CAS:<p>Heparastatin is an inhibitor of heparanase.</p>Formula:C8H11F3N2O5Purezza:98%Colore e forma:SolidPeso molecolare:272.18GRPR antagonist-2
<p>GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) & Pan02 (IC50: 2.5 μM).</p>Formula:C28H32F3N5O4Colore e forma:SolidPeso molecolare:559.58ALK5-IN-82
CAS:<p>ALK5-IN-82 is a potent and selective inhibitor of activin receptor-like kinase 5 (ALK5), demonstrating an IC50 value of 9.1 nM. This compound effectively suppresses the expression of α-smooth muscle actin (α-SMA), collagen I, and the proteinases tissue inhibitor of metalloproteinase 1 (TIMP-1) and matrix metalloproteinase 13 (MMP-13) in human umbilical vein endothelial cells induced by transforming growth factor-β. ALK5-IN-82 shows potential for use in research related to cardiac fibrosis.</p>Formula:C22H19N7OSColore e forma:SolidPeso molecolare:429.50Cinatrin C2
CAS:<p>Cinatrin C2, a phospholipase A2 (PLA2) inhibitor, has an IC50 value of 800 μM and can be extracted from the Circinotrichum falcatisporum strain RF-641.</p>Formula:C18H30O8Colore e forma:SolidPeso molecolare:374.426BM635 mesylate (1493762-74-5 free base)
BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).Formula:C26H33FN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:488.61(1R,3S)-THCCA-Asn
<p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>Formula:C24H24N4O6Colore e forma:SolidPeso molecolare:464.47Dynemicin Q
CAS:<p>Dynemicin Q is an antibiotic that demonstrates potent activity against Gram-positive bacteria.</p>Formula:C28H19NO9Colore e forma:SolidPeso molecolare:513.45Hypnophilin
CAS:<p>Hypnophilin exhibits multiple activities, including effectiveness against Gram-positive bacteria, Gram-negative bacteria, yeasts, molds, and tumors.</p>Formula:C15H20O3Colore e forma:SolidPeso molecolare:248.31820-Deoxysalinomycin
CAS:<p>20-Deoxysalinomycin primarily targets Gram-positive bacteria, with a particular effectiveness against poultry coccidia.</p>Formula:C42H70O10Colore e forma:SolidPeso molecolare:735.00HbF inducer-1
<p>HbF inducer-1 is a fetal hemoglobin inducer which is orally bioavailable.</p>Formula:C18H19N3O3Colore e forma:SolidPeso molecolare:325.36SORT1-IN-1
CAS:<p>SORT1-IN-1 (compound 2) is a SORT1 inhibitor.</p>Formula:C17H13F3N2O4Colore e forma:SolidPeso molecolare:366.29Vicanicin
CAS:<p>Vicanicin is an aryl phenol ether compound found in lichens. It inhibits the expression of Hsp70, modulates intracellular redox-sensitive mechanisms, increases reactive oxygen species (ROS) in cancer cells, alters the Bax/Bcl-2 ratio, activates caspase-3, and induces apoptosis. Vicanicin suppresses cell growth and promotes apoptosis in androgen-sensitive (LNCaP) and androgen-insensitive (DU-145) human prostate cancer cells. It holds potential for prostate cancer research.</p>Formula:C18H16Cl2O5Colore e forma:SolidPeso molecolare:383.223KF-19418
CAS:<p>KF-19418 is a follicle stimulant that directly activates follicles in vitro and promotes hair growth in vivo.</p>Formula:C21H14N4OColore e forma:SolidPeso molecolare:338.368,9-Epoxyeicosatrienoic acid
CAS:<p>8,9-Epoxyeicosatrienoic acid offers unique protective effects on the glomerulus. It inhibits the increase in glomerular albumin permeability caused by circulating permeability factors (FSPF). Additionally, 8,9-Epoxyeicosatrienoic acid is used in research related to glomerular dysfunction.</p>Formula:C20H32O3Colore e forma:SolidPeso molecolare:320.47Antileishmanial agent-6
<p>Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.</p>Formula:C24H26O8Colore e forma:SolidPeso molecolare:442.46Erizepine
CAS:<p>Erizepine, an octopamine receptor 3 (OAR3) antagonist, exhibits a Ki value of 474 nM. This compound is utilized in insect research.</p>Formula:C20H22N2Colore e forma:SolidPeso molecolare:290.4LK-732
CAS:<p>LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.</p>Formula:C25H29N5O3SColore e forma:SolidPeso molecolare:479.59Ro-51
CAS:<p>dual P2X3 and P2X2/3 antagonist</p>Formula:C17H23IN4O4Purezza:98%Colore e forma:SolidPeso molecolare:474.29Aspochalasin M
CAS:<p>Aspochalasin M shows moderate activity on HL-60 cells (IC50=20.0 μ M). Aspochalasin M has research potential in leukemia diseases.</p>Formula:C24H35NO4Colore e forma:SolidPeso molecolare:401.54Melithiazole B
CAS:<p>Melithiazol B is an antibiotic and a potent inhibitor of β-methoxyacrylate (MOA), with both antifungal and cytotoxic properties.</p>Formula:C20H24N2O4S2Colore e forma:SolidPeso molecolare:420.546Peptaibolin
CAS:<p>Peptaibolin exhibits activity against Gram-positive bacteria and yeast. The minimum inhibitory concentration (MIC) for its effect on Bacillus subtilis [ATCC 6633] and Candida albicans is 100 μg/mL.</p>Formula:C31H51N5O6Colore e forma:SolidPeso molecolare:589.77Iodinin
CAS:<p>Iodinin is an antibiotic with antibacterial and antifungal properties.</p>Formula:C12H8N2O4Colore e forma:SolidPeso molecolare:244.203Lactaroviolin
CAS:<p>Lactaroviolin is an aromatic derivative antibiotic that can inhibit the growth of Mycobacterium tuberculosis.</p>Formula:C15H14OColore e forma:SolidPeso molecolare:210.271D6808
<p>D6808: selective c-Met inhibitor, IC50=2.9 nM, induces apoptosis and cell cycle arrest, for NSCLC/gastric cancer research.</p>Formula:C30H25F3N6O2Colore e forma:SolidPeso molecolare:558.55DD04107
CAS:<p>DD04107 inhibits α-CGRP release, targets Synaptotagmin 1 in sensory neurons.</p>Formula:C48H88N14O12SColore e forma:SolidPeso molecolare:1085.36Isobetanin
CAS:<p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>Formula:C24H26N2O13Colore e forma:SolidPeso molecolare:550.47VEGFR-2-IN-17
<p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>Formula:C21H14ClN3O2Colore e forma:SolidPeso molecolare:375.81Chloronectrin
CAS:<p>Chloronectrin exhibits activity against Gram-positive bacteria.</p>Formula:C25H33ClO6Colore e forma:SolidPeso molecolare:464.979FTI-2148
CAS:<p>FTI-2148 blocks RAS-related FT-1 & GGT-1; IC50: 1.4 nM & 1.7 μM.</p>Formula:C24H28N4O3SPurezza:98%Colore e forma:SolidPeso molecolare:452.57Odiparcil
CAS:<p>Odiparcil is an orally active beta-d-thioxyloside analog.</p>Formula:C15H16O6SPurezza:98%Colore e forma:SolidPeso molecolare:324.35Pyrrolomycin A
CAS:<p>Pyrrolomycin A is a pyrrole antibiotic that exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>Formula:C4H2Cl2N2O2Colore e forma:SolidPeso molecolare:180.977Milbemycin α11
CAS:<p>Milbemycin α11 (Meilingmycin A) is an antibiotic known for its ability to eliminate nematodes and mites.</p>Formula:C36H50O9Colore e forma:SolidPeso molecolare:626.781-Deamino-1-hydroxysagamicin
CAS:<p>1-Deamino-1-hydroxysagamicin (AntibioticSUM-3) is an aminoglycoside antibiotic that is effective against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H40N4O8Colore e forma:SolidPeso molecolare:464.554Mevidalen HBA
CAS:<p>Mevidalen (LY3154207), a potent D1 positive allosteric modulator, is in clinical trials for Lewy body dementia.</p>Formula:C31H35Cl2NO6Colore e forma:SolidPeso molecolare:588.52Griseochelin
CAS:<p>Griseochelin exhibits activity against Gram-negative bacteria and inhibits Coccidioides.</p>Formula:C33H60O7Colore e forma:SolidPeso molecolare:568.825Phenazostatin B
CAS:<p>Phenazostatin B is a phenazine derivative known for its neuroprotective properties. It acts by scavenging free radicals, protecting N18-RE 105 neuronal cells from glutamate-induced toxicity, and inhibiting lipid peroxidation. It inhibits glutamate toxicity in N18-RE-105 cells, with an EC50 of 0.33 μg/mL.</p>Formula:C32H26N4O4Colore e forma:SolidPeso molecolare:530.57Fortimicin B
CAS:<p>Fortimicin B exhibits weak antibacterial activity.</p>Formula:C15H32N4O5Colore e forma:SolidPeso molecolare:348.43820-HEDE
CAS:20-HEDE (WIT 002) is a 20-hydroxyeicosatetraenoic acid (20-HETE) antagonist.Formula:C20H36O3Purezza:98%Colore e forma:SolidPeso molecolare:324.50DC41
CAS:<p>DC41 is a CC-1065-based cancer drug, an antibody-linked DNA alkylator.</p>Formula:C37H34ClN5O4SPurezza:98%Colore e forma:SolidPeso molecolare:680.22DLCI-1
CAS:<p>DLCI-1 is a potent and selective oral inhibitor of cytochrome P450 2A6 (CYP2A6), significantly reducing self-administered nicotine doses in both male and female mice.</p>Formula:C12H14N2SColore e forma:SolidPeso molecolare:218.32MRS2279
CAS:<p>Selective, high affinity competitive antagonist of the P2Y1 receptor</p>Formula:C13H18ClN5O8P2Purezza:98%Colore e forma:SolidPeso molecolare:469.71Octahydrocyclopenta[c]pyrrole
CAS:Octahydrocyclopenta[c]pyrrole has demonstrated promising applications in the fields of anti-inflammatory, anti-tumor, and neuroprotection. The unique structure-activity relationship of Octahydrocyclopenta[c]pyrrole offers fresh insights for the design of new drugs.Formula:C7H13NColore e forma:SolidPeso molecolare:111.18SID 125240931
CAS:<p>SID 125240931 is a regulator of fluorine-activated proteins (FAPs). This compound disrupts the binding between fluoride and FAPs.</p>Formula:C19H24N4O3SColore e forma:SolidPeso molecolare:388.48Ledene
CAS:<p>Ledene (Viridiflorene) is an essential oil produced by viridiflorene synthase.</p>Formula:C15H24Purezza:98%Colore e forma:SolidPeso molecolare:204.35DWN-12088 HCl
CAS:<p>DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitor</p>Formula:C15H21Cl4N3OColore e forma:SolidPeso molecolare:401.15ART615
<p>ART615 is a related isomer of ART558. ART615 inhibits Polθ by <10% at 12 μM and is able to act as a control for ART558 (IC50:7.9 nM).</p>Formula:C21H21F3N4O2Colore e forma:SolidPeso molecolare:418.4115:0-18:1 DG
CAS:<p>15:0-18:1 DG is a form of diacylglycerol (DAG). It is produced by the hydrolysis of triacylglycerol (TAG) found in butter. This compound shows potential for research in obesity, cardiovascular diseases, and dietary interventions.</p>Formula:C36H68O5Colore e forma:SolidPeso molecolare:580.922Rafutrombopag
CAS:<p>Rafutrombopag is a thrombopoietin (TPO) agonist.</p>Formula:C25H22N4O5Colore e forma:SolidPeso molecolare:458.47Miyakamide B1
CAS:<p>Miyakamide B1 is an antibiotic with insecticidal properties, capable of inhibiting the growth of brine shrimp. It displays moderate activity against Xanthomonas bacteria and inhibits P388 cells with an IC50 of 8.8 μg/mL.</p>Formula:C31H32N4O4Colore e forma:SolidPeso molecolare:524.61UCN-02
CAS:<p>UCN-02 (7-epi-Hydroxystaurosporine) is a PKC inhibitor produced by Streptomyces N-126 strain, which inhibits PKA.</p>Formula:C28H26N4O4Purezza:98%Colore e forma:SolidPeso molecolare:482.53Resolvin E2
CAS:<p>RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.</p>Formula:C20H30O4Colore e forma:SolidPeso molecolare:334.45ZK-Thiazolidinone
CAS:<p>ZK-Thiazolidinone (TAL), ATP-competitive PLK1 inhibitor, disrupts cell division processes in vitro and in vivo, targeting human/mouse tumors.</p>Formula:C23H26F3N5O2SColore e forma:SolidPeso molecolare:493.55Isoleucyl tRNA synthetase-IN-1
CAS:<p>Isoleucyl tRNA synthetase-IN-1 is a selective and potent inhibitor (Ki: 88 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formula:C23H35N5O7SColore e forma:SolidPeso molecolare:525.62MCTR2
CAS:<p>MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.</p>Formula:C27H40N2O6SColore e forma:SolidPeso molecolare:520.68Nemotin
CAS:<p>Nemotin exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while its effectiveness against Gram-negative bacteria is present but relatively weaker.</p>Formula:C11H8O2Colore e forma:SolidPeso molecolare:172.18Plm IV inhibitor-2
CAS:<p>"Plm IV inhibitor-2: Potent for Plm IV (IC50=24nM), affects Plm II/Plm I; malaria research compound."</p>Formula:C39H54N4O4Colore e forma:SolidPeso molecolare:642.87Fudecalone
CAS:<p>Fudecalone is produced by the Penicillium strain FO-2030. It completely inhibits the coccidian parasite Eimeria Tenella that is resistant to Monensin.</p>Formula:C15H22O3Colore e forma:SolidPeso molecolare:250.33AVE 0991
CAS:<p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>Formula:C29H32N4O5S2Purezza:98.69%Colore e forma:SolidPeso molecolare:580.72GG-43
<p>GG-43 is a potent inhibitor of LIN28. The IC50 value of GG-43 against human LIN28A is 4 μM [1].</p>Formula:C21H21NO3Colore e forma:SolidPeso molecolare:335.4Thiazolo[5,4-c]pyridin-4(5H)-one
CAS:<p>Thiazolo[5,4-c]pyridin-4(5H)-one is a compound used for diagnostic imaging of TDP-43, in PET imaging of neurodegenerative diseases ALS、AD、FTD、LATE.</p>Formula:C22H22FN5O2SPurezza:98.75%Colore e forma:SolidPeso molecolare:439.51Coleon-U-quinone
CAS:<p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>Formula:C20H24O5Colore e forma:SolidPeso molecolare:344.4IACS-8779
CAS:<p>IACS-8779 is a potent STING agonist that efficiently stimulates interferon gene activity and exhibits strong systemic antitumor effects.</p>Formula:C21H25N9O10P2S2Purezza:98%Colore e forma:SolidPeso molecolare:689.55Antiplatelet agent 3
CAS:<p>Antiplatelet agent 3 (Compound K-10) is a compound with antiplatelet aggregation activity, exhibiting IC50 values of 2.55, 3.22, and 2.09 mg/mL for platelet aggregation induced by ADP, AA, and COL, respectively. It holds potential for research in cardiovascular diseases.</p>Formula:C38H32N2O5Colore e forma:SolidPeso molecolare:596.671Cuevaene A
CAS:<p>Cuevaene A can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. It exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and demonstrates moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>Formula:C21H22O5Colore e forma:SolidPeso molecolare:354.396Pyrrolomycin E
CAS:<p>Pyrrolomycin E is a pyrrole-based antibiotic with activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>Formula:C10H5Cl3N2O3Colore e forma:SolidPeso molecolare:307.517VU0463271 quarterhydrate
<p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>Formula:C19H20N4O2S2Colore e forma:SolidPeso molecolare:387O-Desmethyl Midostaurin
CAS:O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.Formula:C34H28N4O4Purezza:98%Colore e forma:SolidPeso molecolare:556.61Chloroquinocin
CAS:<p>Chloroquinocin exhibits moderate activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA).</p>Formula:C17H15ClO5Colore e forma:SolidPeso molecolare:334.751Unoprostone isopropyl
CAS:<p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>Formula:C25H44O5Purezza:98%Colore e forma:SolidPeso molecolare:424.61PRN694
CAS:<p>PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.</p>Formula:C28H35F2N5O2SPurezza:98%Colore e forma:SolidPeso molecolare:543.6710-Hydroxyundeca-2,4,6,8-tetraynamide
CAS:<p>10-Hydroxyundeca-2,4,6,8-tetraynamide is a polyacetylene antibiotic exhibiting activity against Gram-positive and Gram-negative bacteria, yeasts, fungi, as well as cytotoxic properties.</p>Formula:C11H7NO2Colore e forma:SolidPeso molecolare:185.179ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Formula:C23H26Cl2N2O3Colore e forma:SolidPeso molecolare:449.37ER Thermo Yellow
CAS:<p>ER Thermo Yellow is a high-sensitivity (3.9%/°C) fluorescent probe designed for temperature visualization specifically targeting the endoplasmic reticulum.</p>Formula:C27H20BClF5N3O3Peso molecolare:575.72PTP1B-IN-3 diammonium
<p>PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.</p>Formula:C12H13BrF2N3O3PColore e forma:SolidPeso molecolare:396.12(±)-HIP-B
CAS:<p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>Formula:C6H8N2O4Purezza:98%Colore e forma:SolidPeso molecolare:172.14Mycoversilin
CAS:<p>Mycoversilin is an antibiotic with inhibitory activity against dermatophytes and plant pathogenic fungi, but it does not exhibit activity against yeasts and bacteria. It strongly inhibits protein synthesis.</p>Formula:C18H16O8Colore e forma:SolidPeso molecolare:360.315GSK1820795A
CAS:<p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>Formula:C35H34N8Colore e forma:SolidPeso molecolare:566.7FMK-MEA
CAS:<p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>Formula:C21H26FN5O2Purezza:98%Colore e forma:SolidPeso molecolare:399.46Orvepitant
CAS:<p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>Formula:C31H35F7N4O2Colore e forma:SolidPeso molecolare:628.62Chitinovorin A
CAS:<p>Chitinovorin A is a β-lactam antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>Formula:C26H41N9O11SColore e forma:SolidPeso molecolare:687.722EP4 receptor antagonist 2
CAS:<p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>Formula:C27H29N3O5Colore e forma:SolidPeso molecolare:475.54Lucilactaene
CAS:<p>Lucilactaene exhibits potent antimalarial activity and functions as a P53-transfected tumor cell cycle inhibitor. It effectively halts the cell cycle progression of H1299/TSP53 cells at the G1 phase.</p>Formula:C22H27NO6Peso molecolare:401.45Melanoxazal
CAS:<p>Melanoxazal is an inhibitor of melanin biosynthesis, effectively suppressing melanin formation in silkworm larva hemolymph with an IC50 of 30.1 μg/mL, and it also exhibits strong inhibitory effects on mushroom tyrosinase (IC50 of 4.2 μg/mL), while lacking antibacterial activity.</p>Formula:C8H9NO3Peso molecolare:167.16Polyoxin L
CAS:<p>Polyoxin L is a nucleoside-type antifungal antibiotic that is notably effective against rice sheath blight.</p>Formula:C16H23N5O12Peso molecolare:477.38Henagliflozin
CAS:<p>Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.</p>Formula:C22H24ClFO7Colore e forma:SolidPeso molecolare:454.87Haloquinone
CAS:<p>Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.</p>Formula:C17H12O5Colore e forma:SolidPeso molecolare:296.274Griseolutein A
CAS:<p>Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C17H14N2O6Colore e forma:SolidPeso molecolare:342.303Pelagiomicin C
CAS:Pelagiomicin C exhibits activity against both Gram-positive and Gram-negative bacteria.Formula:C17H15N3O5Colore e forma:SolidPeso molecolare:341.318Epicillin
CAS:<p>Epicillin possesses antibacterial activity.</p>Formula:C16H21N3O4SColore e forma:SolidPeso molecolare:351.421FTI 276 TFA
CAS:FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).Formula:C23H28F3N3O5S2Colore e forma:SolidPeso molecolare:547.61Oiligodendrocyte differentiation promoter 1
CAS:<p>Oiligodendrocyte differentiation promoter 1 is a promoter of oiligodendrocyte differentiation .</p>Formula:C25H25Cl2NO5Purezza:98%Colore e forma:SolidPeso molecolare:490.38MK-7445
CAS:<p>MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.</p>Formula:C21H13Cl2N7OColore e forma:SolidPeso molecolare:450.28Monamycin B
CAS:<p>Monamycin B is an ester peptide antibiotic with activity against Gram-positive bacteria.</p>Formula:C33H55N7O8Colore e forma:SolidPeso molecolare:677.83AM-9514
CAS:<p>AM-9514: a potent Glucokinase activator with strong in vitro results, good pharmacokinetics, and efficacy in diabetes.</p>Formula:C18H25N5O4Colore e forma:SolidPeso molecolare:375.42Methymycin
CAS:<p>Methymycin is a macrolide antibiotic with activity against Gram-positive bacteria and some Gram-negative bacteria.</p>Formula:C25H43NO7Colore e forma:SolidPeso molecolare:469.611Cycloepoxydon
CAS:<p>Cycloepoxydon inhibits the NF-KB and AP-1 mediated secretion of alkaline phosphatase (SEAP) induced by Phorbol 12-myristate 13-acetate (PMA), with IC50 values of 1-2 μg/mL (4.2-8.4 μM) and 3-5 μg/mL (12.6-21 μM), respectively.</p>Formula:C12H16O5Colore e forma:SolidPeso molecolare:240.252OncoFAP
CAS:<p>OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.</p>Formula:C21H19F2N5O5Purezza:99.77%Colore e forma:SolidPeso molecolare:459.40Ciprokiren
CAS:<p>Ciprokiren, a renin inhibitor by Roche, halts human renin; IC50: 0.07/0.65 nmol/L. Lowers blood pressure in animals. Preclinical development ceased.</p>Formula:C37H55N5O8SColore e forma:SolidPeso molecolare:729.93Chitinovorin C
CAS:<p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>Formula:C15H20N4O8SColore e forma:SolidPeso molecolare:416.406TRPV1 antagonist 3
<p>TRPV1 antagonist 3 (7q) strongly blocks TRPV1 at 2.66 nM IC50, is selective, 60% bioavailable, and crosses the blood-brain barrier.</p>Formula:C23H25N3OSColore e forma:SolidPeso molecolare:391.53Trk-IN-8
<p>Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).</p>Formula:C18H16F2N6O2Colore e forma:SolidPeso molecolare:386.36ONO-DI-004
CAS:<p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>Formula:C24H38O6Colore e forma:SolidPeso molecolare:422.55(S)-5-hydroxy-6-methoxy Duloxetine maleate
<p>(S)-5-hydroxy-6-methoxy Duloxetine, an active metabolite of the (S)-duloxetine, functions as a serotonin (5-HT) and norepinephrine reuptake inhibitor.</p>Formula:C19H21NO3S·C4H4O4Colore e forma:SolidPeso molecolare:459.51Cinnatriacetin A
CAS:<p>Cinnatriacetin A exhibits activity against Gram-positive bacteria.</p>Formula:C23H20O5Colore e forma:SolidPeso molecolare:376.402Rhodomycin B
CAS:<p>Rhodomycin B exhibits activity against Gram-positive bacteria, while its effects on Gram-negative bacteria and fungi are relatively weak.</p>Formula:C28H33NO10Colore e forma:SolidPeso molecolare:543.562Saframycin B
CAS:<p>Saframycin B exhibits activity against Gram-positive bacteria and has weaker efficacy against mycobacteria.</p>Formula:C28H31N3O8Colore e forma:SolidPeso molecolare:537.561Salfredin C1
CAS:<p>Salfredin C1 is an inhibitor of aldose reductase.</p>Formula:C13H11NO6Colore e forma:SolidPeso molecolare:277.229SAR107375
CAS:<p>SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].</p>Formula:C24H30ClN5O5S2Colore e forma:SolidPeso molecolare:568.11KY-02327 acetate
<p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>Formula:C22H31N3O6Colore e forma:SolidPeso molecolare:433.5Deoxyfrenolicin
CAS:<p>Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.</p>Formula:C18H18O6Colore e forma:SolidPeso molecolare:330.332Namitecan
CAS:Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.Formula:C23H22N4O5Purezza:98%Colore e forma:SolidPeso molecolare:434.44Feigrisolide C
CAS:<p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>Formula:C21H36O7Colore e forma:SolidPeso molecolare:400.5063HKT-IN-1
CAS:<p>3HKT-IN-1 (Compound 17122279) is an inhibitor of Anopheles gambiae 3-hydroxykynurenine transaminase (3HKT) and is utilized in malaria research.</p>Formula:C12H11BrN2O3Colore e forma:SolidPeso molecolare:311.131GW311616
CAS:<p>GW-311616 is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>Formula:C19H31N3O4SColore e forma:SolidPeso molecolare:397.53SARS-CoV-2 nsp3-IN-1
<p>Compound 15c selectively inhibits SARS-CoV-2 nsp3 Mac1 with IC50 of 6.1 μM.</p>Formula:C17H15N5O2Colore e forma:SolidPeso molecolare:321.3311-Demethyltomaymycin
CAS:<p>11-Demethyltomaymycin is an antibiotic that exhibits antiviral activity against Escherichia coli T1 and T3 bacteriophages, along with antibacterial properties against Gram-positive bacteria. Furthermore, it shows cytotoxic effects on leukemia L1210 cells.</p>Formula:C15H18N2O4Colore e forma:SolidPeso molecolare:290.314Sulprostone
CAS:<p>EP3 and EP1 receptor agonist</p>Formula:C23H31NO7SPurezza:98%Colore e forma:White To Off-White SolidPeso molecolare:465.56Chrymutasin B
CAS:<p>Chrymutasin B is a glycoside antitumor antibiotic known for its cytotoxic properties.</p>Formula:C32H31NO13Colore e forma:SolidPeso molecolare:637.587RK-582
CAS:<p>RK-582: oral spiroindolinone tankyrase inhibitor, halts colon cancer growth in COLO-320DM mouse model.</p>Formula:C27H35FN6O3Colore e forma:SolidPeso molecolare:510.6PD-149163
CAS:<p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>Formula:C42H71N9O6Colore e forma:SolidPeso molecolare:798.07Enactin Ⅴa
CAS:<p>EnactinVa is a compound produced by the bacterium Streptomyces roseoviridis and exhibits relatively weak antifungal activity.</p>Formula:C19H38N2O5Colore e forma:SolidPeso molecolare:374.515AKR1C3-IN-8
<p>AKR1C3-IN-8 (Compound 5) is an effective and selective AKR1C3 inhibitor (IC50=0.069 μM). AKR1C3-IN-8 has antitumor activity.</p>Formula:C23H20N4O3Colore e forma:SolidPeso molecolare:400.43Curvularol
CAS:<p>Curvularol exhibits mild antifungal activity but lacks antibacterial effects. At a concentration of 150 ng/mL, it can inhibit the cell cycle progression of normal rat renal cells (G1 phase NRK). Additionally, 100 ng/mL of Curvularol can restore the morphology of deformed NRK cells induced by SRCTS. Curvularol also inhibits protein synthesis.</p>Formula:C15H22O4Colore e forma:SolidPeso molecolare:266.333RIPK1-IN-24
CAS:<p>RIPK1-IN-24 is an inhibitor of receptor-interacting protein kinase 1 (RIPK1) with an IC50 of 1.3 μM. It is utilized in research on inflammatory diseases.</p>Formula:C26H21FN6O2Colore e forma:SolidPeso molecolare:468.48PD-1/PD-L1-IN-16
<p>PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.</p>Formula:C34H30N4O4Colore e forma:SolidPeso molecolare:558.63Ezomycin D2
CAS:<p>Ezomycin D2 is an antifungal antibiotic effective primarily against plant pathogens such as Sclerotinia sclerotiorum and Botrytis cinerea. It helps control diseases like sclerotinia blight and gray mold in crops, as well as candidiasis.</p>Formula:C19H27N5O14Colore e forma:SolidPeso molecolare:549.443Purine phosphoribosyltransferase-IN-1
<p>Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.</p>Formula:C11H15N5Na4O10P2Colore e forma:SolidPeso molecolare:531.17Inactone
CAS:<p>Inactone is a biologically active molecule with a 3-pentanoylimino group that inhibits the large ribosomal subunit.</p>Formula:C15H21NO4Colore e forma:SolidPeso molecolare:279.332ATM-3507 trihydrochloride (1861449-70-8 free base)
<p>ATM-3507 trihydrochloride is a potent tropomyosin inhibitor (IC50s: 3.83-6.84 μM in human melanoma cell lines).</p>Formula:C37H49Cl3FN5O2Purezza:98%Colore e forma:SolidPeso molecolare:721.17MMP408
CAS:<p>MMP408 acts as an inhibitor of MMP-12.</p>Formula:C19H20N2O7SColore e forma:SolidPeso molecolare:420.44Cremimycin
CAS:<p>Cremimycin exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) of 0.2-0.39 μg/mL. Additionally, Cremimycin demonstrates cytotoxic effects on mouse tumor cell lines P388, L1210, IMC, S180, B16, and SS3 in vitro.</p>Formula:C35H53NO9Colore e forma:SolidPeso molecolare:631.797BAY-693
CAS:<p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>Formula:C26H30F3N7O2Colore e forma:SolidPeso molecolare:529.56SX 3202
CAS:<p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>Formula:C17H11BrFN3O4Colore e forma:SolidPeso molecolare:420.19CI-1029
CAS:<p>CI-1029: HIV protease inhibitor, combats mutant strains, high efficacy, good bioavailability in animals.</p>Formula:C28H37NO4SColore e forma:SolidPeso molecolare:483.66Nothramicin
CAS:<p>Nothramicin is an anthracycline antibiotic that exhibits antimycobacterial activity.</p>Formula:C30H37NO11Colore e forma:SolidPeso molecolare:587.615TY 11223
CAS:<p>TY 11223: stable homoisocarbacyclin analog, potently inhibits platelet aggregation with lasting effect and selective activity.</p>Formula:C24H34O5Colore e forma:SolidPeso molecolare:402.52VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Formula:C20H21N3O2Colore e forma:SolidPeso molecolare:335.4Nnc 09-0026
CAS:<p>Nnc 09-0026 is a neuronal calcium channel blocker</p>Formula:C25H35Cl2F3N2OColore e forma:SolidPeso molecolare:507.46CY208-243 Mandelate
CAS:<p>CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.</p>Formula:C27H26N2O3Colore e forma:SolidPeso molecolare:426.52Antidepressant agent 2
<p>Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.</p>Formula:C21H22ClFN2O3SColore e forma:SolidPeso molecolare:436.93KUS121
CAS:<p>KUS121: VCP ATPase activity inhibitor (IC50=330 nM), protects cells from ER stress, assists in cerebral ischemia, and preserves vision in retinitis pigmentosa.</p>Formula:C22H17FN4NaO3SColore e forma:SolidPeso molecolare:459.45Chuangxinmycin
CAS:<p>Chuangxinmycin is an antibiotic that can be isolated from Actinoplanes tsinanensis CPCC 200056. It exhibits antibacterial activity both in vitro and in vivo, making it useful for research related to infections.</p>Formula:C12H11NO2SColore e forma:SolidPeso molecolare:233.286Cytosaminomycin A
CAS:<p>Cytosaminomycin A is an antibiotic with anticoccidial and antibacterial properties.</p>Formula:C22H34N4O8SColore e forma:SolidPeso molecolare:514.592Hynapene A
CAS:<p>Hynapene A exhibits an inhibitory minimum inhibitory concentration (MIC) of 123 μM against Eimeria tenella.</p>Formula:C18H28O5Colore e forma:SolidPeso molecolare:324.412KHK-IN-6
CAS:<p>KHK-IN-6 (compound 33) acts as a KHK inhibitor with an IC50 of 0.6nM.</p>Formula:C23H24F3N5O2SColore e forma:SolidPeso molecolare:491.53TRβ agonist 1
CAS:<p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>Formula:C29H25FN2O8Colore e forma:SolidPeso molecolare:548.52Fosfocytocin
CAS:<p>Fosfocytocin can be found in the Pseudomonas fluorescens strain PK-52 and exhibits very weak antibacterial activity.</p>Formula:C12H20N4O13P2Colore e forma:SolidPeso molecolare:490.254Naphthablin
CAS:<p>Naphthablin is a naphthoquinone compound that inhibits the function of the Abl oncogene. It prevents the morphological transformation of v-ablts-NIH3T3 cells induced by Abl and also suppresses RNA synthesis.</p>Formula:C29H36O8Colore e forma:SolidPeso molecolare:512.591IMP-321
CAS:IMP-321 is a soluble dimeric recombinant form of LAG-3 and first-in-class antigen presenting cell activator.Formula:C56H78N18O14SColore e forma:SolidPeso molecolare:1259.4TLR7/8 antagonist 2
<p>TLR7/8 antagonist 2: potent, orally active, IC50: 4.9 nM (TLR7), 0.6 nM (TLR8); potential for lupus therapy research.</p>Formula:C22H26FN5Colore e forma:SolidPeso molecolare:379.47TRPC5-IN-4
CAS:<p>TRPC5-IN-4: Potent, safe inhibitor; IC50 14.07 nM (TRPC5), 65 nM (TRPC4); non-toxic to liver/kidney cells; for CKD research.</p>Formula:C18H11ClF4N4O3Colore e forma:SolidPeso molecolare:442.75Pateamine A
CAS:<p>Pateamine A: marine-sourced macrolide from Mycale hentscheli; anticancer, antiviral, and translation inhibitor.</p>Formula:C31H45N3O4SColore e forma:SolidPeso molecolare:555.77PLP_Snyder530
<p>PLP_Snyder530, a potent PL pro inhibitor, halts SARS-CoV-2 by triggering protease conformation changes.</p>Formula:C24H24N2O2Colore e forma:SolidPeso molecolare:372.46U 75875
CAS:<p>U 75875 is a protease inhibitor.</p>Formula:C45H61N7O7Colore e forma:SolidPeso molecolare:812.01MAP3K14-IN-173
CAS:<p>MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.</p>Formula:C29H31N7O2Colore e forma:SolidPeso molecolare:509.60E-3030 free acid
CAS:<p>E-3030 free acid, a PPAR agonist, lowers blood glucose, triglycerides, and insulin; boosts adiponectin; reduces apo C-III; and raises lipoprotein lipase.</p>Formula:C22H23ClFNO5Purezza:98%Colore e forma:SolidPeso molecolare:435.87CVS-1578
CAS:<p>CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.</p>Formula:C20H30N6O5SColore e forma:SolidPeso molecolare:466.55CGC 11144
CAS:<p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>Formula:C40H100Cl10N10Colore e forma:SolidPeso molecolare:1075.82Leucomycin A7
CAS:<p>Leucomycin A7 is a component of the leucomycin complex, isolated from *Streptomyces kitasatoensis*. It possesses antibacterial activity, effectively inhibiting the growth of gram-positive bacteria, while its inhibitory effect on gram-negative bacteria is comparatively weaker.</p>Formula:C38H63NO14Colore e forma:SolidPeso molecolare:757.905Minnelide free acid
CAS:<p>Minnelide treats pancreatic cancer, hinders androgen-related prostate growth, shrinks tumors, and improves survival.</p>Formula:C21H27O10PColore e forma:SolidPeso molecolare:470.41α-Prumycin hydrochloride
CAS:<p>α-Prumycin hydrochloride is a carbohydrate antibiotic with antifungal properties and weak antibacterial activity.</p>Formula:C8H19Cl2N3O4Colore e forma:SolidPeso molecolare:292.16KFA1982
CAS:<p>KFA1982 is a novel and potent factor Xa inhibitor.</p>Formula:C28H34ClN3O9S2Colore e forma:SolidPeso molecolare:656.17Carazostatin
CAS:<p>Carazostatin is an antioxidant, free radical scavenger, and potent lipid peroxidation inhibitor.</p>Formula:C20H25NOPurezza:98%Colore e forma:Pale Yellow SolidPeso molecolare:295.42Rezatapopt
CAS:<p>Rezatapopt (PC14586) is a p53 reactivator with antitumor activity for the study of locally advanced or metastatic solid tumors.</p>Formula:C28H31F4N5O2Purezza:98.12%Colore e forma:SolidPeso molecolare:545.57Tribenuron
CAS:<p>Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.</p>Formula:C14H15N5O6SColore e forma:SolidPeso molecolare:381.36Copper(II) ionophore I
CAS:Copper(II) ionophore I is an active compound.Formula:C26H44N2S4Colore e forma:SolidPeso molecolare:512.90Anti-Trypanosoma cruzi agent-1
<p>Anti-Trypanosoma cruzi agent-1 (Compd E5) has a potent anti-Toxoplasma effect.</p>Formula:C23H29N3O5Colore e forma:SolidPeso molecolare:427.49Nemotinic acid
CAS:<p>Nemotinic acid exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while also displaying weaker activity against Gram-negative bacteria.</p>Formula:C11H10O3Colore e forma:SolidPeso molecolare:190.195SARS-CoV-2 nsp14-IN-2
<p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>Formula:C21H21N5O5SColore e forma:SolidPeso molecolare:455.49Cyclo (D-Pro-L-Val)
CAS:<p>Cyclo(D-Pro-L-Val) inhibits the activity of β-glucosidase (β-glycosidase) with an IC50 of 75 μg/mL and exhibits either no inhibitory effects or only weak inhibition on other glycosidases.</p>Formula:C10H16N2O2Colore e forma:SolidPeso molecolare:196.246Terfluranol
CAS:Terfluranol, a benzyl derivative, is utilized as an antitumor medication.Formula:C17H17F3O2Colore e forma:SolidPeso molecolare:310.312,4-Diaminoanisole
CAS:<p>2,4-Diaminoanisole is a carcinogenic aromatic primary amine compound.</p>Formula:C7H10N2OColore e forma:SolidPeso molecolare:138.17Melithiazole K
CAS:<p>Melithiazol K is an antibiotic and functions as a β-methoxyacrylate (MOA) inhibitor, exhibiting strong resistance.</p>Formula:C20H26N2O5S2Colore e forma:SolidPeso molecolare:438.561AMPK Activator SC4
CAS:<p>SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.</p>Formula:C26H18ClN3O4Colore e forma:SolidPeso molecolare:471.89Prohibitin ligand 1
<p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>Formula:C20H22N2OColore e forma:SolidPeso molecolare:306.4EP-7041 HCl
CAS:<p>EP-7041 is a novel, potent, and selective Factor XIa inhibitor.</p>Formula:C19H27ClN4O4Colore e forma:SolidPeso molecolare:410.89MPO-IN-8
CAS:<p>MPO-IN-8, an orally active myeloperoxidase (MPO) inhibitor, effectively inhibits the production of hypochlorous acid in neutrophils and the release of extracellular traps (NETosis). In mice exhibiting gouty arthritis, it reduces swelling, decreases peroxidase activity, and lowers IL-1β levels.</p>Formula:C12H9N3O2Colore e forma:SolidPeso molecolare:227.22Leu-AMS R enantiomer
CAS:<p>Leu-AMS R enantiomer is the R enatiomer of Leu-AMS. Leu-AMS is a potent leucyl-tRNA synthetase (LRS) inhibitor that inhibits the bacteria growth.</p>Formula:C16H25N7O7SPurezza:98%Colore e forma:SolidPeso molecolare:459.481-Deamino-1-hydroxygentamicin C1a
CAS:<p>1-Deamino-1-hydroxygentamicin C1a (AntibioticSU-2) is an aminoglycoside antibiotic effective against both gram-positive and gram-negative bacteria.</p>Formula:C19H38N4O8Colore e forma:SolidPeso molecolare:450.5273-O-Demethyl-2'-N-glylfortimicin B
CAS:<p>3-O-Demethyl-2'-N-glylfortimicin B is a type of aminoglycoside antibiotic.</p>Formula:C16H33N5O6Colore e forma:SolidPeso molecolare:391.463Mollisin
CAS:<p>Mollisin is a quinone antibiotic with antifungal properties.</p>Formula:C14H10Cl2O4Colore e forma:SolidPeso molecolare:313.1334-Diazo-3-methoxy-2,5-cyclohexadien-1-one
CAS:<p>4-Diazo-3-methoxy-2,5-cyclohexadien-1-one demonstrates notable activity against anaerobic bacteria. Minimum inhibitory concentrations (MIC) are 0.4 μg/mL for Clostridium and Bacteroidetes, and 0.2 μg/mL for Haemophilus.</p>Formula:C7H6N2O2Colore e forma:SolidPeso molecolare:150.14PI3K-IN-23
<p>PI3K-IN-23 is a (E)-9-oxooctadec-10-en-12-ynoic acid analogue that promotes glucose uptake (EC50: 7.00 μM).</p>Formula:C24H33NO4SColore e forma:SolidPeso molecolare:431.59RN941
CAS:<p>RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.</p>Formula:C34H34FN7O5Purezza:98%Colore e forma:SolidPeso molecolare:639.68
![Octahydrocyclopenta[c]pyrrole](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT201335.webp&w=3840&q=75)
![Thiazolo[5,4-c]pyridin-4(5H)-one](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT88035.webp&w=3840&q=75)
