Altri inibitori
Questa categoria comprende una vasta gamma di inibitori che non rientrano nelle classificazioni standard ma sono comunque fondamentali per varie ricerche biochimiche e farmacologiche. Questi inibitori possono bersagliare vie, enzimi e interazioni molecolari uniche o meno studiate, fornendo strumenti preziosi per aree di ricerca specializzate. Presso CymitQuimica, offriamo una selezione diversificata di inibitori di alta qualità che coprono molteplici bersagli biologici e discipline di ricerca, permettendoti di esplorare nuove strade terapeutiche e approfondire la tua comprensione dei processi biologici complessi.
Trovati 37827 prodotti di "Altri inibitori"
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Oral antiplatelet agent 1
CAS:<p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>Formula:C23H24N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:468.53VEGFR-2-IN-5 hydrochloride
<p>VEGFR-2-IN-5 hydrochloride is an effective VEGFR2 inhibitor.</p>Formula:C19H25ClN8Colore e forma:SolidPeso molecolare:400.91CV 5975
CAS:<p>CV 5975 is a nonsulfhydryl ACE inhibitor that was investigated for use in hypertension and heart failure.</p>Formula:C22H31N3O5SColore e forma:SolidPeso molecolare:449.56TRPV1 antagonist 3
<p>TRPV1 antagonist 3 (7q) strongly blocks TRPV1 at 2.66 nM IC50, is selective, 60% bioavailable, and crosses the blood-brain barrier.</p>Formula:C23H25N3OSColore e forma:SolidPeso molecolare:391.53GNE-616
CAS:<p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>Formula:C24H23F4N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:537.53Sequoiaflavone
CAS:<p>Sequoiaflavone is a biflavone isolated from Ginkgo biloba.</p>Formula:C31H20O10Colore e forma:SolidPeso molecolare:552.48O-Desmethyl Midostaurin
CAS:O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.Formula:C34H28N4O4Purezza:98%Colore e forma:SolidPeso molecolare:556.61MK-8970
<p>MK-8970 is an acetal carbonate prodrug of raltegravir with enhanced colonic absorption.</p>Formula:C25H29FN6O8Colore e forma:SolidPeso molecolare:560.54Protease-Activated Receptor-1 antagonist 3
<p>PAR-1 antagonist 3: potent (IC50: 7 nM), binds hERG K+ channels (IC50: 9 μM).</p>Formula:C30H34N4O3Colore e forma:SolidPeso molecolare:498.62AL-GDa62
<p>AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).</p>Formula:C24H28FN3OColore e forma:SolidPeso molecolare:393.5AVE-1330A free acid
CAS:<p>AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.</p>Formula:C7H11N3O6SColore e forma:SolidPeso molecolare:265.243'-GMP
CAS:<p>3'-GMP is a nucleotide that can be isolated from the tubers of Helianthus tuberosus L. (Jerusalem artichoke).</p>Formula:C10H14N5O8PColore e forma:SolidPeso molecolare:363.221LPM4870108
<p>LPM4870108: Potent, oral pan-Trk inhibitor, selective over ALK, with anti-tumor effects. TrkC IC50=0.2nM, TrkA IC50=2.4nM.</p>Formula:C20H19FN6O3Colore e forma:SolidPeso molecolare:410.4Mycoversilin
CAS:<p>Mycoversilin is an antibiotic with inhibitory activity against dermatophytes and plant pathogenic fungi, but it does not exhibit activity against yeasts and bacteria. It strongly inhibits protein synthesis.</p>Formula:C18H16O8Colore e forma:SolidPeso molecolare:360.315Albicidin
CAS:<p>Albicidin is a DNA gyrase inhibitor produced by Xanthomonas albilineans.</p>Formula:C44H38N6O12Colore e forma:SolidPeso molecolare:842.818Epicorazine A
CAS:<p>Epicorazine A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE), with a minimum inhibitory concentration (MIC) of 12.5-25 μg/mL. It is also effective against Candida albicans, showing an MIC of 25 μg/mL.</p>Formula:C18H16N2O6S2Colore e forma:SolidPeso molecolare:420.459Oudemansin A
CAS:<p>Oudemansin A is an antibiotic that targets fungi, inhibiting the synthesis of proteins, RNA, and DNA.</p>Formula:C17H22O4Colore e forma:SolidPeso molecolare:290.35L 156903
CAS:<p>L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.</p>Formula:C35H41N7O5SColore e forma:SolidPeso molecolare:671.81Fostriecin (free base)
CAS:<p>Fostriecin inhibits PP2A/PP4 (IC50s = 3.2/3 nM), weakly affects topoisomerase II/PP1 (IC50s = 40/131 μM), doesn't inhibit PP2B, and may modify epigenetics.</p>Formula:C19H27O9PColore e forma:SolidPeso molecolare:430.39RIP1 kinase inhibitor 1
CAS:<p>RIP1 kinase inhibitor 1 is an orally available and brain-penetrating inhibitor of RIP1 kinase with pKi of 9.04.</p>Formula:C24H20ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:461.9OM-153
CAS:<p>OM-153 blocks tankyrase 1 (IC50: 13 nM) and 2 (IC50: 2 nM), stifling WNT signaling and COLO 320DM cell growth.</p>Formula:C28H24FN7O2Colore e forma:SolidPeso molecolare:509.53TCMDC-135051 TFA (2413716-15-9 free base)
<p>TCMDC-135051 TFA is a highly selective and potent inhibitor of protein kinase PfCLK3.</p>Formula:C31H34F3N3O5Purezza:98%Colore e forma:SolidPeso molecolare:585.61Lipohexin
CAS:<p>Lipohexin is a peptide antibiotic that exhibits activity against Gram-positive bacteria. It competitively inhibits human placental proline endopeptidase (proline endopeptidase) with an IC50 of 3.5 μM. Additionally, Lipohexin inhibits proline endopeptidase from Flavobacterium meningosepticum, with an IC50 of 25 μM.</p>Formula:C39H68N6O9Colore e forma:SolidPeso molecolare:764.992Rivenprost
CAS:<p>Rivenprost, selective EP4 agonist (Ki: 0.7 nM), promotes bone growth, osteoblast differentiation, and aids wound healing.</p>Formula:C24H34O6SColore e forma:SolidPeso molecolare:450.59Antiviral agent 6
<p>Antiviral agent 6 showed excellent anti-TSWV effects in vivo (EC50: 188 mg/L).</p>Formula:C23H27BrN2O3S2Colore e forma:SolidPeso molecolare:523.51AX15910
<p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>Formula:C32H38N6O3Colore e forma:SolidPeso molecolare:554.7STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Formula:C17H12N4O4Colore e forma:SolidPeso molecolare:336.3Adiaft
CAS:<p>Adiaftis a bioactive chemical.</p>Formula:C10H11IN2O4Colore e forma:SolidPeso molecolare:350.11Aeruginosin 98-B
CAS:<p>Aeruginosin 98-B, a protease inhibitor, effectively inhibits trypsin, plasmin, and thrombin with IC50 values of 0.6, 7.0, and 10.0 μg/mL, respectively.</p>Formula:C29H46N6O9SColore e forma:SolidPeso molecolare:654.78Efrapeptin F
CAS:<p>Efrapeptin F, from Tolypocladium fungi, inhibits mitochondrial complex V and targets nutrient-deprived tumor cells.</p>Formula:C82H141N18O16Colore e forma:SolidPeso molecolare:1635.11FTI 276 TFA
CAS:FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).Formula:C23H28F3N3O5S2Colore e forma:SolidPeso molecolare:547.61Fonsartan free acid
CAS:<p>Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.</p>Formula:C26H32N4O5S2Purezza:98%Colore e forma:SolidPeso molecolare:544.69Deldeprevir Na
CAS:<p>Deldeprevir Na is an Antiviral Polyprotein cleavage inhibitor. HCV NS3/4A inhibitor.</p>Formula:C45H55F2N6NaO8S2Colore e forma:SolidPeso molecolare:933.08Retelliptine
CAS:Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.Formula:C25H32N4OPurezza:98%Colore e forma:SolidPeso molecolare:404.55Flurandrenolone Acetate
CAS:<p>Flurandrenolone Acetate, a synthetic glucocorticoid derived from Flurandrenolide, is used to study skin issues like eczema and psoriasis.</p>Formula:C26H35FO7Colore e forma:SolidPeso molecolare:478.55Salfredin C3
CAS:<p>Salfredin C3 is an inhibitor of aldose reductase (aldose reductase).</p>Formula:C16H15NO8Colore e forma:SolidPeso molecolare:349.292BI-207524
CAS:<p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>Formula:C35H36ClN5O5Colore e forma:SolidPeso molecolare:642.14CEP-2563
CAS:CEP-2563 is a prodrug of CEP-751. It also used as an antitumor agent, inhibiting protein kinases.Formula:C36H41ClN6O6Purezza:98%Colore e forma:SolidPeso molecolare:689.20Azicemicin A
CAS:<p>Azicemicin A exhibits mild antibacterial activity and shows no acute toxicity when administered via intraperitoneal injection to mice at a dosage of 150 mg/kg.</p>Formula:C23H25NO9Colore e forma:SolidPeso molecolare:459.446Antibiotic MA 144M1
CAS:<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formula:C42H55NO15Colore e forma:SolidPeso molecolare:813.88SHP2-IN-9
<p>SHP2-IN-9: Potent SHP2 inhibitor, IC50=1.174 μM, 85x SHP1 selectivity, crosses blood-brain barrier, hampers cancer growth.</p>Formula:C20H20FN3O2SColore e forma:SolidPeso molecolare:385.4620S Proteasome-IN-4
CAS:<p>20S Proteasome-IN-4: brain-penetrant, parasite-specific, oral, inhibits T.b. brucei proteasome (IC50: 6.3nM), for HAT research.</p>Formula:C20H18ClF2N3O3Colore e forma:SolidPeso molecolare:421.83Anticancer agent 17
<p>Anticancer agent 17 was effective against HeLa cells (IC50: 0.19 μM) and A2780 cells (IC50: 0.09 μM).</p>Formula:C27H34BrN3OColore e forma:SolidPeso molecolare:496.48KMH-233
CAS:<p>KMH-233 effectively blocks LAT1, inhibiting L-leucine uptake and cell growth, boosting betastatin and cisplatin efficacy at 25 μM.</p>Formula:C32H25N7O5Colore e forma:SolidPeso molecolare:587.58Nepaprazole sodium
CAS:<p>Nepaprazole Na (TY-11345), a proton pump inhibitor, may treat gastric ulcers; it reduces H+/K(+)-ATPase activity, with IC50 of 5.8-9.9 microM.</p>Formula:C18H18N3NaO2SColore e forma:SolidPeso molecolare:363.41MK-2748
CAS:<p>MK-2748 is an inhibitor of NS3 protease, hepatitis C virus.</p>Formula:C42H56N6O10SColore e forma:SolidPeso molecolare:836.99LLS30
CAS:<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Formula:C34H33Cl4N5O3Colore e forma:SolidPeso molecolare:701.47GW311616
CAS:<p>GW-311616 is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>Formula:C19H31N3O4SColore e forma:SolidPeso molecolare:397.53GSK1820795A
CAS:<p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>Formula:C35H34N8Colore e forma:SolidPeso molecolare:566.7MDK6465
CAS:<p>MDK6465 (PCSK9-IN-8b), CAS#1900686-46-5, is a liver-targeted PCSK9 synthesis inhibitor.</p>Formula:C27H29ClFN9O4Colore e forma:SolidPeso molecolare:598.03AG-7404
CAS:<p>AG-7404: strong protease inhibitor, fights poliovirus, EC50 0.080-0.674 μM, effective on V-073-resistant strains.</p>Formula:C26H29N5O7Colore e forma:SolidPeso molecolare:523.54TRβ agonist 1
CAS:<p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>Formula:C29H25FN2O8Colore e forma:SolidPeso molecolare:548.52SB 204070 hydrochloride
CAS:<p>SB 204070 hydrochloride is an inhibitor of beta-lactamase, it is isolated from Spondias mombin.</p>Formula:C19H27ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:382.88Lycopodine
CAS:<p>Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of</p>Formula:C16H25NOPurezza:98%Colore e forma:SolidPeso molecolare:247.38KUSC-5037
<p>KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.</p>Formula:C18H17F3N6O2Colore e forma:SolidPeso molecolare:406.13651Anti-ToCV agent 1
<p>Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.</p>Formula:C22H19FN2O5SColore e forma:SolidPeso molecolare:442.46Methysergide maleate
CAS:<p>Methysergide prevents migraines/cluster headaches; treats serotonin syndrome, carcinoid-induced diarrhea; risk of fibrosis limits use.</p>Formula:C25H31N3O6Purezza:98%Colore e forma:White To Off-WhitePeso molecolare:469.54Epithienamycin D
CAS:<p>Epithienamycin D is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C13H16N2O5SColore e forma:SolidPeso molecolare:312.342ERGi-USU-6 mesylate
<p>ERGi-USU-6 (mesylate) is a new selective ERG positive prostate cancer inhibitor with an IC50 value of 0.089 μM that is an ERGi-USU-6 salt derivative.</p>Formula:C14H18N4O4SColore e forma:SolidPeso molecolare:338.38Minnelide free acid
CAS:<p>Minnelide treats pancreatic cancer, hinders androgen-related prostate growth, shrinks tumors, and improves survival.</p>Formula:C21H27O10PColore e forma:SolidPeso molecolare:470.41Hispidospermidin
CAS:<p>Hispidospermidin is a phospholipase C inhibitor.</p>Formula:C25H47N3OColore e forma:SolidPeso molecolare:405.66ONO-AE1-329
CAS:<p>ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.</p>Formula:C22H30O6S2Colore e forma:SolidPeso molecolare:454.6Namitecan
CAS:Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.Formula:C23H22N4O5Purezza:98%Colore e forma:SolidPeso molecolare:434.445(S),6(R)-DiHETE
CAS:<p>5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.</p>Formula:C20H32O4Colore e forma:SolidPeso molecolare:336.47Glutaminyl cyclases-IN-1
<p>Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.</p>Formula:C25H30N6O2SColore e forma:SolidPeso molecolare:478.61Resolvin D1 methyl ester
CAS:<p>Resolvin D1, from docosahexaenoic acid via 15-/5-lipoxygenase, curbs acute inflammation; EC50 ~30 nM. Its methyl ester may enhance bioavailability.</p>Formula:C23H34O5Colore e forma:SolidPeso molecolare:390.51Nonsteroidal aromatase inhibitor 1
<p>Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.</p>Formula:C22H16N4O2Colore e forma:SolidPeso molecolare:368.39ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Formula:C23H26Cl2N2O3Colore e forma:SolidPeso molecolare:449.37p38-α MAPK-IN-5
CAS:<p>p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.</p>Formula:C37H49N11O2Colore e forma:SolidPeso molecolare:679.86Antiangiogenic agent 3
<p>Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.</p>Formula:C19H20O7Colore e forma:SolidPeso molecolare:360.3616(R)-Iloprost
CAS:<p>Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>Formula:C22H32O4Colore e forma:SolidPeso molecolare:360.49Quorum Sensing-IN-1
<p>Quorum Sensing-IN-1 is a small-molecule inhibitor of quorum sensing.</p>Formula:C13H10N2O2S2Colore e forma:SolidPeso molecolare:290.36NTPDase-IN-3
CAS:<p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>Formula:C22H24ClN3OS2Colore e forma:SolidPeso molecolare:446.03Antitumor agent-51
<p>Antitumor agent-51 targets osteosarcoma with 21.9 nM IC50, high selectivity, and low toxicity.</p>Formula:C23H25N5O2SColore e forma:SolidPeso molecolare:435.54Kaitocephalin
CAS:<p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>Formula:C18H21Cl2N3O9Colore e forma:SolidPeso molecolare:494.28ALK5-IN-7
CAS:<p>ALK5-IN-7 inhibits ALK5, useful in TGF-β disease research like cancer, fibrosis, and autoimmune disorders. See WO2021129621A1.</p>Formula:C26H28N4O3SColore e forma:SolidPeso molecolare:476.59SOS1-IN-6
CAS:<p>SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).</p>Formula:C26H28F3N3O2Colore e forma:SolidPeso molecolare:471.51PKG1α activator 3
<p>PKG1α activator 3 is a PKG1α activator (EC50basal/partial=13/0.52 μM).</p>Formula:C27H26Cl2N2O6Colore e forma:SolidPeso molecolare:545.41CVS-1578
CAS:<p>CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.</p>Formula:C20H30N6O5SColore e forma:SolidPeso molecolare:466.55TrxR-IN-5
<p>TrxR-IN-5 (compound 4f) is an effective inhibitor of thioredoxin reductase (TrxR) with an IC₅₀ of 0.16 μM. anti-proliferative and anti-metastatic.</p>Formula:C26H22O3Colore e forma:SolidPeso molecolare:382.46NB-533
CAS:<p>NB-533 is a macrocyclic peptidic BACE-1 inhibitor.</p>Formula:C33H55N3O4Colore e forma:SolidPeso molecolare:557.81MAP3K14-IN-173
CAS:<p>MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.</p>Formula:C29H31N7O2Colore e forma:SolidPeso molecolare:509.60ETX0282
CAS:<p>ETX0282, oral class A/C β-lactamase inhibitor, developed by Entasis with cefpodoxime for bacterial infections.</p>Formula:C13H18FN3O5Colore e forma:SolidPeso molecolare:315.30Canosimibe
CAS:<p>Canosimibe is a cholesterol absorption inhibitor</p>Formula:C44H60FN3O10Colore e forma:SolidPeso molecolare:809.96Polvitolimod
CAS:<p>Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.</p>Formula:C13H14FN5O4Colore e forma:SolidPeso molecolare:323.28Harziphilone
CAS:<p>Harziphilone exhibits mild activity against Gram-positive bacteria and possesses antitumor properties, showing inhibitory effects on lymphocytic leukemia L1210 and leukemia P388 with an IC50 of 0.26 μg/mL. Additionally, Harziphilone inhibits the binding of the Rev protein to [33P]-labeled Rev response element (RRE) RNA, with an IC50 of 2.0 μM.</p>Formula:C15H18O4Colore e forma:SolidPeso molecolare:262.301Lorajmine
CAS:Lorajmine, a monochloroacetyl derivative of ajmaline, is a class Ia antiarrhythmic agent that is rapidly hydrolyzed to ajmaline by plasma and tissue esterases.Formula:C22H27ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:402.91Combretastatin A1 phosphate
CAS:<p>Combretastatin A1 phosphate: potent anti-angiogenic and tumor vascular disruptor, with research potential in pancreatic neuroendocrine tumors.</p>Formula:C18H22O12P2Colore e forma:SolidPeso molecolare:492.31Antiviral agent 15
<p>Compound 15f, a Clofazimine derivative, inhibits rabies (EC50: 1.45 μM) and SARS-CoV-2 (EC50: 14.6 μM).</p>Formula:C27H24FN5OColore e forma:SolidPeso molecolare:453.51Mifepristone methochloride
CAS:<p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>Formula:C30H38ClNO2Colore e forma:SolidPeso molecolare:480.08MB-7133
CAS:<p>MB-7133 is an inhibitor of DNA synthesis.</p>Formula:C17H21N4O8PPurezza:98%Colore e forma:SolidPeso molecolare:440.34Henagliflozin
CAS:<p>Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.</p>Formula:C22H24ClFO7Colore e forma:SolidPeso molecolare:454.87EICAR
CAS:<p>EICAR: IMP dehydrogenase inhibitor with anticancer and antiviral properties, failed in leukemia trials, active against various viruses but not SARS.</p>Formula:C11H13N3O5Colore e forma:SolidPeso molecolare:267.24RORγt inhibitor 2
CAS:<p>RORγt Inhibitor 2, a potent inhibitor of RORγt, exhibits an IC50 of 9.2 nM and is utilized in the study of cancer, inflammation, or autoimmune diseases that are</p>Formula:C31H33F5N2O7SColore e forma:SolidPeso molecolare:672.66A1-Phytoprostane-I
CAS:<p>A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.</p>Formula:C18H28O4Colore e forma:SolidPeso molecolare:308.41Latrunculin M
CAS:<p>Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.</p>Formula:C21H33NO5SColore e forma:SolidPeso molecolare:411.55VRT-18858
CAS:<p>VRT-18858 is a metabolite of VX-740.</p>Formula:C24H25N5O7Colore e forma:SolidPeso molecolare:495.48Dinordrin I diacetate
CAS:<p>Dinordrin I diacetate is an implantation inhibitor and hormone.</p>Formula:C25H32O4Purezza:98%Colore e forma:SolidPeso molecolare:396.52Kahweol linoleate
CAS:<p>Kahweol linoleate, a semi-synthetic from coffee, blocks osteoclast creation, fights cancerous cells, prevents DNA damage, and reduces oxidative stress.</p>Formula:C38H56O4Colore e forma:SolidPeso molecolare:576.85Porothramycin B
CAS:<p>Porothramycin B is an antibiotic with activity against Gram-positive bacteria and anaerobes.</p>Formula:C19H23N3O4Colore e forma:SolidPeso molecolare:357.4049(S)-HEPE
CAS:<p>9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.</p>Formula:C20H30O3Colore e forma:SolidPeso molecolare:318.45FWM-1
<p>FWM-1 blocks SARS-CoV-2 NSP13, hinders ATP binding, with -328.6 kcal/mol binding energy.</p>Formula:C15H11ClN4O4S2Colore e forma:SolidPeso molecolare:410.86M-COPA
CAS:<p>M-COPA disrupts Golgi, blocks MET & Arf1 activation, and inhibits angiogenesis via VEGFR & NF-kB pathways.</p>Formula:C25H34N2O2Colore e forma:SolidPeso molecolare:394.55Lucilactaene
CAS:<p>Lucilactaene exhibits potent antimalarial activity and functions as a P53-transfected tumor cell cycle inhibitor. It effectively halts the cell cycle progression of H1299/TSP53 cells at the G1 phase.</p>Formula:C22H27NO6Peso molecolare:401.45Cilobamine (free base)
CAS:<p>Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.</p>Formula:C17H23Cl2NOColore e forma:SolidPeso molecolare:328.28XR8-89
CAS:<p>XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.</p>Formula:C29H36N4O2SColore e forma:SolidPeso molecolare:504.69GSK3527497 HCl
CAS:<p>GSK3527497: potent TRPV4 inhibitor, IC50=12 nM, targets heart/respiratory issues, for oral/IV use, low-dose effective.</p>Formula:C17H17Cl2FN4O4SColore e forma:SolidPeso molecolare:463.3054EP-7041 HCl
CAS:<p>EP-7041 is a novel, potent, and selective Factor XIa inhibitor.</p>Formula:C19H27ClN4O4Colore e forma:SolidPeso molecolare:410.89ONO-AE1-259 lysine
CAS:<p>ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)</p>Formula:C28H49ClN2O6Colore e forma:SolidPeso molecolare:545.15Alentemol hydrobromide
CAS:<p>Alentemol hydrobromide is a Dopamine agonist.</p>Formula:C19H26BrNOPurezza:98%Colore e forma:SolidPeso molecolare:364.32Agarospirol
CAS:<p>Agarospirol has partial anti-inflammatory activity.</p>Formula:C15H26OPurezza:98%Colore e forma:SolidPeso molecolare:222.37Difeterol
CAS:<p>Difeterol is a biochemical.</p>Formula:C25H29NO2Colore e forma:SolidPeso molecolare:375.50ATX inhibitor 22
<p>ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.</p>Formula:C19H17Cl3F2N2O4SColore e forma:SolidPeso molecolare:513.77Mopivabil
<p>Mopivabil is the angiotensin II receptor antagonist[1].</p>Formula:C14H20O3Colore e forma:SolidPeso molecolare:236.31EP4 receptor antagonist 2
CAS:<p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>Formula:C27H29N3O5Colore e forma:SolidPeso molecolare:475.54Isoleucyl tRNA synthetase-IN-2
CAS:<p>Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formula:C22H33N5O8SColore e forma:SolidPeso molecolare:527.59TrxR-IN-2
<p>TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.</p>Formula:C22H22N4O4Colore e forma:SolidPeso molecolare:406.43Clavalanine
CAS:<p>Clavalanine (Ro 22-5417) is capable of inhibiting various bacteria and fungi.</p>Formula:C8H12N2O4Colore e forma:SolidPeso molecolare:200.192Antitumor agent-50
<p>Antitumor agent-50 (compound 1a) is a thiazolidinone.</p>Formula:C17H14FNO3SColore e forma:SolidPeso molecolare:331.36SARS 3CLpro-IN-1
CAS:<p>SARS 3CLpro-IN-1: stereospecific SARS 3CL protease inhibitor, octahydroisochromene class, IC50 = 95 μM.</p>Formula:C22H38N4O2Colore e forma:SolidPeso molecolare:390.56Hsp90-IN-16
<p>Hsp90-IN-16, a selective HSP90 inhibitor, targets HER2+ cancers with 6 μM IC50 in HCC1954 cells, blocking client proteins and inducing apoptosis.</p>Formula:C30H26FN3O6Colore e forma:SolidPeso molecolare:543.54Antiallergic agent-1
<p>Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.</p>Formula:C27H19F6N5OColore e forma:SolidPeso molecolare:543.46AM-9514
CAS:<p>AM-9514: a potent Glucokinase activator with strong in vitro results, good pharmacokinetics, and efficacy in diabetes.</p>Formula:C18H25N5O4Colore e forma:SolidPeso molecolare:375.42Pegcantratinib
CAS:<p>Pegcantratinib is a tropomyosin receptor kinase inhibitor for treatment for inherited CYLD defective skin tumours.</p>Formula:C32H28N4O7Colore e forma:SolidPeso molecolare:580.59GYKI-53784
CAS:<p>GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.</p>Formula:C19H20N4O3Colore e forma:SolidPeso molecolare:352.39Diheteropeptin
CAS:<p>Diheteropeptin exhibits activity similar to that of transforming growth factor-β and has the ability to inhibit HDAC.</p>Formula:C28H42N4O6Colore e forma:SolidPeso molecolare:530.66Tylophorinidine
CAS:<p>Tylophorinidine is an antifungal agent that has shown to inhibit cell growth.</p>Formula:C22H23NO4Colore e forma:SolidPeso molecolare:365.42DS01080522
<p>DS01080522: PRKACA inhibitor, IC50: kinase 0.8 nM, CREB 66 nM; potential for cancer research.</p>Formula:C23H20Cl2N4O3Colore e forma:SolidPeso molecolare:471.34PAT-347
CAS:<p>PAT-347 is a potent inhibitor of Autotaxin, an enzyme linked to cell survival and diseases like cancer and fibrosis.</p>Formula:C28H21ClF2N2O3SColore e forma:SolidPeso molecolare:538.99Bulgecin A
CAS:<p>Bulgecin A is an inhibitor of binuclear metallo-beta-lactamases and Lytic transglycosolase.</p>Formula:C16H29N3O14S2Colore e forma:SolidPeso molecolare:551.54Steroid sulfatase-IN-4
<p>Steroid sulfatase-IN-4 irreversibly inhibits human STS with a 25 nM IC50, useful for endometriosis research.</p>Formula:C19H17ClN2O5SColore e forma:SolidPeso molecolare:420.87Oxythiamine diphosphate ammonium
<p>Oxythiamin diphosphate ammonium is a potent inhibitor of transketolase (TK).</p>Colore e forma:SolidCarpetimycin B
CAS:<p>Carpetimycin B exhibits potent activity against both Gram-positive and Gram-negative bacteria, including those that produce β-lactamase. Carpetimycin B is also a strong inhibitor of β-lactamase (β-lactamase).</p>Formula:C14H18N2O9S2Colore e forma:SolidPeso molecolare:422.431SARS-CoV-2-IN-23
<p>SARS-CoV-2-IN-23 (compound GRL-0617) is an inhibitor of SARS-COV-2 papain-like protease (PLpro) (IC 50 = 2.3 μM) [1].</p>Formula:C21H22N2OColore e forma:SolidPeso molecolare:318.41Cytosaminomycin C
CAS:<p>Cytosaminomycin C exhibits anti-Eimeria Tenella coccidial activity.</p>Formula:C23H36N4O8Colore e forma:SolidPeso molecolare:496.554Epelmycin D
CAS:<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Formula:C30H35NO11Colore e forma:SolidPeso molecolare:585.599Tandutinib (MLN518) HCl
Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.Formula:C31H43ClN6O4Purezza:98%Colore e forma:SolidPeso molecolare:599.16Moflomycin
CAS:<p>Moflomycin is an anthracycline derivative. It exhibits a higher antileukemic activity compared to other anthracyclines.</p>Formula:C25H25IO10Purezza:98%Colore e forma:SolidPeso molecolare:612.36Pluracidomycin C2
CAS:<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C11H15NO9S2Colore e forma:SolidPeso molecolare:369.37GP-1681
CAS:<p>GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.</p>Formula:C24H30NaO5Purezza:98%Colore e forma:SolidPeso molecolare:421.48Enpp-1-IN-12
<p>ENPP1-IN-12 is a potent, oral ENPP1 inhibitor with a Ki of 41 nM and anti-tumor properties.</p>Formula:C17H19N5O3SColore e forma:SolidPeso molecolare:373.43Glidobactin C
CAS:<p>Glidobactin C (GlbC) is an antitumor antibiotic with activity against pathogenic fungi and yeasts. It exhibits antifungal properties against Candida albicans and Aspergillus fumigatus, with a minimum inhibitory concentration (MIC) of 0.8 μg/mL. Additionally, Glidobactin C prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Formula:C29H48N4O6Colore e forma:SolidPeso molecolare:548.715MB725
CAS:<p>MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.</p>Formula:C18H21IN4O2SColore e forma:SolidPeso molecolare:484.3511-Demethyltomaymycin
CAS:<p>11-Demethyltomaymycin is an antibiotic that exhibits antiviral activity against Escherichia coli T1 and T3 bacteriophages, along with antibacterial properties against Gram-positive bacteria. Furthermore, it shows cytotoxic effects on leukemia L1210 cells.</p>Formula:C15H18N2O4Colore e forma:SolidPeso molecolare:290.314SLN124
<p>SLN124, a GalNAc-siRNA targeting TMPRSS6, may normalize iron balance by restoring ferroregulation.</p>Colore e forma:SolidFR 901537
CAS:<p>FR 901537 is a new aromatase inhibitor with antitumor effects.</p>Formula:C23H29N3O6S2Purezza:98%Colore e forma:SolidPeso molecolare:507.62ORP-101
CAS:<p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>Formula:C60H84N2O8Colore e forma:SolidPeso molecolare:961.32DS89002333
<p>DS89002333: oral PRKACA inhibitor with 0.3 nM IC50, effective against FL-HCC with DNAJB1-PRKACA fusion in xenografts.</p>Formula:C22H20ClF2N3O3Colore e forma:SolidPeso molecolare:447.86YEATS4 binder-1
<p>YEATS4 binder-1(4e) is an effective and selective compound that targets the KAc recognition site within the YEATS structural domain, exhibiting a binding</p>Formula:C23H34N4O3Colore e forma:SolidPeso molecolare:414.54Mesulergine
CAS:<p>Mesulergine is metabolized into dopaminergic agonists.</p>Formula:C18H26N4O2SColore e forma:SolidPeso molecolare:362.49NI-Pano
<p>NI-Pano (CH-03) is a novel hypoxia-activated KDAC inhibitor capable of O2-dependent release of the compound panobinostat.</p>Formula:C26H28N6O4Colore e forma:SolidPeso molecolare:488.54NS2B/NS3-IN-5
<p>Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.</p>Formula:C14H9IN2O3SColore e forma:SolidPeso molecolare:412.2rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formula:C25H24Cl2FN3O3Colore e forma:SolidPeso molecolare:504.38Resorcinomycin B
CAS:<p>Resorcinomycin B is an antibiotic found in [Streptoverticillum roseoverticillatum].</p>Formula:C13H18N4O5Colore e forma:SolidPeso molecolare:310.306Pterulinic acid
CAS:<p>Pterulinic acid is an inhibitor of coenzyme I:coenzyme Q oxidoreductase. It demonstrates IC50 values (μg/mL) of 50 for the mammalian cell line L1210, 20 for HL60, 25 for HeLaS3, and 100 for BHK.</p>Formula:C15H11ClO4Colore e forma:SolidPeso molecolare:290.70BMS-520
CAS:<p>BMS-520: potent oral S1P1 agonist, effective in rat arthritis and mouse multiple sclerosis model.</p>Formula:C23H17F3N4O4Colore e forma:SolidPeso molecolare:470.4Polyoxin G
CAS:<p>Polyoxin G is a nucleoside antifungal antibiotic noted for its significant efficacy against rice sheath blight.</p>Formula:C17H25N5O12Colore e forma:SolidPeso molecolare:491.41Schidigera-genin B
CAS:<p>Schidigera-genin B is a steroidal saponin that can be isolated from Yucca glauca. It exhibits mild antifungal activity.</p>Formula:C27H40O4Colore e forma:SolidPeso molecolare:428.604Pulvilloric acid
CAS:<p>Pulvilloric acid is an antifungal antibiotic produced by the organism Pen. pulvillorum 504.</p>Formula:C15H18O5Colore e forma:SolidPeso molecolare:278.30CB-7646
CAS:<p>CB-7646 is a stable trimelamol (TM) analogue, which is an antitumor agent.</p>Formula:C8H16N6O2Colore e forma:SolidPeso molecolare:228.25Polyoxin J
CAS:<p>Polyoxin J is a nucleoside antifungal antibiotic, notably effective against sheath blight in rice.</p>Formula:C17H25N5O12Peso molecolare:491.41Chitinase-IN-4
<p>Chitinase-IN-4 (compound 8f) is a potent and selective inhibitor of OfChi-h with an IC50 value of 0.1 μM and good insecticidal activity.</p>Formula:C21H24ClN7Colore e forma:SolidPeso molecolare:409.92Defucogilvocarcin V
CAS:<p>Defucogilvocarcin V is an antibiotic with activity against Gram-positive bacteria.</p>Formula:C21H16O5Colore e forma:SolidPeso molecolare:348.349Phenazostatin A
CAS:<p>Phenazostatin A is a phenazine compound known for its neuroprotective properties. It acts by scavenging free radicals, protecting N18-RE 105 neuronal cells from glutamate-induced toxicity, and inhibiting lipid peroxidation. Phenazostatin A inhibits glutamate toxicity in N18-RE-105 cells with an EC50 of 0.34 μg/mL.</p>Formula:C28H20N4O3Colore e forma:SolidPeso molecolare:460.48Dienomycin B
CAS:<p>Dienomycin B exhibits mild antibacterial activity.</p>Formula:C18H23NO2Colore e forma:SolidPeso molecolare:285.38Chitinovorin C
CAS:<p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>Formula:C15H20N4O8SColore e forma:SolidPeso molecolare:416.406Cycloepoxydon
CAS:<p>Cycloepoxydon inhibits the NF-KB and AP-1 mediated secretion of alkaline phosphatase (SEAP) induced by Phorbol 12-myristate 13-acetate (PMA), with IC50 values of 1-2 μg/mL (4.2-8.4 μM) and 3-5 μg/mL (12.6-21 μM), respectively.</p>Formula:C12H16O5Colore e forma:SolidPeso molecolare:240.2521,6-Dihydroxy-2-chlorophenazine
CAS:<p>1,6-Dihydroxy-2-chlorophenazine exhibits weak antifungal and anti-yeast activity.</p>Formula:C12H7ClN2O2Colore e forma:SolidPeso molecolare:246.65Nanaomycin E
CAS:<p>Nanaomycin E is an antibiotic with activity against Gram-positive bacteria and fungi.</p>Formula:C16H14O7Colore e forma:SolidPeso molecolare:318.2784-Chloropyridine
CAS:<p>4-Chloropyridine acts as an inhibitor of Nicotinamide N-methyltransferase (NNMT). Serving as a substrate for NNMT, this compound enhances the electrophilicity at the C4 position through methylation of the pyridine nitrogen. This modification facilitates an aromatic nucleophilic substitution reaction with the non-catalytic cysteine (C159) in NNMT, ultimately leading to suicidal activity inhibition of the enzyme. 4-Chloropyridine is a promising candidate for the development of activity-based probes targeting NNMT functions.</p>Formula:C5H4ClNColore e forma:SolidPeso molecolare:113.55PZ-3022
CAS:<p>PZ-3022 is an orally active, conformational PanK activator that counteracts C3-CoA inhibition. In a mouse model of propionic acidemia, it elevates hepatic CoASH and C2-CoA levels while reducing C3-CoA, making it useful for studying mitochondrial defects in propionic acidemia.</p>Formula:C20H21N5OColore e forma:SolidPeso molecolare:347.41Fusarin C
CAS:<p>Fusarin C is a mutagenic compound found in strains of the Fusarium genus.</p>Formula:C23H29NO7Colore e forma:SolidPeso molecolare:431.479Fosfazinomycin B
CAS:<p>Fosfazinomycin B exhibits activity against plant pathogenic fungi such as the rice blast pathogen (Xanthomonas oryzae).</p>Formula:C10H23N6O6PColore e forma:SolidPeso molecolare:354.3Exfoliamycin
CAS:<p>Exfoliamycin is a naphthoquinone antibiotic found in the Streptomyces strain Exfoliamycin Tu 1424, and it exhibits activity against Gram-positive bacteria.</p>Formula:C22H26O9Colore e forma:SolidPeso molecolare:434.436Oximidine Ⅲ
CAS:<p>Oximidine III is an antitumor antibiotic that selectively inhibits the growth of rat fibroblast 3Y1 cells and induces mutations in various tumor genes. The inhibitory effects of Oximidine III on vH-ras-3Y1, v-src-3Y1 cells, and normal 3Y1 cells have IC50 values of 14 nM, 4.5 nM, and 140 nM, respectively. Additionally, Oximidine III arrests cells with RAS or SRC mutations in the G1 phase of the cell cycle and increases the expression of p21WAF1.</p>Formula:C23H24N2O6Colore e forma:SolidPeso molecolare:424.45Tzc 5665
CAS:<p>Tzc 5665 is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action.</p>Formula:C31H38ClN5O7Colore e forma:SolidPeso molecolare:628.12Bacithrocin B
CAS:<p>Bacithrocin B is a thrombin inhibitor that suppresses the activity of thrombin, Factor Xa, trypsin, and papain, with IC50 values of 84 μM, 17 μM, 1.7 μM, and 0.02 μM, respectively.</p>Formula:C19H29N5O3Colore e forma:SolidPeso molecolare:375.4652-Hydroxygentamicin A3
CAS:<p>2-Hydroxygentamicin A3 is an aminoglycoside antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Formula:C18H36N4O11Colore e forma:SolidPeso molecolare:484.499Matlystatin F
CAS:<p>Matlystatin F is an inhibitor of metalloproteinases (MMP).</p>Formula:C27H44N6O6Colore e forma:SolidPeso molecolare:548.675Carazostatin
CAS:<p>Carazostatin is an antioxidant, free radical scavenger, and potent lipid peroxidation inhibitor.</p>Formula:C20H25NOPurezza:98%Colore e forma:Pale Yellow SolidPeso molecolare:295.42Eponemycin
CAS:<p>Eponemycin is an antibiotic with antitumor properties. It exhibits cytotoxicity against cancer cell lines B16-F10, L1210, P388, and HCT-116, with IC50 values of 0.0017, 0.01, 0.031, and 0.0097 µg/mL, respectively. In B16-F10 and mitomycin C, Eponemycin inhibits DNA synthesis, with IC50 values of 0.1 µg/mL and 0.41 µg/mL, respectively.</p>Formula:C20H34N2O6Colore e forma:SolidPeso molecolare:398.494Dykellic acid
CAS:<p>Dykellic acid is a RhoA inhibitor. It can suppress the migration and motility of B16 cells and inhibit the tubular formation of HUVECs. Dykellic acid shows potential for use in cancer research.</p>Formula:C14H16O4Colore e forma:SolidPeso molecolare:248.274Maltophilin
CAS:<p>Maltophilin is a broad-spectrum antifungal antibiotic that exhibits no antibacterial activity against either Gram-positive or Gram-negative bacteria.</p>Formula:C29H38N2O6Peso molecolare:510.62NTPDase-IN-1
<p>NTPDase-IN-1 selectively inhibits NTPDases 1, 2, 8 with IC50 of 0.05, 0.23, 0.54 μM. Non-competitive, K m 21 μM, used in cancer, immune, infection research.</p>Formula:C18H25N3OS2Colore e forma:SolidPeso molecolare:363.54Exophilin A
CAS:<p>Exophilin A is an antibiotic that exhibits activity against Gram-positive bacteria.</p>Formula:C30H56O10Colore e forma:SolidPeso molecolare:576.76Herbimycin B
CAS:<p>Herbimycin B, an ansamycin antibiotic, functions as an inhibitor of Src family kinases. It exhibits herbicidal effects on most monocotyledonous and dicotyledonous plants and can inhibit the activity of tobacco mosaic virus (TMV), HeLa cells, and Ehrlich cells.</p>Formula:C29H40N2O7Colore e forma:SolidPeso molecolare:528.637KR-67607
CAS:<p>KR-67607, or NTX-101, is a novel 11β-HSD1 inhibitor that protects against eye injury by reducing cortisol and preserving eye structures.</p>Formula:C24H29Cl2F3N4O4SColore e forma:SolidPeso molecolare:597.48Juglomycin A
CAS:<p>Juglomycin A exhibits broad-spectrum antibacterial and anti-mycobacterial activity and can inhibit Ehrlich ascites carcinoma in mice.</p>Formula:C14H10O6Colore e forma:SolidPeso molecolare:274.2263-Methoxy-2,5-toluquinone
CAS:<p>3-Methoxy-2,5-toluquinone is an antimicrobial agent that exhibits moderate antibacterial and antifungal properties.</p>Formula:C8H8O3Colore e forma:SolidPeso molecolare:152.147Anticancer agent 78
<p>Anticancer agent 78: anti-aromatase (IC50=0.9 μM), cytotoxic, potential in breast cancer research.</p>Formula:C19H14BrNO4Colore e forma:SolidPeso molecolare:400.22PD-149163
CAS:<p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>Formula:C42H71N9O6Colore e forma:SolidPeso molecolare:798.07Esorubicin
CAS:<p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>Formula:C27H29NO10Colore e forma:SolidPeso molecolare:527.52FTO-IN-6
CAS:<p>FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).</p>Formula:C14H12N4O6Colore e forma:SolidPeso molecolare:332.27VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Formula:C20H21N3O2Colore e forma:SolidPeso molecolare:335.4Cryptosporiopsin
CAS:<p>Cryptosporiopsin can be isolated from strains of Cryptosporiopsis sp. and Sporormia affinis. It exhibits antimicrobial activity against various basidiomycetes, alga fungi, ascomycetes, and glaucomycetes responsible for wood decay. Additionally, it inhibits the germination of Phytophthora potatoes spores. Cryptosporiopsin also shows some activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C10H10Cl2O4Colore e forma:SolidPeso molecolare:265.09SID 125240931
CAS:<p>SID 125240931 is a regulator of fluorine-activated proteins (FAPs). This compound disrupts the binding between fluoride and FAPs.</p>Formula:C19H24N4O3SColore e forma:SolidPeso molecolare:388.48SAR107375
CAS:<p>SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].</p>Formula:C24H30ClN5O5S2Colore e forma:SolidPeso molecolare:568.11Iodinin
CAS:<p>Iodinin is an antibiotic with antibacterial and antifungal properties.</p>Formula:C12H8N2O4Colore e forma:SolidPeso molecolare:244.203Citreamicin γ
CAS:<p>Citreamicin γ demonstrates activity against aerobic and anaerobic Gram-positive bacteria.</p>Formula:C33H25NO12Colore e forma:SolidPeso molecolare:627.551Melanocin A
CAS:<p>Melanocin A is an inhibitor of melanin biosynthesis. It suppresses the synthesis of melanin and tyrosinase with an IC50 of 9.0 nM and MIC of 0.9 μM. Additionally, Melanocin A exhibits antioxidant properties.</p>Formula:C18H14N2O5Colore e forma:SolidPeso molecolare:338.31
