
Segnalazione citoscheletrica
Gli inibitori della segnalazione del citoscheletro sono composti che interrompono le vie di segnalazione che regolano il citoscheletro, cruciale per la forma, la motilità, la divisione delle cellule e il trasporto intracellulare. Questi inibitori vengono utilizzati per studiare la dinamica delle proteine del citoscheletro, come actina e tubulina, e il loro ruolo in processi come la migrazione cellulare, l'adesione e la metastasi del cancro. Gli inibitori della segnalazione del citoscheletro sono preziosi nella ricerca sulla biologia cellulare, sul cancro e sulla neurobiologia. Presso CymitQuimica, offriamo una gamma completa di inibitori della segnalazione del citoscheletro di alta qualità per supportare le tue ricerche in questi ambiti.
Trovati 1602 prodotti per "Segnalazione citoscheletrica".
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Adropin (34-76) (human, mouse, rat)
CAS:Adropin (34-76) (human, mouse, rat) is a peptide that attenuates liver fibrosis and insulin resistance. Cost-effective and quality-assured.Formula:C190H293N55O68S2Purezza:94.23% - 99.95%Colore e forma:White SolidPeso molecolare:4499.82Entasobulin
CAS:Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.Formula:C26H18ClN3O2Purezza:98.40%Colore e forma:SolidPeso molecolare:439.89Bosutinib
CAS:Bosutinib (SKI-606) is a synthetic quinolone derivative and dual kinase inhibitor that targets both Abl (IC50: 1 nM) and Src (IC50: 1.2 nM) kinases.Formula:C26H29Cl2N5O3Purezza:98.98% - 99.93%Colore e forma:Yellow SolidPeso molecolare:530.45Dasatinib monohydrate
CAS:Dasatinib monohydrate, an oral SRC-kinase inhibitor, counters imatinib-resistant chronic myeloid leukemia.Formula:C22H28ClN7O3SPurezza:99.68% - >99.99%Colore e forma:White SolidPeso molecolare:506.03Mps1-IN-3
CAS:Mps1-IN-3 is an effective and selective inhibitor of MPS1 kinase (IC50: 50 nM).Formula:C26H31N7O4SPurezza:99.25%Colore e forma:SolidPeso molecolare:537.63Ref: TM-T16130
2mg34,00€5mg54,00€1mL*10mM (DMSO)64,00€10mg87,00€25mg149,00€50mg255,00€100mg384,00€200mg538,00€Meclofenamic acid sodium
CAS:Meclofenamic acid sodium (Movens), a non-steroidal anti-inflammatory agent, has properties of antipyretic and antigranulation activities.Formula:C14H10Cl2NNaO2Purezza:98% - 98.96%Colore e forma:SolidPeso molecolare:318.14RWJ 50271
CAS:RWJ 50271 inhibits LFA-1/ICAM-1 interaction with IC50 5.0 μM in HL60 cells.Formula:C18H17F3N4O2SPurezza:99.09%Colore e forma:White SolidPeso molecolare:410.41Ref: TM-T12783
1mg120,00€5mg295,00€1mL*10mM (DMSO)326,00€10mg447,00€25mg707,00€50mg964,00€100mg1.243,00€200mg1.693,00€Larazotide acetate
CAS:Larazotide acetate is a synthetic peptide. It functions as a tight junction regulator and reverses leaky junctions to their normally closed state.Formula:C34H59N9O12Purezza:95.53% - 99.42%Colore e forma:Purple LiquidPeso molecolare:785.89TTBK1-IN-2
CAS:TTBK1-IN-2, a TTBK1 inhibitor with IC50s of 0.24/4.22 µM, lowers TDP-43 phosphorylation in vitro and in mice.Formula:C18H13ClN4OPurezza:99.83%Colore e forma:SolidPeso molecolare:336.77Ref: TM-T60086
1mg77,00€5mg159,00€1mL*10mM (DMSO)167,00€10mg226,00€25mg378,00€50mg537,00€100mg718,00€200mg964,00€PKC β pseudosubstrate acetate
PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) is a selective cell-permeable inhibitor of PKC.Purezza:95.42%Colore e forma:SoildA-3 hydrochloride
CAS:A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.Formula:C12H14Cl2N2O2SPurezza:99.32%Colore e forma:SolidPeso molecolare:321.22Dasatinib
CAS:Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.Formula:C22H26ClN7O2SPurezza:99.59% - 99.86%Colore e forma:Pale-Yellow SolidPeso molecolare:488.01CC-99677
CAS:CC-99677 (Gamcemetinib) is a MK2 inhibitor targeting autoimmune diseases; potent in rat assays with IC50=156.3 nM & EC50=89 nM.Formula:C22H20ClN5O3SPurezza:99.59%Colore e forma:SolidPeso molecolare:469.94CCT251545
CAS:CCT251545 is an potent and oral-bioavailable WNT signaling inhibitor(IC50 of 5 nM in 7dF3 cells).Formula:C23H24ClN5OPurezza:98.29% - 98.69%Colore e forma:White SolidPeso molecolare:421.92ADH-1 trifluoroacetate
CAS:ADH-1 trifluoroacetate (Exherin trifluoroacetate) is a cyclic pentapeptide vascular-targeting agent with potential antineoplastic and antiangiogenic activities.Formula:C24H35F3N8O8S2Purezza:90.08% - 99.98%Colore e forma:White SolidPeso molecolare:684.71Imatinib Mesylate
CAS:Imatinib Mesylate (STI-571) is a tyrosine kinase receptor inhibitor with antineoplastic activity (IC50s: 0.6 μM, 0.1 μM and 0.1 μM for v-Abl, c-Kit and PDGFR,Formula:C29H31N7O·CH4SO3Purezza:98% - >99.99%Colore e forma:White SolidPeso molecolare:589.71AS1949490
CAS:AS1949490, a selective SHIP-2 inhibitor with IC50 of 620 nM, boosts glucose metabolism by upregulating GLUT1 in L6 myotubes.Formula:C20H18ClNO2SPurezza:99.94%Colore e forma:SolidPeso molecolare:371.88Ref: TM-T14327
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg119,00€25mg236,00€50mg380,00€100mg555,00€Delcasertib
CAS:Delcasertib (KAI-9803) is a potent and selective inhibitor of δ-protein kinase C (δPKC).Formula:C120H199N45O34S2Purezza:99.96%Colore e forma:SolidPeso molecolare:2880.28Ref: TM-T11740
1mg192,00€5mg485,00€10mg700,00€25mg1.063,00€50mg1.459,00€1mL*10mM (DMSO)1.603,00€100mg1.963,00€BNC105
CAS:BNC105 is a tubulin polymerization inhibitor. It has potent antiproliferative and tumor vascular disrupting properties.Formula:C20H20O7Purezza:96.57%Colore e forma:SolidPeso molecolare:372.37Ref: TM-T14694
1mg79,00€5mg152,00€1mL*10mM (DMSO)167,00€10mg215,00€25mg351,00€50mg494,00€100mg665,00€200mg893,00€Spiperone
CAS:Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.Formula:C23H26FN3O2Purezza:99.34% - 99.91%Colore e forma:SolidPeso molecolare:395.47
