
Antiparassitari
Gli antiparassitari sono composti progettati per trattare e prevenire le infezioni parassitarie inibendo la crescita e la sopravvivenza dei parassiti. Questa categoria include una gamma di agenti antiparassitari destinati esclusivamente all'uso in laboratorio e non per il consumo umano. Questi prodotti sono essenziali per scopi di ricerca, consentendo agli scienziati di studiare i cicli di vita dei parassiti, i meccanismi d'azione e lo sviluppo della resistenza. L'uso di antiparassitari in ambienti di laboratorio aiuta nella scoperta e nell'ottimizzazione di nuovi trattamenti per le malattie parassitarie, contribuendo ai progressi nella parassitologia medica e veterinaria. I ricercatori si affidano a questi prodotti per migliorare la comprensione delle infezioni parassitarie e sviluppare terapie più efficaci.
Trovati 703 prodotti di "Antiparassitari"
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Antileishmanial agent-16
CAS:Antileishmanial agent-16 (compound 14c), an anti-Leishmania agent, exhibits potent activity against Leishmania major promastigotes (IC50 = 0.59 µM) andFormula:C27H37N5O4Purezza:98%Colore e forma:SolidPeso molecolare:495.61DDD85646
CAS:DDD85646 is an inhibitor of T. brucei N-myristoyltransferase with a Ki of 1.44 nM, an IC50 of 2 nM and an EC50 of 2 nM. The IC50 of hNMT is 4 nM.Formula:C21H24Cl2N6O2SPurezza:97.8% - 99.76%Colore e forma:SolidPeso molecolare:495.43Ref: TM-T27135
1mg96,00€5mg266,00€10mg399,00€25mg677,00€50mg940,00€100mg1.293,00€1mL*10mM (DMSO)290,00€Phylloflavan
CAS:Phylloflavan, an antileishmanial compound, exhibits an intracellular half maximal effective concentration (EC50) of 3.2 nM in RAW 264.7 cells and inhibits theFormula:C26H26O10Purezza:98%Colore e forma:SolidPeso molecolare:498.48Antileishmanial agent-17
CAS:Antileishmanial agent-17, a coumarin hybrid, exhibits potent antileishmanial activity (IC50 <0.78 μM) while proving non-toxic to normal VERO cells.Formula:C27H37N5O5Purezza:98%Colore e forma:SolidPeso molecolare:511.61ELQ-596
CAS:ELQ-596, a quinolone derivative, exhibits antimicrobial activity against several protozoan parasites, including the intraerythrocytic parasites Plasmodium and Babesia. ELQ-596 attenuates babesiosis in immunosuppressed mice [1].Formula:C24H17ClF3NO3Colore e forma:SolidPeso molecolare:459.84UCB7362
CAS:UCB7362 (GLXC-26743) is an orally available and potent plasmepsin X (PMX) inhibitor with anti-malarial activity.UCB7362 inhibits parasite reproduction.Formula:C25H26ClN5O3Purezza:97.67%Colore e forma:SolidPeso molecolare:479.96Propamidine
CAS:Propamidine acts as a covalent inhibitor of TMPRSS2 and exhibits antibacterial properties. [1]Formula:C17H20N4O2Purezza:98%Colore e forma:SolidPeso molecolare:312.37EDI048
CAS:EDI048, also known as compound 1.16, is an orally active inhibitor of Cryptosporidium PI4K, utilized in the study of cryptosporidiosis [1].Formula:C25H21ClN4O4Purezza:98%Colore e forma:SolidPeso molecolare:476.91BTG 502
CAS:BTG 502 is an alkylamide insecticide that binds to voltage-gated sodium channels, antagonising the activation of sodium channels by Batrachotoxin (BTX).Formula:C21H24BrNOPurezza:99.30%Colore e forma:SolidPeso molecolare:386.33Antileishmanial agent-23
CAS:Antileishmanial agent-23 (compound G1/9), a potent and selective trypanothione reductase (TR) inhibitor, exhibits an IC50 of 2.24 ± 0.52 μM.Formula:C20H17N3O4S2Purezza:98%Colore e forma:SolidPeso molecolare:427.5Eugenitin
CAS:Eugenitin, a polyketide from Mycoleptodiscus indicus, exhibits inhibitory activity against Leishmania major with an LD50 of 39.9 μM and demonstrates lowFormula:C12H12O4Purezza:98%Colore e forma:SolidPeso molecolare:220.22OfChi-h-IN-2
CAS:OfChi-h-IN-2 (compound TQ19) is a potent inhibitor of OfChi-h, exhibiting a K i of 0.33 μM, and significantly impairs the growth and development of OstriniaFormula:C25H28ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:481.98FIKK9.1-IN-1
CAS:FIKK9.1-IN-1 (Compound 1), an antimalarial agent (IC50: 2.68 μg/mL), serves as a FIKK9.1 inhibitor by interacting with the ATP-binding residues within FIKK9.1,Formula:C22H22N2SePurezza:98%Colore e forma:SolidPeso molecolare:393.38Z-Pro-Pro-CHO
CAS:Z-Pro-Pro-CHO acts as a prolyl oligopeptidase inhibitor with half-maximal inhibitory concentrations (IC50) of 0.16 μM for human prolyl oligopeptidase and 0.01Formula:C18H22N2O4Purezza:98%Colore e forma:SolidPeso molecolare:330.38Fervenulin
CAS:<p>Fervenulin, from Streptomyces sp. CMU-MH021, halts egg hatch (MIC: 30 μg/mL) and kills J2 larvae (MIC: 120 μg/mL) of M. incognita.</p>Formula:C7H7N5O2Purezza:99.75%Colore e forma:SolidPeso molecolare:193.16Myrrhterpenoid O
CAS:Unfortunately, you did not provide the description of the chemical compound that needs to be rewritten.Formula:C16H20O3Purezza:98%Colore e forma:SolidPeso molecolare:260.33SID 26681509
CAS:SID 26681509 is a selective, reversible and competitive human cathepsin L inhibitor (IC50 of 56 nM).Formula:C27H33N5O5SPurezza:99.18%Colore e forma:SolidPeso molecolare:539.65Ref: TM-T12909
1mg66,00€5mg144,00€10mg216,00€25mg437,00€50mg652,00€100mg930,00€1mL*10mM (DMSO)172,00€Dehydroemetine
CAS:Dehydroemetine, a synthetic emetine, treats amoebic infections and leishmaniasis, and resists metronidazole amoebiosis.Formula:C29H38N2O4Purezza:98.68% - 99.68%Colore e forma:SolidPeso molecolare:478.62GSK3186899
CAS:GSK3186899 is an inhibitor of Cdc2-related kinase 12 with an EC50 of 1.4 μM for L. donovani.Formula:C19H28F3N7O3SPurezza:98.35% - 99.61%Colore e forma:SolidPeso molecolare:491.53ZY-19489
CAS:<p>ZY-19489: Antimalarial, potential single-dose cure, FDA orphan drug status.</p>Formula:C24H32FN9Purezza:>99.99%Colore e forma:SoildPeso molecolare:465.57
