
Antiparassitari
Gli antiparassitari sono composti progettati per trattare e prevenire le infezioni parassitarie inibendo la crescita e la sopravvivenza dei parassiti. Questa categoria include una gamma di agenti antiparassitari destinati esclusivamente all'uso in laboratorio e non per il consumo umano. Questi prodotti sono essenziali per scopi di ricerca, consentendo agli scienziati di studiare i cicli di vita dei parassiti, i meccanismi d'azione e lo sviluppo della resistenza. L'uso di antiparassitari in ambienti di laboratorio aiuta nella scoperta e nell'ottimizzazione di nuovi trattamenti per le malattie parassitarie, contribuendo ai progressi nella parassitologia medica e veterinaria. I ricercatori si affidano a questi prodotti per migliorare la comprensione delle infezioni parassitarie e sviluppare terapie più efficaci.
Trovati 701 prodotti di "Antiparassitari"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
GNF179
CAS:GNF179 is an optimized 8,8-dimethyl IP analog.Formula:C22H23ClFN5OPurezza:98.9%Colore e forma:SolidPeso molecolare:427.9Lotilaner
CAS:Lotilaner is a parasiticide.Formula:C20H14Cl3F6N3O3SPurezza:99.56%Colore e forma:SolidPeso molecolare:596.76CpNMT-IN-1
<p>CpNMT-IN-1 (Compound 11e) is an inhibitor of N-myristoyltransferase (CpNMT) with an IC50 value of 2.5 μM. It also inhibits the growth of microsporidia, demonstrating an EC50 value of 6.9 μM.</p>Formula:C25H25ClN4O4SColore e forma:SolidPeso molecolare:513.008AAP4
AAP4 is a potent inhibitor of OfChi-h and OfHex1, exhibiting Ki values of 29.3 nM and 4.9 μM, respectively. It also demonstrates insecticidal activity against the lepidopteran pest Ostrinia furnacalis.Formula:C21H23BrClN7Colore e forma:SolidPeso molecolare:488.811Ile-AMS TFA
Ile-AMS TFA exhibits activity against P. falciparum, with an ABSIC50 value of 1.19 nM.Formula:C18H27F3N8O8SColore e forma:SolidPeso molecolare:572.52Alkaline tryptase-IN-1
Alkaline tryptase-IN-1 (compound H-13) is an insecticide that targets alkaline trypsin-like enzymes. It has lethal concentration (LC50) values of 8.72, 13.77, 14.17, 12.96, and 12.35 μg/mL against Schizaphis graminum, Sitobion avenae, Brevicoryne brassicae, Aphis gossypii, Aphis spiraecola, and Myzus persicae, respectively.Formula:C29H33BrN2O2SColore e forma:SolidPeso molecolare:553.55TSO-13
<p>TSO-13 is an inhibitor of the major cysteine protease Cruzipain found in Trypanosoma cruzi, with an IC50 of 2.2 μM. In Vero cells, TSO-13 also suppresses T. cruzi, exhibiting an IC50 of 1.9 μM.</p>Formula:C32H36N4O4S2Colore e forma:SolidPeso molecolare:604.78Azlocillin sodium salt
CAS:<p>Azlocillin sodium, an acylampicillin, is a broad-spectrum antibiotics</p>Formula:C20H22N5NaO6SPurezza:97.63% - 98.302%Colore e forma:SolidPeso molecolare:483.47Antiparasitic agent-26
<p>Antiparasitic agent-26 (Compound 8) is an antiparasitic compound that effectively inhibits the growth of Naegleria fowleri, with an IC50 of 22.87 μM (trophozoite stage) and 25.16 μM (cyst stage). It exerts its antiparasitic effects by inducing programmed cell death, which includes cytosolic calcium accumulation, mitochondrial membrane potential collapse, ATP synthesis inhibition, ROS accumulation, and chromatin condensation. Antiparasitic agent-26 can be utilized in research on primary amoebic meningoencephalitis (PAM).</p>Colore e forma:Odour SolidAntitrypanosomal agent 23
Antitrypanosomal agent 23 is an antiparasitic compound effective against intracellular amastigotes of Trypanosoma cruzi in LLC-MK2 and C2C12 cells, demonstrating activity with IC50 values of 0.10 and 0.11 μM, respectively. It also acts as a weak inhibitor of recombinant Trypanosoma cruzi sialyltransferase (TcTS) with an IC50 of 1.1 mM.Formula:C14H16N4O7Colore e forma:SolidPeso molecolare:352.1019Febrifugine dihydrochloride
CAS:Febrifugine dihydrochloride (Propyldazine hydrochloride) is a biochemical with therapeutic activity regarding malaria, cancer, fibrosis and inflammatoryFormula:C16H21Cl2N3O3Purezza:98.27% - 99.85%Colore e forma:SolidPeso molecolare:374.26SpdSyn binder-1
CAS:SpdSyn binder-1 weakly inhibits malaria by binding to Plasmodium falciparum's spermidine synthase. Used for research.Formula:C21H22N4OPurezza:99.5%Colore e forma:SolidPeso molecolare:346.43Norselic acid B
CAS:Norselic acid B is a naturally occurring compound that can be isolated from the sponge Crella sp. collected in Antarctica. It demonstrates activity against Leishmania parasites.Formula:C29H44O4Colore e forma:SolidPeso molecolare:456.657Dixanthogen
CAS:Dixanthogen (Auligen) is an ectoparasiticide. Dixanthogen is a thiocarbonyl compound.Formula:C6H10O2S4Purezza:95% - 98%Colore e forma:SolidPeso molecolare:242.4Antiproliferative agent-56
Antiproliferative agent-56 (Compound 31) is an antimalarial agent that inhibits the Pf3D7 strain of the malaria parasite Plasmodium falciparum with an IC50 of >12.5 (48h) and 0.03 μM (98h), displaying slow-acting characteristics.Colore e forma:Odour SolidNitroxynil
CAS:Nitroxynil is an anthelmintic for adult/immature parasites, mainly used in Fasciola hepatica studies.Formula:C7H3IN2O3Purezza:99.76%Colore e forma:SolidPeso molecolare:290.01Antimalarial agent 43
Antimalarial agent 43 (compound 16c) is an antimalarial compound that exhibits an IC50 value of 0.0151 μM against the 3D7 strain.Colore e forma:Odour SolidSulfadiazine
CAS:<p>Sulfadiazine, a short-acting sulfonamide, blocks bacterial folic acid synthesis; used with pyrimethamine to treat toxoplasmosis in AIDS, newborns.</p>Formula:C10H10N4O2SPurezza:99.32%Colore e forma:White To Slightly Yellow Crystalline PowderPeso molecolare:250.28Nicarbazin
CAS:Nicarbazin (Nicoxin) is an equimolar complex of 4, 4'-Dinitrocarbanilide and 2-Hydroxy-4, 6-dimethylpyrimidine. A coccidiostat for poultry.Formula:C19H18N6O6Purezza:99.54%Colore e forma:Crystals Yellow Or Greenish Yellow Powder Odorless With A Bit Of SmellPeso molecolare:426.38Amprolium
CAS:Amprolium is a veterinary coccidiostat that interferes with THIAMINE metabolism.Formula:C14H19N4·ClPurezza:98%Colore e forma:SolidPeso molecolare:278.79

