
Recettori accoppiati alla proteina G e recettori 7-TM
I recettori accoppiati alle proteine G (GPCR) e i recettori a 7 domini transmembrana (7-TM) sono una grande famiglia di proteine di membrana che svolgono ruoli chiave nella comunicazione cellulare e nella trasduzione del segnale. Questi recettori sono coinvolti in un'ampia gamma di processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la regolazione ormonale. I GPCR sono bersagli principali nella scoperta di farmaci, rendendoli essenziali per la ricerca in farmacologia e medicina. Presso CymitQuimica, offriamo un'ampia selezione di reagenti e composti di alta qualità correlati ai GPCR e ai recettori 7-TM per supportare la tua ricerca e gli sforzi di sviluppo di farmaci.
Trovati 5875 prodotti per "Recettori accoppiati alla proteina G e recettori 7-TM".
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Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Formula:C19H29ClN2O4Purezza:99.49%Colore e forma:SolidPeso molecolare:384.9Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Formula:C31H33N3O4Purezza:99.66%Colore e forma:SolidPeso molecolare:511.61Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFormula:C17H19N3·HClPurezza:98% - 99.53%Colore e forma:White SolidPeso molecolare:301.82Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purezza:99.35%Colore e forma:White SolidPeso molecolare:335.87Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formula:C15H23N3O4SPurezza:98.20% - 99.88%Colore e forma:White SolidPeso molecolare:341.43Cefaclor monohydrate
CAS:Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.Formula:C15H16ClN3O5SPurezza:97.36% - 99.9%Colore e forma:White SolidPeso molecolare:385.82AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formula:C17H14O5Purezza:97.59%Colore e forma:SolidPeso molecolare:298.29Ref: TM-T14148
1mg34,00€5mg63,00€1mL*10mM (DMSO)67,00€10mg92,00€25mg165,00€50mg250,00€100mg401,00€200mg580,00€(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H10FNO2Purezza:97.82%Colore e forma:SolidPeso molecolare:195.19Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Formula:C19H23Cl2N5OPurezza:99.5% - 99.52%Colore e forma:SolidPeso molecolare:408.33Ticlopidine hydrochloride
CAS:Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Formula:C14H15Cl2NSPurezza:99.83% - 99.97%Colore e forma:White PowderPeso molecolare:300.25Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purezza:99.85% - 99.99%Colore e forma:SolidPeso molecolare:367.50Azatadine dimaleate
CAS:Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Formula:C28H30N2O8Purezza:99.7% - >99.99%Colore e forma:SolidPeso molecolare:522.55Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formula:C22H21Cl3N4OPurezza:98% - 99.91%Colore e forma:White SolidPeso molecolare:463.79Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFormula:C19H25F3N2O6Purezza:99.92% - 99.94%Colore e forma:White SolidPeso molecolare:434.41Ref: TM-T1077
1mL*10mM (DMSO)35,00€10mg49,00€25mg65,00€50mg80,00€100mg109,00€200mg161,00€500mg263,00€Salmeterol
CAS:Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.Formula:C25H37NO4Purezza:99.2% - 99.9%Colore e forma:SolidPeso molecolare:415.57Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formula:C22H23N3O2Purezza:99.29% - 99.97%Colore e forma:White SolidPeso molecolare:361.44Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purezza:99.43% - 99.62%Colore e forma:White SolidPeso molecolare:448.39Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purezza:99.98%Colore e forma:SolidPeso molecolare:231.65Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurezza:99.44% - 99.84%Colore e forma:SolidPeso molecolare:307.39Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purezza:99.16% - 99.86%Colore e forma:SolidPeso molecolare:266.55
