Derivati delle Benzodiazepine
Le benzodiazepine sono composti organici con un nucleo biciclico fuso di benzodiazepina, ampiamente utilizzati nello sviluppo di farmaci con proprietà ansiolitiche, sedative, anticonvulsivanti e miorilassanti. I loro derivati includono strutture modificate che ne migliorano la selettività e il profilo farmacocinetico, consentendo la creazione di nuove molecole con applicazioni terapeutiche avanzate. Questi composti sono impiegati nella formulazione di API per il trattamento dei disturbi del sonno, dell’ansia, dell’epilessia e degli spasmi muscolari. Inoltre, i derivati delle benzodiazepine sono fondamentali nella ricerca di nuovi agenti psicotropi e nell’ottimizzazione dei trattamenti neurologici.
Presso CymitQuimica, offriamo derivati delle benzodiazepine di alta purezza per applicazioni in sintesi chimica, sviluppo farmaceutico e neuroscienze.
Trovati 333 prodotti di "Derivati delle Benzodiazepine"
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3-AMINO-1-METHYL-5-PHENYL-1H-BENZO[E][1,4]DIAZEPIN-2(3H)-ONE
CAS:Purezza:95.0%Colore e forma:SolidPeso molecolare:265.3160095214844Defluoro 8-Hydroxy Flumazenil
CAS:Prodotto controllatoFormula:C15H15N3O4Colore e forma:NeatPeso molecolare:301.30(R)-3-amino-9-fluoro-5-phenyl-1H-benzo[e][1,4]diazepin-2(3H)-one
Purezza:97%Peso molecolare:269.27899169921875Ref: 10-F790109
1gPrezzo su richiesta50mgPrezzo su richiesta100mgPrezzo su richiesta250mgPrezzo su richiesta2H-1,4-Benzodiazepin-2-one, 3-amino-1,3-dihydro-5-phenyl-, (3S)-
CAS:Purezza:98%Peso molecolare:251.289Cloxazolam
CAS:Prodotto controllato<p>Applications Cloxazolam is a benzodiazepine derivative with anxiolytic, hypnotic and antihypertensive properties used as an anti-anxiety drug. It is metabolized into the active metabolite Delorezepam (D230675). Controlled Substance.<br>References Oliveira-Silva, D. et al.: Biomed. Chrom., 23, 1266 (2009); Kamioka, T. et al.: Psychopharmacol., 52, 17 (1977); Fischer-Cornelssen, K.A. et al.: Arzneim.-Forsch., 31, 1757 (1981);<br></p>Formula:C17H14Cl2N2O2Colore e forma:NeatPeso molecolare:349.213-Amino-5-phenyl-1H-benzo[e][1,4]diazepin-2(3H)-one
CAS:Purezza:95.0%Peso molecolare:251.289001464843757-bromo-5-phenyl-1,3-dihydro-2H-benzo[e][1,4]diazepin-2-one
CAS:Purezza:95.0%Peso molecolare:315.17001342773447-methyl-5-phenyl-1,3,4,5-tetrahydro-2H-benzo[e][1,4]diazepin-2-one
CAS:Purezza:95.0%Peso molecolare:252.317001342773444-(2-Benzoyl-4-chlorophenyl)-5-methyl-4H-1,2,4-triazole-3-carboxaldehyde
CAS:Prodotto controllatoFormula:C17H12ClN3O2Colore e forma:NeatPeso molecolare:325.758-Chloro-5,6-dihydro-5-methyl-6-oxo-4H-Imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic Acid Ethyl Ester
CAS:Prodotto controllato<p>Impurity Flumazenil EP Impurity F<br>Applications 8-Chloro-5,6-dihydro-5-methyl-6-oxo-4H-Imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic Acid Ethyl Ester is an impurity of Flumazenil (F500450), an imidazodiazepine which selectively blocks the central effects of classic benzodiazepines.<br>References Hunkeler, W., et al.: Nature, 290, 514 (1981), Pole, P., et al.: Arch. Pharmacol., 316, 317 (1981), Timm, U., et al.: Arzneim.-Forsch., 33, 358 (1983),<br></p>Formula:C15H14ClN3O3Colore e forma:NeatPeso molecolare:319.743-Amino-6-bromo-4-(2-pyridinyl)-2(1H)-quinolinone(>90%)
CAS:Prodotto controllato<p>Stability Air Sensitive<br>Applications 3-Amino-6-bromo-4-(2-pyridinyl)-2(1H)-quinolinone is an impurity of Bromazepam (B678500); a controlled substance (depressant) and anxiolytic.<br>References Schwartz, M.A., et al.: J. Pharm. Sci., 62, 1776 (1973); Chalmers, P., et al.: Anesthesia, 39, 370 (1984); Hassan, M.M., et al.: Anal. Profiles Drug Subs., 16, 1 (1987)<br></p>Formula:C14H10BrN3OPurezza:>90%Colore e forma:Light Brown To BrownPeso molecolare:316.15Alprazolam 5-Oxide
CAS:Prodotto controllato<p>Applications A metabolite of Alprazolam (A575650).<br>References Schwartz, M.A., et al.: J. Pharmacol. Exp. Ther., 149, 423 (1965), Childress, S.J., et al.: J. Pharm. Sci., 53, 577 (1964), Gall, M., et al.: J. Med. Chem., 21, 1290 (1978)<br></p>Formula:C17H13ClN4OColore e forma:NeatPeso molecolare:324.767-Chloro-1,3-dihydro-5-phenyl-2H-1,4-benzodiazepine-2-thione
CAS:Prodotto controllato<p>Applications 7-Chloro-1,3-dihydro-5-phenyl-2H-1,4-benzodiazepine-2-thione (cas# 4547-02-8) is a positive allosteric modulator for the muscarinic M1 receptor, which could be a potential treament for the Alzheimer's disease or Schizophrenia.<br>References Flohr, A., et al.: Bioorg. Med. Chem. Lett., 27, 5415 (2017)<br></p>Formula:C15H11ClN2SColore e forma:BeigePeso molecolare:286.7792Bromazepam-d4
CAS:Prodotto controllato<p>Applications Controlled substance (depressant). Anxiolytic. Labelled Bromazepam.<br>References Schwartz, M.A., et al.: J. Pharm. Sci., 62, 1776 (1973), Chalmers, P., et al.: Anesthesia, 39, 370 (1984), Hassan, M.M., et al.: Anal. Profiles Drug Subs., 16, 1 (1987),<br></p>Formula:C142H4H6BrN3OColore e forma:NeatPeso molecolare:320.18Clobazam-13C6 (1 mg/ml in Acetonitrile)
CAS:Prodotto controllatoFormula:C6C10H13ClN2O2Colore e forma:ColourlessPeso molecolare:306.702-Amino-5-nitro-2'-chlorobenzophenone
CAS:<p>Impurity Clonazepam EP Impurity A<br>Applications 2-Amino-5-nitro-2'-chlorobenzophenone (Clonazepam EP Impurity A) is an impurity of Clonazepam (C587080).<br></p>Formula:C13H9ClN2O3Colore e forma:NeatPeso molecolare:276.68Flunitrazepam
CAS:Prodotto controllato<p>Applications Flunitrazepam is used as an hypnotic. This is a controlled substance (depressant).<br>References Sternbach, L.H., et al.: J. Med. Chem., 6, 261 (1963), Eidelberg, E., et al.: Neurology, 5, 223 (1965), Caplan, Y., et al.: J. Anal. Toxicol., 25, 396 (2001), Wood, M., et al.: Forensic Sci. Int., 150, 227 (2005),<br></p>Formula:C16H12FN3O3Colore e forma:Off-WhitePeso molecolare:313.283-Amino-4-(2-chlorophenyl)-6-nitro-2(1H)-quinolinone (Clonazepam Impurity)
CAS:<p>Impurity Clonazepam EP Impurity B<br>Applications 3-Amino-4-(2-chlorophenyl)-6-nitro-2(1H)-quinolinone (Clonazepam EP Impurity B) is an impurity of Clonazepam (C587080), antiepileptic agent with anxiolytic and antimanic properties.<br>References Mayer, W., et al.: Pharmazie, 29, 700 (1974), Blum, et al.: Arzneim.-Forsch., 23, 377 (1973), Winslow, W.C., et al.: Anal. Profiles Drug Subs., 6, 61 (1977)<br></p>Formula:C15H10ClN3O3Colore e forma:Yellow BrownPeso molecolare:315.717-Amino Clonazepam
CAS:Prodotto controllato<p>Applications The major metabolite of Clonazepam (C587080).<br>References Clark, D., et al.: Drugs, 29, 342 (1985), Colmenero, J., et al.: Antimicrob. Agents Chemother., 38, 2798 (1994), Grant, D., et al.: Pharmacology, 61, 204 (2000), Negrusz, A., et al.: Anal. Bioanal. Chem., 376, 1198 (2003),<br></p>Formula:C15H12ClN3OColore e forma:YellowPeso molecolare:285.73Methyl Clonazepam
CAS:Prodotto controllato<p>Applications Shows sedative and anxiolytic properties. Impairment of psychomotor performance reported. Activity blocked by flumazenil.<br>References Doumont, A., et al.: Psychopharmacology, 87, 130 (1985), Psychopharmacology, 94(4), 501 (1988)<br></p>Formula:C16H12ClN3O3Colore e forma:YellowPeso molecolare:329.74
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