Derivati delle Benzodiazepine
Le benzodiazepine sono composti organici con un nucleo biciclico fuso di benzodiazepina, ampiamente utilizzati nello sviluppo di farmaci con proprietà ansiolitiche, sedative, anticonvulsivanti e miorilassanti. I loro derivati includono strutture modificate che ne migliorano la selettività e il profilo farmacocinetico, consentendo la creazione di nuove molecole con applicazioni terapeutiche avanzate. Questi composti sono impiegati nella formulazione di API per il trattamento dei disturbi del sonno, dell’ansia, dell’epilessia e degli spasmi muscolari. Inoltre, i derivati delle benzodiazepine sono fondamentali nella ricerca di nuovi agenti psicotropi e nell’ottimizzazione dei trattamenti neurologici.
Presso CymitQuimica, offriamo derivati delle benzodiazepine di alta purezza per applicazioni in sintesi chimica, sviluppo farmaceutico e neuroscienze.
Trovati 333 prodotti di "Derivati delle Benzodiazepine"
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9-Nitro-3,4-dihydro-1H-benzo[e][1,4]diazepin-5(2H)-one
CAS:Formula:C9H9N3O3Purezza:95.0%Peso molecolare:207.1898-Amino-4-Boc-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C14H21N3O2Purezza:97%Peso molecolare:263.3417-Fluoro-3,4-dihydro-1H-benzo[e][1,4]diazepine-2,5-dione
CAS:Formula:C9H7FN2O2Purezza:97.0%Colore e forma:SolidPeso molecolare:194.1654-Boc-2,3,4,5-Tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C14H20N2O2Purezza:97.0%Colore e forma:SolidPeso molecolare:248.3264-Boc-9-Methyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C15H22N2O2Purezza:97.0%Peso molecolare:262.3538-Chloro-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C9H11ClN2Purezza:97.0%Colore e forma:SolidPeso molecolare:182.653-(Piperidin-4-yl)-1,3,4,5-tetrahydro-2H-benzo[d][1,3]diazepin-2-one
CAS:Purezza:97%Peso molecolare:245.3260044-Boc-7-Methyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C15H22N2O2Purezza:97.0%Peso molecolare:262.3532,3,4,5-Tetrahydro-1H-benzo[e][1,4]diazepine
CAS:Formula:C9H12N2Purezza:97.0%Colore e forma:White to yellow/orange crystalline powderPeso molecolare:148.2098-Bromo-3,4-dihydro-1H-benzo[e][1,4]diazepin-5(2H)-one
CAS:Formula:C9H9BrN2OPurezza:97.0%Peso molecolare:241.0881,2,4,5-Tetrahydro-benzo[e][1,4]diazepin-3-one
CAS:Formula:C9H10N2OPurezza:97.0%Colore e forma:SolidPeso molecolare:162.1922,3,4,5-TETRAHYDRO-1H-BENZO[E][1,4]DIAZEPIN-8-YLAMINE 2HCL
CAS:Formula:C9H15Cl2N3Purezza:97.0%Peso molecolare:236.143-Amino-4-(2-fluorophenyl)-1-methyl-6-nitroquinolin-2(1H)-one
CAS:Prodotto controllatoFormula:C16H12FN3O3Colore e forma:NeatPeso molecolare:313.283-Methyl Clobazam
CAS:Prodotto controllato<p>Applications 3-Methyl Clobazam is a metabolite of Clobazam (C582500), a benzodiazepine psychotherapeutic agent that has proven efficacy against multiple seizure types. An anxiolytic; anticonvulsant.<br>References Gastaut, H., et al.: Epilepsia, 20, 437 (1979); Guberman, A., et al.: Can J. Neurol. Sci., 17, 311 (1990); Munn, R., et al.: Pediatr. Neurol. 9, 465 (1993)<br></p>Formula:C17H15ClN2O2Colore e forma:NeatPeso molecolare:314.773,3-Dimethyl Clobazam
Prodotto controllatoFormula:C18H17ClN2O2Colore e forma:NeatPeso molecolare:328.792-(2-Aminoacetamido)-5-nitro-2'-chlorobenzophenone Hydrochloride (Clonazepam Impurity)
CAS:Prodotto controllatoFormula:C15H12ClN3O4·ClHColore e forma:WhitePeso molecolare:370.18747-Aminonorflunitrazepam
CAS:Prodotto controllatoFormula:C15H12FN3OColore e forma:Light YellowPeso molecolare:269.27N,N-Dimethylformamide Diethyl Acetal
CAS:Prodotto controllato<p>Stability Moisture Sensitive<br>Applications N,N-Dimethylformamide Diethyl Acetal is used as a reagent in the design of EGF-R tyrosine kinase inhibitors. Also used in the synthesis of aminopyridine derivatives.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Traxler, P. et al.: J. Med. Chem., 40, 3601 (1997); Cheikh, N. et al.: Tetrahedron, 69, 1234 (2013);<br></p>Formula:C7H17NO2Colore e forma:NeatPeso molecolare:147.22Flumazenil Carboxylic Acid-D3
Prodotto controllato<p>Applications Flumazenil Carboxylic Acid-D3 is an isotope labelled form of Flumazenil Carboxylic Acid (F500455); a derivative of Flumazenil (F500455), a benzodiazepine antagonist that can prevent or abolish (at the receptor level) the effects of a benzodiazepine.<br>References Brogden, R. & Goa, K.: Drugs, 35, 448 (1988); Klotz, U. & Kanto, J.: Clin. Pharmacokinet., 14, 1 (1988)<br></p>Formula:C13H7D3FN3O3Colore e forma:NeatPeso molecolare:278.252-Amino-5-nitrobenzophenone
CAS:Prodotto controllatoFormula:C13H10N2O3Colore e forma:NeatPeso molecolare:242.233-Amino-6-chloro-3,4-dihydro-2-methyl-4-phenyl-4-quinazolinol
CAS:Prodotto controllatoFormula:C15H14ClN3OColore e forma:NeatPeso molecolare:287.742-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine
CAS:Prodotto controllato<p>Applications 2-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine is an impurity of Alprazolam (A575650.<br>References Hester, J.B., et al.: J. Org. Chem., 44, 2688, (1979); Anjaneyulu, Y., et al.: Asian. J. Chem., 19, 3375 (2007);<br></p>Formula:C17H15ClN4OColore e forma:White To Off-WhitePeso molecolare:326.782-Bromo-N-[4-bromo-2-(2-pyridinylcarbonyl)phenyl]-acetamide
CAS:Prodotto controllato<p>Applications 2-Bromo-N-[4-bromo-2-(2-pyridinylcarbonyl)phenyl]-acetamide is a derivative of 2-(2-Amino-5-bromobenzoyl)pyridine (A601785); an intermediate in the preparation of Bromazepam (B678500).<br>References Panderi, I., et al.: J. Pharm. Biomed. Anal., 17, 327 (1998); El-Haj, B., et al.: J. Anal. Toxicol., 25, 316 (2001); Hansen, S., et al.: J. Pharm. Biomed. Anal., 39, 322 (2005)<br></p>Formula:C14H10Br2N2O2Colore e forma:NeatPeso molecolare:398.05N-(4-Bromo-2-picolinoylphenyl)-2-chloroacetamide
CAS:Prodotto controllato<p>Applications N-(4-Bromo-2-picolinoylphenyl)-2-chloroacetamide is a derivative of 2-(2-Amino-5-bromobenzoyl)pyridine (A601785); an intermediate in the preparation of Bromazepam (B678500).<br>References Panderi, I., et al.: J. Pharm. Biomed. Anal., 17, 327 (1998); El-Haj, B., et al.: J. Anal. Toxicol., 25, 316 (2001); Hansen, S., et al.: J. Pharm. Biomed. Anal., 39, 322 (2005)<br></p>Formula:C14H10BrClN2O2Colore e forma:Light Yellow To BeigePeso molecolare:353.60Alprazolam 5,6-Epoxide
CAS:Prodotto controllato<p>Applications Alprazolam derivative.<br>References Hester, J. et al., J. of Med. Chem. 23, 643 (1980)<br></p>Formula:C17H13ClN4OColore e forma:NeatPeso molecolare:324.772-(2-Amino-5-bromobenzoyl)pyridine
CAS:<p>2-(2-Amino-5-bromobenzoyl)pyridine (2ABBP) is a chemical compound with the molecular formula C10H7BrN3. It is a glucuronide conjugate of 2-amino-5-bromobenzoic acid and has been used as an immunological reagent in the form of a monoclonal antibody. 2ABBP binds to dryopteris, which is a plant species that contains polyphenols called pteridines. 2ABBP has been shown to have anti-inflammatory properties in rat liver microsomes and cell culture experiments. The mechanism of action may involve inhibition of cyclooxygenase enzymes, which are involved in prostaglandin synthesis. 2ABBP also binds to human serum albumin and chaperones, proteins that bind other proteins or small molecules. The biological activity of 2ABBP may be due to its ability to form coval</p>Formula:C12H9BrN2OPurezza:Min. 95%Peso molecolare:277.12 g/molClobazam CIV
CAS:Prodotto controllatoClobazam (inn) and methyprylon (inn)Formula:C16H13ClN2O2Colore e forma:White Crystalline PowderPeso molecolare:300.066567-Amino Clonazepam-d4
CAS:Prodotto controllato<p>Applications A labelled major metabolite of Clonazepam (C587080).<br>References Clark, D., et al.: Drugs, 29, 342 (1985), Colmenero, J., et al.: Antimicrob. Agents Chemother., 38, 2798 (1994), Grant, D., et al.: Pharmacology, 61, 204 (2000), Negrusz, A., et al.: Anal. Bioanal. Chem., 376, 1198 (2003),<br></p>Formula:C152H4H8ClN3OColore e forma:NeatPeso molecolare:289.75
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![2,3,4,5-TETRAHYDRO-1H-BENZO[E][1,4]DIAZEPIN-8-YLAMINE 2HCL](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2F10%2Fthumb-webp%2FF304019.webp&w=3840&q=75)
![2-Bromo-N-[4-bromo-2-(2-pyridinylcarbonyl)phenyl]-acetamide](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FB680675.webp&w=3840&q=75)
