Sulfonamidi e Derivati
Le sulfonamidi sono composti che contengono un gruppo funzionale sulfonamidico (-SO₂NH₂), in cui un atomo di zolfo è legato a un gruppo amminico. Furono tra i primi antibiotici sintetici utilizzati in medicina, inibendo la sintesi dell’acido folico nei batteri, conferendo loro proprietà antimicrobiche. Sono utilizzate principalmente per trattare infezioni batteriche, sebbene il loro impiego sia diminuito a causa della resistenza antimicrobica. Oltre al loro uso come antibiotici, le sulfonamidi trovano applicazioni nel trattamento di malattie come la malaria e le malattie infiammatorie intestinali.
Presso CymitQuimica, offriamo sulfonamidi e i loro derivati ad alta purezza per la ricerca in microbiologia e lo sviluppo farmaceutico.
Trovati 2589 prodotti di "Sulfonamidi e Derivati"
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1-(N-(2,2,2-trifluoroethyl)sulfamoyl)piperidine-4-carboxylic acid
CAS:Formula:C8H13F3N2O4SPurezza:95.0%Peso molecolare:290.261-(Piperidine-1-sulfonyl)piperazine
CAS:Formula:C9H19N3O2SPurezza:98.0%Colore e forma:SolidPeso molecolare:233.331-(N-(2,2,2-trifluoroethyl)sulfamoyl)piperidine-3-carboxylic acid
CAS:Formula:C8H13F3N2O4SPurezza:95.0%Peso molecolare:290.262-Methyl-2H-1,2-benzothiazin-4(3H)-one 1,1-Dioxide
CAS:Prodotto controllato<p>Applications 2-Methyl-2H-1,2-benzothiazin-4(3H)-one 1,1-Dioxide is an intermediate used in the synthesis of Amido Methyl Meloxicam (A576790), which is an impurity of Meloxicam (M216100).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Lazer, E., et al.: J. Med. Chem., 40, 980 (1997),<br></p>Formula:C9H9NO3SColore e forma:NeatPeso molecolare:211.24Ibuprofen-13C6
CAS:<p>Applications Labelled Ibuprofen, a selective cyclooxygenase inhibitor (IC50=14.9uM). Inhibits PGH synthase-1 and PGH synthase-2 with comparable potency.<br>References Busson, M., et al.: J. Int. Med Res., 14, 53 (1986), Meade, E.A., et al.: J. Biol. Chem., 268, 6610 (1993), Davies, N.M., et al.: Clin. Pharmacokinet., 34, 101 (1998),<br></p>Formula:C713C6H18O2Colore e forma:NeatPeso molecolare:212.24Dehydro Indapamide-d3
CAS:Prodotto controllatoFormula:C16H11D3ClN3O3SColore e forma:NeatPeso molecolare:366.845-Desmethyl-6-methyl Glipizide
CAS:Prodotto controllato<p>Impurity Glipizide EP Impurity E<br>Applications 5-Desmethyl-6-methyl Glipizide (Glipizide EP Impurity E) is a Glipizide (G410225) impurity.<br>References Hoizey, G., et al.: Clin. Chem., 51, 1666 (2005), Singh, S., et al.: J. Pharm. Biomed. Anal., 41, 1037 (2006),<br></p>Formula:C21H27N5O4SColore e forma:NeatPeso molecolare:445.54Bumetanide 3-(Butyl(nitroso)amino) (1 mg/mL in Methanol)
CAS:Prodotto controllatoFormula:C17H19N3O6SColore e forma:ColourlessPeso molecolare:393.41Bumetanide 3-(Butyl(nitroso)amino)-d5
CAS:Prodotto controllatoFormula:C17D5H14N3O6SColore e forma:NeatPeso molecolare:398.445O-Methyl Piroxicam
CAS:Prodotto controllatoFormula:C16H15N3O4SColore e forma:NeatPeso molecolare:345.372-Methyl-4-(1-methylethoxy)-N-2-pyridinyl-2H-1,2-benzothiazine-3-carboxamide 1,1-Dioxide
CAS:Prodotto controllato<p>Applications 2-Methyl-4-(1-methylethoxy)-N-2-pyridinyl-2H-1,2-benzothiazine-3-carboxamide 1,1-Dioxide is an impurity of Piroxicam (P510000), a non-steroidal anti-inflammatory with long half-life.<br>References Carty, T.J., et al.: Prostaglandins, 47, 55 (1980); Brogden, R.N., et al.: Drugs, 22, 165 (1981); Mihalic, M., et al.: Anal. Profiles Drug Subs., 15, 509 (1986); Laneauville., O., et al.: J. Pharmacol. Exp. Ther., 271, 927 (1994)<br></p>Formula:C18H19N3O4SColore e forma:NeatPeso molecolare:373.43[2-[4-(Aminosulfonyl)phenyl]ethyl]carbamic Acid Ethyl Ester
CAS:Prodotto controllato<p>Impurity Glipizide EP Impurity F<br>Applications [2-[4-(Aminosulfonyl)phenyl]ethyl]carbamic Acid Ethyl Ester (Glipizide EP Impurity F) is a Glipizide (G410225) impurity.<br></p>Formula:C11H16N2O4SColore e forma:NeatPeso molecolare:272.323-[(4-Aminophenyl)sulfonyl]benzenamine
CAS:Prodotto controllato<p>Applications 3-[(4-Aminophenyl)sulfonyl]benzenamine is an impurity of Dapsone (D193250), an antibacterial used in the treatment of dermatitis herpetiformis.<br>References Francis, J., et al.: Br. J. Pharmacol., 5, 565 (1950); Uetrecht, J., et al.: Clin. Dermatol., 7, 111 (1989); Reszka, K., et al.: Chem. Res. Toxicol., 22, 1137 (2009); Santos, J., et al.: Bioorg. Med. Chem., 17, 3795 (2009);Varma, M., et al.: J. Med. Chem., 52, 4844 (2009)<br></p>Formula:C12H12N2O2SColore e forma:NeatPeso molecolare:248.301N-Acetylsulfathiazole-d4 (Major)
CAS:Prodotto controllato<p>Applications A deuterated metabolite of the drug Sulfathiazole.<br></p>Formula:C112H4H7N3O3S2Colore e forma:NeatPeso molecolare:301.38Glimepiride-d4 (phenylethyl-a,a,b,b-d4) (cis/trans)
CAS:Prodotto controllato<p>Applications Glimepiride-d4 (phenylethyl-a,a,b,b-d4) (cis/trans) is a useful isotopically labeled compound of Glimepiride (G410150)<br></p>Formula:C24H30D4N4O5SColore e forma:NeatPeso molecolare:244.2O-Desmethyl Indomethacin-d4
CAS:Prodotto controllato<p>Applications The major labelled metabolite of Indomethacin.<br>References Lewis, R., et al.: J. Clin. Invest., 53, 1607 (1974), Alvan, G., et al.: Clin. Pharmacol. Ther., 18, 364 (1975), Mungall, D., et al.: J. Pharm. Sci., 73, 1000 (1984), Baldwin, S., et al.: Xenobiotica, 25, 261 (1995),<br></p>Formula:C18H10D4ClNO4Colore e forma:NeatPeso molecolare:347.79Sulfamethoxazole-d4 β-D-Glucuronide
CAS:Prodotto controllato<p>Applications The main labelled metabolite of Sulfamethoxazole.<br>References Altenburger, R., et al.: Environ. Toxicol. Chem., 19, 2341 (2000), Pascoe, R., et al.: Anal. Chem., 73, 6014 (2001), Zhaohua, H., et al.: Eur. J. Med. Chem., 36, 863 (2001),<br></p>Formula:C16H15D4N3O9SColore e forma:NeatPeso molecolare:433.43Tiafenacil
CAS:<p>Applications Tiafenacil is a uracil herbicide used as a pesticide for the prevention and control of plants.<br>References Peng, X., et al. Faming Zhuanli Shenqing, 68pp Patent 2018 CODEN:CNXXEV<br></p>Formula:C19H18ClF4N3O5SColore e forma:Off White SolidPeso molecolare:511.87Indomethacin 1-Glycerin Ester
CAS:<p>Applications Indometacin 1-Glycerin Ester was synthesized and evaluated for anti-flammatory activity in the rate paw carrageenin edema essay.<br>References Paris, Gerard. , et al.: J. Med. Chem, 23, 9 (1980)<br></p>Formula:C22H22ClNO6Colore e forma:NeatPeso molecolare:431.87Metolazone
CAS:Prodotto controllato<p>Applications A diruetic. An antihypertensive.<br>References Curry, C.L., et al.: Clin. Ther., 9, 47 (1986), Kiyingi, A., et al.: Lancet, 335, 29 (1990)<br></p>Formula:C16H16ClN3O3SColore e forma:NeatPeso molecolare:365.83Sulfadiazine Silver Salt
CAS:Prodotto controllato<p>Applications Coordination compound. Antibacterial.<br>References Bohni, et al.: Chemotherapy, 14, 195 (1969), Carr, et al.: Antimicrob. Agents Chemother., 4, 585 (1973), Stober, H., et al.: Anal. Profiles Drug Subs., 11, 523 (1982),<br></p>Formula:C10H9N4O2S·AgColore e forma:NeatPeso molecolare:357.14Benzeneacetonitrile
CAS:Prodotto controllato<p>Applications Benzeneacetonitrile is a volatile compound released from apple trees infested with light brown apple moth larvae. It is also used in the synthesis of phenobarbital (P316760), methylphenidate (M325880), and other amphetamines.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Suckling, D. et al.: J. Agr. Food. Chem., 60, 9562 (2012); Cuevas-G. et al.: Int. J. Food. Sci. Technol., 47, 1378 (2012)<br></p>Formula:C8H7NColore e forma:NeatPeso molecolare:117.15(4R,6S)-5,6-Dihydro-6-methyl-4H-thieno[2,3-b]thiopyran-4-ol 7,7-Dioxide
CAS:Prodotto controllato<p>Applications (4R,6S)-4H-Thieno[2,3-b]thiopyran-4-ol, 5,6-dihydro-6-methyl-,7,7-dioxide is an analog of topically-active carbonic anhydrase inhibitor MK-507 also commonly known as Dorzolamide (D535100).<br>References Blacklock, T., et al.: J. Org. Chem., 58, 1672 (1993); Tempkin, O., et al.: Tetrahedron: Asym., 7, 2721 (1996)<br></p>Formula:C8H10O3S2Colore e forma:NeatPeso molecolare:218.29Sulfamethizole-d4
CAS:Prodotto controllato<p>Applications Isotope Labelled Sulfamethizole is a sulfonamide based antibiotic that exhibit bactericidal activities towards gram-negative bacteria. Sulfamehizole was shown to be effective in treating gram-negative Bacillus AmpC enzyme in elderly patients with lower respiratory tract infection and as well as against microbs responsible for tuberculosis.<br>References Mondelli, M., et al.: J. Molec. Struct., 1036, 180 (2013); Leelakrishnana, S., et al.: Adv. App. Sci. Res., 3, 3502 (2012); Ghoreishi, S.M., et al.: Anal. Lett., 46, 323 (2012);<br></p>Formula:C92H4H6N4O2S2Colore e forma:NeatPeso molecolare:274.36N-Nitroso Aceclofenac
Prodotto controllatoFormula:C16H12Cl2N2O5Colore e forma:NeatPeso molecolare:383.183N-Nitroso Furosemide-d5
Prodotto controllatoFormula:C12D5H5ClN3O6SColore e forma:NeatPeso molecolare:364.7738-Isopropyl Etodolac
CAS:Prodotto controllato<p>Impurity Etodolac EP Impurity D<br>Applications 8-Isopropyl Etodolac (Etodolac EP Impurity D) is an impurity in the synthesis of Etodolac (E933100), may have use in the treatment of myeloma. COX-1/COX-2/β-catenin inhibitors, or anti-inflammatory agent.<br>References Humber, L.G., et al.: Med. Res. Rev., 7, 1 (1987); Balfour, J.A, et al.: Drugs, 42, 274 (1991); Kato, et al.: J. Pharm. Pharmacol., 53 1679 (2001);<br></p>Formula:C18H23NO3Colore e forma:NeatPeso molecolare:301.38Benzoxazolemethanesulfonamide-N-(6-methyl-hexanoate)
CAS:Prodotto controllato<p>Applications Intermediate of Zonisamide-N-(6-hexanoic acid).<br></p>Formula:C15H20N2O5SColore e forma:NeatPeso molecolare:340.394-Hydroxy Triamterene Sulfate-d4, Sodium Salt
CAS:Prodotto controllato<p>Applications Isotope labelled 4-hydroxy triamterene sulfate sodium salt a metabolite of Triamterne, a diuretic agent.<br>References Vollmer, G., et al.: Arzneim.-Forsch., 31, 529 (1981), Gilfrich, H.J., et al.: Eur. J. Clin. Pharmacol., 25, 237 (1983),<br></p>Formula:C12H6D4N7NaO4SColore e forma:NeatPeso molecolare:375.333-Azabicyclo[3.3.0]octane Hydrochloride
CAS:Prodotto controllato<p>Applications 3-Azabicyclo[3.3.0]octane Hydrochloride is a reactant in the preparation of substituted pyrimidines derivatives as novel hedgehog signaling pathway inhibitors.<br>References Xin, M. et al.: Med. Chem. Res., 23, 3784 (2014); Xin, M. et al.: Bioorg. Med. Chem. Lett., 24, 983 (2014);<br></p>Formula:C7H13N·ClHColore e forma:White To Light YellowPeso molecolare:147.651-[1-(4-Chlorobenzoyl)-5-hydroxy-2-methyl-1H-indole-3-acetate]β-D-Glucopyranuronic Acid
CAS:Prodotto controllato<p>Stability Hygroscopic, Moisture Sensitive<br>Applications 1-[1-(4-Chlorobenzoyl)-5-hydroxy-2-methyl-1H-indole-3-acetate]β-D-Glucopyranuronic Acid is an analog of Indomethacin Acyl-β-D-glucuronide a metabolite of Indomethacin (I641000). Acyl glucuronides have been implicated in the toxicity of many xenobiotics and marketed drugs.<br>References Abid, A., et al.: Biochem. Pharmacol., 50, 557 (1995), Gamage, N., et al.: Toxicol. Sci., 90, 5 (2006), Cerveny, L., et al.: Drug Metab. Dispos., 35, 1032 (2007), Hayeshi, R., et al.: Eur. J. Pharm. Sci., 35, 383 (2008),<br></p>Formula:C24H22ClNO10Colore e forma:NeatPeso molecolare:519.894-Amino-4'-chlorodiphenyl Sulfone
CAS:Prodotto controllato<p>Applications 4-Amino-4'-chlorodiphenyl sulfone is a substituted 4-aminodiphenylsulfone as Escherichia coli dihydropteroate synthase inhibitor.<br>References Lopez de Compadre, R.L., et al.: J. Med. Chem., 31, 2315 (1988),<br></p>Formula:C12H10ClNO2SColore e forma:Off-White To Light YellowPeso molecolare:267.73rac-trans Dorzolamide Hydrochloride
CAS:Prodotto controllato<p>Applications rac-trans Dorzolamide is an impurity of Dorzolamide (D535100).<br>References Casini, A., et al.: Bioorg. Med. Chem. Lett., 13, 841 (2003), Clare, B., et al.: Bioorg. Med. Chem., 13, 2197 (2005),<br></p>Formula:C10H17ClN2O4S3Colore e forma:NeatPeso molecolare:360.9Dapsone N-β-D-Glucuronide Sodium Salt
CAS:Prodotto controllato<p>Stability Hygroscopic, unstable in solution<br>Applications Dapsone N-β-D-Glucuronide is the glucuronide conjugate and main urinary metabolite of the antibacterial Dapsone (D193250).<br>References Andoh, B.Y.A. et al.: Xenobiotica, 4, 571 (1974); Ogiya, S. et al.: Yakug. Zas., 81, 349 (1961);<br></p>Formula:C18H19N2NaO8SColore e forma:NeatPeso molecolare:446.41Indomethacin 1-Menthol ester
CAS:Prodotto controllato<p>Applications Indomethacin terpenoids' esters were synthesized and assessed both in vitro and in vivo as indomethacin dermal prodrugs.<br>References Bonina,, Francesco. , et al.: European Journal of Pharmaceutical Sciences, 14, 123 (2001),<br></p>Formula:C29H34ClNO4Colore e forma:NeatPeso molecolare:496.0385-Amino-3-(4-sulfonylphenyl)salicyclic Acid Sodium Salt
CAS:Prodotto controllato<p>Stability Hygroscopic<br>Applications 5-Amino-3-(4-sulfonylphenyl)salicyclic Acid Sodium Salt is an impurity of mesalamine (M258100), which is the active metabolite of Sulfasalazine (S699084). Anti-inflammatory (gastrointestinal).<br>References Friedman, G., et al.: Am. J. Gastroenterol., 81, 141 (1986); Tursi A., Expert Opin. Pharmacother., 6, 69 (2005);<br></p>Formula:C13H11NO6S•x(Na)Colore e forma:NeatPeso molecolare:309.29 + x(22.99)8-Propyl Etodolac
CAS:Prodotto controllato<p>Impurity Etodolac EP Impurity E<br>Applications 8-Propyl Etodolac (Etodolac EP Impurity E) is an impurity in the synthesis of Etodolac (E933100), may have use in the treatment of myeloma. COX-1/COX-2/β-catenin inhibitors.<br>References Humber, L.G., et al.: Med. Res. Rev., 7, 1 (1987); Balfour, J.A, et al.: Drugs, 42, 274 (1991); Kato, et al.: J. Pharm. Pharmacol., 53 1679 (2001);<br></p>Formula:C18H23NO3Colore e forma:NeatPeso molecolare:301.38trans-Carboxy Glimepiride-d5
CAS:Prodotto controllato<p>Applications An active labelled metabolite of Glimepiride (G410150).<br>References Groop, L., et al.: Diabetes Care, 15, 737 (1992), Muller, G., et al.: Diabetes, 42, 1852 (1993), Kramer, W., et al.: Biochem. Biophys. Acta, 119, 278 (1994),<br></p>Formula:C24H27D5N4O7SColore e forma:NeatPeso molecolare:525.63Gliclazide Impurity D
CAS:<p>Applications Gliclazide Impurity D is a manufacturing impurity of the drug Gliclazide (G409875) which is a sulfonylurea hypoglycemic agent and is used as an antidiabetic.<br>References Duhault, J., et al.: Arzneimittel-Forsch., 22, 1686 (1972), Holmes, B., et al.: Drugs, 27, 301 (1984),<br></p>Formula:C15H20N2O3SColore e forma:NeatPeso molecolare:308.3959Ethyl 4-[2-(5-Chloro-2-methoxybenzamido)ethyl]benzene Sulfonamide Carbamate
CAS:Prodotto controllatoFormula:C19H21ClN2O6SColore e forma:NeatPeso molecolare:440.90Methyl 5-Methoxy-2-methylindole-3-acetate
CAS:Prodotto controllato<p>Applications Intermediate in the preparation of Indomethacin<br>References Kalgutkar, A.S., et al.: Bioorg. Med. Chem., 13, 6810 (2005),<br></p>Formula:C13H15NO3Colore e forma:NeatPeso molecolare:233.26(S)-4-Hydroxy-2-(3-methoxypropyl)-3,4-dihydro-2H-thieno[3,2-e][1,2]thiazine-6-sulfonamide 1,1-Dioxide
CAS:Prodotto controllato<p>Applications (S)-4-Hydroxy-2-(3-methoxypropyl)-3,4-dihydro-2H-thieno[3,2-e][1,2]thiazine-6-sulfonamide 1,1-Dioxide has been used as a reactant for the preparation of Brinzolamide (AL-4862) [B677600], a topical carbonic anhydrase inhibitor.<br>References Conrow, R.E., et. al.: Org. Process Res. Dev., 3, 114 (1999)<br></p>Formula:C10H16N2O6S3Colore e forma:NeatPeso molecolare:356.44Hydroxy Gliclazide
CAS:Prodotto controllato<p>Applications The major hydroxylated metabolite of Gliclazide (G409875).<br>References Miyazaki, H., et al.: Eur. J. Drug Metab. Pharmacokinet., 8, 117 (1983), Rieutord, A., et al.: Xenobiotica, 25, 1345 (1995),<br></p>Formula:C15H21N3O4SColore e forma:NeatPeso molecolare:339.41Mefenamic Acyl-β-D-glucuronide
CAS:Prodotto controllato<p>Stability Hygroscopic<br>Applications Mefenamic acid metabolite.<br>References Besunder, J., et al.: Clin. Pharmacokinet., 14, 261 (1988), Smith, P., et al.: Drug Metab. Dipos., 18, 639 (1990), Kraus, D., et al.: Clin. Pharmacol. Ther., 54, 351 (1993), Sato, J., et al.: Biol. Pharm. Bull., 16, 811 (1993),<br></p>Formula:C21H23NO8Colore e forma:NeatPeso molecolare:417.412-Nitrophenyl Phenyl Sulfide
CAS:Prodotto controllato<p>Applications 2-Nitrophenyl Phenyl Sulfide is used in the study of non-nucleoside reverse transcriptase inhibitors of HIV-1.<br>References Chan, J., et al.: J. Med. Chem., 44, 1866 (2001); McMahon, J., et al.: Antimicro. Agents Chemother., 37, 754 (1993)<br></p>Formula:C12H9NO2SColore e forma:NeatPeso molecolare:231.273-Methoxy Acetaminophen-d3
CAS:Prodotto controllato<p>Applications 3-Methoxy Acetaminophen-d3 is deuterium labeled 3-Methoxy Acetaminophen (M226050). 3-Methoxy Acetaminophen is a metabolite of Acetaminophen (A161220), an analgesic and antipyretic agent used as a pain reliever to treat headache, muscle aches, and arthritis (1,2,3).<br>References (1) McGill, M. R. and Jaeschke, H. Pharm Res. 30, 2174 (2013)(2) Fairbrother, J.E., et al.: Anal. Profiles Drug Subs., 3, 1 (1974) (3) Hinson, J.A., et al.: Rev. Biochem. Toxicol., 2, 103 (1980)<br></p>Formula:C92H3H8NO3Colore e forma:NeatPeso molecolare:184.207bis(4-Nitrophenyl) Sulfone
CAS:Prodotto controllato<p>Applications BIS(4-NITROPHENYL) SULFONE (cas# 1156-50-9) is a useful research chemical.<br></p>Formula:C12H8N2O6SColore e forma:NeatPeso molecolare:308.26
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![1-[1-(4-Chlorobenzoyl)-5-hydroxy-2-methyl-1H-indole-3-acetate]β-D-Glucopyranuronic A…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FC429115.webp&w=3840&q=75)
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