Informazioni sul prodotto
Nome:Ticlopidine N-oxide
Sinonimi:
- 5-[(2-Chlorophenyl)methyl]-4,5,6,7-tetrahydrothieno[3,2-c]pyridine 5-oxide
Marchio:Biosynth
Descrizione:Ticlopidine N-oxide is a metabolite of ticlopidine, an anti-platelet drug. Ticlopidine N-oxide has been shown to be a competitive inhibitor of cytochrome P450 enzymes. The molecule is linear and the active site contains chlorophenyl groups that are oriented in a way that allows for the formation of the n-oxide form. X-ray crystallography studies have shown that ticlopidine N-oxide binds to the thiol group of cytochrome P450 enzymes, forming a covalent bond. This inhibits protein synthesis by preventing the transfer of electrons from NADH to cytochrome P450, which is required for metabolism. Ticlopidine N-oxide also forms dimers with other molecules, which may be responsible for its anti-inflammatory properties.
Avviso:I nostri prodotti sono destinati esclusivamente ad uso di laboratorio. Per qualsiasi altro utilizzo, vi preghiamo di contattarci.
Proprietà chimiche
Peso molecolare:279.79 g/mol
Formula:C14H14ClNOS
Purezza:Min. 95%