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CymitQuimica ha oltre 25 partner, tra i quali spicca il fornitore TargetMol

CymitQuimica ha oltre 25 partner, tra i quali spicca il fornitore TargetMol

We have reached an agreement with TargetMol: CymitQuimica clients will benefit for a 20% discount on all TargetMol products until the end of the year.On our website you can find the products offered by this partner, which has become one of the world's most recognised compound libraries and small molecule inhibitors supplier. TargetMol offers approximately 120 compound libraries and a wide range of chemical products and kits for life sciences.

Finisce il 31 dic( 8 giorni restanti )

prodotti per pagina.111930 prodotti in questa promozione.
  • Justicidin B

    CAS:
    Justicidin B: anticancer, proapoptotic, inhibits bone resorption & platelets, antiviral, fungicidal, antiprotozoal.
    Formula:C21H16O6
    Colore e forma:Solid
    Peso molecolare:364.35
  • D-threo-PDMP

    CAS:
    D-threo-PDMP inhibits glucoceramide synthase, cutting cell surface glycosphingolipids and hindering neurite growth.
    Formula:C23H38N2O3
    Colore e forma:Solid
    Peso molecolare:390.56
  • JNJ-49095397

    CAS:
    <p>JNJ-49095397 (RV568) is a p38 MAPK-α and p38 MAPK-γ kinase inhibitor for the study of respiratory syncytial virus infection.</p>
    Formula:C34H36N6O4
    Purezza:98.33% - 99.04%
    Colore e forma:Solid
    Peso molecolare:592.69
  • PKCiota-IN-1

    CAS:
    <p>PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).</p>
    Formula:C25H22FN5O
    Colore e forma:Solid
    Peso molecolare:427.47
  • FITM

    CAS:
    FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).
    Formula:C18H18FN5OS
    Purezza:97.25%
    Colore e forma:Solid
    Peso molecolare:371.43
  • Azaphilone-9

    CAS:
    <p>AZA-9 inhibits cancer growth by blocking HuR-ARE RNA binding; IC50=1.2μM.</p>
    Formula:C21H23BrO5
    Colore e forma:Solid
    Peso molecolare:435.31
  • TNKS1/2-IN-1

    CAS:
    <p>TNKS1/2-IN-1: potent inhibitor for cancer, fibrosis research; pIC50 7.1-8.2.</p>
    Formula:C26H23F4N3O4
    Colore e forma:Solid
    Peso molecolare:517.47
  • VEGFR-3-IN-1

    CAS:
    VEGFR-3-IN-1, a potent VEGFR3 inhibitor (IC50=110.4 nM), hinders tumor growth and VEGFR3 signaling, affecting HDLEC and MDA-MB cell proliferation/migration.
    Formula:C29H29ClF3N7OS
    Purezza:99.95%
    Colore e forma:Solid
    Peso molecolare:616.1
  • Naloxonazine

    CAS:
    <p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>
    Formula:C38H42N4O6
    Colore e forma:Solid
    Peso molecolare:650.76
  • IMD-vanillin

    CAS:
    IMD-vanillin is a novel compound characterized as an imidazoquinolinone-derived dimer with NF-κB immunomodulatory properties.
    Formula:C37H45N7O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:651.8
  • IMD-catechol

    CAS:
    IMD-catechol: an imidazoquinolinone-based dimer with NF-κB activity; improves CT26 cancer treatment, low toxicity.
    Formula:C31H34N6O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:538.64
  • CDK4/6-IN-15

    CAS:
    CDK4/6-IN-15: Oral, selective CDK4/6 inhibitor, halts cancer cell growth, G1 arrest, suppresses Rb phosphorylation.
    Formula:C21H27FN8S
    Colore e forma:Solid
    Peso molecolare:442.56
  • 18:0-22:6 DG

    CAS:
    1-Stearoyl-2-docosahexaenoyl-sn-glycerol (18:0-22:6 DG) is a diacylglycerol capable of binding to RasGRP and modulating the activation of MAP kinases.
    Formula:C43H72O5
    Colore e forma:Solid
    Peso molecolare:669.03
  • EC330

    CAS:
    EC330, a novel steroidal LIF inhibitor showed cytotoxicity in various cancer cell lines and NCI-60 cell line panel at low nano-molar range.
    Formula:C30H32F2O2
    Purezza:97.83%
    Colore e forma:Solid
    Peso molecolare:462.57
  • NCGC00138783


    NCGC00138783 blocks CD47/SIRPα interaction; IC50 of 50 µM.
    Formula:C30H28F7N7O5S
    Colore e forma:Solid
    Peso molecolare:731.64
  • TRK/ALK-IN-1


    TRK/ALK-IN-1: Potent dual TRK & ALK inhibitor; IC50s: 2.2nM (TRKA), 9.3nM (ALK WT), 38nM (ALK L1196M); cancer research potential.
    Formula:C31H35ClF2N8O2S
    Colore e forma:Solid
    Peso molecolare:657.18
  • Triphen diol

    CAS:
    Triphen diol, a phenol diol, fights pancreatic cancer & cholangiocarcinoma, inducing apoptosis via caspase-dependent & -independent paths.
    Formula:C22H20O4
    Colore e forma:Solid
    Peso molecolare:348.39
  • ChemR23-IN-3


    <p>ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.</p>
    Formula:C31H33N5O5S2
    Colore e forma:Solid
    Peso molecolare:619.75
  • Epothilone E

    CAS:
    <p>Epothilone E, a derivative of epothilone, functions by inhibiting microtubule protein activity, thereby halting cell division and exhibiting anti-tumor</p>
    Formula:C26H39NO7S
    Colore e forma:Solid
    Peso molecolare:509.66
  • Aramchol

    CAS:
    Aramchol (C20-FABAC), a mix of arachidic & cholic acid, lessens cholesterol crystallization & dissolves crystals in bile.
    Formula:C44H79NO5
    Purezza:≥95%
    Colore e forma:Solid
    Peso molecolare:702.1
  • eIF4A3-IN-17

    CAS:
    <p>eIF4A3-IN-17, a silvestrol analogue, disrupts eIF4F assembly; EC50: 0.9-15 nM. Used in cancer pathogenesis research.</p>
    Formula:C28H25NO7
    Colore e forma:Solid
    Peso molecolare:487.5
  • eIF4A3-IN-18

    CAS:
    eIF4A3-IN-18, a silvestrol analogue with EC50s: 0.8/35/2 nM, inhibits eIF4F complex and is cytotoxic (LC50: 0.06 nM) for cancer research.
    Formula:C29H28N2O6
    Colore e forma:Solid
    Peso molecolare:500.54
  • Palazestrant

    CAS:
    Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor.
    Formula:C28H36FN3O
    Purezza:97.55%
    Colore e forma:Solid
    Peso molecolare:449.6
  • G4/HDAC-IN-1


    <p>G4/HDAC-IN-1, a G4/HDAC dual inhibitor, IC50 1.1 µM, blocks TNBC growth, useful in cancer research.</p>
    Formula:C36H49ClFN7O4
    Colore e forma:Solid
    Peso molecolare:698.27
  • JBSNF-000028


    <p>JBSNF-000028: potent oral NNMT inhibitor; IC50s—human 0.033 μM, monkey 0.19 μM, mouse 0.21 μM; aids insulin sensitivity &amp; weight loss.</p>
    Formula:C11H13N3
    Purezza:99.23%
    Colore e forma:Solid
    Peso molecolare:187.24
  • hDHODH-IN-11

    CAS:
    hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.
    Formula:C24H23N3O3
    Colore e forma:Solid
    Peso molecolare:401.46
  • Miridesap

    CAS:
    <p>Miridesap (GSK2315698) rapidly depletes SAP in blood, cerebrospinal fluid, and amyloid deposits via liver clearance.</p>
    Formula:C16H24N2O6
    Purezza:≥95%
    Colore e forma:Solid
    Peso molecolare:340.37
  • 15-PGDH-IN-1

    CAS:
    15-PGDH-IN-1: potent oral 15-PGDH inhibitor, IC50=3nM, useful for tissue repair research.
    Formula:C24H22N4O2
    Colore e forma:Solid
    Peso molecolare:398.46
  • CDK4/6-IN-14

    CAS:
    CDK4/6-IN-14: potent CDK4/6 inhibitor, IC50s 10/16 nM, >60-fold selectivity over CDKs 1/2/7/9, selective across 205 kinases.
    Formula:C24H27ClFN7O
    Colore e forma:Solid
    Peso molecolare:483.97
  • Dynamin IN-1

    CAS:
    Dynamin IN-1 is a potent dynamin inhibitor with an IC 50 value of 1.0 µM .
    Formula:C23H24N2O
    Colore e forma:Solid
    Peso molecolare:344.45
  • Zidesamtinib

    CAS:
    <p>Zidesamtinib (NVL-520) is a ROS1 fusion and resistance mutation inhibitor that inhibits ROS1 and can be used to study non-small cell lung cancer.</p>
    Formula:C22H22FN7O
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:419.455
  • Fazamorexant

    CAS:
    Fazamorexant (YZJ-1139) is a powerful orexin receptor antagonist effective for insomnia research.
    Formula:C25H25FN4O2
    Colore e forma:Solid
    Peso molecolare:432.49
  • Gumelutamide

    CAS:
    Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.
    Formula:C22H21ClN6O
    Colore e forma:Solid
    Peso molecolare:420.89
  • Darizmetinib

    CAS:
    Darizmetinib (HRX215) is an MKK4 inhibitor.
    Formula:C21H17F2N5O3S
    Purezza:98.03% - 99.57%
    Colore e forma:Solid
    Peso molecolare:457.45
  • DRAK1/2-IN-1

    CAS:
    DRAK1/2-IN-1 is a potent inhibitor targeting both DRAK1 and DRAK2, displaying dissociation constants (Kd) of 1 µM and 6 µM, respectively.
    Formula:C22H24N2O3S
    Colore e forma:Solid
    Peso molecolare:396.5
  • BCR-ABL-IN-7

    CAS:
    BCR-ABL-IN-7 is an inhibitor of ABL kinase activity in WT and T315I mutants.BCR-ABL-IN-7 can be used in chronic myeloid leukemia (CML) research.
    Formula:C19H16FN3O3S
    Purezza:98.28%
    Colore e forma:Solid
    Peso molecolare:385.41
  • NUCC-0000323

    CAS:
    NUCC-0000323: potent SOD1 inhibitor, curbs expression, used in ALS research.
    Formula:C15H13BrN4S
    Colore e forma:Solid
    Peso molecolare:361.26
  • THZ2

    CAS:
    THZ2 (CDK7-IN-1), an analog of THZ1, is a potent and selective CDK7 inhibitor(IC50:13.9 nM),with the potential to treat Triple-negative breast cancer (TNBC).
    Formula:C31H28ClN7O2
    Purezza:98.28%
    Colore e forma:Solid
    Peso molecolare:566.05
  • Falcarindiol

    CAS:
    Falcarindiol is an orally active natural polyacetylene compound, anti-inflammatory and antiproliferative. inhibits NO production, suppressing iNOS expression.
    Formula:C17H24O2
    Purezza:99.38%
    Colore e forma:Solid
    Peso molecolare:260.37
  • Sycosterol A


    <p>Sycosterol A is an α-synuclein (α-syn) inhibitory sterol .</p>
    Formula:C27H48O9S
    Colore e forma:Solid
    Peso molecolare:548.73
  • Anserinone B

    CAS:
    Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).
    Formula:C11H14O4
    Colore e forma:Solid
    Peso molecolare:210.23
  • Dictyostatin

    CAS:
    Dictyostatin: potent microtubule stabilizer & anticancer agent with antiproliferative effects; researched for tauopathies.
    Formula:C32H52O6
    Colore e forma:Solid
    Peso molecolare:532.75
  • Inuviscolide

    CAS:
    Inuviscolide induces apoptosis, G2/M arrest in melanoma, and has anti-cancer, anti-inflammatory effects.
    Formula:C15H20O3
    Colore e forma:Solid
    Peso molecolare:248.32
  • ZINC00640089

    CAS:
    <p>ZINC00640089: Selective LCN2 inhibitor; curbs SUM149 cell growth and AKT activity; useful for IBC research.</p>
    Formula:C20H13F3N2O2
    Purezza:98.41% - 99.80%
    Colore e forma:Solid
    Peso molecolare:370.32
  • Actinoquinol

    CAS:
    Actinoquinol, a compound effective in absorbing UVB radiation, plays a crucial role in protecting the human eye from photooxidative and other oxidative
    Formula:C11H11NO4S
    Colore e forma:Solid
    Peso molecolare:253.27
  • KG-501

    CAS:
    KG-501 (Naphthol AS-E phosphate) is a cAMP response element-binding protein (CREB) inhibitor(IC50 : 6.89 μM).
    Formula:C17H13ClNO5P
    Purezza:97.81%
    Colore e forma:Solid
    Peso molecolare:377.72
  • Rosolic Acid

    CAS:
    Rosolic Acid activates Nrf2, boosts angiogenesis, reduces inflammation, deters apoptosis, aids pancreatic cells, and shields ECs from stress.
    Formula:C19H14O3
    Colore e forma:Solid
    Peso molecolare:290.31
  • (S)-JDQ-443

    CAS:
    <p>(S)-JDQ-443, an isomer of JDQ-443, is a selective, potent oral KRAS G12C inhibitor with antitumor properties.</p>
    Formula:C29H28ClN7O
    Colore e forma:Solid
    Peso molecolare:526.03
  • Octotiamine

    CAS:
    Octotiamine (TATD), a Vitamin B1 analogue and component of the vitamin complex, is utilized in research related to Vitamin B1 deficiency.
    Formula:C23H36N4O5S3
    Colore e forma:Solid
    Peso molecolare:544.75
  • Aflibercept

    CAS:
    <p>Aflibercept has a wide range of applications in life science related research.</p>
    Colore e forma:Liquid
  • TGFβRI-IN-6

    CAS:
    <p>TGFβRI-IN-6 is a potent TGFβRI inhibitor with an IC50 value of 0.55 nM.TGFβRI-IN-6 has the potential to enhance anti-tumour immunity.</p>
    Formula:C17H10F4N6
    Colore e forma:Solid
    Peso molecolare:374.3
  • Cyprodenate

    CAS:
    Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.
    Formula:C13H25NO2
    Colore e forma:Solid
    Peso molecolare:227.34
  • c-Met-IN-16

    CAS:
    c-Met-IN-16 is a c-Met inhibitor that can be used for cancer research .
    Formula:C21H17F2N9O
    Colore e forma:Solid
    Peso molecolare:449.42
  • LEM-14-1189

    CAS:
    <p>LEM-14-1189 inhibits NSD1/2/3 (IC50: 418/111/60 μM), targets nuclear receptors, and may treat cancer and blood diseases.</p>
    Formula:C35H34N6O5S2
    Purezza:98.06%
    Colore e forma:Solid
    Peso molecolare:682.81
  • FT011

    CAS:
    <p>FT011, a direct anti-fibrotic agent,attenuates cardiac remodelling and dysfunction in experimental diabetic cardiomyopathy.</p>
    Formula:C20H17NO5
    Purezza:98.98%
    Colore e forma:Solid
    Peso molecolare:351.35
  • DPNB-ABT594


    DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.
    Formula:C31H46ClN3O11
    Colore e forma:Solid
    Peso molecolare:672.16
  • eeAChE-IN-2

    CAS:
    eeAChE-IN-2 is a potent inhibitor of eeAChE, exhibiting inhibitory potency with an IC50 of 2 nM.
    Formula:C37H40N8O5S
    Colore e forma:Solid
    Peso molecolare:708.83
  • (Rac)-SHIN2

    CAS:
    (Rac)-SHIN2 is a serine hydroxymethyltransferase (SHMT) inhibitor for the study of T-cell acute lymphoblastic leukemia (T-ALL).
    Formula:C23H26N4O3
    Purezza:98.165% - 99.48%
    Colore e forma:Solid
    Peso molecolare:406.48
  • Masofaniten

    CAS:
    Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the study of prostate and breast cancer.
    Formula:C24H24Cl2N4O4S
    Purezza:98.42% - 98.66%
    Colore e forma:Solid
    Peso molecolare:535.44
  • IMD-ferulic


    <p>IMD-ferulic, a compound that forms covalent bonds, acts as an NF-κB modulator, enhancing the adjuvanticity of small molecule immune potentiators.</p>
    Formula:C36H41N7O4
    Colore e forma:Solid
    Peso molecolare:635.76
  • photoCORM-1


    photoCORM-1: a CORM with real-time CO monitoring via color change, exhibits cellular uptake and anti-tumor activity.
    Formula:C33H32Cl2N2O6
    Colore e forma:Solid
    Peso molecolare:623.52
  • photoCORM-2

    CAS:
    photoCORM-2 releases CO, changes color for real-time monitoring, has good cellular uptake, and anti-tumor properties.
    Formula:C17H13NO3
    Colore e forma:Solid
    Peso molecolare:279.29
  • hGGPPS-IN-3

    CAS:
    13h (hGGPPS-IN-3), a strong C2-ThP-BPs hGGPPS blocker, triggers MM cell apoptosis and shows in vivo anti-myeloma effects.
    Formula:C21H19BrN4O7P2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:613.31
  • β-Estradiol 17-acetate

    CAS:
    <p>β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) is a metabolite of estradiol.</p>
    Formula:C20H26O3
    Purezza:98.11% - 99.88%
    Colore e forma:Solid
    Peso molecolare:314.42
  • BAY 1214784

    CAS:
    <p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>
    Formula:C29H26ClF4N3O5S2
    Colore e forma:Solid
    Peso molecolare:672.11
  • Bis-Pro-5FU

    CAS:
    Bis-Pro-5FU enhances oral uptake and safety of 5-FU, an anti-cancer drug for colorectal and pancreatic tumors.
    Formula:C10H7FN2O2
    Colore e forma:Solid
    Peso molecolare:206.17
  • Hsp90-IN-17

    CAS:
    Hsp90-IN-17 (Example 5) is an inhibitor of HSP90, applicable in researching proliferative diseases, including cancer and neurodegenerative conditions.
    Formula:C21H20N4O7
    Colore e forma:Solid
    Peso molecolare:440.41
  • HIF-2α-IN-7

    CAS:
    HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.
    Formula:C18H9F6NO2
    Colore e forma:Solid
    Peso molecolare:385.26
  • L-Afegostat

    CAS:
    <p>L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.</p>
    Formula:C6H13NO3
    Colore e forma:Solid
    Peso molecolare:147.17
  • PF-06455943

    CAS:
    PF-06455943: LRRK2 inhibitor, IC50=3nM, PET radioligand, used for ADME/neuro PK & Parkinson's research.
    Formula:C17H14FN5O
    Colore e forma:Solid
    Peso molecolare:323.32
  • GDC-0575

    CAS:
    <p>GDC-0575 (ARRY-575) is a highly-selective oral small-molecule Chk1 inhibitor(IC50 of 1.2 nM).</p>
    Formula:C16H20BrN5O
    Purezza:≥95%
    Colore e forma:Solid
    Peso molecolare:378.27
  • SIRT2-IN-11

    CAS:
    SIRT2-IN-11 (AEM1), a SIRT2 inhibitor (IC50 18.5μM), induces apoptosis and affects p53, used in cancer research.
    Formula:C21H22N2O
    Colore e forma:Solid
    Peso molecolare:318.41
  • eIF4A3-IN-9

    CAS:
    eIF4A3-IN-9, a silvestrol analogue, disrupts eIF4F complex assembly; EC50s: 29/450/80 nM (myc/tub-LUC, MB-231 cells); for cancer research.
    Formula:C28H27NO8
    Colore e forma:Solid
    Peso molecolare:505.52
  • METTL3-IN-1

    CAS:
    <p>METTL3-IN-1 is a polyheterocyclic compound, acts as METTL3 inhibitor .</p>
    Formula:C25H24FN5O2
    Colore e forma:Solid
    Peso molecolare:445.49
  • METTL3-IN-2

    CAS:
    METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.
    Formula:C25H26N8O
    Colore e forma:Solid
    Peso molecolare:454.53
  • METTL3-IN-3

    CAS:
    METTL3-IN-3 is a polyheterocyclic compound, acts as METTL3 inhibitor .
    Formula:C26H28BrFN6O2
    Colore e forma:Solid
    Peso molecolare:555.44
  • PF-07054894

    CAS:
    PF-07054894: potent CCR6 antagonist, targets GPCR, for inflammatory bowel disease research.
    Formula:C24H30N6O4
    Colore e forma:Solid
    Peso molecolare:466.53
  • cis-ccc_R08

    CAS:
    cis-ccc_R08 infection . cis-ccc_R08 is a cccDNA (covalently closed circular DNA) inhibitor .
    Formula:C22H19ClO6
    Colore e forma:Solid
    Peso molecolare:414.84
  • PARP10-IN-2

    CAS:
    <p>PARP10-IN-2 is a potent inhibitor of PARP10, a mono-ADP-ribosyltransferase, with an IC50 value of 3.64 μM for human PARP10.PARP10-IN-2 also inhibited PARP2 and</p>
    Formula:C14H10N2O2
    Purezza:99.27%
    Colore e forma:Solid
    Peso molecolare:238.24
  • PCSK9-IN-13

    CAS:
    PCSK9-IN-13 is a potent inhibitor of PCSK9, effectively preventing the binding of PCSK9 to low-density lipoprotein (LDL) receptors through its mechanism of
    Formula:C30H33N5O2
    Colore e forma:Solid
    Peso molecolare:495.62
  • Vemtoberant

    CAS:
    Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.
    Formula:C29H37N3O8S2
    Colore e forma:Solid
    Peso molecolare:619.75
  • BDP5290

    CAS:
    BDP5290 is a potent inhibitor of both ROCK and MRCK(IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively.)
    Formula:C17H18ClN7O
    Purezza:97.22%
    Colore e forma:Solid
    Peso molecolare:371.82
  • HSP90-IN-20

    CAS:
    HSP90-IN-20, a potent inhibitor of HSP90, exhibits an IC50 of ≤10 μM, indicating its potential application in cancer research.
    Formula:C26H32N4O4
    Colore e forma:Solid
    Peso molecolare:464.56
  • NLRP3-IN-14

    CAS:
    NLRP3-IN-14, potent selective NLRP3 inhibitor, KD 5.87μM; IC50 0.131μM for IL-1β; for inflammation research.
    Formula:C27H28N2O4
    Colore e forma:Solid
    Peso molecolare:444.52
  • NLRP3-IN-15

    CAS:
    NLRP3-IN-15: potent, selective NLRP3 inflammasome inhibitor; IC50 0.114 μM for IL-1β; for inflammation research.
    Formula:C22H19NO4
    Colore e forma:Solid
    Peso molecolare:361.39
  • NLRP3-IN-16

    CAS:
    NLRP3-IN-16: potent NLRP3 inflammasome inhibitor; IC50=0.065μM; curbs IL-1β; used in inflammation studies.
    Formula:C25H25NO5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:419.47
  • THRX-144644

    CAS:
    THRX-144644: lung-specific ALK5 inhibitor, 0.14 nM IC50, no systemic TGFβ toxicity.
    Formula:C26H28ClF2N7
    Colore e forma:Solid
    Peso molecolare:512
  • ONO-0740556

    CAS:
    ONO-0740556 is a potent agonist of the Gi-coupled human lysophosphatidic acid receptor 1 (LPA1), exhibiting an EC50 value of 0.26 nM.
    Formula:C20H34NO6P
    Colore e forma:Solid
    Peso molecolare:415.46
  • NLRP3-IN-13

    CAS:
    <p>NLRP3-IN-13 is an NLRP3 inhibitor that inhibits NLRP3-associated inflammation.NLRP3-IN-13 can be used in the study of neurological disorders and inflammation.</p>
    Formula:C19H15N3O3S
    Purezza:99.16%
    Colore e forma:Solid
    Peso molecolare:365.41
  • MALT1-IN-11

    CAS:
    <p>MALT1-IN-11: MALT1 inhibitor, IC50 &lt;10-100 nM, reduces IL10, for cancer/autoimmune research.</p>
    Formula:C20H16F4N8O
    Colore e forma:Solid
    Peso molecolare:460.39
  • CU-CPT9b

    CAS:
    <p>CU-CPT9b (TLR8-specific antagonist 1) is an antagonist of toll-like receptor 8 (TLR8; Kd = 21 nM).</p>
    Formula:C16H13NO2
    Purezza:98.1%
    Colore e forma:Solid
    Peso molecolare:251.28
  • c-Met-IN-14

    CAS:
    c-Met-IN-14: selective c-Met kinase inhibitor, IC50 2.89 nM, anticancer, stops G2/M phase, induces A549 cell apoptosis.
    Formula:C34H38ClFN4O7S
    Colore e forma:Solid
    Peso molecolare:701.2
  • PARP1-IN-12


    PARP1-IN-12: potent PARP1 inhibitor, IC50 2.99 nM, triggers cell apoptosis, G2/M arrest, induces DSBs in BRCA-deficient cells.
    Formula:C43H56FN5O5
    Colore e forma:Solid
    Peso molecolare:741.93
  • PARP7-IN-12

    CAS:
    PARP7-IN-12, a potent inhibitor targeting PARP7, exhibits an IC50 of 7.836 nM. This compound is applicable in cancer research.
    Formula:C23H27ClF3N5O5
    Colore e forma:Solid
    Peso molecolare:545.94
  • PARP-2-IN-3

    CAS:
    <p>PARP-2-IN-3 is used in the study of breast cancer as a PARP-2 inhibitor with antitumor activity that induces apoptosis (apoptosis) and necrosis in cancer cells.</p>
    Formula:C20H20ClN3O3
    Purezza:99.33%
    Colore e forma:Solid
    Peso molecolare:385.84
  • hCAIX-IN-16

    CAS:
    hCAIX-IN-16 (Compound 12d), an inhibitor of hCA IX, exhibits inhibition constants (K i) of 190.0 nM for hCA IX and 187.9 nM for hCA XII.
    Formula:C20H20N8O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:436.49
  • hCAIX-IN-15

    CAS:
    hCAIX-IN-15 is a potent inhibitor of human carbonic anhydrase IX (hCA IX) with an inhibition constant (Ki) of 38.8 nM, exhibiting broad-spectrum anticancer
    Formula:C18H14FN7O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:411.41
  • LIXIVAPTAN

    CAS:
    Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
    Formula:C27H21ClFN3O2
    Purezza:98.36%
    Colore e forma:Solid
    Peso molecolare:473.93
  • hCAIX-IN-14

    CAS:
    hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .
    Formula:C11H17ClN6O2S
    Colore e forma:Solid
    Peso molecolare:332.81
  • HDAC6-IN-14


    HDAC6-IN-14, an inhibitor of HDAC6 (HDAC), exhibits high selectivity with an IC50 value of 42 nM, demonstrating over 100-fold selectivity compared to HDAC1,
    Formula:C24H30FN3O4
    Colore e forma:Solid
    Peso molecolare:443.51