(-)-(2R,5S)-1-Allyl-2,5-dimethylpiperazine

CAS: 155836-78-5

Ref. 3D-FA17303

Product Information

• Name: (-)-(2R,5S)-1-Allyl-2,5-dimethylpiperazine
• Synonyms: (2R,5S)-2,5-Dimethyl-1-(2-propen-1-yl)piperazine(2R-trans)-2,5-Dimethyl-1-(2-propenyl)piperazine, (2R,5S)-1-Allyl-2,5-dimethylpiperazine, (2R,5S)-2,5-Dimethyl-1-(2-propen-1-yl)piperazine, (2R,5S)-2,5-Dimethyl-1-Prop-2-En-1-Ylpiperazine, Piperazine, 2,5-dimethyl-1-(2-propen-1-yl)-, (2R,5S)-, Piperazine, 2,5-dimethyl-1-(2-propenyl)-, (2R,5S)-, Piperazine, 2,5-dimethyl-1-(2-propenyl)-, (2R-trans)-

Description

(-)-(2R,5S)-1-Allyl-2,5-dimethylpiperazine is a novel analog of benzyl alcohols that binds to the delta opioid receptor. The compound was found to be an agonist in vitro and in vivo. It showed no affinity for other opioid receptors or for the benzodiazepine receptor. (-)-(2R,5S)-1-Allyl-2,5-dimethylpiperazine was found to have high affinity for the human cloned delta opioid receptor with a Ki value of 0.6 nM. This compound is also a potent alkylate inhibitor with an IC50 of 6 microM against ethoxy radical formation and an IC50 of 25 microM against lipid peroxidation induced by H2O2.

• Brand: Biosynth

Chemical properties

• Molecular weight: 154.25 g/mol
• Formula: C₉H₁₈N₂
• Purity: Min. 95%