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Apoptose

Apoptose

Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.

Subcategorias de "Apoptose"

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Foram encontrados 5592 produtos de "Apoptose"

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  • Tauroursodeoxycholate

    CAS:
    <p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>
    Fórmula:C26H45NO6S
    Pureza:98.77% - 99.93%
    Cor e Forma:White Solid
    Peso molecular:499.7
  • PEAQX

    CAS:
    <p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>
    Fórmula:C17H17BrN3O5P
    Pureza:98% - 99.9%
    Cor e Forma:Solid
    Peso molecular:454.21
  • AR42

    CAS:
    <p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>
    Fórmula:C18H20N2O3
    Pureza:98.46% - 98.96%
    Cor e Forma:Solid
    Peso molecular:312.36
  • Emricasan

    CAS:
    <p>Emricasan (IDN-6556) is a pan-caspase inhibitor with irreversible properties.</p>
    Fórmula:C26H27F4N3O7
    Pureza:98.13% - 99%
    Cor e Forma:Solid
    Peso molecular:569.5
  • Aloperine

    CAS:
    <p>Aloperine exhibits anti-inflammatory, antibacterial, antiviral, and anti-tumor properties.</p>
    Fórmula:C15H24N2
    Pureza:98% - 99.88%
    Cor e Forma:Yellow Crystalline Powder
    Peso molecular:232.36
  • 1400W dihydrochloride

    CAS:
    <p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>
    Fórmula:C10H17Cl2N3
    Pureza:98% - 99.94%
    Cor e Forma:Solid
    Peso molecular:250.17
  • Bilobalide

    CAS:
    <p>Bilobalide ((-)-Bilobalide), a bioactive from Gingko Biloba, is active on hypoxia-induced alterations.</p>
    Fórmula:C15H18O8
    Pureza:98.81% - 99.92%
    Cor e Forma:White Solid
    Peso molecular:326.3
  • Ipatasertib

    CAS:
    <p>Ipatasertib (GDC-0068) is a selective, ATP-competitive pan-Akt inhibitor that can lead to p53-independent PUMA activation.Cost-effective and quality-assured.</p>
    Fórmula:C24H32ClN5O2
    Pureza:98.28% - 99.21%
    Cor e Forma:Solid
    Peso molecular:458
  • Sulforaphane

    CAS:
    <p>Sulforaphane is a natural isothiocyanate that activates Nrf2. Sulforaphane has antitumor and anti-inflammatory activities. Cost-effective and quality-assured.</p>
    Fórmula:C6H11NOS2
    Pureza:95% - 99.79%
    Cor e Forma:Light Yellow Liquid
    Peso molecular:177.29
  • Nω-Hydroxy-nor-L-Arginine Dihydrochloride

    CAS:
    <p>Nω-Hydroxy-nor-L-Arginine Dihydrochloride is a competitive and reversible inhibitor of arginase</p>
    Fórmula:C5H14Cl2N4O3
    Pureza:99.12% - 99.84%
    Cor e Forma:Solid
    Peso molecular:249.10
  • ZZW-115 hydrochloride

    CAS:
    <p>ZZW-115 hydrochloride inhibits the activity of NUPR1.</p>
    Fórmula:C24H34Cl3F3N4S
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:573.97
  • Chromium picolinate

    CAS:
    <p>Chromium picolinate causes DNA damage and mutation. It is an activator of p38.</p>
    Fórmula:C18H12CrN3O6
    Pureza:99.64%
    Cor e Forma:Violet-Red Crystalline Powder
    Peso molecular:418.30
  • Thalidomide-NH-PEG1-NH2 hydrochloride

    CAS:
    <p>Thalidomide-NH-PEG1-NH2 hydrochloride (4-[(2-(2-Aminoethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione HCl) is a synthetic E3 ligase ligand-</p>
    Fórmula:C17H21ClN4O5
    Pureza:97.13%
    Cor e Forma:Solid
    Peso molecular:396.83
  • Trolox

    CAS:
    <p>Trolox is a vitamin E analogue, used in reducing oxidative stress or damage.</p>
    Fórmula:C14H18O4
    Pureza:98.90% - 99.90%
    Cor e Forma:White To Fainly Beige Crystalline Powder
    Peso molecular:250.29
  • Thalidomide-NH-CH2-COOH

    CAS:
    <p>Thalidomide-NH-CH2-COOH ((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)glycine) is a synthesized E3 ligase ligand-linker conjugate containing a</p>
    Fórmula:C15H13N3O6
    Pureza:96.3800%
    Cor e Forma:Solid
    Peso molecular:331.28
  • Tetrahydroxyquinone monohydrate

    CAS:
    <p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>
    Fórmula:C6H6O7
    Cor e Forma:Solid
    Peso molecular:190.11
  • Apocynin

    CAS:
    <p>Apocynin (NSC 2146) is a specific NADPH-oxidase inhibitor (IC50: 10 μM).</p>
    Fórmula:C9H10O3
    Pureza:99.71% - 99.98%
    Cor e Forma:Yellowish To Brown Powder
    Peso molecular:166.17
  • Alda-1

    CAS:
    <p>Alda-1 activates ALDH2*1 and ALDH2*2, permeates cells, and targets mitochondrial aldehyde dehydrogenase 2.</p>
    Fórmula:C15H11Cl2NO3
    Pureza:98.5% - 99.63%
    Cor e Forma:Solid
    Peso molecular:324.16
  • Metamizole magnesium

    CAS:
    <p>Metamizole magnesium (Metamizolemagnesiumsalt) is a pain reliever, which can antispasmodic.</p>
    Fórmula:C26H32MgN6O8S2
    Pureza:93.51%
    Cor e Forma:Solid
    Peso molecular:645.01
  • ARRY 520 hydrochloride

    CAS:
    <p>'ARRY 520 hydrochloride: a KSP inhibitor causing apoptosis and strong anti-proliferative effects.'</p>
    Fórmula:C20H23ClF2N4O2S
    Pureza:98.06% - 99.62%
    Cor e Forma:Solid
    Peso molecular:456.94
  • Eltrombopag Olamine

    CAS:
    <p>Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin</p>
    Fórmula:C29H36N6O6
    Pureza:99.59% - 99.89%
    Cor e Forma:Solid
    Peso molecular:564.63
  • HA15

    CAS:
    <p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>
    Fórmula:C23H22N4O3S2
    Pureza:99.77% - 99.86%
    Cor e Forma:Solid
    Peso molecular:466.58
  • ISRIB (trans-isomer)

    CAS:
    <p>ISRIB (trans-isomer) is a potent inhibitor of PERK that rescues protein translation and prevents SG formation in the presence of P-eIF2α. Cost effective and quality assured.</p>
    Fórmula:C22H24Cl2N2O4
    Pureza:97.86% - 99.27%
    Cor e Forma:Solid
    Peso molecular:451.34
  • Thalidomide 4-fluoride

    CAS:
    <p>Thalidomide 4-fluoride (E3 ligase Ligand 4) (Cereblon ligand 4) is the Thalidomide-based Cereblon ligand.</p>
    Fórmula:C13H9FN2O4
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:276.22
  • Thalidomide-O-amido-C6-NH2 hydrochloride

    CAS:
    <p>Thalidomide-O-amido-C6-NH2 HCl, a cereblon ligand-linker for PROTAC synthesis.</p>
    Fórmula:C21H27ClN4O6
    Pureza:97.33%
    Cor e Forma:Solid
    Peso molecular:466.915
  • CA-4948

    CAS:
    <p>CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity.</p>
    Fórmula:C24H25N7O5
    Pureza:99.35% - 99.88%
    Cor e Forma:Solid
    Peso molecular:491.5
  • Tenovin-6

    CAS:
    <p>Tenovin-6 is a p53 transcriptional activity agonist.</p>
    Fórmula:C25H34N4O2S
    Pureza:97.71% - >99.99%
    Cor e Forma:Solid
    Peso molecular:454.63
  • Dacarbazine citrate

    CAS:
    <p>Dacarbazine citrate treats lymphatic cancers, malignant melanoma, islet cell carcinoma, and soft tissue sarcoma.</p>
    Fórmula:C12H18N6O8
    Cor e Forma:Solid
    Peso molecular:374.31
  • FOXO4-DRI acetate


    <p>FOXO4-DRI acetate is a bioactive chemical.</p>
    Fórmula:C36H64N14O14S
    Pureza:99.10%
    Cor e Forma:Solid
    Peso molecular:5358.06
  • Periplocin

    CAS:
    <p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>
    Fórmula:C36H56O13
    Pureza:99.66% - 99.74%
    Cor e Forma:Solid
    Peso molecular:696.82
  • TrxR1-IN-B19

    CAS:
    <p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>
    Fórmula:C21H22O5
    Pureza:98.6%
    Cor e Forma:Solid
    Peso molecular:354.4
  • Thalidomide-O-amido-C3-NH2 TFA

    CAS:
    <p>Thalidomide-based E3 ligase linker for PROTAC tech; cereblon ligand conjugate.</p>
    Fórmula:C20H21F3N4O8
    Pureza:98.47%
    Cor e Forma:Solid
    Peso molecular:502.4
  • Thalidomide-O-COOH

    CAS:
    <p>Thalidomide-O-COOH is a Cereblon ligand for CRBN protein recruitment and PROTAC construction with a linker.</p>
    Fórmula:C15H12N2O7
    Pureza:98% - 98.29%
    Cor e Forma:Solid
    Peso molecular:332.27
  • Methoxychlor

    CAS:
    <p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>
    Fórmula:C16H15Cl3O2
    Pureza:98.82% - ≥95%
    Cor e Forma:Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment If
    Peso molecular:345.65
  • Liproxstatin-1 hydrochloride

    CAS:
    <p>Liproxstatin-1 hydrochloride is a high-potency ferroptosis inhibitor capable of effectively preventing ferroptotic cell death, with an IC50 value of 22 nM [1].</p>
    Fórmula:C19H22Cl2N4
    Cor e Forma:Solid
    Peso molecular:377.31
  • GSK778 hydrochloride

    CAS:
    <p>GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to 143 nM, effective in cancer models.</p>
    Fórmula:C30H34ClN5O3
    Pureza:97.26% - 98.35%
    Cor e Forma:Solid
    Peso molecular:548.08
  • Thalidomide-4-OH

    CAS:
    <p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>
    Fórmula:C13H10N2O5
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:274.23
  • Thalidomide-NH-C4-NH-Boc

    CAS:
    <p>Thalidomide-NH-C4-NH-Boc is a cereblon-based E3 ligase ligand-linker for PROTACs.</p>
    Fórmula:C22H28N4O6
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:444.48
  • Difurazon hydrochloride

    CAS:
    <p>Difurazon HCl: a mutagenic antibacterial and growth promoter, used for bacillary dysentery in feed.</p>
    Fórmula:C14H13ClN6O6
    Pureza:98.51%
    Cor e Forma:Solid
    Peso molecular:396.74
  • Methoxyamine HCl

    CAS:
    <p>Methoxyamine HCl targets DNA repair sites, potentially increasing DNA breaks and enhancing alkylating agents' anti-cancer effects.</p>
    Fórmula:CH6ClNO
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:83.51
  • Alogliptin Benzoate

    CAS:
    <p>Alogliptin Benzoate, a potent DPP-4 inhibitor with &gt;10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>
    Fórmula:C25H27N5O4
    Pureza:99.94% - >99.99%
    Cor e Forma:White Powder
    Peso molecular:461.51
  • OICR-9429

    CAS:
    <p>OICR-9429 blocks WDR5 binding to MLL/Histone 3, hindering acute myeloid leukemia cell growth in vitro.</p>
    Fórmula:C29H32F3N5O3
    Pureza:97.07% - 99.93%
    Cor e Forma:Solid
    Peso molecular:555.59
  • Thalidomide-O-amido-PEG3-C2-NH2 TFA

    CAS:
    <p>Synthetic E3 ligase ligand-linker, Thalidomide-O-amido-PEG3-C2-NH2 TFA, used in PROTAC with cereblon ligand and PEG.</p>
    Fórmula:C25H31F3N4O11
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:620.54
  • Bigelovin

    CAS:
    <p>Bigelovin: RXRα agonist, inhibits mTOR via ROS, induces apoptosis/autophagy, anti-tumor sesquiterpene from Inula sp.</p>
    Fórmula:C17H20O5
    Pureza:99.61% - 99.72%
    Cor e Forma:Solid
    Peso molecular:304.34
  • KRCA-0008

    CAS:
    <p>KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability.</p>
    Fórmula:C30H37ClN8O4
    Pureza:96.19%
    Cor e Forma:Solid
    Peso molecular:609.12
  • Perhexiline

    CAS:
    <p>Perhexiline: oral CPT1/2 inhibitor, limits fat metabolism, crosses BBB, anti-cancer, induces liver cell apoptosis, for cancer/cardio research.</p>
    Fórmula:C19H35N
    Cor e Forma:Solid
    Peso molecular:277.49
  • Ketorolac hemicalcium

    CAS:
    <p>Ketorolac hemicalcium: NSAID, COX-1/COX-2 inhibitor (IC50: 20/120 nM), treats eye inflammation &amp; pain, used in cancer research.</p>
    Fórmula:C30H24CaN2O6
    Cor e Forma:Solid
    Peso molecular:548.608
  • Thalidomide-propargyl

    CAS:
    <p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>
    Fórmula:C16H12N2O5
    Pureza:95.14%
    Cor e Forma:Solid
    Peso molecular:312.28
  • Thalidomide-NH-C6-NH2 hydrochloride

    CAS:
    <p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>
    Fórmula:C19H25ClN4O4
    Pureza:99.27%
    Cor e Forma:Solid
    Peso molecular:408.88
  • Britannin

    CAS:
    <p>Britannin, a sesquiterpene lactone, inhibits proliferation and induces apoptosis through the mitochondrial signaling pathway in human breast cancer cells.</p>
    Fórmula:C19H26O7
    Pureza:98% - 99.98%
    Cor e Forma:Solid
    Peso molecular:366.41
  • Verteporfin

    CAS:
    <p>Verteporfin (BPD-MA) is a YAP inhibitor that inhibits YAP-TEAD interactions.</p>
    Fórmula:C41H42N4O8
    Pureza:95.37% - 99.82%
    Cor e Forma:Dark Green To Black Solid
    Peso molecular:718.79
  • Sulfaphenazole

    CAS:
    <p>Sulfaphenazole (Plisulfan) is an inhibitor of CYP2C9 (Ki: 0.3 μM) that demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki: 63/29 μM for</p>
    Fórmula:C15H14N4O2S
    Pureza:97.53% - 99.67%
    Cor e Forma:Solid
    Peso molecular:314.36
  • PK11000

    CAS:
    <p>PK11000 is a p53 targeting compound, has anti-tumor activities through activation of unstable p53.</p>
    Fórmula:C6H5ClN2O4S
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:236.63
  • Abacavir monosulfate

    CAS:
    <p>Abacavir monosulfate: oral HIV inhibitor, anticancer; crosses blood-brain barrier, suppresses telomerase.</p>
    Fórmula:C14H20N6O5S
    Cor e Forma:Solid
    Peso molecular:384.41
  • Benidipine hydrochloride

    CAS:
    <p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>
    Fórmula:C28H32ClN3O6
    Pureza:99.80%
    Cor e Forma:Solid
    Peso molecular:542.03
  • (ZE)-SU9516

    CAS:
    <p>(ZE)-SU9516 is a selectively potent ATP-competitive inhibitor of CDKs.</p>
    Fórmula:C13H11N3O2
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:241.25
  • Diclofenac Potassium

    CAS:
    <p>Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.</p>
    Fórmula:C14H10Cl2KNO2
    Pureza:99.51%
    Cor e Forma:White To Yellowish Crystalline Powder
    Peso molecular:334.24
  • Thalidomide-O-amido-PEG2-C2-NH2 TFA

    CAS:
    <p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>
    Fórmula:C23H27F3N4O10
    Pureza:95.74% - 99%
    Cor e Forma:Solid
    Peso molecular:576.48
  • IMT1

    CAS:
    <p>IMT1 (Propanamide, N,N-dimethyl-2-[[4-(2-methylphenyl)-2-oxo-2H-1-benzopyran-7-yl]oxy]-) has anticancer activity.</p>
    Fórmula:C21H21NO4
    Pureza:98.07% - 98.14%
    Cor e Forma:Solid
    Peso molecular:351.4
  • Cystamine dihydrochloride

    CAS:
    <p>Cystamine dihydrochloride is a radiation-protective agent. It also protects against carbon tetrachloride liver damage.</p>
    Fórmula:C4H14Cl2N2S2
    Pureza:98.91% - 99.81%
    Cor e Forma:White Powder
    Peso molecular:225.19
  • MS7972

    CAS:
    <p>MS7972 is CREBBP inhibitor that blocks human p53 and CREB binding protein association. MS7972 can almost completely block this BRD interaction at 50 μM</p>
    Fórmula:C14H13NO2
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:227.26
  • KX2-361

    CAS:
    <p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>
    Fórmula:C24H24FN3O2
    Pureza:99.64% - 99.68%
    Cor e Forma:Solid
    Peso molecular:405.46
  • Fipronil

    CAS:
    <p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>
    Fórmula:C12H4Cl2F6N4OS
    Pureza:97.21%
    Cor e Forma:Solid Powder
    Peso molecular:437.15
  • Ralimetinib dimesylate

    CAS:
    <p>Ralimetinib dimesylate (LY2228820 dimesylate) is a orally available, p38 MAPK inhibitor with potential anti-inflammatory and antineoplastic activities.</p>
    Fórmula:C24H29FN6·2CH4O3S
    Pureza:98% - 99.38%
    Cor e Forma:Solid
    Peso molecular:612.74
  • Pomolic acid

    CAS:
    <p>Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-</p>
    Fórmula:C30H48O4
    Pureza:96.84% - 99.79%
    Cor e Forma:Solid
    Peso molecular:472.7
  • Crebanine

    CAS:
    <p>Crebanine mitigates arrhythmias, increases aconitine tolerance in rats, lacks effect on ouabain-induce arrhythmias, and shows anti-cancer properties.</p>
    Fórmula:C20H21NO4
    Pureza:99.17% - 99.77%
    Cor e Forma:Solid
    Peso molecular:339.39
  • DEL-22379

    CAS:
    <p>DEL-22379 is a water-soluble ERK dimerization inhibitor with IC50 of ~0.5 μM.</p>
    Fórmula:C26H28N4O3
    Pureza:99.3% - 99.53%
    Cor e Forma:Solid
    Peso molecular:444.53
  • Cilengitide

    CAS:
    <p>Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.</p>
    Fórmula:C27H40N8O7
    Pureza:98% - 99.8%
    Cor e Forma:Solid
    Peso molecular:588.66
  • Rabeprazole sodium

    CAS:
    <p>Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.</p>
    Fórmula:C18H20N3NaO3S
    Pureza:98% - 99.912%
    Cor e Forma:White Or Off White Crystalline Powder
    Peso molecular:381.42
  • Deltamethrin

    CAS:
    <p>Deltamethrin, a pyrethroid insecticide, causes reversible hind limb rigidity in rats and is used for crop protection and disease control.</p>
    Fórmula:C22H19Br2NO3
    Pureza:99.25% - 99.85%
    Cor e Forma:White To Off-White Crystals Or Powder
    Peso molecular:505.20
  • Mitochonic acid 5

    CAS:
    <p>MA-5, derived from a plant hormone, binds mitochondria and reduces heart/kidney damage, aiding mitochondrial disease survival.</p>
    Fórmula:C18H13F2NO3
    Pureza:98.85%
    Cor e Forma:Solid
    Peso molecular:329.3
  • Nutlin-3

    CAS:
    <p>Nutlin-3 is an MDM2 antagonist that inhibits MDM2-p53 interaction and activates p53. Nutlin-3 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C30H30Cl2N4O4
    Pureza:98.13% - 99.89%
    Cor e Forma:Solid
    Peso molecular:581.49
  • Desmorpholinyl Navitoclax-NH-Me

    CAS:
    <p>Desmorpholinyl Navitoclax-NH-Me (Desmorpholinyl ABT-263-NH-Me) is a Bcl-xL inhibitor, which can be employed alongside a CRBN ligand to synthesize XZ739, a</p>
    Fórmula:C44H51ClF3N5O5S3
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:918.55
  • Avadomide HCl

    CAS:
    <p>Avadomide (CC-122), an oral drug, targets CRBN, degrades Ikaros/Aiolos, and mimics interferon, showing antitumor effects in DLBCL.</p>
    Fórmula:C14H15ClN4O3
    Cor e Forma:Solid
    Peso molecular:322.75
  • NAE-IN-M22

    CAS:
    <p>NAE-IN-M22: Selective, potent NEDD8 enzyme inhibitor; blocks cancer cell growth; induces apoptosis in A549 cells; effective in vivo.</p>
    Fórmula:C20H24Cl2N2
    Pureza:97.65%
    Cor e Forma:Solid
    Peso molecular:363.32
  • Anagrelide hydrochloride

    CAS:
    <p>Anagrelide hydrochloride (BL4162A) serves as a treatment for essential thrombocytosis.</p>
    Fórmula:C10H7Cl2N3O·HCl
    Pureza:99.58%
    Cor e Forma:Off-White Powder
    Peso molecular:292.55
  • NSC622608

    CAS:
    <p>NSC622608, a VISTA ligand, modulates T-cell tumor attacks as an immune checkpoint.</p>
    Fórmula:C9H12BrN3OS2
    Pureza:98.48%
    Cor e Forma:Solid
    Peso molecular:322.24
  • Lercanidipine hydrochloride

    CAS:
    <p>Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class.</p>
    Fórmula:C36H41N3O6·HCl
    Pureza:99.86% - 99.91%
    Cor e Forma:Pale-Yellow Powder
    Peso molecular:648.19
  • 4-Oxofenretinide

    CAS:
    <p>4-Oxofenretinide (3-Keto fenretinide) , a recently identified fenretinide metabolite, induces marked G2-M cell cycle arrest and apoptosis.</p>
    Fórmula:C26H31NO3
    Pureza:96.89%
    Cor e Forma:Solid
    Peso molecular:405.53
  • Ibuprofen Lysine

    CAS:
    <p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>
    Fórmula:C19H32N2O4
    Pureza:99.26%
    Cor e Forma:Coa
    Peso molecular:352.47
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Fórmula:C14H17ClN2
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:248.75
  • Bardoxolone Methyl

    CAS:
    <p>Bardoxolone Methyl (TP-155) is a synthetic triterpenoid that acts as an activator of the Nrf2 pathway and an inhibitor of the NF-κB pathway with potential anti-</p>
    Fórmula:C32H43NO4
    Pureza:97.81% - 99.09%
    Cor e Forma:Solid
    Peso molecular:505.69
  • RA375

    CAS:
    <p>RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than RA190 due to nitro rings and chloroacetamide.</p>
    Fórmula:C30H25ClN4O7
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:588.99
  • SRT 2183

    CAS:
    <p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>
    Fórmula:C27H24N4O2S
    Pureza:97.86%
    Cor e Forma:Solid
    Peso molecular:468.57
  • 2-Bromohexadecanoic acid

    CAS:
    <p>2-Bromohexadecanoic acid (2-BP) is a PPARδ agonist, and a palmitoylation inhibitor, inhibiting DHHC-mediated palmitoylation. Cost-effective and quality-assured.</p>
    Fórmula:C16H31BrO2
    Pureza:97% - 98.3%
    Cor e Forma:White Crystalline Powder
    Peso molecular:335.32
  • Vildagliptin dihydrate

    CAS:
    <p>Vildagliptin dihydrate: potent, selective DPP-IV inhibitor with 3.5 nM IC50, high oral bioavailability, effective against hyperglycemia.</p>
    Fórmula:C17H29N3O4
    Cor e Forma:Solid
    Peso molecular:339.436
  • Mycophenolic acid sodium

    CAS:
    <p>Mycophenolic acid sodium inhibits IMPDH with EC50 of 0.24 μM, has antiviral, immunosuppressive, antiangiogenic, and antitumor properties.</p>
    Fórmula:C17H19NaO6
    Cor e Forma:Solid
    Peso molecular:342.323
  • Decursin

    CAS:
    <p>Decursin: potential antiepileptic, hepatoprotective, anti-cancer, anti-amnesic; affects NOX activation, PKCα/MAPK/NF-κB pathways, AChE.</p>
    Fórmula:C19H20O5
    Pureza:97.22% - 99.84%
    Cor e Forma:Solid
    Peso molecular:328.36
  • Deguelin

    CAS:
    <p>Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.</p>
    Fórmula:C23H22O6
    Pureza:96.39% - 99.29%
    Cor e Forma:Solid
    Peso molecular:394.42
  • JQ-1 (carboxylic acid)

    CAS:
    <p>JQ-1 (carboxylic acid) is a cell-permeable BRD4 inhibitor with IC50s of 77 nM for BRD4(1) and 33 nM for BRD4(2)</p>
    Fórmula:C19H17ClN4O2S
    Pureza:99.14% - 99.9%
    Cor e Forma:Solid
    Peso molecular:400.88
  • Avitinib

    CAS:
    <p>Avitinib (AC0010), also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth factor receptor (EGFR) mutant-selective inhibitor,</p>
    Fórmula:C26H26FN7O2
    Pureza:99.81% - >99.99%
    Cor e Forma:Solid
    Peso molecular:487.53
  • Pantoprazole sodium

    CAS:
    <p>Pantoprazole sodium is a proton pump inhibitor that irreversibly blocks gastric acid secretion by bonding with H+/K+-ATPase.</p>
    Fórmula:C16H14F2N3NaO4S
    Pureza:96.92% - 99.81%
    Cor e Forma:White To Off-White Solid
    Peso molecular:405.35
  • Ζ-Stat

    CAS:
    <p>ζ-Stat (NSC37044), a specific and atypical inhibitor of PKC-ζ with an IC50 of 5 μM, demonstrates the ability to inhibit proliferation and induce apoptosis in</p>
    Fórmula:C10H8O10S3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:384.36
  • Thalidomide-O-amido-PEG-C2-NH2 hydrochloride

    CAS:
    <p>Thalidomide-O-amido-PEG-C2-NH2 HCl is a cereblon ligand-linker for PROTAC synthesis.</p>
    Fórmula:C19H23ClN4O7
    Pureza:95%
    Cor e Forma:Solid
    Peso molecular:454.862
  • Mirdametinib

    CAS:
    <p>Mirdametinib (PD325901) is an MEK inhibitor (IC50=0.33 nM) with selective, non-ATP-competitive, and oral activity.</p>
    Fórmula:C16H14F3IN2O4
    Pureza:99.11% - 99.63%
    Cor e Forma:White Powder
    Peso molecular:482.19
  • Darapladib

    CAS:
    <p>Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.</p>
    Fórmula:C36H38F4N4O2S
    Pureza:99.82% - >99.99%
    Cor e Forma:Solid
    Peso molecular:666.77
  • BTR-1

    CAS:
    <p>5-Benzylidene-3-ethyl rhodanine(BTR-1 (5-Benzylidene-3-ethyl rhodanine)) is an active anti-cancer agent. BTR-1 activates apoptosis and induces cell death.</p>
    Fórmula:C12H11NOS2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:249.35
  • Picrocrocin

    CAS:
    <p>Picrocrocin is a natural product</p>
    Fórmula:C16H26O7
    Pureza:98.4%
    Cor e Forma:Solid
    Peso molecular:330.37
  • 4-Methylbenzylidene camphor

    CAS:
    <p>4-Methylbenzylidene camphor: UVB blocker in sunscreens, cosmetics; exhibits estrogenic activity.</p>
    Fórmula:C18H22O
    Pureza:99.92%
    Cor e Forma:White Solid
    Peso molecular:254.37
  • GDC-0623

    CAS:
    <p>GDC-0623 (RG 7421) is a potent and ATP-uncompetitive MEK1 inhibitor with Ki of 0.13 nM. Phase 1.</p>
    Fórmula:C16H14FIN4O3
    Pureza:98.95% - 99.02%
    Cor e Forma:Solid
    Peso molecular:456.21