
Apoptose
Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.
Subcategorias de "Apoptose"
- ASK(6 produtos)
- BCL(11 produtos)
- Caspase(125 produtos)
- FOXO1(3 produtos)
- IAP(66 produtos)
- Mdm2(12 produtos)
- PD-1/PD-L1(125 produtos)
- PDK(9 produtos)
- PERK(25 produtos)
- Serina/treonina quinase(15 produtos)
- Survivina(13 produtos)
- TNF(92 produtos)
- c-RET(51 produtos)
- p53(62 produtos)
Exibir 6 mais subcategorias
Foram encontrados 5592 produtos de "Apoptose"
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Tauroursodeoxycholate
CAS:<p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>Fórmula:C26H45NO6SPureza:98.77% - 99.93%Cor e Forma:White SolidPeso molecular:499.7PEAQX
CAS:<p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>Fórmula:C17H17BrN3O5PPureza:98% - 99.9%Cor e Forma:SolidPeso molecular:454.21AR42
CAS:<p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>Fórmula:C18H20N2O3Pureza:98.46% - 98.96%Cor e Forma:SolidPeso molecular:312.36Emricasan
CAS:<p>Emricasan (IDN-6556) is a pan-caspase inhibitor with irreversible properties.</p>Fórmula:C26H27F4N3O7Pureza:98.13% - 99%Cor e Forma:SolidPeso molecular:569.5Aloperine
CAS:<p>Aloperine exhibits anti-inflammatory, antibacterial, antiviral, and anti-tumor properties.</p>Fórmula:C15H24N2Pureza:98% - 99.88%Cor e Forma:Yellow Crystalline PowderPeso molecular:232.361400W dihydrochloride
CAS:<p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>Fórmula:C10H17Cl2N3Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:250.17Bilobalide
CAS:<p>Bilobalide ((-)-Bilobalide), a bioactive from Gingko Biloba, is active on hypoxia-induced alterations.</p>Fórmula:C15H18O8Pureza:98.81% - 99.92%Cor e Forma:White SolidPeso molecular:326.3Ipatasertib
CAS:<p>Ipatasertib (GDC-0068) is a selective, ATP-competitive pan-Akt inhibitor that can lead to p53-independent PUMA activation.Cost-effective and quality-assured.</p>Fórmula:C24H32ClN5O2Pureza:98.28% - 99.21%Cor e Forma:SolidPeso molecular:458Sulforaphane
CAS:<p>Sulforaphane is a natural isothiocyanate that activates Nrf2. Sulforaphane has antitumor and anti-inflammatory activities. Cost-effective and quality-assured.</p>Fórmula:C6H11NOS2Pureza:95% - 99.79%Cor e Forma:Light Yellow LiquidPeso molecular:177.29Nω-Hydroxy-nor-L-Arginine Dihydrochloride
CAS:<p>Nω-Hydroxy-nor-L-Arginine Dihydrochloride is a competitive and reversible inhibitor of arginase</p>Fórmula:C5H14Cl2N4O3Pureza:99.12% - 99.84%Cor e Forma:SolidPeso molecular:249.10ZZW-115 hydrochloride
CAS:<p>ZZW-115 hydrochloride inhibits the activity of NUPR1.</p>Fórmula:C24H34Cl3F3N4SPureza:99.97%Cor e Forma:SolidPeso molecular:573.97Chromium picolinate
CAS:<p>Chromium picolinate causes DNA damage and mutation. It is an activator of p38.</p>Fórmula:C18H12CrN3O6Pureza:99.64%Cor e Forma:Violet-Red Crystalline PowderPeso molecular:418.30Thalidomide-NH-PEG1-NH2 hydrochloride
CAS:<p>Thalidomide-NH-PEG1-NH2 hydrochloride (4-[(2-(2-Aminoethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione HCl) is a synthetic E3 ligase ligand-</p>Fórmula:C17H21ClN4O5Pureza:97.13%Cor e Forma:SolidPeso molecular:396.83Trolox
CAS:<p>Trolox is a vitamin E analogue, used in reducing oxidative stress or damage.</p>Fórmula:C14H18O4Pureza:98.90% - 99.90%Cor e Forma:White To Fainly Beige Crystalline PowderPeso molecular:250.29Thalidomide-NH-CH2-COOH
CAS:<p>Thalidomide-NH-CH2-COOH ((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)glycine) is a synthesized E3 ligase ligand-linker conjugate containing a</p>Fórmula:C15H13N3O6Pureza:96.3800%Cor e Forma:SolidPeso molecular:331.28Tetrahydroxyquinone monohydrate
CAS:<p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>Fórmula:C6H6O7Cor e Forma:SolidPeso molecular:190.11Apocynin
CAS:<p>Apocynin (NSC 2146) is a specific NADPH-oxidase inhibitor (IC50: 10 μM).</p>Fórmula:C9H10O3Pureza:99.71% - 99.98%Cor e Forma:Yellowish To Brown PowderPeso molecular:166.17Alda-1
CAS:<p>Alda-1 activates ALDH2*1 and ALDH2*2, permeates cells, and targets mitochondrial aldehyde dehydrogenase 2.</p>Fórmula:C15H11Cl2NO3Pureza:98.5% - 99.63%Cor e Forma:SolidPeso molecular:324.16Metamizole magnesium
CAS:<p>Metamizole magnesium (Metamizolemagnesiumsalt) is a pain reliever, which can antispasmodic.</p>Fórmula:C26H32MgN6O8S2Pureza:93.51%Cor e Forma:SolidPeso molecular:645.01ARRY 520 hydrochloride
CAS:<p>'ARRY 520 hydrochloride: a KSP inhibitor causing apoptosis and strong anti-proliferative effects.'</p>Fórmula:C20H23ClF2N4O2SPureza:98.06% - 99.62%Cor e Forma:SolidPeso molecular:456.94Eltrombopag Olamine
CAS:<p>Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin</p>Fórmula:C29H36N6O6Pureza:99.59% - 99.89%Cor e Forma:SolidPeso molecular:564.63HA15
CAS:<p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>Fórmula:C23H22N4O3S2Pureza:99.77% - 99.86%Cor e Forma:SolidPeso molecular:466.58ISRIB (trans-isomer)
CAS:<p>ISRIB (trans-isomer) is a potent inhibitor of PERK that rescues protein translation and prevents SG formation in the presence of P-eIF2α. Cost effective and quality assured.</p>Fórmula:C22H24Cl2N2O4Pureza:97.86% - 99.27%Cor e Forma:SolidPeso molecular:451.34Thalidomide 4-fluoride
CAS:<p>Thalidomide 4-fluoride (E3 ligase Ligand 4) (Cereblon ligand 4) is the Thalidomide-based Cereblon ligand.</p>Fórmula:C13H9FN2O4Pureza:99.12%Cor e Forma:SolidPeso molecular:276.22Thalidomide-O-amido-C6-NH2 hydrochloride
CAS:<p>Thalidomide-O-amido-C6-NH2 HCl, a cereblon ligand-linker for PROTAC synthesis.</p>Fórmula:C21H27ClN4O6Pureza:97.33%Cor e Forma:SolidPeso molecular:466.915CA-4948
CAS:<p>CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity.</p>Fórmula:C24H25N7O5Pureza:99.35% - 99.88%Cor e Forma:SolidPeso molecular:491.5Tenovin-6
CAS:<p>Tenovin-6 is a p53 transcriptional activity agonist.</p>Fórmula:C25H34N4O2SPureza:97.71% - >99.99%Cor e Forma:SolidPeso molecular:454.63Dacarbazine citrate
CAS:<p>Dacarbazine citrate treats lymphatic cancers, malignant melanoma, islet cell carcinoma, and soft tissue sarcoma.</p>Fórmula:C12H18N6O8Cor e Forma:SolidPeso molecular:374.31FOXO4-DRI acetate
<p>FOXO4-DRI acetate is a bioactive chemical.</p>Fórmula:C36H64N14O14SPureza:99.10%Cor e Forma:SolidPeso molecular:5358.06Periplocin
CAS:<p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>Fórmula:C36H56O13Pureza:99.66% - 99.74%Cor e Forma:SolidPeso molecular:696.82TrxR1-IN-B19
CAS:<p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>Fórmula:C21H22O5Pureza:98.6%Cor e Forma:SolidPeso molecular:354.4Thalidomide-O-amido-C3-NH2 TFA
CAS:<p>Thalidomide-based E3 ligase linker for PROTAC tech; cereblon ligand conjugate.</p>Fórmula:C20H21F3N4O8Pureza:98.47%Cor e Forma:SolidPeso molecular:502.4Thalidomide-O-COOH
CAS:<p>Thalidomide-O-COOH is a Cereblon ligand for CRBN protein recruitment and PROTAC construction with a linker.</p>Fórmula:C15H12N2O7Pureza:98% - 98.29%Cor e Forma:SolidPeso molecular:332.27Methoxychlor
CAS:<p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>Fórmula:C16H15Cl3O2Pureza:98.82% - ≥95%Cor e Forma:Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment IfPeso molecular:345.65Liproxstatin-1 hydrochloride
CAS:<p>Liproxstatin-1 hydrochloride is a high-potency ferroptosis inhibitor capable of effectively preventing ferroptotic cell death, with an IC50 value of 22 nM [1].</p>Fórmula:C19H22Cl2N4Cor e Forma:SolidPeso molecular:377.31GSK778 hydrochloride
CAS:<p>GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to 143 nM, effective in cancer models.</p>Fórmula:C30H34ClN5O3Pureza:97.26% - 98.35%Cor e Forma:SolidPeso molecular:548.08Thalidomide-4-OH
CAS:<p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>Fórmula:C13H10N2O5Pureza:99.59%Cor e Forma:SolidPeso molecular:274.23Thalidomide-NH-C4-NH-Boc
CAS:<p>Thalidomide-NH-C4-NH-Boc is a cereblon-based E3 ligase ligand-linker for PROTACs.</p>Fórmula:C22H28N4O6Pureza:98.87%Cor e Forma:SolidPeso molecular:444.48Difurazon hydrochloride
CAS:<p>Difurazon HCl: a mutagenic antibacterial and growth promoter, used for bacillary dysentery in feed.</p>Fórmula:C14H13ClN6O6Pureza:98.51%Cor e Forma:SolidPeso molecular:396.74Methoxyamine HCl
CAS:<p>Methoxyamine HCl targets DNA repair sites, potentially increasing DNA breaks and enhancing alkylating agents' anti-cancer effects.</p>Fórmula:CH6ClNOPureza:≥98%Cor e Forma:SolidPeso molecular:83.51Alogliptin Benzoate
CAS:<p>Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>Fórmula:C25H27N5O4Pureza:99.94% - >99.99%Cor e Forma:White PowderPeso molecular:461.51OICR-9429
CAS:<p>OICR-9429 blocks WDR5 binding to MLL/Histone 3, hindering acute myeloid leukemia cell growth in vitro.</p>Fórmula:C29H32F3N5O3Pureza:97.07% - 99.93%Cor e Forma:SolidPeso molecular:555.59Thalidomide-O-amido-PEG3-C2-NH2 TFA
CAS:<p>Synthetic E3 ligase ligand-linker, Thalidomide-O-amido-PEG3-C2-NH2 TFA, used in PROTAC with cereblon ligand and PEG.</p>Fórmula:C25H31F3N4O11Pureza:99.82%Cor e Forma:SolidPeso molecular:620.54Bigelovin
CAS:<p>Bigelovin: RXRα agonist, inhibits mTOR via ROS, induces apoptosis/autophagy, anti-tumor sesquiterpene from Inula sp.</p>Fórmula:C17H20O5Pureza:99.61% - 99.72%Cor e Forma:SolidPeso molecular:304.34KRCA-0008
CAS:<p>KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability.</p>Fórmula:C30H37ClN8O4Pureza:96.19%Cor e Forma:SolidPeso molecular:609.12Perhexiline
CAS:<p>Perhexiline: oral CPT1/2 inhibitor, limits fat metabolism, crosses BBB, anti-cancer, induces liver cell apoptosis, for cancer/cardio research.</p>Fórmula:C19H35NCor e Forma:SolidPeso molecular:277.49Ketorolac hemicalcium
CAS:<p>Ketorolac hemicalcium: NSAID, COX-1/COX-2 inhibitor (IC50: 20/120 nM), treats eye inflammation & pain, used in cancer research.</p>Fórmula:C30H24CaN2O6Cor e Forma:SolidPeso molecular:548.608Thalidomide-propargyl
CAS:<p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>Fórmula:C16H12N2O5Pureza:95.14%Cor e Forma:SolidPeso molecular:312.28Thalidomide-NH-C6-NH2 hydrochloride
CAS:<p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>Fórmula:C19H25ClN4O4Pureza:99.27%Cor e Forma:SolidPeso molecular:408.88Britannin
CAS:<p>Britannin, a sesquiterpene lactone, inhibits proliferation and induces apoptosis through the mitochondrial signaling pathway in human breast cancer cells.</p>Fórmula:C19H26O7Pureza:98% - 99.98%Cor e Forma:SolidPeso molecular:366.41Verteporfin
CAS:<p>Verteporfin (BPD-MA) is a YAP inhibitor that inhibits YAP-TEAD interactions.</p>Fórmula:C41H42N4O8Pureza:95.37% - 99.82%Cor e Forma:Dark Green To Black SolidPeso molecular:718.79Sulfaphenazole
CAS:<p>Sulfaphenazole (Plisulfan) is an inhibitor of CYP2C9 (Ki: 0.3 μM) that demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki: 63/29 μM for</p>Fórmula:C15H14N4O2SPureza:97.53% - 99.67%Cor e Forma:SolidPeso molecular:314.36PK11000
CAS:<p>PK11000 is a p53 targeting compound, has anti-tumor activities through activation of unstable p53.</p>Fórmula:C6H5ClN2O4SPureza:99.70%Cor e Forma:SolidPeso molecular:236.63Abacavir monosulfate
CAS:<p>Abacavir monosulfate: oral HIV inhibitor, anticancer; crosses blood-brain barrier, suppresses telomerase.</p>Fórmula:C14H20N6O5SCor e Forma:SolidPeso molecular:384.41Benidipine hydrochloride
CAS:<p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>Fórmula:C28H32ClN3O6Pureza:99.80%Cor e Forma:SolidPeso molecular:542.03(ZE)-SU9516
CAS:<p>(ZE)-SU9516 is a selectively potent ATP-competitive inhibitor of CDKs.</p>Fórmula:C13H11N3O2Pureza:99.59%Cor e Forma:SolidPeso molecular:241.25Diclofenac Potassium
CAS:<p>Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.</p>Fórmula:C14H10Cl2KNO2Pureza:99.51%Cor e Forma:White To Yellowish Crystalline PowderPeso molecular:334.24Thalidomide-O-amido-PEG2-C2-NH2 TFA
CAS:<p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>Fórmula:C23H27F3N4O10Pureza:95.74% - 99%Cor e Forma:SolidPeso molecular:576.48IMT1
CAS:<p>IMT1 (Propanamide, N,N-dimethyl-2-[[4-(2-methylphenyl)-2-oxo-2H-1-benzopyran-7-yl]oxy]-) has anticancer activity.</p>Fórmula:C21H21NO4Pureza:98.07% - 98.14%Cor e Forma:SolidPeso molecular:351.4Cystamine dihydrochloride
CAS:<p>Cystamine dihydrochloride is a radiation-protective agent. It also protects against carbon tetrachloride liver damage.</p>Fórmula:C4H14Cl2N2S2Pureza:98.91% - 99.81%Cor e Forma:White PowderPeso molecular:225.19MS7972
CAS:<p>MS7972 is CREBBP inhibitor that blocks human p53 and CREB binding protein association. MS7972 can almost completely block this BRD interaction at 50 μM</p>Fórmula:C14H13NO2Pureza:99.78%Cor e Forma:SolidPeso molecular:227.26KX2-361
CAS:<p>KX2-361 is a orally bioavailable small molecule dual Src/tubulin inhibitor that provides long term survival in a murine model of glioblastoma</p>Fórmula:C24H24FN3O2Pureza:99.64% - 99.68%Cor e Forma:SolidPeso molecular:405.46Fipronil
CAS:<p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>Fórmula:C12H4Cl2F6N4OSPureza:97.21%Cor e Forma:Solid PowderPeso molecular:437.15Ralimetinib dimesylate
CAS:<p>Ralimetinib dimesylate (LY2228820 dimesylate) is a orally available, p38 MAPK inhibitor with potential anti-inflammatory and antineoplastic activities.</p>Fórmula:C24H29FN6·2CH4O3SPureza:98% - 99.38%Cor e Forma:SolidPeso molecular:612.74Pomolic acid
CAS:<p>Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-</p>Fórmula:C30H48O4Pureza:96.84% - 99.79%Cor e Forma:SolidPeso molecular:472.7Crebanine
CAS:<p>Crebanine mitigates arrhythmias, increases aconitine tolerance in rats, lacks effect on ouabain-induce arrhythmias, and shows anti-cancer properties.</p>Fórmula:C20H21NO4Pureza:99.17% - 99.77%Cor e Forma:SolidPeso molecular:339.39DEL-22379
CAS:<p>DEL-22379 is a water-soluble ERK dimerization inhibitor with IC50 of ~0.5 μM.</p>Fórmula:C26H28N4O3Pureza:99.3% - 99.53%Cor e Forma:SolidPeso molecular:444.53Cilengitide
CAS:<p>Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.</p>Fórmula:C27H40N8O7Pureza:98% - 99.8%Cor e Forma:SolidPeso molecular:588.66Rabeprazole sodium
CAS:<p>Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.</p>Fórmula:C18H20N3NaO3SPureza:98% - 99.912%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:381.42Deltamethrin
CAS:<p>Deltamethrin, a pyrethroid insecticide, causes reversible hind limb rigidity in rats and is used for crop protection and disease control.</p>Fórmula:C22H19Br2NO3Pureza:99.25% - 99.85%Cor e Forma:White To Off-White Crystals Or PowderPeso molecular:505.20Mitochonic acid 5
CAS:<p>MA-5, derived from a plant hormone, binds mitochondria and reduces heart/kidney damage, aiding mitochondrial disease survival.</p>Fórmula:C18H13F2NO3Pureza:98.85%Cor e Forma:SolidPeso molecular:329.3Nutlin-3
CAS:<p>Nutlin-3 is an MDM2 antagonist that inhibits MDM2-p53 interaction and activates p53. Nutlin-3 has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C30H30Cl2N4O4Pureza:98.13% - 99.89%Cor e Forma:SolidPeso molecular:581.49Desmorpholinyl Navitoclax-NH-Me
CAS:<p>Desmorpholinyl Navitoclax-NH-Me (Desmorpholinyl ABT-263-NH-Me) is a Bcl-xL inhibitor, which can be employed alongside a CRBN ligand to synthesize XZ739, a</p>Fórmula:C44H51ClF3N5O5S3Pureza:99.87%Cor e Forma:SolidPeso molecular:918.55Avadomide HCl
CAS:<p>Avadomide (CC-122), an oral drug, targets CRBN, degrades Ikaros/Aiolos, and mimics interferon, showing antitumor effects in DLBCL.</p>Fórmula:C14H15ClN4O3Cor e Forma:SolidPeso molecular:322.75NAE-IN-M22
CAS:<p>NAE-IN-M22: Selective, potent NEDD8 enzyme inhibitor; blocks cancer cell growth; induces apoptosis in A549 cells; effective in vivo.</p>Fórmula:C20H24Cl2N2Pureza:97.65%Cor e Forma:SolidPeso molecular:363.32Anagrelide hydrochloride
CAS:<p>Anagrelide hydrochloride (BL4162A) serves as a treatment for essential thrombocytosis.</p>Fórmula:C10H7Cl2N3O·HClPureza:99.58%Cor e Forma:Off-White PowderPeso molecular:292.55NSC622608
CAS:<p>NSC622608, a VISTA ligand, modulates T-cell tumor attacks as an immune checkpoint.</p>Fórmula:C9H12BrN3OS2Pureza:98.48%Cor e Forma:SolidPeso molecular:322.24Lercanidipine hydrochloride
CAS:<p>Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class.</p>Fórmula:C36H41N3O6·HClPureza:99.86% - 99.91%Cor e Forma:Pale-Yellow PowderPeso molecular:648.194-Oxofenretinide
CAS:<p>4-Oxofenretinide (3-Keto fenretinide) , a recently identified fenretinide metabolite, induces marked G2-M cell cycle arrest and apoptosis.</p>Fórmula:C26H31NO3Pureza:96.89%Cor e Forma:SolidPeso molecular:405.53Ibuprofen Lysine
CAS:<p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>Fórmula:C19H32N2O4Pureza:99.26%Cor e Forma:CoaPeso molecular:352.471-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Fórmula:C14H17ClN2Pureza:98.27%Cor e Forma:SolidPeso molecular:248.75Bardoxolone Methyl
CAS:<p>Bardoxolone Methyl (TP-155) is a synthetic triterpenoid that acts as an activator of the Nrf2 pathway and an inhibitor of the NF-κB pathway with potential anti-</p>Fórmula:C32H43NO4Pureza:97.81% - 99.09%Cor e Forma:SolidPeso molecular:505.69RA375
CAS:<p>RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than RA190 due to nitro rings and chloroacetamide.</p>Fórmula:C30H25ClN4O7Pureza:99.56%Cor e Forma:SolidPeso molecular:588.99SRT 2183
CAS:<p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>Fórmula:C27H24N4O2SPureza:97.86%Cor e Forma:SolidPeso molecular:468.572-Bromohexadecanoic acid
CAS:<p>2-Bromohexadecanoic acid (2-BP) is a PPARδ agonist, and a palmitoylation inhibitor, inhibiting DHHC-mediated palmitoylation. Cost-effective and quality-assured.</p>Fórmula:C16H31BrO2Pureza:97% - 98.3%Cor e Forma:White Crystalline PowderPeso molecular:335.32Vildagliptin dihydrate
CAS:<p>Vildagliptin dihydrate: potent, selective DPP-IV inhibitor with 3.5 nM IC50, high oral bioavailability, effective against hyperglycemia.</p>Fórmula:C17H29N3O4Cor e Forma:SolidPeso molecular:339.436Mycophenolic acid sodium
CAS:<p>Mycophenolic acid sodium inhibits IMPDH with EC50 of 0.24 μM, has antiviral, immunosuppressive, antiangiogenic, and antitumor properties.</p>Fórmula:C17H19NaO6Cor e Forma:SolidPeso molecular:342.323Decursin
CAS:<p>Decursin: potential antiepileptic, hepatoprotective, anti-cancer, anti-amnesic; affects NOX activation, PKCα/MAPK/NF-κB pathways, AChE.</p>Fórmula:C19H20O5Pureza:97.22% - 99.84%Cor e Forma:SolidPeso molecular:328.36Deguelin
CAS:<p>Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.</p>Fórmula:C23H22O6Pureza:96.39% - 99.29%Cor e Forma:SolidPeso molecular:394.42JQ-1 (carboxylic acid)
CAS:<p>JQ-1 (carboxylic acid) is a cell-permeable BRD4 inhibitor with IC50s of 77 nM for BRD4(1) and 33 nM for BRD4(2)</p>Fórmula:C19H17ClN4O2SPureza:99.14% - 99.9%Cor e Forma:SolidPeso molecular:400.88Avitinib
CAS:<p>Avitinib (AC0010), also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth factor receptor (EGFR) mutant-selective inhibitor,</p>Fórmula:C26H26FN7O2Pureza:99.81% - >99.99%Cor e Forma:SolidPeso molecular:487.53Pantoprazole sodium
CAS:<p>Pantoprazole sodium is a proton pump inhibitor that irreversibly blocks gastric acid secretion by bonding with H+/K+-ATPase.</p>Fórmula:C16H14F2N3NaO4SPureza:96.92% - 99.81%Cor e Forma:White To Off-White SolidPeso molecular:405.35Ζ-Stat
CAS:<p>ζ-Stat (NSC37044), a specific and atypical inhibitor of PKC-ζ with an IC50 of 5 μM, demonstrates the ability to inhibit proliferation and induce apoptosis in</p>Fórmula:C10H8O10S3Pureza:99.85%Cor e Forma:SolidPeso molecular:384.36Thalidomide-O-amido-PEG-C2-NH2 hydrochloride
CAS:<p>Thalidomide-O-amido-PEG-C2-NH2 HCl is a cereblon ligand-linker for PROTAC synthesis.</p>Fórmula:C19H23ClN4O7Pureza:95%Cor e Forma:SolidPeso molecular:454.862Mirdametinib
CAS:<p>Mirdametinib (PD325901) is an MEK inhibitor (IC50=0.33 nM) with selective, non-ATP-competitive, and oral activity.</p>Fórmula:C16H14F3IN2O4Pureza:99.11% - 99.63%Cor e Forma:White PowderPeso molecular:482.19Darapladib
CAS:<p>Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.</p>Fórmula:C36H38F4N4O2SPureza:99.82% - >99.99%Cor e Forma:SolidPeso molecular:666.77BTR-1
CAS:<p>5-Benzylidene-3-ethyl rhodanine(BTR-1 (5-Benzylidene-3-ethyl rhodanine)) is an active anti-cancer agent. BTR-1 activates apoptosis and induces cell death.</p>Fórmula:C12H11NOS2Pureza:98%Cor e Forma:SolidPeso molecular:249.35Picrocrocin
CAS:<p>Picrocrocin is a natural product</p>Fórmula:C16H26O7Pureza:98.4%Cor e Forma:SolidPeso molecular:330.374-Methylbenzylidene camphor
CAS:<p>4-Methylbenzylidene camphor: UVB blocker in sunscreens, cosmetics; exhibits estrogenic activity.</p>Fórmula:C18H22OPureza:99.92%Cor e Forma:White SolidPeso molecular:254.37GDC-0623
CAS:<p>GDC-0623 (RG 7421) is a potent and ATP-uncompetitive MEK1 inhibitor with Ki of 0.13 nM. Phase 1.</p>Fórmula:C16H14FIN4O3Pureza:98.95% - 99.02%Cor e Forma:SolidPeso molecular:456.21
