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Apoptose

Apoptose

Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.

Subcategorias de "Apoptose"

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Foram encontrados 5592 produtos de "Apoptose"

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  • Obatoclax Mesylate

    CAS:
    <p>Obatoclax Mesylate (GX15-070) is a Bcl-2 antagonist (Ki: 0.22 μM) and can induce apoptosis with up-regulation of Bim, induced cytochrome c release, and</p>
    Fórmula:C20H19N3O·CH4O3S
    Pureza:99.58% - 99.88%
    Cor e Forma:Solid
    Peso molecular:413.49
  • Ibandronate sodium monohydrate

    CAS:
    <p>Ibandronate sodium monohydrate (BM-210955) is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.</p>
    Fórmula:C9H24NNaO8P2
    Pureza:99.62%
    Cor e Forma:White Crystalline Powder
    Peso molecular:359.23
  • Neobavaisoflavone

    CAS:
    <p>Neobavaisoflavone: DNA polymerase inhibitor, potential for treating bone loss, anti-inflammatory, reduces ROS, RNS, cytokines in macrophages.</p>
    Fórmula:C20H18O4
    Pureza:99.31% - 99.87%
    Cor e Forma:Solid
    Peso molecular:322.35
  • RGX-202

    CAS:
    <p>RGX-202 (β-GPA) is an orally active inhibitor of the SLC6A8 transport protein. RGX-202 is a creatine analog that alters skeletal muscle energy expenditure.</p>
    Fórmula:C4H9N3O2
    Pureza:99.67% - 99.8%
    Cor e Forma:Solid
    Peso molecular:131.13
  • PD173955

    CAS:
    <p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>
    Fórmula:C21H16Cl2N4OS
    Pureza:98.52% - 98.99%
    Cor e Forma:Solid
    Peso molecular:443.35
  • Nobiletin

    CAS:
    <p>Nobiletin: a citrus-derived flavone with anti-inflammatory and anti-cancer properties; water-insoluble, very weak acid.</p>
    Fórmula:C21H22O8
    Pureza:98.65% - 99.76%
    Cor e Forma:Solid
    Peso molecular:402.39
  • Bioymifi

    CAS:
    <p>Bioymifi (DR5 Activator), a novel TRAIL activator, binds to DR5's ECD, inducing DR5 aggregation and stimulating cell apoptosis. Cost-effective and quality-assured.</p>
    Fórmula:C22H12BrN3O4S
    Pureza:98% - 99.79%
    Cor e Forma:Solid
    Peso molecular:494.32
  • Oncrasin-1

    CAS:
    <p>Oncrasin 1 is a potent inhibitor of anticancer that kills various human lung cancer cells with K-Ras mutations at low or submicromolar concentrations</p>
    Fórmula:C16H12ClNO
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:269.73
  • Rilmenidine hemifumarate

    CAS:
    <p>Rilmenidine hemifumarate (S-3341 hemifumarate) is an I1 imidazoline receptor and α2-adrenergic receptor agonist that induces autophagy.</p>
    Fórmula:C10H16N2OC4H4O4
    Pureza:98.14%
    Cor e Forma:Solid
    Peso molecular:238.28
  • CA-5f

    CAS:
    <p>CA-5f is a potent late-stage macroautophagy/autophagy inhibitor via inhibiting autophagosome-lysosome fusion.</p>
    Fórmula:C24H24N2O3
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:388.46
  • 2,5-dimethyl Celecoxib

    CAS:
    <p>2,5-dimethyl Celecoxib, a derivative targeting mPGES-1, inhibits PGE2 synthesis in inflammation.</p>
    Fórmula:C18H16F3N3O2S
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:395.4
  • Pinoresinol

    CAS:
    <p>Pinoresinol ((+)-Pinoresinol) has antiinflammatory, hepatoprotective, and fungicidal activities, it can protect pial microcirculation from I-reperfusion injury</p>
    Fórmula:C20H22O6
    Pureza:98.67%
    Cor e Forma:Solid
    Peso molecular:358.39
  • BX-912

    CAS:
    <p>BX-912 inhibits PDK1 with IC50 of 12 nM; over 10x more selective versus C-Kit, EGFR, PKA, PKC.</p>
    Fórmula:C20H23BrN8O
    Pureza:98.29% - 99.34%
    Cor e Forma:Solid
    Peso molecular:471.35
  • CCT128930 hydrochloride

    CAS:
    <p>CCT128930 hydrochloride: Potent AKT inhibitor (IC50=6 nM), 28x selective over PKA, 20x over p70S6K, induces cell cycle arrest &amp; DNA damage.</p>
    Fórmula:C18H21Cl2N5
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:378.3
  • L-Asparaginase

    CAS:
    <p>L-Asparaginase, an enzyme for acute lymphoblastic leukemia treatment, is administered via injection.</p>
    Fórmula:NA
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:N/A
  • Elesclomol

    CAS:
    <p>Elesclomol (STA-4783) is an oxidative stress inducer and a highly lipophilic copper ion carrier.</p>
    Fórmula:C19H20N4O2S2
    Pureza:97.17% - 99.51%
    Cor e Forma:Solid
    Peso molecular:400.52
  • HO-3867

    CAS:
    <p>HO-3867, an analog of curcumin, is a sspecific STAT3 inhibitor.</p>
    Fórmula:C28H30F2N2O2
    Pureza:91.18% - 99.21%
    Cor e Forma:Solid
    Peso molecular:464.55
  • LRRK2-IN-1

    CAS:
    <p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>
    Fórmula:C31H38N8O3
    Pureza:98% - 98.82%
    Cor e Forma:Solid
    Peso molecular:570.69
  • S-trityl-L-Cysteine

    CAS:
    <p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>
    Fórmula:C22H21NO2S
    Pureza:97.02%
    Cor e Forma:Almost White To Light Yellow Granular Powder
    Peso molecular:363.47
  • NSC 95397

    CAS:
    <p>NSC 95397 is a potent inhibitor of Cdc25 dual specificity phosphatase(Ki of 32, 96, and 40 nM for Cdc25A, Cdc25B, and Cdc25C, respectively).</p>
    Fórmula:C14H14O4S2
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:310.39
  • SKI II

    CAS:
    <p>SKI II is a selective non-ATP S1P receptor inhibitor with an IC50 of 0.5 μM; it doesn't inhibit PKCα, PI3K, or ERK2.</p>
    Fórmula:C15H11ClN2OS
    Pureza:99.34% - 99.93%
    Cor e Forma:Solid
    Peso molecular:302.78
  • STF-118804

    CAS:
    <p>STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 &lt;10 nM.</p>
    Fórmula:C25H23N3O4S
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:461.53
  • Pracinostat

    CAS:
    <p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>
    Fórmula:C20H30N4O2
    Pureza:99.15% - 99.67%
    Cor e Forma:Solid
    Peso molecular:358.48
  • SKI-178

    CAS:
    <p>SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM.</p>
    Fórmula:C21H22N4O4
    Pureza:97.09%
    Cor e Forma:Solid
    Peso molecular:394.42
  • Clodronate disodium tetrahydrate

    CAS:
    <p>Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.</p>
    Fórmula:CH10Cl2Na2O10P2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:360.92
  • CM-272

    CAS:
    <p>CM-272 is a dual G9a/DNA methyltransferases (DNMTs) inhibitor.</p>
    Fórmula:C28H38N4O3
    Pureza:97.83%
    Cor e Forma:Solid
    Peso molecular:478.63
  • Trifloxystrobin

    CAS:
    <p>Trifloxystrobin is a fungicide against R. solani in sugar beets with EC50s: 23.0 μg/L for Daphnia neonates, 1.7 μg/L for embryos.</p>
    Fórmula:C20H19F3N2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:408.37
  • JKE-1674

    CAS:
    <p>JKE-1674 is an orally active glutathione peroxidase 4 (GPX4) inhibitor and the active metabolite of ML-210.Cost-effective and quality-assured.</p>
    Fórmula:C20H20Cl2N4O4
    Pureza:98.02% - 98.4%
    Cor e Forma:Solid
    Peso molecular:451.3
  • QNZ

    CAS:
    <p>QNZ (EVP4593) (EVP4593) is an effective inhibitor of NF-κB activation and TNF-α production. The IC50 of QNZ for NF-κB and TNF-α is11 nM and 7 nM, respectively.</p>
    Fórmula:C22H20N4O
    Pureza:99.17% - 99.18%
    Cor e Forma:White Solid
    Peso molecular:356.42
  • Thalidomide-O-C4-NH2 hydrochloride

    CAS:
    <p>Thalidomide-linker 9: a cereblon ligand, E3 ligase conjugate for PROTAC tech.</p>
    Fórmula:C17H20ClN3O5
    Pureza:98.33%
    Cor e Forma:Solid
    Peso molecular:381.81
  • Laquinimod sodium

    CAS:
    <p>Laquinimod (ABR-215062) sodium is an oral agent for MS, halting neurodegeneration and inflammation.</p>
    Fórmula:C19H16ClN2NaO3
    Cor e Forma:Solid
    Peso molecular:378.79
  • Thalidomide-PEG4-Propargyl

    CAS:
    <p>Thalidomide-PEG4-Propargyl is a synthetic E3 ligase ligand for PROTAC with a cereblon ligand and linker.</p>
    Fórmula:C24H28N2O9
    Pureza:97.46%
    Cor e Forma:Solid
    Peso molecular:488.49
  • SKLB-163

    CAS:
    <p>SKLB-163 acts by downregulating RhoGDI, activating JNK-1 signaling pathway and caspase-3, and reducing phosphorylated Akt and p44/42 MAPK.</p>
    Fórmula:C18H16ClN3O2S2
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:405.92
  • Mitoxantrone diacetate

    CAS:
    <p>Mitoxantrone diacetate hinders topoisomerase II &amp; PKC, fights tumors &amp; orthopoxviruses (IC50: 8.5μM, EC50: 0.25-0.8μM).</p>
    Fórmula:C26H36N4O10
    Cor e Forma:Solid
    Peso molecular:564.592
  • ONO-8130

    CAS:
    <p>ONO-8130 is an orally available antagonist of EP1 receptor.</p>
    Fórmula:C25H28N2O5S2
    Pureza:97.82%
    Cor e Forma:Solid
    Peso molecular:500.63
  • Chelerythrine

    CAS:
    <p>1.</p>
    Fórmula:C21H18NO4
    Pureza:98.36%
    Cor e Forma:Solid
    Peso molecular:348.37
  • Tofacitinib Citrate

    CAS:
    <p>Tofacitinib Citrate (CP-690550 citrate) is a a potent, cell-permeable inhibitor of JAK1/2/3 (IC50s: 1/20/112 nM).</p>
    Fórmula:C22H28N6O8
    Pureza:99.19% - 99.75%
    Cor e Forma:Solid
    Peso molecular:504.49
  • Benzoylpaeoniflorin

    CAS:
    <p>1. Benzoylpaeoniflorin is active against cyclooxygenase-1 and cyclooxygenase-2 enzymes.</p>
    Fórmula:C30H32O12
    Pureza:95.86% - 97.28%
    Cor e Forma:Solid
    Peso molecular:584.57
  • Cinchonine monohydrochloride hydrate

    CAS:
    <p>Cinchonine monohydrochloride hydrate: natural antimalarial, inhibits platelet aggregation &amp; cancer cell growth, blocks fat cell formation.</p>
    Fórmula:C19H25ClN2O2
    Cor e Forma:Solid
    Peso molecular:348.87
  • C5 Lenalidomide

    CAS:
    <p>C5 Lenalidomide is an chemical weith inconclusive biological activity.</p>
    Fórmula:C13H13N3O3
    Pureza:99.4%
    Cor e Forma:Solid
    Peso molecular:259.26
  • Kinetin riboside

    CAS:
    <p>Kinetin riboside (N6-Furfuryladenosine) can induce apoptosis in cancer cells. It inhibits the proliferation of HCT-15 cells(IC50 of 2.5 μM)</p>
    Fórmula:C15H17N5O5
    Pureza:98.17%
    Cor e Forma:White Solid
    Peso molecular:347.33
  • Dacomitinib

    CAS:
    <p>Dacomitinib (PF299) is an oral selective inhibitor of EGFR, ERBB2, ERBB4 with IC50s: 6, 45.7, 73.7 nM.</p>
    Fórmula:C24H25ClFN5O2
    Pureza:99.4% - 99.72%
    Cor e Forma:Solid
    Peso molecular:469.94
  • Shield-1

    CAS:
    <p>Shield-1 is a specific, high-affinity, and cell-permeable ligand for FK506-binding protein 12 (FKBP).Cost-effective and quality-assured.</p>
    Fórmula:C42H56N2O10
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:748.9
  • Tazemetostat

    CAS:
    <p>Tazemetostat (EPZ6438): Oral EZH2 inhibitor, blocks histone H3K27 methylation, potential cancer therapy.</p>
    Fórmula:C34H44N4O4
    Pureza:98.24% - ≥95%
    Cor e Forma:Solid
    Peso molecular:572.74
  • Nerol

    CAS:
    <p>Nerol (Neryl alcohol) is a monoterpene found in many essential oils, such as lemon balm and hop.Nerol can lessened the severity of ouabain-triggered arrhythmias</p>
    Fórmula:C10H18O
    Pureza:98.59%
    Cor e Forma:Colorless Oily Liquid Liquid
    Peso molecular:154.25
  • Ricolinostat

    CAS:
    <p>Ricolinostat (Rocilinostat) is an orally bioavailable, specific inhibitor of histone deacetylase 6 (HDAC6) with potential antineoplastic activity.</p>
    Fórmula:C24H27N5O3
    Pureza:97.17% - 99.76%
    Cor e Forma:Solid
    Peso molecular:433.5
  • BAY 61-3606 HCl

    CAS:
    <p>BAY 61-3606 HCl: a reversible Syk inhibitor, halts mast cell degranulation, cytokines, and sensitizes MCF-7 cells to TRAIL-induced apoptosis.</p>
    Fórmula:C20H19ClN6O3
    Cor e Forma:Solid
    Peso molecular:426.86
  • FB23-2

    CAS:
    <p>FB23-2 is a potent and selective mRNA N6-methyladenosine (m6A) demethylase FTO inhibitor(IC50 : 2.6 μM).</p>
    Fórmula:C18H15Cl2N3O3
    Pureza:97.29% - ≥95%
    Cor e Forma:Solid
    Peso molecular:392.24
  • Phenoxyethanol

    CAS:
    <p>Phenoxyethanol (NSC-1864) is germicidal. It often used together with quaternary ammonium compounds.</p>
    Fórmula:C8H10O2
    Pureza:99.47%
    Cor e Forma:Clear To Practically Clear Colourless Liquid
    Peso molecular:138.16
  • Hederacolchiside A1

    CAS:
    <p>Hederacolchiside A1 exhibits anti-leishmanial and anticancer activities by disrupting cell membranes and inducing apoptosis via the PI3K/Akt/mTOR pathway.</p>
    Fórmula:C47H76O16
    Pureza:98.76% - 99.92%
    Cor e Forma:Solid
    Peso molecular:897.1
  • Calcium dobesilate

    CAS:
    <p>Calcium dobesilate(CaD) has angioprotective properties and protects endothelial cells partly by ameliorating HG induced inflammation.</p>
    Fórmula:C6H5O5SCa0
    Pureza:98.39%
    Cor e Forma:White Or Almost Powder
    Peso molecular:229.2
  • ZYN57939

    CAS:
    <p>ZYN57939 (MTR-106), an RNA polymerase I inhibitor, treats related diseases with a 0.855 μM IC50 against HT-29 cells.</p>
    Fórmula:C28H27N7O2S
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:525.62
  • Cladribine

    CAS:
    <p>Cladribine (2CdA), an adenosine deaminase inhibitor, is utilized in the treatment of lymphoproliferative diseases.</p>
    Fórmula:C10H12ClN5O3
    Pureza:99.58% - >99.99%
    Cor e Forma:White Crystalline Solid
    Peso molecular:285.69
  • Talampanel

    CAS:
    <p>Talampanel (LY-300164), an oral selective AMPA receptor antagonist, exhibits anti-seizure and neuroprotective properties.</p>
    Fórmula:C19H19N3O3
    Pureza:98.3%
    Cor e Forma:Solid
    Peso molecular:337.37
  • Glycochenodeoxycholic acid sodium salt

    CAS:
    <p>GCDCA, a bile acid-glycine salt, is a secondary bile acid from colonic microbes.</p>
    Fórmula:C26H42NNaO5
    Pureza:95.48% - 99.82%
    Cor e Forma:Solid
    Peso molecular:471.61
  • Birinapant

    CAS:
    <p>Birinapant (TL32711) is a synthetic small molecule that is both a peptidomimetic of second mitochondrial-derived activator of caspases (SMAC) and inhibitor of</p>
    Fórmula:C42H56F2N8O6
    Pureza:97.08% - ≥95%
    Cor e Forma:Solid
    Peso molecular:806.94
  • σ1 Receptor antagonist-1

    CAS:
    <p>σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist.</p>
    Fórmula:C21H23NOS
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:337.48
  • Tenovin-6 Hydrochloride

    CAS:
    <p>Tenovin-6 HCl: Inhibits SIRT1 (21µM), SIRT2 (10µM), HDAC8; potent p53 activator.</p>
    Fórmula:C25H35ClN4O2S
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:491.09
  • Azoramide

    CAS:
    <p>Azoramide, a small-molecule modulator, has the antidiabetic activity of unfolded protein response.</p>
    Fórmula:C15H17ClN2OS
    Pureza:99.08% - 99.85%
    Cor e Forma:Solid
    Peso molecular:308.83
  • AZD3759 hydrochloride

    CAS:
    <p>AZD3759 hydrochloride is an oral, CNS-penetrant EGFR inhibitor with IC50s of 0.2/0.3/0.2 nM.</p>
    Fórmula:C22H24Cl2FN5O3
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:496.36
  • Ciprofloxacin hydrochloride monohydrate

    CAS:
    <p>Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) is a fluoroquinolone antibiotic with potent antibacterial activity.</p>
    Fórmula:C17H21ClFN3O4
    Pureza:99.23% - 99.85%
    Cor e Forma:White Or Yellowish Crystalline Powder
    Peso molecular:385.82
  • Tenovin-3

    CAS:
    <p>Tenovin-3 acts as a p53 activator.</p>
    Fórmula:C18H21N3OS
    Pureza:99.72% - ≥95%
    Cor e Forma:Solid
    Peso molecular:327.44
  • A-419259

    CAS:
    <p>A-419259 (RK-20449) is an apoptosis inducer that selectively inhibits the Src family of kinases, including Src,LCK, and Lyn, with an IC50=3 to 9 nM.</p>
    Fórmula:C29H34N6O
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:482.62
  • PKD-IN-1 dihydrochloride (956121-30-5 free base)

    CAS:
    <p>CRT0066101 dihydrochloride is an inhibitor of PKD.</p>
    Fórmula:C18H21Cl3N4O
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:415.75
  • Tauroursodeoxycholate

    CAS:
    <p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>
    Fórmula:C26H45NO6S
    Pureza:98.77% - 99.93%
    Cor e Forma:White Solid
    Peso molecular:499.7
  • PEAQX

    CAS:
    <p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>
    Fórmula:C17H17BrN3O5P
    Pureza:98% - 99.9%
    Cor e Forma:Solid
    Peso molecular:454.21
  • AR42

    CAS:
    <p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>
    Fórmula:C18H20N2O3
    Pureza:98.46% - 98.96%
    Cor e Forma:Solid
    Peso molecular:312.36
  • Emricasan

    CAS:
    <p>Emricasan (IDN-6556) is a pan-caspase inhibitor with irreversible properties.</p>
    Fórmula:C26H27F4N3O7
    Pureza:98.13% - 99%
    Cor e Forma:Solid
    Peso molecular:569.5
  • Aloperine

    CAS:
    <p>Aloperine exhibits anti-inflammatory, antibacterial, antiviral, and anti-tumor properties.</p>
    Fórmula:C15H24N2
    Pureza:98% - 99.88%
    Cor e Forma:Yellow Crystalline Powder
    Peso molecular:232.36
  • 1400W dihydrochloride

    CAS:
    <p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>
    Fórmula:C10H17Cl2N3
    Pureza:98% - 99.94%
    Cor e Forma:Solid
    Peso molecular:250.17
  • Bilobalide

    CAS:
    <p>Bilobalide ((-)-Bilobalide), a bioactive from Gingko Biloba, is active on hypoxia-induced alterations.</p>
    Fórmula:C15H18O8
    Pureza:98.81% - 99.92%
    Cor e Forma:White Solid
    Peso molecular:326.3
  • Ipatasertib

    CAS:
    <p>Ipatasertib (GDC-0068) is a selective, ATP-competitive pan-Akt inhibitor that can lead to p53-independent PUMA activation.Cost-effective and quality-assured.</p>
    Fórmula:C24H32ClN5O2
    Pureza:98.28% - 99.21%
    Cor e Forma:Solid
    Peso molecular:458
  • Nω-Hydroxy-nor-L-Arginine Dihydrochloride

    CAS:
    <p>Nω-Hydroxy-nor-L-Arginine Dihydrochloride is a competitive and reversible inhibitor of arginase</p>
    Fórmula:C5H14Cl2N4O3
    Pureza:99.12% - 99.84%
    Cor e Forma:Solid
    Peso molecular:249.10
  • Tetrahydroxyquinone monohydrate

    CAS:
    <p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>
    Fórmula:C6H6O7
    Cor e Forma:Solid
    Peso molecular:190.11
  • Alda-1

    CAS:
    <p>Alda-1 activates ALDH2*1 and ALDH2*2, permeates cells, and targets mitochondrial aldehyde dehydrogenase 2.</p>
    Fórmula:C15H11Cl2NO3
    Pureza:98.5% - 99.63%
    Cor e Forma:Solid
    Peso molecular:324.16
  • Eltrombopag Olamine

    CAS:
    <p>Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin</p>
    Fórmula:C29H36N6O6
    Pureza:99.59% - 99.89%
    Cor e Forma:Solid
    Peso molecular:564.63
  • HA15

    CAS:
    <p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>
    Fórmula:C23H22N4O3S2
    Pureza:99.77% - 99.86%
    Cor e Forma:Solid
    Peso molecular:466.58
  • Thalidomide-O-amido-C6-NH2 hydrochloride

    CAS:
    <p>Thalidomide-O-amido-C6-NH2 HCl, a cereblon ligand-linker for PROTAC synthesis.</p>
    Fórmula:C21H27ClN4O6
    Pureza:97.33%
    Cor e Forma:Solid
    Peso molecular:466.915
  • Dacarbazine citrate

    CAS:
    <p>Dacarbazine citrate treats lymphatic cancers, malignant melanoma, islet cell carcinoma, and soft tissue sarcoma.</p>
    Fórmula:C12H18N6O8
    Cor e Forma:Solid
    Peso molecular:374.31
  • FOXO4-DRI acetate


    <p>FOXO4-DRI acetate is a bioactive chemical.</p>
    Fórmula:C36H64N14O14S
    Pureza:99.10%
    Cor e Forma:Solid
    Peso molecular:5358.06
  • Periplocin

    CAS:
    <p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>
    Fórmula:C36H56O13
    Pureza:99.66% - 99.74%
    Cor e Forma:Solid
    Peso molecular:696.82
  • TrxR1-IN-B19

    CAS:
    <p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>
    Fórmula:C21H22O5
    Pureza:98.6%
    Cor e Forma:Solid
    Peso molecular:354.4
  • Thalidomide-O-amido-C3-NH2 TFA

    CAS:
    <p>Thalidomide-based E3 ligase linker for PROTAC tech; cereblon ligand conjugate.</p>
    Fórmula:C20H21F3N4O8
    Pureza:98.47%
    Cor e Forma:Solid
    Peso molecular:502.4
  • Methoxychlor

    CAS:
    <p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>
    Fórmula:C16H15Cl3O2
    Pureza:98.82% - ≥95%
    Cor e Forma:Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment If
    Peso molecular:345.65
  • Thalidomide-NH-C4-NH-Boc

    CAS:
    <p>Thalidomide-NH-C4-NH-Boc is a cereblon-based E3 ligase ligand-linker for PROTACs.</p>
    Fórmula:C22H28N4O6
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:444.48
  • Bigelovin

    CAS:
    <p>Bigelovin: RXRα agonist, inhibits mTOR via ROS, induces apoptosis/autophagy, anti-tumor sesquiterpene from Inula sp.</p>
    Fórmula:C17H20O5
    Pureza:99.61% - 99.72%
    Cor e Forma:Solid
    Peso molecular:304.34
  • Thalidomide-propargyl

    CAS:
    <p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>
    Fórmula:C16H12N2O5
    Pureza:95.14%
    Cor e Forma:Solid
    Peso molecular:312.28
  • Thalidomide-NH-C6-NH2 hydrochloride

    CAS:
    <p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>
    Fórmula:C19H25ClN4O4
    Pureza:99.27%
    Cor e Forma:Solid
    Peso molecular:408.88
  • Benidipine hydrochloride

    CAS:
    <p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>
    Fórmula:C28H32ClN3O6
    Pureza:99.80%
    Cor e Forma:Solid
    Peso molecular:542.03
  • (ZE)-SU9516

    CAS:
    <p>(ZE)-SU9516 is a selectively potent ATP-competitive inhibitor of CDKs.</p>
    Fórmula:C13H11N3O2
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:241.25
  • Diclofenac Potassium

    CAS:
    <p>Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.</p>
    Fórmula:C14H10Cl2KNO2
    Pureza:99.51%
    Cor e Forma:White To Yellowish Crystalline Powder
    Peso molecular:334.24
  • Pomolic acid

    CAS:
    <p>Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-</p>
    Fórmula:C30H48O4
    Pureza:96.84% - 99.79%
    Cor e Forma:Solid
    Peso molecular:472.7
  • Cilengitide

    CAS:
    <p>Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.</p>
    Fórmula:C27H40N8O7
    Pureza:98% - 99.8%
    Cor e Forma:Solid
    Peso molecular:588.66
  • Desmorpholinyl Navitoclax-NH-Me

    CAS:
    <p>Desmorpholinyl Navitoclax-NH-Me (Desmorpholinyl ABT-263-NH-Me) is a Bcl-xL inhibitor, which can be employed alongside a CRBN ligand to synthesize XZ739, a</p>
    Fórmula:C44H51ClF3N5O5S3
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:918.55
  • Lercanidipine hydrochloride

    CAS:
    <p>Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class.</p>
    Fórmula:C36H41N3O6·HCl
    Pureza:99.86% - 99.91%
    Cor e Forma:Pale-Yellow Powder
    Peso molecular:648.19
  • 4-Oxofenretinide

    CAS:
    <p>4-Oxofenretinide (3-Keto fenretinide) , a recently identified fenretinide metabolite, induces marked G2-M cell cycle arrest and apoptosis.</p>
    Fórmula:C26H31NO3
    Pureza:96.89%
    Cor e Forma:Solid
    Peso molecular:405.53
  • Ibuprofen Lysine

    CAS:
    <p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>
    Fórmula:C19H32N2O4
    Pureza:99.26%
    Cor e Forma:Coa
    Peso molecular:352.47
  • RA375

    CAS:
    <p>RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than RA190 due to nitro rings and chloroacetamide.</p>
    Fórmula:C30H25ClN4O7
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:588.99
  • SRT 2183

    CAS:
    <p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>
    Fórmula:C27H24N4O2S
    Pureza:97.86%
    Cor e Forma:Solid
    Peso molecular:468.57
  • Deguelin

    CAS:
    <p>Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.</p>
    Fórmula:C23H22O6
    Pureza:96.39% - 99.29%
    Cor e Forma:Solid
    Peso molecular:394.42