
Apoptose
Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.
Subcategorias de "Apoptose"
- ASK(6 produtos)
- BCL(11 produtos)
- Caspase(125 produtos)
- FOXO1(3 produtos)
- IAP(66 produtos)
- Mdm2(12 produtos)
- PD-1/PD-L1(125 produtos)
- PDK(9 produtos)
- PERK(25 produtos)
- Serina/treonina quinase(15 produtos)
- Survivina(13 produtos)
- TNF(92 produtos)
- c-RET(51 produtos)
- p53(62 produtos)
Exibir 6 mais subcategorias
Foram encontrados 5592 produtos de "Apoptose"
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Obatoclax Mesylate
CAS:<p>Obatoclax Mesylate (GX15-070) is a Bcl-2 antagonist (Ki: 0.22 μM) and can induce apoptosis with up-regulation of Bim, induced cytochrome c release, and</p>Fórmula:C20H19N3O·CH4O3SPureza:99.58% - 99.88%Cor e Forma:SolidPeso molecular:413.49Ibandronate sodium monohydrate
CAS:<p>Ibandronate sodium monohydrate (BM-210955) is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.</p>Fórmula:C9H24NNaO8P2Pureza:99.62%Cor e Forma:White Crystalline PowderPeso molecular:359.23Neobavaisoflavone
CAS:<p>Neobavaisoflavone: DNA polymerase inhibitor, potential for treating bone loss, anti-inflammatory, reduces ROS, RNS, cytokines in macrophages.</p>Fórmula:C20H18O4Pureza:99.31% - 99.87%Cor e Forma:SolidPeso molecular:322.35RGX-202
CAS:<p>RGX-202 (β-GPA) is an orally active inhibitor of the SLC6A8 transport protein. RGX-202 is a creatine analog that alters skeletal muscle energy expenditure.</p>Fórmula:C4H9N3O2Pureza:99.67% - 99.8%Cor e Forma:SolidPeso molecular:131.13PD173955
CAS:<p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>Fórmula:C21H16Cl2N4OSPureza:98.52% - 98.99%Cor e Forma:SolidPeso molecular:443.35Nobiletin
CAS:<p>Nobiletin: a citrus-derived flavone with anti-inflammatory and anti-cancer properties; water-insoluble, very weak acid.</p>Fórmula:C21H22O8Pureza:98.65% - 99.76%Cor e Forma:SolidPeso molecular:402.39Bioymifi
CAS:<p>Bioymifi (DR5 Activator), a novel TRAIL activator, binds to DR5's ECD, inducing DR5 aggregation and stimulating cell apoptosis. Cost-effective and quality-assured.</p>Fórmula:C22H12BrN3O4SPureza:98% - 99.79%Cor e Forma:SolidPeso molecular:494.32Oncrasin-1
CAS:<p>Oncrasin 1 is a potent inhibitor of anticancer that kills various human lung cancer cells with K-Ras mutations at low or submicromolar concentrations</p>Fórmula:C16H12ClNOPureza:99.75%Cor e Forma:SolidPeso molecular:269.73Rilmenidine hemifumarate
CAS:<p>Rilmenidine hemifumarate (S-3341 hemifumarate) is an I1 imidazoline receptor and α2-adrenergic receptor agonist that induces autophagy.</p>Fórmula:C10H16N2OC4H4O4Pureza:98.14%Cor e Forma:SolidPeso molecular:238.28CA-5f
CAS:<p>CA-5f is a potent late-stage macroautophagy/autophagy inhibitor via inhibiting autophagosome-lysosome fusion.</p>Fórmula:C24H24N2O3Pureza:99.69%Cor e Forma:SolidPeso molecular:388.462,5-dimethyl Celecoxib
CAS:<p>2,5-dimethyl Celecoxib, a derivative targeting mPGES-1, inhibits PGE2 synthesis in inflammation.</p>Fórmula:C18H16F3N3O2SPureza:99.85%Cor e Forma:SolidPeso molecular:395.4Pinoresinol
CAS:<p>Pinoresinol ((+)-Pinoresinol) has antiinflammatory, hepatoprotective, and fungicidal activities, it can protect pial microcirculation from I-reperfusion injury</p>Fórmula:C20H22O6Pureza:98.67%Cor e Forma:SolidPeso molecular:358.39BX-912
CAS:<p>BX-912 inhibits PDK1 with IC50 of 12 nM; over 10x more selective versus C-Kit, EGFR, PKA, PKC.</p>Fórmula:C20H23BrN8OPureza:98.29% - 99.34%Cor e Forma:SolidPeso molecular:471.35CCT128930 hydrochloride
CAS:<p>CCT128930 hydrochloride: Potent AKT inhibitor (IC50=6 nM), 28x selective over PKA, 20x over p70S6K, induces cell cycle arrest & DNA damage.</p>Fórmula:C18H21Cl2N5Pureza:98.55%Cor e Forma:SolidPeso molecular:378.3L-Asparaginase
CAS:<p>L-Asparaginase, an enzyme for acute lymphoblastic leukemia treatment, is administered via injection.</p>Fórmula:NAPureza:97%Cor e Forma:SolidPeso molecular:N/AElesclomol
CAS:<p>Elesclomol (STA-4783) is an oxidative stress inducer and a highly lipophilic copper ion carrier.</p>Fórmula:C19H20N4O2S2Pureza:97.17% - 99.51%Cor e Forma:SolidPeso molecular:400.52HO-3867
CAS:<p>HO-3867, an analog of curcumin, is a sspecific STAT3 inhibitor.</p>Fórmula:C28H30F2N2O2Pureza:91.18% - 99.21%Cor e Forma:SolidPeso molecular:464.55LRRK2-IN-1
CAS:<p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>Fórmula:C31H38N8O3Pureza:98% - 98.82%Cor e Forma:SolidPeso molecular:570.69S-trityl-L-Cysteine
CAS:<p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>Fórmula:C22H21NO2SPureza:97.02%Cor e Forma:Almost White To Light Yellow Granular PowderPeso molecular:363.47NSC 95397
CAS:<p>NSC 95397 is a potent inhibitor of Cdc25 dual specificity phosphatase(Ki of 32, 96, and 40 nM for Cdc25A, Cdc25B, and Cdc25C, respectively).</p>Fórmula:C14H14O4S2Pureza:98.66%Cor e Forma:SolidPeso molecular:310.39SKI II
CAS:<p>SKI II is a selective non-ATP S1P receptor inhibitor with an IC50 of 0.5 μM; it doesn't inhibit PKCα, PI3K, or ERK2.</p>Fórmula:C15H11ClN2OSPureza:99.34% - 99.93%Cor e Forma:SolidPeso molecular:302.78STF-118804
CAS:<p>STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 <10 nM.</p>Fórmula:C25H23N3O4SPureza:98.66%Cor e Forma:SolidPeso molecular:461.53Pracinostat
CAS:<p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>Fórmula:C20H30N4O2Pureza:99.15% - 99.67%Cor e Forma:SolidPeso molecular:358.48SKI-178
CAS:<p>SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM.</p>Fórmula:C21H22N4O4Pureza:97.09%Cor e Forma:SolidPeso molecular:394.42Clodronate disodium tetrahydrate
CAS:<p>Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.</p>Fórmula:CH10Cl2Na2O10P2Pureza:98%Cor e Forma:SolidPeso molecular:360.92CM-272
CAS:<p>CM-272 is a dual G9a/DNA methyltransferases (DNMTs) inhibitor.</p>Fórmula:C28H38N4O3Pureza:97.83%Cor e Forma:SolidPeso molecular:478.63Trifloxystrobin
CAS:<p>Trifloxystrobin is a fungicide against R. solani in sugar beets with EC50s: 23.0 μg/L for Daphnia neonates, 1.7 μg/L for embryos.</p>Fórmula:C20H19F3N2O4Pureza:99.49%Cor e Forma:SolidPeso molecular:408.37JKE-1674
CAS:<p>JKE-1674 is an orally active glutathione peroxidase 4 (GPX4) inhibitor and the active metabolite of ML-210.Cost-effective and quality-assured.</p>Fórmula:C20H20Cl2N4O4Pureza:98.02% - 98.4%Cor e Forma:SolidPeso molecular:451.3QNZ
CAS:<p>QNZ (EVP4593) (EVP4593) is an effective inhibitor of NF-κB activation and TNF-α production. The IC50 of QNZ for NF-κB and TNF-α is11 nM and 7 nM, respectively.</p>Fórmula:C22H20N4OPureza:99.17% - 99.18%Cor e Forma:White SolidPeso molecular:356.42Thalidomide-O-C4-NH2 hydrochloride
CAS:<p>Thalidomide-linker 9: a cereblon ligand, E3 ligase conjugate for PROTAC tech.</p>Fórmula:C17H20ClN3O5Pureza:98.33%Cor e Forma:SolidPeso molecular:381.81Laquinimod sodium
CAS:<p>Laquinimod (ABR-215062) sodium is an oral agent for MS, halting neurodegeneration and inflammation.</p>Fórmula:C19H16ClN2NaO3Cor e Forma:SolidPeso molecular:378.79Thalidomide-PEG4-Propargyl
CAS:<p>Thalidomide-PEG4-Propargyl is a synthetic E3 ligase ligand for PROTAC with a cereblon ligand and linker.</p>Fórmula:C24H28N2O9Pureza:97.46%Cor e Forma:SolidPeso molecular:488.49SKLB-163
CAS:<p>SKLB-163 acts by downregulating RhoGDI, activating JNK-1 signaling pathway and caspase-3, and reducing phosphorylated Akt and p44/42 MAPK.</p>Fórmula:C18H16ClN3O2S2Pureza:99.23%Cor e Forma:SolidPeso molecular:405.92Mitoxantrone diacetate
CAS:<p>Mitoxantrone diacetate hinders topoisomerase II & PKC, fights tumors & orthopoxviruses (IC50: 8.5μM, EC50: 0.25-0.8μM).</p>Fórmula:C26H36N4O10Cor e Forma:SolidPeso molecular:564.592ONO-8130
CAS:<p>ONO-8130 is an orally available antagonist of EP1 receptor.</p>Fórmula:C25H28N2O5S2Pureza:97.82%Cor e Forma:SolidPeso molecular:500.63Tofacitinib Citrate
CAS:<p>Tofacitinib Citrate (CP-690550 citrate) is a a potent, cell-permeable inhibitor of JAK1/2/3 (IC50s: 1/20/112 nM).</p>Fórmula:C22H28N6O8Pureza:99.19% - 99.75%Cor e Forma:SolidPeso molecular:504.49Benzoylpaeoniflorin
CAS:<p>1. Benzoylpaeoniflorin is active against cyclooxygenase-1 and cyclooxygenase-2 enzymes.</p>Fórmula:C30H32O12Pureza:95.86% - 97.28%Cor e Forma:SolidPeso molecular:584.57Cinchonine monohydrochloride hydrate
CAS:<p>Cinchonine monohydrochloride hydrate: natural antimalarial, inhibits platelet aggregation & cancer cell growth, blocks fat cell formation.</p>Fórmula:C19H25ClN2O2Cor e Forma:SolidPeso molecular:348.87C5 Lenalidomide
CAS:<p>C5 Lenalidomide is an chemical weith inconclusive biological activity.</p>Fórmula:C13H13N3O3Pureza:99.4%Cor e Forma:SolidPeso molecular:259.26Kinetin riboside
CAS:<p>Kinetin riboside (N6-Furfuryladenosine) can induce apoptosis in cancer cells. It inhibits the proliferation of HCT-15 cells(IC50 of 2.5 μM)</p>Fórmula:C15H17N5O5Pureza:98.17%Cor e Forma:White SolidPeso molecular:347.33Dacomitinib
CAS:<p>Dacomitinib (PF299) is an oral selective inhibitor of EGFR, ERBB2, ERBB4 with IC50s: 6, 45.7, 73.7 nM.</p>Fórmula:C24H25ClFN5O2Pureza:99.4% - 99.72%Cor e Forma:SolidPeso molecular:469.94Shield-1
CAS:<p>Shield-1 is a specific, high-affinity, and cell-permeable ligand for FK506-binding protein 12 (FKBP).Cost-effective and quality-assured.</p>Fórmula:C42H56N2O10Pureza:99.08%Cor e Forma:SolidPeso molecular:748.9Tazemetostat
CAS:<p>Tazemetostat (EPZ6438): Oral EZH2 inhibitor, blocks histone H3K27 methylation, potential cancer therapy.</p>Fórmula:C34H44N4O4Pureza:98.24% - ≥95%Cor e Forma:SolidPeso molecular:572.74Nerol
CAS:<p>Nerol (Neryl alcohol) is a monoterpene found in many essential oils, such as lemon balm and hop.Nerol can lessened the severity of ouabain-triggered arrhythmias</p>Fórmula:C10H18OPureza:98.59%Cor e Forma:Colorless Oily Liquid LiquidPeso molecular:154.25Ricolinostat
CAS:<p>Ricolinostat (Rocilinostat) is an orally bioavailable, specific inhibitor of histone deacetylase 6 (HDAC6) with potential antineoplastic activity.</p>Fórmula:C24H27N5O3Pureza:97.17% - 99.76%Cor e Forma:SolidPeso molecular:433.5BAY 61-3606 HCl
CAS:<p>BAY 61-3606 HCl: a reversible Syk inhibitor, halts mast cell degranulation, cytokines, and sensitizes MCF-7 cells to TRAIL-induced apoptosis.</p>Fórmula:C20H19ClN6O3Cor e Forma:SolidPeso molecular:426.86FB23-2
CAS:<p>FB23-2 is a potent and selective mRNA N6-methyladenosine (m6A) demethylase FTO inhibitor(IC50 : 2.6 μM).</p>Fórmula:C18H15Cl2N3O3Pureza:97.29% - ≥95%Cor e Forma:SolidPeso molecular:392.24Phenoxyethanol
CAS:<p>Phenoxyethanol (NSC-1864) is germicidal. It often used together with quaternary ammonium compounds.</p>Fórmula:C8H10O2Pureza:99.47%Cor e Forma:Clear To Practically Clear Colourless LiquidPeso molecular:138.16Hederacolchiside A1
CAS:<p>Hederacolchiside A1 exhibits anti-leishmanial and anticancer activities by disrupting cell membranes and inducing apoptosis via the PI3K/Akt/mTOR pathway.</p>Fórmula:C47H76O16Pureza:98.76% - 99.92%Cor e Forma:SolidPeso molecular:897.1Calcium dobesilate
CAS:<p>Calcium dobesilate(CaD) has angioprotective properties and protects endothelial cells partly by ameliorating HG induced inflammation.</p>Fórmula:C6H5O5SCa0Pureza:98.39%Cor e Forma:White Or Almost PowderPeso molecular:229.2ZYN57939
CAS:<p>ZYN57939 (MTR-106), an RNA polymerase I inhibitor, treats related diseases with a 0.855 μM IC50 against HT-29 cells.</p>Fórmula:C28H27N7O2SPureza:99.81%Cor e Forma:SolidPeso molecular:525.62Cladribine
CAS:<p>Cladribine (2CdA), an adenosine deaminase inhibitor, is utilized in the treatment of lymphoproliferative diseases.</p>Fórmula:C10H12ClN5O3Pureza:99.58% - >99.99%Cor e Forma:White Crystalline SolidPeso molecular:285.69Talampanel
CAS:<p>Talampanel (LY-300164), an oral selective AMPA receptor antagonist, exhibits anti-seizure and neuroprotective properties.</p>Fórmula:C19H19N3O3Pureza:98.3%Cor e Forma:SolidPeso molecular:337.37Glycochenodeoxycholic acid sodium salt
CAS:<p>GCDCA, a bile acid-glycine salt, is a secondary bile acid from colonic microbes.</p>Fórmula:C26H42NNaO5Pureza:95.48% - 99.82%Cor e Forma:SolidPeso molecular:471.61Birinapant
CAS:<p>Birinapant (TL32711) is a synthetic small molecule that is both a peptidomimetic of second mitochondrial-derived activator of caspases (SMAC) and inhibitor of</p>Fórmula:C42H56F2N8O6Pureza:97.08% - ≥95%Cor e Forma:SolidPeso molecular:806.94σ1 Receptor antagonist-1
CAS:<p>σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist.</p>Fórmula:C21H23NOSPureza:99.8%Cor e Forma:SolidPeso molecular:337.48Tenovin-6 Hydrochloride
CAS:<p>Tenovin-6 HCl: Inhibits SIRT1 (21µM), SIRT2 (10µM), HDAC8; potent p53 activator.</p>Fórmula:C25H35ClN4O2SPureza:99.36%Cor e Forma:SolidPeso molecular:491.09Azoramide
CAS:<p>Azoramide, a small-molecule modulator, has the antidiabetic activity of unfolded protein response.</p>Fórmula:C15H17ClN2OSPureza:99.08% - 99.85%Cor e Forma:SolidPeso molecular:308.83AZD3759 hydrochloride
CAS:<p>AZD3759 hydrochloride is an oral, CNS-penetrant EGFR inhibitor with IC50s of 0.2/0.3/0.2 nM.</p>Fórmula:C22H24Cl2FN5O3Pureza:99.62%Cor e Forma:SolidPeso molecular:496.36Ciprofloxacin hydrochloride monohydrate
CAS:<p>Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) is a fluoroquinolone antibiotic with potent antibacterial activity.</p>Fórmula:C17H21ClFN3O4Pureza:99.23% - 99.85%Cor e Forma:White Or Yellowish Crystalline PowderPeso molecular:385.82Tenovin-3
CAS:<p>Tenovin-3 acts as a p53 activator.</p>Fórmula:C18H21N3OSPureza:99.72% - ≥95%Cor e Forma:SolidPeso molecular:327.44A-419259
CAS:<p>A-419259 (RK-20449) is an apoptosis inducer that selectively inhibits the Src family of kinases, including Src,LCK, and Lyn, with an IC50=3 to 9 nM.</p>Fórmula:C29H34N6OPureza:99.48%Cor e Forma:SolidPeso molecular:482.62PKD-IN-1 dihydrochloride (956121-30-5 free base)
CAS:<p>CRT0066101 dihydrochloride is an inhibitor of PKD.</p>Fórmula:C18H21Cl3N4OPureza:99.5%Cor e Forma:SolidPeso molecular:415.75Tauroursodeoxycholate
CAS:<p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>Fórmula:C26H45NO6SPureza:98.77% - 99.93%Cor e Forma:White SolidPeso molecular:499.7PEAQX
CAS:<p>PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so 1A/2B (IC50: 29,600 nM).</p>Fórmula:C17H17BrN3O5PPureza:98% - 99.9%Cor e Forma:SolidPeso molecular:454.21AR42
CAS:<p>AR42 (OSU-HDAC42) is an HDAC inhibitor (IC50: 30 nM).</p>Fórmula:C18H20N2O3Pureza:98.46% - 98.96%Cor e Forma:SolidPeso molecular:312.36Emricasan
CAS:<p>Emricasan (IDN-6556) is a pan-caspase inhibitor with irreversible properties.</p>Fórmula:C26H27F4N3O7Pureza:98.13% - 99%Cor e Forma:SolidPeso molecular:569.5Aloperine
CAS:<p>Aloperine exhibits anti-inflammatory, antibacterial, antiviral, and anti-tumor properties.</p>Fórmula:C15H24N2Pureza:98% - 99.88%Cor e Forma:Yellow Crystalline PowderPeso molecular:232.361400W dihydrochloride
CAS:<p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>Fórmula:C10H17Cl2N3Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:250.17Bilobalide
CAS:<p>Bilobalide ((-)-Bilobalide), a bioactive from Gingko Biloba, is active on hypoxia-induced alterations.</p>Fórmula:C15H18O8Pureza:98.81% - 99.92%Cor e Forma:White SolidPeso molecular:326.3Ipatasertib
CAS:<p>Ipatasertib (GDC-0068) is a selective, ATP-competitive pan-Akt inhibitor that can lead to p53-independent PUMA activation.Cost-effective and quality-assured.</p>Fórmula:C24H32ClN5O2Pureza:98.28% - 99.21%Cor e Forma:SolidPeso molecular:458Nω-Hydroxy-nor-L-Arginine Dihydrochloride
CAS:<p>Nω-Hydroxy-nor-L-Arginine Dihydrochloride is a competitive and reversible inhibitor of arginase</p>Fórmula:C5H14Cl2N4O3Pureza:99.12% - 99.84%Cor e Forma:SolidPeso molecular:249.10Tetrahydroxyquinone monohydrate
CAS:<p>Anticataract compound; redox-active; forms ROS via semiquinone radical cycle.</p>Fórmula:C6H6O7Cor e Forma:SolidPeso molecular:190.11Alda-1
CAS:<p>Alda-1 activates ALDH2*1 and ALDH2*2, permeates cells, and targets mitochondrial aldehyde dehydrogenase 2.</p>Fórmula:C15H11Cl2NO3Pureza:98.5% - 99.63%Cor e Forma:SolidPeso molecular:324.16Eltrombopag Olamine
CAS:<p>Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin</p>Fórmula:C29H36N6O6Pureza:99.59% - 99.89%Cor e Forma:SolidPeso molecular:564.63HA15
CAS:<p>HA15 targets BiP/GRP78/HSPA5, showing anti-cancer effects on all tested melanoma cells, resistant or patient-derived.</p>Fórmula:C23H22N4O3S2Pureza:99.77% - 99.86%Cor e Forma:SolidPeso molecular:466.58Thalidomide-O-amido-C6-NH2 hydrochloride
CAS:<p>Thalidomide-O-amido-C6-NH2 HCl, a cereblon ligand-linker for PROTAC synthesis.</p>Fórmula:C21H27ClN4O6Pureza:97.33%Cor e Forma:SolidPeso molecular:466.915Dacarbazine citrate
CAS:<p>Dacarbazine citrate treats lymphatic cancers, malignant melanoma, islet cell carcinoma, and soft tissue sarcoma.</p>Fórmula:C12H18N6O8Cor e Forma:SolidPeso molecular:374.31FOXO4-DRI acetate
<p>FOXO4-DRI acetate is a bioactive chemical.</p>Fórmula:C36H64N14O14SPureza:99.10%Cor e Forma:SolidPeso molecular:5358.06Periplocin
CAS:<p>Periplocin fights lung cancer, induces apoptosis, stunts growth via beta-catenin/Tcf, and treats rheumatoid arthritis/traditional ailments.</p>Fórmula:C36H56O13Pureza:99.66% - 99.74%Cor e Forma:SolidPeso molecular:696.82TrxR1-IN-B19
CAS:<p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>Fórmula:C21H22O5Pureza:98.6%Cor e Forma:SolidPeso molecular:354.4Thalidomide-O-amido-C3-NH2 TFA
CAS:<p>Thalidomide-based E3 ligase linker for PROTAC tech; cereblon ligand conjugate.</p>Fórmula:C20H21F3N4O8Pureza:98.47%Cor e Forma:SolidPeso molecular:502.4Methoxychlor
CAS:<p>Methoxychlor, an organochlorine pesticide, is thought to be an endocrine disrupter that affects Ca2 homeostasis and cell viability in different cell models.</p>Fórmula:C16H15Cl3O2Pureza:98.82% - ≥95%Cor e Forma:Colorless Crystals (Technical Grey Powder) To The Environment Immediate Steps Should Be Taken To Limit Its Spread To The Environment IfPeso molecular:345.65Thalidomide-NH-C4-NH-Boc
CAS:<p>Thalidomide-NH-C4-NH-Boc is a cereblon-based E3 ligase ligand-linker for PROTACs.</p>Fórmula:C22H28N4O6Pureza:98.87%Cor e Forma:SolidPeso molecular:444.48Bigelovin
CAS:<p>Bigelovin: RXRα agonist, inhibits mTOR via ROS, induces apoptosis/autophagy, anti-tumor sesquiterpene from Inula sp.</p>Fórmula:C17H20O5Pureza:99.61% - 99.72%Cor e Forma:SolidPeso molecular:304.34Thalidomide-propargyl
CAS:<p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>Fórmula:C16H12N2O5Pureza:95.14%Cor e Forma:SolidPeso molecular:312.28Thalidomide-NH-C6-NH2 hydrochloride
CAS:<p>Pomalidomide-C6-NH2 HCl is a synthetic conjugate for PROTAC, combining CRBN ligand and linker.</p>Fórmula:C19H25ClN4O4Pureza:99.27%Cor e Forma:SolidPeso molecular:408.88Benidipine hydrochloride
CAS:<p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>Fórmula:C28H32ClN3O6Pureza:99.80%Cor e Forma:SolidPeso molecular:542.03(ZE)-SU9516
CAS:<p>(ZE)-SU9516 is a selectively potent ATP-competitive inhibitor of CDKs.</p>Fórmula:C13H11N3O2Pureza:99.59%Cor e Forma:SolidPeso molecular:241.25Diclofenac Potassium
CAS:<p>Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.</p>Fórmula:C14H10Cl2KNO2Pureza:99.51%Cor e Forma:White To Yellowish Crystalline PowderPeso molecular:334.24Pomolic acid
CAS:<p>Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-</p>Fórmula:C30H48O4Pureza:96.84% - 99.79%Cor e Forma:SolidPeso molecular:472.7Cilengitide
CAS:<p>Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.</p>Fórmula:C27H40N8O7Pureza:98% - 99.8%Cor e Forma:SolidPeso molecular:588.66Desmorpholinyl Navitoclax-NH-Me
CAS:<p>Desmorpholinyl Navitoclax-NH-Me (Desmorpholinyl ABT-263-NH-Me) is a Bcl-xL inhibitor, which can be employed alongside a CRBN ligand to synthesize XZ739, a</p>Fórmula:C44H51ClF3N5O5S3Pureza:99.87%Cor e Forma:SolidPeso molecular:918.55Lercanidipine hydrochloride
CAS:<p>Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class.</p>Fórmula:C36H41N3O6·HClPureza:99.86% - 99.91%Cor e Forma:Pale-Yellow PowderPeso molecular:648.194-Oxofenretinide
CAS:<p>4-Oxofenretinide (3-Keto fenretinide) , a recently identified fenretinide metabolite, induces marked G2-M cell cycle arrest and apoptosis.</p>Fórmula:C26H31NO3Pureza:96.89%Cor e Forma:SolidPeso molecular:405.53Ibuprofen Lysine
CAS:<p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>Fórmula:C19H32N2O4Pureza:99.26%Cor e Forma:CoaPeso molecular:352.47RA375
CAS:<p>RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than RA190 due to nitro rings and chloroacetamide.</p>Fórmula:C30H25ClN4O7Pureza:99.56%Cor e Forma:SolidPeso molecular:588.99SRT 2183
CAS:<p>SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).</p>Fórmula:C27H24N4O2SPureza:97.86%Cor e Forma:SolidPeso molecular:468.57Deguelin
CAS:<p>Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.</p>Fórmula:C23H22O6Pureza:96.39% - 99.29%Cor e Forma:SolidPeso molecular:394.42
