Receptor CGRP
Os receptores de CGRP estão envolvidos na transmissão da dor e na regulação do fluxo sanguíneo. O CGRP é um neuropeptídeo que desempenha um papel crítico na fisiopatologia da enxaqueca, dilatando os vasos sanguíneos e modulando as vias de sinalização da dor. Alvejar os receptores de CGRP tornou-se uma abordagem promissora no desenvolvimento de terapias para enxaqueca. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de CGRP para apoiar sua pesquisa em manejo da dor, neurobiologia e saúde vascular.
Foram encontrados 51 produtos de "Receptor CGRP"
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Erenumab
CAS:<p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>Pureza:99.43% (SEC-HPLC) - > 95%Cor e Forma:LiquidPeso molecular:146.2 kDaPHM-27 (human) acetate
<p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>Fórmula:C137H215F3N34O42SPureza:99.20%Cor e Forma:SoildPeso molecular:3099.44Vazegepant
CAS:<p>Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.</p>Fórmula:C36H46N8O3Pureza:98.61%Cor e Forma:SolidPeso molecular:638.80(3R,5R,6S)-Atogepant
<p>(3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.</p>Fórmula:C29H23F6N5O3Cor e Forma:SolidPeso molecular:603.52PHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Fórmula:C135H214N34O40SPureza:98%Cor e Forma:SolidPeso molecular:2985.44Adrenomedullin (AM) (22-52), human TFA
<p>Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.</p>Fórmula:C161H253N46F3O50Pureza:98%Cor e Forma:SolidPeso molecular:3690.06Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:<p>CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.</p>Fórmula:C163H267N51O50S2Pureza:98%Cor e Forma:SolidPeso molecular:3805.31Adrenomedullin (11-50), rat
CAS:<p>Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.</p>Fórmula:C194H304N58O59S4Pureza:98%Cor e Forma:SolidPeso molecular:4521.17HTL22562
CAS:<p>HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.</p>Fórmula:C40H49N11O5Cor e Forma:SolidPeso molecular:763.904α-CGRP(human)
CAS:<p>Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.</p>Fórmula:C163H267N51O49S2Pureza:98%Cor e Forma:SolidPeso molecular:3789.33Adrenomedullin (16-31), human
CAS:<p>Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).</p>Fórmula:C82H129N25O21S2Pureza:98%Cor e Forma:SolidPeso molecular:1865.19Cagrilintide
CAS:<p>Cagrilintide: a long-acting amylin analogue, potential obesity treatment, reduces appetite and weight.</p>Fórmula:C194H312N54O59S2Cor e Forma:SolidPeso molecular:4409.01α-CGRP(human) TFA
<p>α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as a</p>Fórmula:C165H268F3N51O51S2Cor e Forma:SolidPeso molecular:3903.33Adrenomedullin (16-31), human TFA
<p>Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.</p>Fórmula:C84H130F3N25O23S2Cor e Forma:SolidPeso molecular:1979.21Adrenotensin (human)
CAS:<p>Adrenotensin: human 153-185 fragment of Adrenomedullin precursor, a 52-amino acid peptide in CGRP hormone family.</p>Fórmula:C143H224N42O43Cor e Forma:SolidPeso molecular:3219.56Calcitonin Gene Related Peptide (CGRP) II, rat TFA
<p>Rat CGRP II TFA: potent vasodilator and CGRP receptor activator for cardiovascular research.</p>Fórmula:C165H268F3N51O52S2Cor e Forma:SolidPeso molecular:3919.33Olcegepant hydrochloride
CAS:<p>Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.</p>Fórmula:C38H48Br2ClN9O5Pureza:99.69%Cor e Forma:SolidPeso molecular:906.11Cagrilintide acetate
<p>.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.</p>Fórmula:C196H316N54O61S2Pureza:99.88%Cor e Forma:SolidPeso molecular:4469.06β-CGRP (mouse)
<p>β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.</p>Fórmula:C165H265N49O55S2Cor e Forma:SolidPeso molecular:3879.29CGRP 8-37 (rat)
CAS:<p>CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.</p>Fórmula:C138H224N42O41Pureza:99.28%Cor e Forma:SolidPeso molecular:3127.51Adrenomedullin (AM) (22-52), human acetate
<p>Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an</p>Fórmula:C161H256N46O50Pureza:99.42%Cor e Forma:SolidPeso molecular:3636.09α-CGRP (mouse, rat) TFA
<p>α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions and</p>Fórmula:C162H262N50O52S2·C2HF3O2Pureza:98%Cor e Forma:SolidCalcitonin-13C6,15N4 TFA
<p>Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.</p>Fórmula:C1401C5H240N4315NO48S2·5C2HF3O2Cor e Forma:SolidPeso molecular:4007.93Galcanezumab
CAS:<p>Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:144.08 kDaCGRP antagonist 6
<p>CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.</p>Cor e Forma:Odour SolidAdrenomedullin (1-50), rat
CAS:<p>Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.</p>Fórmula:C248H381N77O75S5Pureza:98%Cor e Forma:SolidPeso molecular:5729.5Adrenomedullin (AM) (22-52), human
CAS:<p>Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.</p>Fórmula:C159H252N46O48Pureza:98%Cor e Forma:SolidPeso molecular:3576.04HCGRP-(8-37)
CAS:<p>Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist</p>Fórmula:C139H230N44O38Pureza:98%Cor e Forma:SolidPeso molecular:3125.59Calcitonin (human)
CAS:<p>Endogenous calcitonin receptor agonist. Lowers systemic blood calcium levels and inhibits bone resorption.</p>Fórmula:C151H226N40O45S3Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:3417.87α-CGRP, rat
CAS:<p>Endogenous neuropeptide, potent vasodilator</p>Fórmula:C162H262N50O52S2Pureza:98%Cor e Forma:SolidPeso molecular:3806.25β-CGRP, human
CAS:<p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>Fórmula:C162H267N51O48S3Pureza:98%Cor e Forma:SolidPeso molecular:3793.41SUN B8155
CAS:<p>SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.</p>Fórmula:C14H15N3O3Pureza:99.38% - 99.38%Cor e Forma:SolidPeso molecular:273.29Telcagepant
CAS:<p>Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.</p>Fórmula:C26H27F5N6O3Pureza:98.98% - 98.98%Cor e Forma:SolidPeso molecular:566.52Calcitonin (salmon)
CAS:<p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>Fórmula:C145H240N44O48S2Pureza:99.41% - 99.80%Cor e Forma:PowderPeso molecular:3431.85Rimegepant
CAS:<p>View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.</p>Fórmula:C28H28F2N6O3Pureza:99.1% - 99.99%Cor e Forma:SolidPeso molecular:534.56BCTC
CAS:<p>BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)</p>Fórmula:C20H25ClN4OPureza:99.21%Cor e Forma:SolidPeso molecular:372.89Calcitonin(salmon) Acetate(47931-85-1(free base))
<p>Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5</p>Fórmula:C145H240N44O48S2Pureza:99.29%Cor e Forma:SolidPeso molecular:3431.85Olcegepant
CAS:<p>Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4</p>Fórmula:C38H47Br2N9O5Pureza:96.08% - 97.24%Cor e Forma:SolidPeso molecular:869.65HCGRP-(8-37) acetate
<p>HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.</p>Fórmula:C141H234N44O40Pureza:99.29%Cor e Forma:SolidPeso molecular:3185.64Vazegepant hydrochloride
CAS:<p>Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.</p>Fórmula:C36H47ClN8O3Pureza:98.93%Cor e Forma:SolidPeso molecular:675.3β-CGRP, human acetate
<p>β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor</p>Fórmula:C164H271N51O50S3Pureza:99.35%Cor e Forma:SolidPeso molecular:3853.46Atogepant
CAS:<p>Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.</p>Fórmula:C29H23F6N5O3Pureza:99.66%Cor e Forma:SolidPeso molecular:603.52Fremanezumab
CAS:<p>Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.</p>Pureza:95% - 95%Cor e Forma:LiquidEptinezumab
CAS:<p>Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.</p>Pureza:95% - 95%Cor e Forma:LiquidSB 268262
CAS:<p>CGRP1 antagonist</p>Fórmula:C18H15N3O4S2Pureza:98%Cor e Forma:SolidPeso molecular:401.46CGRP antagonist 1
CAS:<p>CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the</p>Fórmula:C29H26N4O4Pureza:99.55%Cor e Forma:SolidPeso molecular:494.54Ubrogepant
CAS:<p>Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.</p>Fórmula:C29H26F3N5O3Pureza:99.452% - 99.78%Cor e Forma:SolidPeso molecular:549.54MK-3207
CAS:<p>MK-3207 is a potent, oral CGRP receptor antagonist with high selectivity for human and monkey receptors, inhibiting blood flow in vivo.</p>Fórmula:C31H29F2N5O3Cor e Forma:SolidPeso molecular:557.59MK-3207 Hydrochloride
CAS:<p>MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.</p>Fórmula:C31H30ClF2N5O3Pureza:98.19%Cor e Forma:SolidPeso molecular:594.05BI-44370
CAS:<p>BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.</p>Fórmula:C35H47N5O6Cor e Forma:SolidPeso molecular:633.78MK-8825
CAS:<p>MK-8825 is a CGRP receptor antagonist.</p>Fórmula:C31H30F2N6O3Cor e Forma:SolidPeso molecular:572.61
