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Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

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Foram encontrados 8595 produtos de "Metabolismo"

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  • ZK53

    CAS:
    <p>ZK53 is a mitochondrial casein hydrolysing protease P (HsClpP) activator that induces apoptosis and inhibits the hydrolysis of alpha-casein by HsClpP.</p>
    Fórmula:C19H20BrF2N3O
    Pureza:97.8% - 99.36%
    Cor e Forma:Soild
    Peso molecular:424.28
  • α-Glucosidase-IN-80


    <p>α-Glucosidase-IN-80 (Compound 10n) is a potent competitive inhibitor of α-glucosidase, with an IC50 of 48.4 μM. It exhibits favorable pharmacokinetic properties and toxicity profiles, making it suitable for research in diabetes-related conditions.</p>
    Fórmula:C24H24N8OS2
    Cor e Forma:Solid
    Peso molecular:504.63
  • 12-Hydroxynevirapine

    CAS:
    <p>12-Hydroxynevirapine, major Nevirapine metabolite; non-toxic but liver/skin SULTs convert it to reactive 12-Sulphoxy-nevirapine.</p>
    Fórmula:C15H14N4O2
    Cor e Forma:Solid
    Peso molecular:282.3
  • 1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol

    CAS:
    <p>1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol is a quinoxaline derivative and endogenous metabolite applicable to biochemical experiments and drug synthesis research.</p>
    Fórmula:C12H14N2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:250.25
  • Lysylcysteine TFA


    <p>Lysylcysteine (L-Lysyl-L-cysteine)TFA is a dipeptide composed of lysine and cysteine.</p>
    Fórmula:C13H21F6N3O7S
    Cor e Forma:Solid
    Peso molecular:477.10044
  • CMI977

    CAS:
    <p>CMI977 is a potent inhibitor of 5-Lipoxygenase (5-LO).</p>
    Fórmula:C16H19FN2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:322.33
  • Monaschromone

    CAS:
    <p>Monaschromone, a polyketide, hinders B. cinerea, A. solani, M. oryzae, G. saubinettii growth; MICs 6.25-12.5 μM.</p>
    Fórmula:C11H12O4
    Cor e Forma:Solid
    Peso molecular:208.21
  • MCU-i11

    CAS:
    <p>MCU-i11 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.</p>
    Fórmula:C28H28N4O5S
    Pureza:98.3%
    Cor e Forma:Solid
    Peso molecular:532.61
  • MTHFD2-IN-1


    <p>MTHFD2-IN-1 (compound 12) is a potent inhibitor of methylenetetrahydrofolate dehydrogenase (MTHFD2) [1].</p>
    Fórmula:C24H21NO6
    Cor e Forma:Solid
    Peso molecular:419.43
  • DSPE-PEG2000-CSTSMLKAC


    <p>DSPE-PEG2000-CSTSMLKAC is a PEG compound composed of DSPE and CSTSMLKAC. CSTSMLKAC can mediate phage selective homing to ischemic heart tissue. DSPE-PEG2000-CSTSMLKAC is suitable for drug delivery.</p>
    Cor e Forma:Odour Solid
  • Casein Kinase 2 Substrate Peptide

    CAS:
    <p>CK2 Substrate Peptide, C-terminus linked to EDANS, used for CK2 activity assays.</p>
    Fórmula:C45H73N19O24
    Cor e Forma:Solid
    Peso molecular:1264.17
  • CT140


    <p>CT140 is a human IgG4 monoclonal antibody (mAb) that specifically targets PAI-1. The suggested isotype control for this compound is Human IgG4 kappa, Isotype Control.</p>
    Cor e Forma:Odour Liquid
  • Captopril EP Impurity E

    CAS:
    <p>Captopril EP Impurity E, an ACE inhibitor with antihypertensive properties, has an IC50 of 0.025 μM.</p>
    Fórmula:C9H15NO3
    Cor e Forma:Solid
    Peso molecular:185.22
  • DSPE-PEG3000-LyP-1


    <p>DSPE-PEG3000-LyP-1 is a PEG compound composed of DSPE and a nine-residue peptide (LyP-1). The LyP-1 component specifically targets tumor-associated lymphatics and macrophages.</p>
    Cor e Forma:Odour Solid
  • PTP1B-IN-22

    CAS:
    <p>PTP1B-IN-22 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor that inhibits glucose uptake in skeletal muscle L6 myotubes.</p>
    Fórmula:C16H12N2O3S2
    Pureza:98.35%
    Cor e Forma:Soild
    Peso molecular:344.41
  • IDO1/TDO-IN-8


    <p>IDO1/TDO-IN-8 (Compound CZ-17) is a dual IDO1 and TDO inhibitor capable of crossing the blood-brain barrier, with EC50 values of 0.33 μM and 1.78 μM, respectively. It modulates the kynurenine pathway of tryptophan metabolism, reducing the kynurenine/tryptophan ratio. IDO1/TDO-IN-8 has neuroprotective effects, alleviating motor dysfunction and improving depressive behavior, making it relevant for research into Parkinson's disease with comorbid depression.</p>
    Fórmula:C17H14N2S
    Cor e Forma:Solid
    Peso molecular:278.37
  • Equilenin

    CAS:
    <p>Equilenin (E 400) is a natural estrogen that is an endocrine disruptor and has been used in breast cancer research.</p>
    Fórmula:C18H18O2
    Pureza:99.4%
    Cor e Forma:Solid
    Peso molecular:266.33
  • Nor-Acetildenafil

    CAS:
    <p>Nor-Acetildenafil is a derivative of Acetildenafil, a synthetic phosphodiesterase inhibitor.</p>
    Fórmula:C24H32N6O3
    Cor e Forma:Solid
    Peso molecular:452.55
  • Risperidone E-oxime

    CAS:
    <p>Risperidone E-oxime: Risperidone impurity, 5-HT2 &amp; dopamine D2 blocker (Ki: 4.8, 5.9 nM), P-Glycoprotein inhibitor.</p>
    Fórmula:C23H28F2N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:430.49
  • UDP-α-D-Glucose sodium hydrate


    <p>UDP-α-D-Glucose sodium hydrate is an endogenous metabolite and a pyrimidine nucleotide sugar, involved in glycosylation reactions during metabolic</p>
    Fórmula:C15H24N2Na2O18P2
    Cor e Forma:Solid
    Peso molecular:628.28