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Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

Exibir 34 mais subcategorias

Foram encontrados 8595 produtos de "Metabolismo"

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  • Dopropidil

    CAS:
    <p>Dopropidil: anti-angina calcium regulator with anti-ischemic properties in animal models.</p>
    Fórmula:C20H35NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:321.5
  • SA57

    CAS:
    <p>SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).</p>
    Fórmula:C17H23ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:338.83
  • FSG67

    CAS:
    <p>FSG67 is an inhibitor of glycerol 3-phosphate acyltransferase (IC 50 =24 μM) [1].</p>
    Fórmula:C16H25NO4S
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:327.44
  • α-2,3-sialyltransferase-IN-1

    CAS:
    <p>α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).</p>
    Fórmula:C28H45NO6
    Pureza:98% - 98%
    Cor e Forma:Solid
    Peso molecular:491.66
  • Gemlapodect

    CAS:
    <p>Gemlapodect (RO554965), a phosphodiesterase 10A (PDE10A) inhibitor, is utilized in schizophrenia research.</p>
    Fórmula:C22H21N7O3
    Cor e Forma:Solid
    Peso molecular:431.45
  • Aminopeptidase-IN-1

    CAS:
    <p>Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.</p>
    Fórmula:C18H16N2O6
    Pureza:98.37%
    Cor e Forma:Solid
    Peso molecular:356.33
  • Albaconazole

    CAS:
    <p>Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.</p>
    Fórmula:C20H16ClF2N5O2
    Pureza:99.27%
    Cor e Forma:Solid
    Peso molecular:431.82
  • DHODH-IN-17

    CAS:
    <p>DHODH-IN-17 is a human DHODH inhibitor with an IC50 of 0.40 μM.</p>
    Fórmula:C12H9ClN2O2
    Pureza:99.41% - 99.52%
    Cor e Forma:Solid
    Peso molecular:248.67
  • Ipenoxazone

    CAS:
    <p>Ipenoxazone is an effective and centrally acting muscle relaxant.</p>
    Fórmula:C22H34N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:358.52
  • Hexazinone

    CAS:
    <p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>
    Fórmula:C12H20N4O2
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:252.31
  • 7-Biopterin

    CAS:
    <p>7-Biopterin, a 7-substituted pterin, forms non-enzymatically and elevates in urine of hyperphenylalaninemics with PCBD mutations.</p>
    Fórmula:C9H11N5O3
    Cor e Forma:Solid
    Peso molecular:237.22
  • Dexecadotril

    CAS:
    <p>Dexecadotril is a powerful and selective neprilysin inhibitor. It behaves as a prodrug of the enantiomer of thiorphan.</p>
    Fórmula:C21H23NO4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:385.48
  • EN40

    CAS:
    <p>EN40, as a covalent ligand, is a selective inhibitor of aldehyde dehydrogenase 3A1 (IC50: 2 uM).</p>
    Fórmula:C13H15NO2
    Cor e Forma:Solid
    Peso molecular:217.26
  • KD-027

    CAS:
    <p>KD-027 is a novel and long-acting PDE5A(phosphodiesterase 5A) inhibitor with potential antihypertensive activity.</p>
    Fórmula:C25H35N7O6S
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:561.65
  • RO-28-1675

    CAS:
    <p>RO-28-1675 is a direct and selective glucokinase activator, the GK/GKRP complex,insulin secretion and type 2 diabetes.</p>
    Fórmula:C18H22N2O3S2
    Pureza:98.13%
    Cor e Forma:Solid
    Peso molecular:378.51
  • AGI-026

    CAS:
    <p>AGI-026 (AGI-12026) is a novel and potent dual inhibitor of the mutant isocitrate dehydrogenase mIDH1/2 blood-brain barrier, reduce d-2-hydroxyglutarate (2-HG).</p>
    Fórmula:C18H15F6N7
    Pureza:99.79% - 99.86%
    Cor e Forma:Solid
    Peso molecular:443.35
  • TTA-A8

    CAS:
    <p>TTA-A8 is an antagonist of T-type calcium channel.</p>
    Fórmula:C22H21F3N4O2
    Pureza:99.22%
    Cor e Forma:Solid
    Peso molecular:430.42
  • Amiquinsin

    CAS:
    <p>Amiquinsin is a drug with hypotensive effect.</p>
    Fórmula:C11H12N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:204.23
  • GT 949

    CAS:
    <p>GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).</p>
    Fórmula:C30H37N7O2
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:527.66
  • XY101

    CAS:
    <p>XY101 is a selective, metabolically stable and orally available agonist of RORγ inverse(IC50 of 30 nM and a Kd of 380 nM).</p>
    Fórmula:C25H20F7NO4S
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:563.48
  • Teglarinad chloride

    CAS:
    <p>Teglarinad chloride (GMX-1777 chloride) is an inhibitor of NAMPT with antitumor activity that acts by interfering with DNA repair and inhibiting angiogenesis.</p>
    Fórmula:C30H43Cl2N5O8
    Pureza:98.09%
    Cor e Forma:Solid
    Peso molecular:672.6
  • ROR agonist-1

    CAS:
    <p>Potent RORC2 inverse agonist, ROR agonist-1, inhibits IL-17A in TH17 cells, pIC50=7.5, orally active.</p>
    Fórmula:C21H20F6N2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:526.45
  • Radamide

    CAS:
    <p>Radamide is an inhibitor of Grp94.</p>
    Fórmula:C18H18ClNO8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:411.79
  • AE0047 Hydrochloride

    CAS:
    <p>AE0047 Hydrochloride is a blocker of calcium, and used in the research of the hypertensive disease.</p>
    Fórmula:C41H43ClN4O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:723.26
  • WAY-213613

    CAS:
    <p>WAY-213613: Potent GLT-1/EAAT2 inhibitor (IC50: 85 nM), selective over EAAT1/EAAT3; inactive at glutamate receptors.</p>
    Fórmula:C16H13BrF2N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:415.19
  • tHGA

    CAS:
    <p>tHGA is a potent inhibitor of lipoxygenase.</p>
    Fórmula:C18H24O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:304.38
  • 2614W94

    CAS:
    2614W94 is a selective inhibitor of MAO-A with IC50 of 5 nM and Ki of 1.6 nM.
    Fórmula:C15H11F3O4S
    Pureza:99.6%
    Cor e Forma:Solid
    Peso molecular:344.31
  • 20(S)-Hydroxycholesterol

    CAS:
    <p>20(S)-Hydroxycholesterol (20α-Hydroxycholesterol) is an allosteric activator of the oncoprotein smoothened (Smo).</p>
    Fórmula:C27H46O2
    Pureza:99.25% - 99.79%
    Cor e Forma:Solid
    Peso molecular:402.65
  • Lovastatin hydroxy acid sodium

    CAS:
    <p>Lovastatin Sodium is an HMG-CoA reductase inhibitor.</p>
    Fórmula:C24H38NaO6
    Cor e Forma:Solid
    Peso molecular:445.54
  • SCH 42495

    CAS:
    <p>SCH 42495 is an orally active neutral metalloendopeptidase inhibitor. SCH 42495 is the orally active ethyl ester prodrug of SCH 42354.</p>
    Fórmula:C20H29NO4S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:411.58
  • Dehydronitrosonisoldipine

    CAS:
    <p>Dehydronitrosonisoldipine blocks SARM1, slows axon decay &amp; cADPR synthesis; useful in neurodegeneration research.</p>
    Fórmula:C20H22N2O5
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:370.4
  • PDE5-IN-5

    CAS:
    <p>PDE5-IN-5 is a selective inhibitor of phosphodiesterase 5 (PDE5) (IC50: 2.0 nM).</p>
    Fórmula:C23H20BrN3O4
    Cor e Forma:Solid
    Peso molecular:482.33
  • N-Acetylserine

    CAS:
    <p>N-Acetylserine (N-Acetyl-L-serine) serves as the physiological inducer of cysteine biosynthesis by binding to the CysB apoprotein and stimulating cysJIH</p>
    Fórmula:C5H9NO4
    Pureza:99.28%
    Cor e Forma:Solid
    Peso molecular:147.13
  • AZD-3289

    CAS:
    <p>AZD-3289, a potent BACE1 inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>
    Fórmula:C24H14F5N5
    Cor e Forma:Solid
    Peso molecular:467.39
  • D-Erythro-dihydrosphingosine

    CAS:
    <p>D-Erythro-dihydrosphingosine (C18-Dihydrosphingosine) inhibits arachidonic acid release and cPLA2α activity.</p>
    Fórmula:C18H39NO2
    Pureza:99.50% - 99.88%
    Cor e Forma:Solid
    Peso molecular:301.51
  • Oxycinchophen

    CAS:
    <p>Oxycinchophen: Quinoline-based anti-rheumatic with P-selectin inhibition, DHOD blockade, and anti-inflammatory impacts on vascular muscle.</p>
    Fórmula:C16H11NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:265.26
  • Autotaxin-IN-1

    CAS:
    <p>Autotaxin-IN-1: strong inhibitor for osteoarthritis pain; IC50=2.2 nM; good PK and PK/PD.</p>
    Fórmula:C21H23N7O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:405.45
  • MLS000536924

    CAS:
    <p>MLS000536924 is a potent and selective competitive human epithelial 15-lipoxygenase-2 inhibitor.</p>
    Fórmula:C16H15N3S
    Cor e Forma:Solid
    Peso molecular:281.38
  • Indolapril hydrochloride

    CAS:
    <p>Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.</p>
    Fórmula:C24H35ClN2O5
    Cor e Forma:Solid
    Peso molecular:467
  • Fadrozole HCl hydrate

    CAS:
    <p>Fadrozole is a selective inhibitor of aromatase. It also effective in the treatment of estrogen-dependent diseases including breast cancer.</p>
    Fórmula:C14H13N3ClHH2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:268.74
  • Vilazodone carboxylic acid

    CAS:
    <p>Vilazodone carboxylic acid is a vilazodone metabolite observed in both urine and plasma.</p>
    Fórmula:C26H26N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:442.51
  • Tralkoxydim

    CAS:
    <p>Tralkoxydim (Tralkoxydime) is an alkyl ketone herbicide. Tralkoxydim works as an ACCase inhibitor.</p>
    Fórmula:C20H27NO3
    Pureza:97.44%
    Cor e Forma:Solid
    Peso molecular:329.43
  • ML368

    CAS:
    <p>ML368 is a selective inhibitor of CYP3A4.</p>
    Fórmula:C26H18N6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:430.46
  • MMV-667492

    CAS:
    <p>MMV-667492 is an effective inhibitor of Ezrin.</p>
    Fórmula:C17H19N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:313.35
  • Palmostatin B

    CAS:
    <p>Palmostatin B is a modulator of Ras-signaling that acts by targeting acyl protein thioesterase 1 (APT1) and 2 (APT2) in cells.</p>
    Fórmula:C23H36O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:376.53
  • Rev 6207

    CAS:
    <p>Rev 6207 is a non-sulfhydryl ACE-inhibitor.</p>
    Fórmula:C21H31N3O5
    Cor e Forma:Solid
    Peso molecular:405.49
  • hCAIX-IN-5

    CAS:
    <p>hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of &gt;10000, &gt;10000, 130.7, and 829.1 nM, respectively.</p>
    Fórmula:C18H12FNO3
    Pureza:99.26%
    Cor e Forma:Solid
    Peso molecular:309.29
  • Afegostat D-Tartrate

    CAS:
    <p>Afegostat D-Tartrate: pharmacological chaperone, reversibly binds acid-β-glucosidase in ER with high affinity.</p>
    Fórmula:C10H19NO9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:297.26
  • AVX-001

    CAS:
    <p>AVX-001, a cytosolic phospholipase A2 (cPLA2) inhibitor, is used potentially for the treatment of psoriasis.</p>
    Fórmula:C21H29F3OS
    Cor e Forma:Solid
    Peso molecular:386.51
  • (Z)-10-Hydroxynortriptyline

    CAS:
    <p>(Z)-10-Hydroxynortriptyline ((Z)-10-Hydroxy Nortriptyline) is a norepinephrine reuptake inhibitor with antidepressant activity.</p>
    Fórmula:C19H21NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:279.38
  • L-651392

    CAS:
    <p>L-651392 is an inhibitor of leukotriene.</p>
    Fórmula:C14H10BrNO3S
    Cor e Forma:Solid
    Peso molecular:352.2
  • LGE-899

    CAS:
    <p>LGE-899 (Sonidegib metabolite M48) is a main metabolite of Sonidegib which is an inhibitor of the hedgehog pathway.</p>
    Fórmula:C15H11F3O3
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:296.24
  • 1-Methyluric acid

    CAS:
    <p>1-Methyluric acid (1-Methylurate) acts on the bladder mucosa and increases the levels of insulin, triglycerides, cholesterol, and blood glucose.</p>
    Fórmula:C6H6N4O3
    Pureza:98.05%
    Cor e Forma:Solid
    Peso molecular:182.14
  • PDE7-IN-2

    CAS:
    <p>PDE7-IN-2 is an inhibitor of phosphodiesterase 7 (IC50 = 2.1 µM) and can be used in Parkinson's disease studies.</p>
    Fórmula:C14H11ClN2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:322.77
  • IDO inhibitor 1

    CAS:
    <p>IDO inhibitor 1 is an potent inhibitor of indoleamine-2,3 dioxygenase (IDO) ( IC50 &lt;100 nM).with potential immunomodulating and antineoplastic activities.</p>
    Fórmula:C11H13BrFN7O4S
    Pureza:99.805%
    Cor e Forma:Solid
    Peso molecular:438.23
  • 4-Desmethyl Istradefylline

    CAS:
    <p>4-Desmethyl Istradefylline: a metabolite of Istradefylline, a strong, selective oral adenosine A2A receptor blocker, Ki 2.2 nM, used in Parkinson's.</p>
    Fórmula:C19H22N4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:370.40
  • Clofenamide

    CAS:
    <p>Clofenamide is a low-ceiling sulfonamide diuretic.</p>
    Fórmula:C6H7ClN2O4S2
    Cor e Forma:Solid
    Peso molecular:270.71
  • ONO-6126

    CAS:
    <p>ONO-6126 has anti-inflammatory activity and can inhibit Phosphodiesterase and PDE4 in the treatment of respiratory diseases.</p>
    Fórmula:C20H27N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:373.45
  • Telotristat besilate

    CAS:
    <p>Telotristat besilate is an inhibitor of tryptophan hydroxylase.</p>
    Fórmula:C31H28ClF3N6O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:705.11
  • LG 101506

    CAS:
    <p>RXR modulator</p>
    Fórmula:C25H34F2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:420.53
  • Quinaprilat

    CAS:
    <p>Quinaprilat inhibits angiotensin converting enzyme.</p>
    Fórmula:C23H26N2O5
    Pureza:98%
    Cor e Forma:Crystalline Solid
    Peso molecular:410.46
  • L 30

    CAS:
    <p>L 30 is a blocker of the sodium channel.</p>
    Fórmula:C15H24N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:248.36
  • Quinalizarin

    CAS:
    <p>Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.</p>
    Fórmula:C14H8O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:272.21
  • IHMT-PI3Kδ-372

    CAS:
    <p>IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can be used in studies about chronic obstructive pulmonary disease.</p>
    Fórmula:C26H23F2N7O2
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:503.5
  • Ciraparantag

    CAS:
    <p>Ciraparantag inhibits thrombin, factor Xa, and reverses various anticoagulants.</p>
    Fórmula:C22H48N12O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:512.7
  • SHP836

    CAS:
    <p>SHP836 is an inhibitor of SHP2 allosteric (IC50: 12 μM for the full-length SHP2).</p>
    Fórmula:C16H19Cl2N5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.26
  • 4-Acetylsimvastatin

    CAS:
    <p>4-Acetylsimvastatin is acetylated simvastatin. Simvastatin is a competitive inhibitor of HMG-CoA reductase (Ki: 0.2 nM).</p>
    Fórmula:C27H40O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:460.6
  • SCH-51866

    CAS:
    <p>SCH-51866 is a PDE1 and PDE5 phosphodiesterase inhibitor with IC50 value of 0.070 μM and IC50 0.060 μM respectively.</p>
    Fórmula:C19H18F3N5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:389.37
  • hCA I-IN-1

    CAS:
    <p>hCA I-IN-1 inhibits hCA I (Ki: 38.3 nM), II (Ki: 716.4 nM), IX (Ki: 940.1 nM), XII (Ki: 192.8 nM).</p>
    Fórmula:C27H23N5O4S
    Cor e Forma:Solid
    Peso molecular:513.57
  • Manninotrionate

    CAS:
    <p>Manninotrionate, an antitumor agent, linked to BSA; rabbit antiserum made, doesn't agglutinate Ehrlich tumor cells with alpha-D-galactosyl groups.</p>
    Fórmula:C18H32KO17
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:559.535
  • Lith-O-Asp

    CAS:
    <p>Lith-O-Asp is a sialytransferase (ST) inhibitor,(IC50s:12-37 μM).</p>
    Fórmula:C28H45NO6
    Cor e Forma:Solid
    Peso molecular:491.66
  • LH65.3

    CAS:
    <p>LH65.3 is an inhibitor of S. typhimurium infection on the activity of DUSP3, DUSP11, and DUSP27.</p>
    Fórmula:C21H20N2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:412.46
  • Glyoxalase I inhibitor

    CAS:
    <p>Glyoxalase I inhibitor, a candidate for anticancer agents, is a potent Glyoxalase I (GLO1) inhibitor.</p>
    Fórmula:C21H30BrClN4O8S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:613.91
  • PF-4191834

    CAS:
    <p>PF-4191834: Non-iron, non-redox 5-LOX inhibitor, IC50 = 229 nM, 300x selective over 12/15-LOX, inactive on COX enzymes.</p>
    Fórmula:C22H23N3O2S
    Pureza:99.83% - 99.98%
    Cor e Forma:Solid
    Peso molecular:393.5
  • Prolyl Endopeptidase Inhibitor 1

    CAS:
    <p>Prolyl Endopeptidase Inhibitor 1 is a potent inhibitor of prolyl endopeptidase (PEP; PE)(Ki : 15 nM) , has anti-amnesic effect.</p>
    Fórmula:C15H24N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:296.36
  • Cgp 8065

    CAS:
    <p>Cgp 8065 is a filaricidal compound, a dithiocarbamate-derivative of amoscanate.</p>
    Fórmula:C16H15N3O4S2
    Cor e Forma:Solid
    Peso molecular:377.44
  • MAGL-IN-1

    CAS:
    <p>MAGL-IN-1 is a selective and potent monoacylglycerol lipase (MAGL) inhibitor with an IC50 of 80 nM.</p>
    Fórmula:C22H24FNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:369.43
  • Argininic acid

    CAS:
    <p>Argininic acid is an α-amino acid used in the biosynthesis of proteins.</p>
    Fórmula:C6H13N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:175.19
  • Atreleuton

    CAS:
    <p>Atreleuton (ABT-761), reversible oral 5-LO inhibitor, selectively blocks leukotriene formation.</p>
    Fórmula:C16H15FN2O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:318.37
  • ALDH1A1-IN-3

    CAS:
    <p>ALDH1A1-IN-3 selectively inhibits ALDH1A1, enhances HepG2 glucose consumption for metabolic research.</p>
    Fórmula:C31H36F3N5O4
    Cor e Forma:Solid
    Peso molecular:599.64
  • 4,5,6,7-Tetrabromobenzimidazole

    CAS:
    <p>4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].</p>
    Fórmula:C7H2Br4N2
    Cor e Forma:Solid
    Peso molecular:433.72
  • ML387

    CAS:
    <p>ML387 is an inhibitor of human NAD(+)- dependent 15- hydroxyprostaglandin dehydrogenase.</p>
    Fórmula:C20H21N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:335.4
  • MR 16728 hydrochloride

    CAS:
    <p>stimulates the release of acetylcholine from synaptosomes</p>
    Fórmula:C23H37ClN2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:393.01
  • ML404

    CAS:
    <p>ML404 is the mitochondrial permeability transition pore inhibitor.</p>
    Fórmula:C17H13ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:328.75
  • Mesopram

    CAS:
    <p>PDE4 inhibitor, orally active</p>
    Fórmula:C14H19NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:265.3
  • β-Amino Acid Imagabalin Hydrochloride

    CAS:
    <p>β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.</p>
    Fórmula:C9H20ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:209.71
  • IHVR-11029

    CAS:
    <p>IHVR-11029 inhibits ER α-glucosidase, combats hemorrhagic fever viruses, and hinders enveloped virus morphogenesis.</p>
    Fórmula:C18H27F2NO5
    Cor e Forma:Solid
    Peso molecular:375.41
  • Ro 41-0960

    CAS:
    <p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>
    Fórmula:C13H8FNO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:277.2
  • ATX inhibitor 20

    CAS:
    <p>ATX inhibitor 20 is a potent inhibitor of ATX (IC50: 2.3 nM).</p>
    Fórmula:C31H34FN5O3
    Cor e Forma:Solid
    Peso molecular:543.63
  • HZ52

    CAS:
    <p>HZ52: Potent reversible 5-LO inhibitor; IC50 0.7 μM; blocks LTs in human leukocytes.</p>
    Fórmula:C24H26ClN3O2S
    Cor e Forma:Solid
    Peso molecular:456
  • (Rac)-RK-682

    CAS:
    <p>(Rac)-RK-682 racemate; inhibits PTP-1B, LMW-PTP, CDC-25B with IC50s: 8.6, 12.4, 0.7 µM respectively.</p>
    Fórmula:C21H36O5
    Cor e Forma:Solid
    Peso molecular:368.51
  • Adenosine 5'-phosphosulfate (sodium salt)

    CAS:
    <p>Adenosine 5'-phosphosulfate (sodium salt) (APS) is a key intermediate in sulphur metabolism and a substrate for adenosine 5'-phosphosulfate kinase (APSK).</p>
    Fórmula:C10H12N5Na2O10PS
    Cor e Forma:Solid
    Peso molecular:471.24
  • PDE2/PDE10-IN-1

    CAS:
    <p>PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).</p>
    Fórmula:C15H10ClN5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:295.73
  • NCX 1000

    CAS:
    <p>NCX 1000 is a liver-specific NO donor compound,NCX 1000 derived from ursodeoxycholic acid (UDCA).</p>
    Fórmula:C38H55NO10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:685.84
  • Rosuvastatin lactone

    CAS:
    <p>Tilavonemab (ABBV-8E12) is a monoclonal antibody that binds to the N-terminus of the human microtubule-associated protein tau.</p>
    Fórmula:C22H26FN3O5S
    Cor e Forma:Solid
    Peso molecular:463.52
  • CYP11B2-IN-1

    CAS:
    <p>CYP11B2-IN-1 是一种有效的选择性 CYP11B2 抑制剂,对 CYP11B2 和 CYP11B1 的 IC50 分别为 2.3 nM 和 142 nM。</p>
    Fórmula:C18H18FN3O
    Pureza:99.79% - 99.89%
    Cor e Forma:Solid
    Peso molecular:311.35
  • TDP1 Inhibitor-1

    CAS:
    <p>TDP1 Inhibitor-1 is a potent inhibitor of Tyrosyl-DNA Phosphodiesterase 1 (TDP1) (IC50 of 7 μM).</p>
    Fórmula:C26H26N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:446.49
  • L 669262

    CAS:
    <p>L 669262 is a potent inhibitor of HMG-CoA reductase.</p>
    Fórmula:C25H36O6
    Cor e Forma:Solid
    Peso molecular:432.55
  • ALRT 1550

    CAS:
    <p>ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.</p>
    Fórmula:C23H32O2
    Cor e Forma:Solid
    Peso molecular:340.5
  • MMG-0358

    CAS:
    <p>MMG-0358 is a novel potent IDO1 inhibitor, showing low cytotoxicity and higher selectivity for IDO1 over TDO enzyme.</p>
    Fórmula:C8H6ClN3O
    Cor e Forma:Solid
    Peso molecular:195.61
  • Asterriquinol D dimethyl ether

    CAS:
    <p>Asterriquinol D dimethyl ether inhibits mouse myeloma (IC50: 28 μg/mL) and Tritrichomonas foetus.</p>
    Fórmula:C26H24N2O4
    Cor e Forma:Solid
    Peso molecular:428.48
  • DSHN

    CAS:
    <p>DSHN activates SHP, boosting its mRNA and protecting it from ubiquitination and degradation.</p>
    Fórmula:C15H17NO5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:323.36
  • Abiraterone metabolite 1

    CAS:
    <p>Abiraterone metabolite 1, a derivative of abiraterone, inhibits CYP17A1, halts androgen formation, aiding in prostate cancer treatment.</p>
    Fórmula:C24H33NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:351.52
  • EP6

    CAS:
    <p>EP6 blocks 5-LO, key in the AA cascade, reducing leukotrienes to curb inflammation and allergies.</p>
    Fórmula:C24H30N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:390.52
  • NEP-IN-2

    CAS:
    <p>NEP-IN-2 is an inhibitor of neutral endopeptidase. It also is used in the research of proliferation in atherosclerosis, restenosis.</p>
    Fórmula:C16H23NO3S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:341.49
  • BML-111

    CAS:
    <p>inhibits leukotriene B4 (LTB4)-induced polymorphonuclear neutrophils (PMN) chemotaxis</p>
    Fórmula:C8H16O5
    Cor e Forma:Solid
    Peso molecular:192.21
  • MPO-IN-4

    CAS:
    <p>MPO-IN-4, a potent MPO inhibitor (IC50=25 nM), also inhibits TPO (IC50=2.2 μM), but not MGMT.</p>
    Fórmula:C12H11N5
    Cor e Forma:Solid
    Peso molecular:225.25
  • Dapaconazole

    CAS:
    <p>Dapaconazole is used as a drug candidate for antifungals.</p>
    Fórmula:C19H15Cl2F3N2O
    Cor e Forma:Solid
    Peso molecular:415.24
  • 6-Hydroxyluteolin

    CAS:
    <p>6-Hydroxyluteolin, a flavonoid compound extracted from Salvia amarissima Ortega, inhibits aldose reductase (AR) and has antimicrobial activity.</p>
    Fórmula:C15H10O7
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:302.24
  • RG 6866

    CAS:
    RG 6866 is a inhibitor of 5-lipoxygenase.
    Fórmula:C16H17NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:271.31
  • SDZ-MKS 492

    CAS:
    <p>SDZ-MKS 492 is a selective type III isozyme cyclic nucleotide phosphodiesterase inhibitor.</p>
    Fórmula:C20H27N5O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.46
  • MMPX

    CAS:
    <p>calmodulin-sensitive cyclic GMP phosphodiesterase inhibitor</p>
    Fórmula:C12H18N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:266.3
  • OMDM-4

    CAS:
    <p>OMDM-4 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 17.7 μM).</p>
    Fórmula:C29H43NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:453.66
  • Acetaldophosphamide

    CAS:
    <p>Acetaldophosphamide is a novel stable aldophosphamide analog.</p>
    Fórmula:C11H21Cl2N2O6P
    Cor e Forma:Solid
    Peso molecular:379.17
  • Senazodan hydrochloride

    CAS:
    <p>Senazodan hydrochloride (Senazodan HCl) is a Ca2+ sensitizer and phosphodiesterase 3 (PDE3) inhibitor used in the study of cardiovascular diseases.</p>
    Fórmula:C15H15ClN4O
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:302.76
  • CP-532623

    CAS:
    <p>CP-532623, a close structural analog of Torcetrapib, is a CETP inhibitor with highly lipophilic properties. It elevates high-density lipoprotein cholesterol.</p>
    Fórmula:C27H27F9N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:598.5
  • HM-50316

    CAS:
    <p>HM-50316 is a High affinity FABP4 inhibitor (Ki &lt; 1 nM).</p>
    Fórmula:C29H23ClN2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:515.02
  • Prinoxodan

    CAS:
    <p>Prinoxodan is an inhibitor of phosphodiesterase.</p>
    Fórmula:C13H14N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:258.28
  • p18SMI-21

    CAS:
    <p>p18SMI-21 is a novel INK4C inhibitor. It also specifically blocking the bioactivity of p18 protein.</p>
    Fórmula:C10H14N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:258.29
  • Trimoxamine hydrochloride

    CAS:
    <p>Trimoxamine hydrochloride is an antihypertensive.</p>
    Fórmula:C15H24ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:301.81
  • LY 221068

    CAS:
    <p>LY 221068 is a potent antioxidant with anti-inflammatory activity.</p>
    Fórmula:C20H30N2O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:362.53
  • PF-06424439

    CAS:
    <p>PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).</p>
    Fórmula:C22H26ClN7O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:439.94
  • BI 689648

    CAS:
    <p>BI 689648 is a highly selective inhibitor of aldosterone synthase(CYP11B1 and CYP11B2 with IC50s of 310 and 2.1 nM, respectively).</p>
    Fórmula:C16H18N4O2
    Cor e Forma:Solid
    Peso molecular:298.34
  • SHP2-IN-13

    CAS:
    <p>SHP2-IN-13 is an orally active, highly selective allosteric inhibitor targeting the SHP2 “tunnel site,” exhibiting an IC50 of 83.0 nM.</p>
    Fórmula:C16H21N7O
    Cor e Forma:Solid
    Peso molecular:327.38
  • DNS-8254

    CAS:
    <p>DNS-8254: Potent, selective PDE2 inhibitor, enhances memory (IC50=8 nM), effective in rat memory tests.</p>
    Fórmula:C18H15BrF3N5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:454.24
  • HIF-1α inhibitor-1

    CAS:
    <p>HIF-1α inhibitor-1 is a HIF-1 alpha inhibitor.</p>
    Fórmula:C15H11N3O4
    Cor e Forma:Solid
    Peso molecular:297.27
  • CD2665

    CAS:
    <p>CD2665 is an orally active antagonist of retinoic acid receptor (RAR). For RARγ and RARβ, the Kis are 110 nM and 306 nM.</p>
    Fórmula:C31H34O5
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:486.6
  • SCH 42495 racemate

    CAS:
    <p>SCH 42495 racemate is the racemate of SCH 42495. SCH 42495 is an orally active neutral inhibitor of metalloendopeptidase (NEP), with antihypertensive effect.</p>
    Fórmula:C20H29NO4S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:411.58
  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Fórmula:C20H21N3O
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:319.4
  • RORγt Inverse agonist 8

    CAS:
    <p>RORγt Inverse agonist 8 is a potent, selective, orally bioavailable RORγt inverse agonist(human RORγt-LBD with an IC50 of 19 nM).</p>
    Fórmula:C26H33N7O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:475.59
  • Theodrenaline

    CAS:
    <p>Theodrenaline is a cardiac stimulant, also acts as an agent of anti-hypotensive together with cafedrine.</p>
    Fórmula:C17H21N5O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:375.38
  • (1S,2S,3R)-DT-061

    CAS:
    <p>(1S,2S,3R)-DT-061 is an enantiomer of DT-061 which is an orally bioavailable activator of PP2A.</p>
    Fórmula:C25H23F3N2O5S
    Cor e Forma:Solid
    Peso molecular:520.52
  • SWE101

    CAS:
    <p>SWE101 is a potent human and rat soluble epoxide hydrolase (sEH)-P inhibitor(IC50s of 4 μM and 2.8 μM, respectively).</p>
    Fórmula:C19H15Cl2NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:376.23
  • IDO-IN-11

    CAS:
    <p>IDO-IN-11 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.18 μM (Kinase) and 0.014 μM (Hela Cell).</p>
    Fórmula:C19H23BrFN7O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:544.4
  • 11β-HSD1-IN-1

    CAS:
    <p>11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1, IC50: 52 nM), and used for the treatment of pain.</p>
    Fórmula:C18H14ClF4N3O
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:399.77
  • BDM14471

    CAS:
    <p>BDM14471 is a selective inhibitor of hydroxamate PfAM1.</p>
    Fórmula:C17H15FN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:314.31
  • hCAIX/XII-IN-2

    CAS:
    <p>Compound 6a: Selective hCAIX/XII inhibitor; Ki: 30 nM (hCAIX), 3.6 nM (hCAXII); &gt;10,000 nM (hCAI/II).</p>
    Fórmula:C19H14N2O4
    Cor e Forma:Solid
    Peso molecular:334.33
  • DO-264

    CAS:
    <p>DO-264 is an inhibitor of autohydrolase structural domain 12 (ABHD12) and an inhibitor of cellular LysoPS degradation that enhances LPS-induced phagocytosis.</p>
    Fórmula:C23H20Cl2F3N5O2S
    Pureza:97.72% - 99.95%
    Cor e Forma:Solid
    Peso molecular:558.4
  • UK51656

    CAS:
    <p>UK51656 is an antagonist of calcium (IC50: 4 nM).</p>
    Fórmula:C22H28ClN3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:465.93
  • N-Methylmoranoline

    CAS:
    <p>N-Methylmoranoline is an inhibitor of α-glucosidase.</p>
    Fórmula:C7H15NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:177.2
  • Utibapril

    CAS:
    <p>Utibapril is an inhibitor of angiotensin-converting enzyme (ACE) with antihypertensive activities.</p>
    Fórmula:C22H31N3O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:449.56
  • 5β-​Dutasteride

    CAS:
    <p>5β-Dutasteride is the S configuration of Dutasteride. It is a potent inhibitor of both 5 alpha-reductase isozymes.</p>
    Fórmula:C27H30F6N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:528.53
  • IDO1-IN-2

    CAS:
    <p>IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity.</p>
    Fórmula:C15H17FN6O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:364.33
  • TC-E 5005

    CAS:
    <p>PDE10A inhibitor</p>
    Fórmula:C15H18N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:270.33
  • ML218

    CAS:
    <p>ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.</p>
    Fórmula:C19H26Cl2N2O
    Pureza:99.2% - 99.45%
    Cor e Forma:Solid
    Peso molecular:369.33
  • MB-07729

    CAS:
    <p>MB-07729 inhibits fructose-1,6-bisphosphate with IC50: 189 nM (rat), 121 nM (monkey), 31 nM (human) for diabetes research.</p>
    Fórmula:C12H15N2O5PS
    Pureza:99.54% - 99.64%
    Cor e Forma:Solid
    Peso molecular:330.3
  • Acarbose sulfate

    CAS:
    <p>Acarbose sulfate is an anti-diabetic drug and is an inhibitor of alpha-glucosidase.</p>
    Fórmula:C25H45NO22S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:743.68
  • 11β-HSD1-IN-12

    CAS:
    <p>11β-HSD1-IN-12 is an 11β-HSD1 inhibitor.11β-HSD1-IN-12 is implicated in the conversion of glucocorticoids in vivo and can be used to study metabolic syndrome</p>
    Fórmula:C19H27ClN2O3S
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:398.95
  • AGI-14100

    CAS:
    <p>AGI-14100 is a novel and orally available mIDH1 inhibitor.AGI-14100 is used for the treatment of primary human myeloid leukemia.</p>
    Fórmula:C29H22ClF4N5O3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:599.96
  • PF-04822163

    CAS:
    <p>PF-04822163 is a potent inhibitor of PDE1 with IC50 value of 0.0024 μM.</p>
    Fórmula:C19H17ClN2O2
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:340.8
  • MAGLi 432

    CAS:
    <p>MAGLi 432: Potent MAGL inhibitor, selective and reversible. IC50: 4.2 nM (human), 3.1 nM (mouse). Useful for neurological disorder research.</p>
    Fórmula:C22H24BrClN2O2
    Cor e Forma:Solid
    Peso molecular:463.8
  • SLC26A3-IN-3

    CAS:
    <p>SLC26A3-IN-3 (compound 4az), a potent SLC26A3 inhibitor with an IC50 of 40 nM, is utilized for constipation and cystic fibrosis research [1].</p>
    Fórmula:C20H17IO5
    Cor e Forma:Solid
    Peso molecular:464.25
  • p-Valerylphenol

    CAS:
    p-Valerylphenol (NSC-49186) can be used to synthesize acylphenoxyacetic acid compounds.
    Fórmula:C11H14O2
    Pureza:99.87%
    Cor e Forma:White To Light Beige Powder
    Peso molecular:178.23
  • (3S,5S)-Pitavastatin calcium

    CAS:
    <p>(3S,5S)-Pitavastatin calcium is the 3-epimer of Pitavastatin which is a potent HMG-CoA reductase inhibitor.</p>
    Fórmula:C25H26CaFNO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:463.562
  • SPK-601

    CAS:
    <p>SPK-601 is an inhibitor of phosphatidylcholine-specific phospholipase C.</p>
    Fórmula:C11H16KOS2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:267.47
  • IDO-IN-16

    CAS:
    <p>IDO-IN-16 (compound 5) is an IDO inhibitor (IC50: 36 nM).</p>
    Fórmula:C22H21F3N4O
    Cor e Forma:Solid
    Peso molecular:414.42
  • Tenuazonic acid

    CAS:
    <p>Tenuazonic acid, a nonhost-selective mycotoxin from Alternaria alternate, inhibits PSII by blocking electron transport at D1 protein.</p>
    Fórmula:C10H15NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:197.23
  • Propaquizafop

    CAS:
    <p>Propaquizafop, a phenoxyisopropionic acid derivative, is used as a herbicide.</p>
    Fórmula:C22H22ClN3O5
    Pureza:98%
    Cor e Forma:Colourless-To-Brown Crystals
    Peso molecular:443.88
  • Antitumor agent-87

    CAS:
    <p>Antitumor agent-87: potent, high CYP1A1 affinity (Ki 0.23µM), antiproliferative, arrests G2/M cell cycle.</p>
    Fórmula:C22H28N2O6S
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:448.53
  • CX08005

    CAS:
    <p>CX08005 inhibits PTP1B, cuts liver fat, and improves microcirculation in NAFLD.</p>
    Fórmula:C28H39NO4
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:453.61
  • Acetylhydrolase-IN-1

    CAS:
    <p>Acetylhydrolase-IN-1 is an inhibitor of the esterase 1-Alkyl-2-acetylglycerophosphocholine (Alkylacetyl-GPC: acetylhydrolase).</p>
    Fórmula:C23H48NO7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:481.6
  • M77976

    CAS:
    <p>M77976 inhibits PDK4 with an IC50 of 648 μM, targeting obesity and diabetes research.</p>
    Fórmula:C17H16N2O3
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:296.32
  • Disulfamide

    CAS:
    <p>Disulfamide: Oral carbonic anhydrase inhibitor, IC50 0.07 μM, diuretic by blocking Na+/HCO3- reabsorption.</p>
    Fórmula:C7H9ClN2O4S2
    Pureza:98.1%
    Cor e Forma:Solid
    Peso molecular:284.74
  • RORγt/DHODH-IN-2

    CAS:
    <p>RORγt/DHODH-IN-2 (compound 1) is a potent dual RORγt/DHODH inhibitor that can be used in the study of inflammatory bowel disease (IBD).</p>
    Fórmula:C25H30N4OS
    Cor e Forma:Solid
    Peso molecular:434.6
  • VU0155056

    CAS:
    <p>VU0155056 is a dual PLD1/2 inhibitor with IC50 &lt; 1 µM in cellular assays, inhibits breast cancer cell invasion.</p>
    Fórmula:C25H26N4O2
    Pureza:98.6% - 99.15%
    Cor e Forma:Solid
    Peso molecular:414.5
  • MB05032

    CAS:
    <p>MB05032 is a fructose-,-bisphosphatase inhibitor that inhibits gluconeogenesis and may reduce d-lactate-triggered ETosis.</p>
    Fórmula:C11H15N2O4PS
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:302.29
  • SHP504

    CAS:
    <p>SHP504 is an inhibitor of SHP2 phosphatase and acts on SHP21-525 (IC50: 21 μM).</p>
    Fórmula:C23H15ClN4O4
    Cor e Forma:Solid
    Peso molecular:446.84
  • McN3716

    CAS:
    <p>McN3716 is a carnitine palmitoyltransferase I (CPT-1) inhibitor for the study of metabolic diseases.</p>
    Fórmula:C18H34O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:298.46
  • Hydroxythiohomosildenafil

    CAS:
    <p>Hydroxythiohomosildenafil, an analogue of sildenafil, is a phosphodiesterase-5 (PDE-5) inhibitor.</p>
    Fórmula:C23H32N6O4S2
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:520.67
  • Glyoxalase I inhibitor 1

    CAS:
    <p>Glyoxalase I inhibitor 1 is a potent inhibitor of glyoxalase I (GLO1) (IC50: 26 nM).</p>
    Fórmula:C30H27FN6O4S
    Cor e Forma:Solid
    Peso molecular:586.64
  • (+)-Cembrene A

    CAS:
    <p>(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM.</p>
    Fórmula:C20H32
    Cor e Forma:Solid
    Peso molecular:272.47
  • AVE-8134

    CAS:
    <p>AVE-8134 is an agonist of PPARα. For human and rodent PPARα receptor, the EC50 values are 100 and 3000 nM, respectively.</p>
    Fórmula:C22H23NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:381.42
  • LY 269415

    CAS:
    <p>LY 269415 is an anti-inflammatory agent with antioxidant properties in vitro and could be beneficial as therapeutic agents in inflammatory arthritis.</p>
    Fórmula:C19H28N2O2S
    Cor e Forma:Solid
    Peso molecular:348.5
  • Methyl-3β-hydroxycholenate

    CAS:
    <p>Methyl-3β-hydroxycholenate (Methyl 3beta-hydroxychol-5-enoate) is a modulator of RORγ.</p>
    Fórmula:C25H40O3
    Pureza:98.78%
    Cor e Forma:Solid
    Peso molecular:388.58
  • K134

    CAS:
    <p>K134 is an inhibitor of phosphodiesterase 3. The IC50s of K134 for PDE3A, PDE3B, PDE5, PDE2 and PDE4 are 0.1, 0.28, 12.1, &gt;300 and &gt;300 μM, respectively.</p>
    Fórmula:C22H29N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:399.48
  • UK-371804 HCl

    CAS:
    <p>UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-</p>
    Fórmula:C14H17Cl2N5O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:422.29
  • Muristerone A

    CAS:
    <p>Muristerone A is a phytoecdysteroid analog of ecdysone and a potent ecdysteroid receptor agonist with a K d of 1 nM [1].</p>
    Fórmula:C27H44O8
    Cor e Forma:Solid
    Peso molecular:496.63
  • IDO/TDO-IN-1

    CAS:
    <p>IDO/TDO-IN-1 is an orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50s: 9.7 and 47 nM).</p>
    Fórmula:C25H24FN5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:413.49
  • SK-216

    CAS:
    <p>SK-216,PAI-1 inhibitor. Reduces tumor angiogenesis. Inhibits VEGF-induced endothelial cell migration. Alleviates pulmonary fibrosis.</p>
    Fórmula:C29H29NNa2O6
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:533.52
  • MLS000544460

    CAS:
    <p>MLS000544460 is a highly selective and reversible Eya2 phosphatase inhibitor (Kd: 2.0 μM, IC50: 4 μM).MLS000544460 exhibits inhibitory effects on Eya2</p>
    Fórmula:C17H12FN3O2S
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:341.36
  • Cronidipine

    CAS:
    <p>Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>
    Fórmula:C30H32ClN3O8
    Pureza:99.47%
    Cor e Forma:Solid
    Peso molecular:598.04
  • hCAI/II-IN-6

    CAS:
    <p>hCAI/II-IN-6 is a selective and orally active inhibitor of human carbonic anhydrase (CA).</p>
    Fórmula:C19H24N4O3S
    Pureza:97.07%
    Cor e Forma:Solid
    Peso molecular:388.48
  • Lonapalene

    CAS:
    <p>Lonapalene is a topically effective inhibitor of 5-lipoxygenase.</p>
    Fórmula:C16H15ClO6
    Pureza:98.67% - 99.33%
    Cor e Forma:Solid
    Peso molecular:338.74
  • Dasantafil

    CAS:
    <p>Dasantafil (SCH446132) is a small molecule phosphodiesterase-5A (PDE5A) inhibitor used to treat genitourinary disorders and study erectile dysfunction.</p>
    Fórmula:C22H28BrN5O5
    Pureza:99.4% - 99.50%
    Cor e Forma:Solid
    Peso molecular:522.39
  • Phosphatase-IN-1

    CAS:
    <p>Phosphatase-IN-1 is a phosphatidic acid phosphatase (Pah) inhibitor with antifungal activity for the study of rice blast and ruderalia.</p>
    Fórmula:C16H16Cl2FNO2
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:344.21
  • SBI-425

    CAS:
    <p>SBI-425: orally available TNAP inhibitor, enhances cardiovascular health &amp; survival, no bone impact.</p>
    Fórmula:C13H12ClN3O4S
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:341.77
  • IPN60090

    CAS:
    <p>IPN60090: potent oral GLS1 inhibitor, IC50 of 31 nM, potential for anticancer and immunomodulation.</p>
    Fórmula:C24H27F3N8O3
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:532.52
  • Imanixil

    CAS:
    <p>Imanixil boosts LDLR, cuts cholesterol and VLDL production, reducing atherosclerosis.</p>
    Fórmula:C17H17F3N6O2
    Pureza:>99.99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:394.35
  • Tamolarizine

    CAS:
    <p>Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.</p>
    Fórmula:C27H32N2O3
    Pureza:98.17%
    Cor e Forma:Soild
    Peso molecular:432.55
  • Pradefovir

    CAS:
    <p>Pradefovir (Remofovir) is a prodrug for chronic HBV, converting to PMEA in the liver with a Km of 60 μM and clearance of 359 ml/min.</p>
    Fórmula:C17H19ClN5O4P
    Pureza:97.50%
    Cor e Forma:Solid
    Peso molecular:423.79
  • Nanterinone

    CAS:
    <p>Nanterinone: oral phosphodiesterase inhibitor, improves acute heart failure hemodynamics.</p>
    Fórmula:C15H15N3O
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:253.3
  • Rbin-2

    CAS:
    <p>Rbin-2: Potent, selective Midasin inhibitor; reversible, cell-permeable; halts eukaryotic ribosome assembly.</p>
    Fórmula:C13H11BrN4S
    Pureza:98.75%
    Cor e Forma:Solid
    Peso molecular:335.22
  • CM037

    CAS:
    <p>CM037 (A-37) is a selective ALDH1A1 (acetaldehyde dehydrogenase 1A1) inhibitor (IC50; 4.6 µM) with antitumor activity and may be used in studies to eliminate</p>
    Fórmula:C21H25N3O3S2
    Pureza:99.34%
    Cor e Forma:Solid
    Peso molecular:431.57
  • CYP1B1-IN-4

    CAS:
    <p>CYP1B1-IN-4: 2,4-diarylthiazole, selective CYP1B1 inhibitor (IC50=0.2 nM), low cytotoxicity, stable in liver microsomes.</p>
    Fórmula:C18H14N2O2S
    Pureza:98.74%
    Cor e Forma:Solid
    Peso molecular:322.38
  • Tiapamil hydrochloride

    CAS:
    <p>Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity used in the study of angina pectoris.</p>
    Fórmula:C26H38ClNO8S2
    Pureza:99.17%
    Cor e Forma:Solid
    Peso molecular:592.16
  • alphaSYN-IN-NAB2

    CAS:
    <p>alphaSYN-IN-NAB2: a NAB2 gene protein guarding neurons against alpha-SYN harm; aids endosomal transport, cell processes, and can study various diseases.</p>
    Fórmula:C23H20ClN3O
    Pureza:98.49%
    Cor e Forma:Solid
    Peso molecular:389.88
  • Izonsteride

    CAS:
    <p>Izonsteride (LY320236) is a selective and potent 5alpha reductase inhibitor with dual action on the type I and type II isoforms of the enzyme.Izonsteride is</p>
    Fórmula:C24H26N2OS2
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:422.61
  • HTS07545

    CAS:
    <p>HTS07545, an SQOR inhibitor (IC50: 30nM), slows H2S breakdown, researched for heart failure.</p>
    Fórmula:C22H18N2O3
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:358.39
  • Qc1

    CAS:
    <p>Qc1 is an inhibitor of threonine dehydrogenase (TDH) inhibitor and can be used in studies about metabolic diseases.</p>
    Fórmula:C23H16F3N3O2S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:455.45
  • Atibeprone

    CAS:
    <p>Atibeprone is a MAO-B inhibitor with antidepressant activity for the study of Parkinson's disease.</p>
    Fórmula:C17H18N2O3S
    Pureza:99.18% - 99.86%
    Cor e Forma:Solid
    Peso molecular:330.4