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Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

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Foram encontrados 8597 produtos de "Metabolismo"

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  • HLF1-11

    CAS:
    <p>HLF1-11: human lactoferrin peptide, antimicrobial, inhibits MPO, steers monocytes to macrophages, boosts immunity.</p>
    Fórmula:C56H95N25O14S
    Cor e Forma:Solid
    Peso molecular:1374.58
  • HIV-1 inhibitor-58


    <p>HIV-1 Inhibitor-58 (Compound 10c) is a non-nucleoside reverse transcriptase inhibitor with broad-spectrum antiviral properties, effective against both wild-type</p>
    Fórmula:C26H24N6O2
    Cor e Forma:Solid
    Peso molecular:452.51
  • L-739750 2HCl


    <p>L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.</p>
    Fórmula:C23H41Cl2N3O6S2
    Pureza:98.69% - 99.16%
    Cor e Forma:Soild
    Peso molecular:590.62
  • PDE1-IN-8


    <p>PDE1-IN-8 (Compound 3f) acts as an inhibitor of PDE1, with an IC50 of 11 nM. It hinders cAMP and cGMP signaling pathways, impeding the differentiation and proliferation of cells into myofibroblasts, and demonstrates antifibrotic effects in the Bleomycin-induced rat model of pulmonary fibrosis.</p>
    Fórmula:C17H11Cl2N3OS2
    Cor e Forma:Solid
    Peso molecular:408.32
  • N,S-Bis-Fmoc-Glutathione

    CAS:
    <p>N,S-Bis-Fmoc-Glutathione is a potent inhibitor of glyoxalase II, exhibiting a K i of 0.32 mM [1].</p>
    Fórmula:C40H37N3O10S
    Cor e Forma:Solid
    Peso molecular:751.8
  • NDH-1 inhibitor-1

    CAS:
    <p>NDH-1 inhibitor-1 is an effective NDH-1 inhibitor, which can inhibit bovine SMP (mitochondrial granules), potato SMP and Escherichia coli, with pI50 values of &lt;</p>
    Fórmula:C20H19NO3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:321.37
  • PFKFB3-IN-2

    CAS:
    <p>PFKFB3-IN-2 is a 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 (PFKFB3) inhibitor.</p>
    Fórmula:C14H11NO7S
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:337.3
  • Pectin

    CAS:
    <p>Pectin, a plant cell wall derived heteropolysaccharide, forms nanoparticles for delivery and acts as an antimicrobial adsorbent.</p>
    Cor e Forma:Solid
  • SHP2-IN-37


    <p>SHP2-IN-37 (compound C5) is a potent allosteric inhibitor selective for SHP2, with an IC50 of 0.023 μM. It exhibits antiproliferative effects on KYSE-520 and MV-411 cells, with IC50 values of 6.97 μM and 0.67 μM, respectively.</p>
    Fórmula:C19H22Cl2N4O2S
    Cor e Forma:Solid
    Peso molecular:440.08405
  • FCPR03

    CAS:
    <p>FCPR03 is a selective inhibitor of phosphodiesterase 4 (PDE4) with IC50s of 31 nM, 47 nM, and 60 nM for PDE4B1, PDE4D7, and PDE4 catalytic domain, respectively.</p>
    Fórmula:C15H19F2NO3
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:299.31
  • 3-​Oxocholic acid

    CAS:
    <p>3-Oxocholic acid(3-Ketocholic acid) is the metabolite of bile acid and the main product of bile degradation by Clostridium perfringens in the intestine.3-</p>
    Fórmula:C24H38O5
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:406.56
  • (S)-Salsolidine

    CAS:
    <p>(S)-Salsolidine is a MAO inhibitor with Ki 63μM; its R enantiomer is more effective, Ki 26μM.</p>
    Fórmula:C12H17NO2
    Cor e Forma:Solid
    Peso molecular:207.27
  • Histamine glutarimide

    CAS:
    <p>Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.</p>
    Fórmula:C10H13N3O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:207.23
  • PK-10


    <p>PK-10, when combined with Fluconazole, exhibits potent synergistic antifungal activity against multiple Fluconazole-resistant Candida albicans strains.</p>
    Fórmula:C35H36F3N5O
    Cor e Forma:Solid
    Peso molecular:599.69
  • Dimethylaminomicheliolide HCl

    CAS:
    <p>Dimethylaminomicheliolide HCl has potential anti-inflammatory and anti-tumor activity and inhibits the proliferation of glioblastoma cells by targeting pyruvate</p>
    Fórmula:C17H28ClNO3
    Pureza:99.55%
    Cor e Forma:Soild
    Peso molecular:329.86
  • DSPE-PEG5000-R8


    <p>DSPE-PEG5000-R8 is a PEG compound composed of DSPE and the cell-penetrating peptide (R8). It is utilized for drug delivery applications.</p>
    Cor e Forma:Odour Solid
  • Kahalalide A

    CAS:
    <p>Kahalalide A has antimycobacterial activity isolated from the mollusk Elysia rufescens.</p>
    Fórmula:C46H67N7O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:894.08
  • GLX481369


    <p>GLX481369 is a redox-active substance that functions as an NOX4 inhibitor, exhibiting antioxidant effects [1].</p>
    Fórmula:C21H24ClN7O
    Cor e Forma:Solid
    Peso molecular:425.91
  • SPL-334

    CAS:
    <p>SPL-334 is an inhibitor of S-nitrosoglutathione reductase.</p>
    Fórmula:C22H15N3O3S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.50
  • Coenzyme A

    CAS:
    <p>Coenzyme A is an obligatory cofactor in all living cells synthesized from pantothenate (Vitamin B5), adenosine triphosphate (ATP), and cysteine.</p>
    Fórmula:C21H36N7O16P3S
    Pureza:93.84%
    Cor e Forma:Solid
    Peso molecular:767.53
  • FR106969

    CAS:
    <p>FR106969 is a platelet activating factor antagonist isolated from fungus with anti-inflammatory activity.</p>
    Fórmula:C16H22N2O3S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:354.49
  • Dextranase

    CAS:
    <p>Dextranase, a glucan hydrolase, breaks down α-(1,6)-glucosidic bonds in dextran, useful in food, sugar modification, medicine, and more.</p>
    Cor e Forma:Solid
  • Prolylglutamic acid

    CAS:
    <p>Prolylglutamic acid (H-Pro-Glu-OH) is a proline-glutamic acid dipeptide and endogenous metabolite, targeting the LipY lipase of pathogenic mycobacteria.</p>
    Fórmula:C10H16N2O5
    Cor e Forma:Solid
    Peso molecular:244.24
  • Isomer-Turosteride


    <p>Isomer-Turosteride, a novel 5α-reductase inhibitor, reduces prostate DHT and has anticancer properties without raising T levels.</p>
    Fórmula:C27H45N3O3
    Pureza:98.94%
    Cor e Forma:Solid
    Peso molecular:459.67
  • N-Fmoc-D-glutamine

    CAS:
    <p>N-Fmoc-D-glutamine is Fmoc-protected alpha-glutamine. Alpha-glutamine is an α-amino acid and the most abundant free amino acid in human blood.</p>
    Fórmula:C20H20N2O5
    Pureza:99.14%
    Peso molecular:368.38
  • Coprosterol

    CAS:
    <p>Coprosterol is a stanol formed from the biohydrogenation of cholesterol as a biomarker for the presence of human faecal matter in the environment.</p>
    Fórmula:C27H48O
    Cor e Forma:Solid
    Peso molecular:388.67
  • 1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol

    CAS:
    <p>1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol is a quinoxaline derivative and endogenous metabolite applicable to biochemical experiments and drug synthesis research.</p>
    Fórmula:C12H14N2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:250.25
  • L-Proline-15N

    CAS:
    <p>L-Proline-15N is an isotopically labeled amino acid suitable for metabolic research, aiding in the exploration of amino acid metabolism pathways and mechanisms.</p>
    Fórmula:C5H9NO2
    Cor e Forma:Solid
    Peso molecular:116.12
  • GQ-16

    CAS:
    <p>GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.</p>
    Fórmula:C19H16BrNO3S
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:418.3
  • 17β-HSD10-IN-1

    CAS:
    <p>17β-HSD10-IN-1 is a 17β-hydroxysteroid dehydrogenase type 10 inhibitor with blood-brain permeability and potency for the study of Alzheimer's disease.</p>
    Fórmula:C16H13ClN4O3S
    Pureza:98.47%
    Cor e Forma:Soild
    Peso molecular:376.82
  • Mavodelpar free acid hydrochloride


    <p>Mavodelpar free acid hydrochloride (Pparδ agonist HCl) is a potent PPARδ agonist.</p>
    Fórmula:C31H31ClFNO5
    Pureza:98.13%
    Cor e Forma:Soild
    Peso molecular:552.03
  • LH10


    <p>LH10 is an FXR agonist based on fexaramine, with an EC50 of 0.14 μM. It offers hepatoprotective effects, mitigating conditions such as cholestasis induced by alpha naphthylisothiocyanate (ANIT), acute liver injury caused by APAP, and non-alcoholic steatohepatitis (NASH).</p>
    Fórmula:C34H33N3O2
    Cor e Forma:Solid
    Peso molecular:515.64
  • (+)-Menthofuran


    <p>(+)-Menthofuran is a useful organic compound for research related to life sciences and the catalog number is T125544.</p>
    Fórmula:C10H14O
    Cor e Forma:Solid
    Peso molecular:150.221
  • γ-glutamyltransferase

    CAS:
    <p>γ-glutamyltransferase (GGT) is an enzyme located on the outer surface of the cell membrane. It maintains physiological concentrations of intracellular glutathione and cellular defense against oxidative stress by cleaving extracellular glutathione and increasing the availability of amino acids. γ-glutamyltransferase can be utilized as a biomaterial or organic compound in life science-related research.</p>
    Cor e Forma:Solid
  • Beauverolide Ja

    CAS:
    <p>Beauverolide Ja: cyclotetradepsipeptide, CaM inhibitor; Kd 0.078 μM, Ki 0.39 μM; from Isaria fumosorosea.</p>
    Fórmula:C35H46N4O5
    Cor e Forma:Solid
    Peso molecular:602.76
  • Cefetamet Hydrochloride

    CAS:
    <p>Cefetamet is a potent antibiotic to treat respiratory and urinary tract infections.</p>
    Fórmula:C14H16ClN5O5S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.89
  • (±)-threo-3-Methylglutamic acid

    CAS:
    <p>glutamate transport blocker</p>
    Fórmula:C6H11NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:161.16
  • ML162-yne

    CAS:
    <p>ML162-yne is an effective GPX4 inhibitor affinity probe with click chemistry properties. The compound contains an alkyne group capable of reacting with azide-containing molecules through a copper-catalyzed azide-alkyne cycloaddition reaction (CuAAc), making it suitable for protein labeling and related studies.</p>
    Fórmula:C25H22Cl2N2O3S
    Cor e Forma:Solid
    Peso molecular:501.43
  • Neogen

    CAS:
    <p>Neogen, also known as Jadinol PU, is a drug potentially for the restoration of the immune system and hemopoiesis after cytostatics treatment.</p>
    Fórmula:C22H30N4O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:446.50
  • AUPF02

    CAS:
    <p>AUPF02, a 5-aryluracil derivative, is an effective anti-breast cancer compound with an IC50 value of 23.4 µM against MCF-7 cells.</p>
    Fórmula:C14H9F5N2O
    Cor e Forma:Solid
    Peso molecular:316.23
  • PF-1355

    CAS:
    <p>PF-1355 (PF 06281355) is a selective 2-thiouracil mechanism-based MPO inhibitor. PF-1355 is used for treatment of vasculitic diseases.</p>
    Fórmula:C14H15N3O4S
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:321.35
  • α-Amylase-IN-4


    <p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>
    Cor e Forma:Odour Solid
  • TRH Precursor Peptide


    <p>Thyrotropin Releasing Hormone Precursor Peptide</p>
    Fórmula:C42H75N19O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1006.17
  • EDDA

    CAS:
    <p>Ethylenediaminediacetic acid is derived from two molecules of glycine linked by amines.</p>
    Fórmula:C6H12N2O4
    Cor e Forma:Solid
    Peso molecular:176.17
  • Bazinaprine

    CAS:
    <p>Bazinaprine is a selective, reversible monoamine oxidase inhibitor (MAOI) that is a candidate compound for the treatment of depression.</p>
    Fórmula:C17H19N5O
    Pureza:99.65% - 99.93%
    Cor e Forma:Solid
    Peso molecular:309.37
  • Fmoc-L-Proline

    CAS:
    <p>Fmoc-L-Proline (Fmoc-Pro-OH) is a proline derivative.</p>
    Fórmula:C20H19NO4
    Pureza:99.22%
    Cor e Forma:Solid
    Peso molecular:337.37
  • Nedosiran sodium

    CAS:
    <p>Nedosiran sodium, a GalNAc-dsRNA conjugate, is engineered to suppress the synthesis of the hepatic lactate dehydrogenase (LDH) enzyme.</p>
    Cor e Forma:Solid
  • 2-Pentyl-1H-benzo[d]imidazole

    CAS:
    <p>2-Pentyl-1H-benzo[d]imidazole is a micromolar level inhibitor of Cytochrome P450 1A1 and 2B1 and has antibacterial activity against Fusarium verticillioides.</p>
    Fórmula:C12H16N2
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:188.27
  • Thalifendine chloride

    CAS:
    <p>Thalifendine chloride is a metabolite of berberine,the methoxy group at the C-10 position undergoes demethylation by CYP51. cytotoxicity against P-388 cells.</p>
    Fórmula:C19H16ClNO4
    Cor e Forma:Solid
    Peso molecular:357.79
  • FASN-IN-4 tosylate

    CAS:
    <p>FASN-IN-4 tosylate: Fatty acid synthase inhibitor, IC50 10 nM; blocks SARS-CoV-2, EC50 18.6 nM.</p>
    Fórmula:C33H35N3O7S2
    Cor e Forma:Solid
    Peso molecular:649.78
  • [(3R)-3-Hydroxydodecanoyl]-L-carnitine

    CAS:
    <p>[(3R)-3-Hydroxydodecanoyl]-L-carnitine is an endogenous metabolite[1].</p>
    Fórmula:C19H37NO5
    Cor e Forma:Solid
    Peso molecular:359.50
  • CC618

    CAS:
    <p>CC618 is a selective PPARβ/δ antagonist with an IC50 of 10.0 μM.</p>
    Fórmula:C20H15F6N3O3S2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:523.47
  • Nattokinase

    CAS:
    <p>Nattokinase is a serine protease derived from nattō, oral, fibrinolytic/anticoagulant properties. It degrades fibrin, fibrinolytic substrates, and PAI-1.</p>
    Cor e Forma:Solid
  • PR280


    <p>PR280 is a potent inhibitor of dihydroceramide desaturase 1 (Des1) with an IC50 of 700 nM. It forms hydrogen bonds with amino acid residues of Des1, while its cyclopropenone group may coordinate with the iron center, stabilizing its binding at Des1's active site. This inhibits the ceramide biosynthesis pathway, preventing dihydroceramide (dhCer) from converting into ceramide. PR280 can be used in research related to sphingolipid metabolism disorders, including cancer and metabolic diseases.</p>
    Fórmula:C27H49NO4
    Peso molecular:451.36616
  • Butyryl-Coenzyme A trisodium


    <p>Butyryl-Coenzyme A (trisodium) is a microbial metabolite that can be synthesized into butyric acid or butyrate.</p>
    Fórmula:C25H39N7Na3O17P3S
    Peso molecular:903.10291
  • Conagenin

    CAS:
    <p>Conagenin is a small molecular immunomodulator isolated by Streptomyces roseosporus.</p>
    Fórmula:C10H19NO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:249.26
  • γ-Acetylenic GABA hydrochloride

    CAS:
    <p>γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.</p>
    Fórmula:C6H10ClNO2
    Pureza:99.28% - 99.64%
    Cor e Forma:Solid
    Peso molecular:163.6
  • PDE12-IN-1

    CAS:
    <p>PDE12-IN-1, a potent PDE12 inhibitor with a pIC50 of 9.1, increases 2-5A, has a pEC50 of 7.7, and shows antiviral properties.</p>
    Fórmula:C31H27BrFN5O3
    Cor e Forma:Solid
    Peso molecular:616.491
  • N-acetyl Dapsone

    CAS:
    <p>N-acetyl Dapsone is an anti-inflammatory and antimicrobial compound widely used in the treatment of leprosy, malaria, acne and various immune disorders.</p>
    Fórmula:C14H14N2O3S
    Pureza:99.86%
    Cor e Forma:White
    Peso molecular:290.34
  • CB 300919

    CAS:
    <p>CB 300919, a quinazoline antitumor, inhibits CH1 ovarian tumor growth (IC50: 2 nM) over 96h.</p>
    Fórmula:C32H34ClN7O2
    Cor e Forma:Solid
    Peso molecular:584.11
  • SGK1-IN-3 hydrochloride


    <p>SGK1-IN-3 hydrochloride (compound 3a) is an efficacious, orally bioavailable SGK1 inhibitor. The serine/threonine kinase SGK1 acts as an activator of the β-catenin pathway and strongly stimulates cartilage degradation, being upregulated under genomic control in diseased osteoarthritic cartilage. SGK1-IN-3 hydrochloride holds potential for osteoarthritis research.</p>
    Fórmula:C23H21Cl3N6O3S
    Peso molecular:566.04614
  • Transketolase-IN-6


    <p>Transketolase-IN-6 (Compound 6bj) serves as a lead compound for herbicides. It achieves approximately 80% root inhibition in redroot pigweed (Amaranthus retroflexus) and green foxtail (Setaria viridis). Moreover, Transketolase-IN-6 is an effective inhibitor of transketolase (TK).</p>
    Fórmula:C23H27ClN6O
    Peso molecular:438.19349
  • AChE/BChE-IN-17


    <p>AChE/BChE-IN-17 (compound 8m) is a potent inhibitor of AChE and BChE, displaying IC50 values of 125.06 nM and 119.68 nM, respectively. Additionally, AChE/BChE-IN-17 inhibits α-glucosidase, with an IC50 of 41050 nM.</p>
    Fórmula:C28H25N3O4
    Peso molecular:467.18451
  • α-Glucosidase-IN-67


    <p>α-Glucosidase-IN-67 (compound 5k) is a potent inhibitor of α-glucosidase, exhibiting IC50 values of 0.31 µM for α-glucosidase and 4.51 µM for α-amylase. This compound shows potential for research in type 2 diabetes.</p>
    Fórmula:C24H22BrN3O3S
    Peso molecular:511.05653
  • CAXII-IN-2


    <p>CAXII-IN-2 (compound 3j) is a highly effective inhibitor of CAXII. It demonstrates inhibitory activity against CA IX and CAXII, with Ki values of 27.4 nM and 4.0 nM, respectively.</p>
    Fórmula:C16H13FNO4P
    Cor e Forma:Solid
    Peso molecular:333.05662
  • (±)14-HDHA

    CAS:
    <p>(±)14-HDHA is an oxidized metabolite of DHA and can be further oxidized to the 14-oxoDHA, 14-HDoHE inhibits LPS-induced IL-6 mRNA expression.</p>
    Fórmula:C22H32O3
    Cor e Forma:Solid
    Peso molecular:344.49
  • 9(S)-HODE cholesteryl ester

    CAS:
    <p>9(S)-HODE cholesteryl ester, from atherosclerotic lesions, has an uncertain origin and serves as a standard for chiral ester analysis.</p>
    Fórmula:C45H76O3
    Cor e Forma:Solid
    Peso molecular:665.1
  • α-Amylase/α-Glucosidase-IN-11


    <p>α-Amylase/α-Glucosidase-IN-11 (Compound 5d) is an isoxazoline-indigo hybrid with notable antidiabetic properties. It acts as a competitive inhibitor of the key digestive enzymes α-amylase (IC50 = 30.39 μM) and α-glucosidase (IC50 = 65.1 μM). Additionally, it does not penetrate the blood-brain barrier.</p>
    Fórmula:C33H40ClN5O5
    Peso molecular:621.2718
  • ROC-0929

    CAS:
    <p>ROC-0929 (13a) is a selective sPLA2 inhibitor with IC50 of 80 nM, targeting hGX and blocking ERK1/2, p-38 phosphorylation for inflammation research.</p>
    Fórmula:C30H31N3O6S
    Cor e Forma:Solid
    Peso molecular:561.65
  • Phosphoramidon

    CAS:
    <p>Phosphoramidon inhibits metallo-endopeptidase, endothelin-converting enzyme, and thermolysin; derived from Streptomyces tanashiensis culture.</p>
    Fórmula:C23H34N3O10P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:543.5
  • Acetildenafil

    CAS:
    <p>Acetildenafil is an analog of the phosphodiesterase inhibitor sildenafil.</p>
    Fórmula:C25H34N6O3
    Cor e Forma:Off-White To Pale Yelow Solid
    Peso molecular:466.58
  • Diaphorase

    CAS:
    <p>Diaphorase from anaerobic sludge catalyzes RDX biotransformation via denitrification.</p>
    Cor e Forma:Solid
  • Impurity F of Calcipotriol

    CAS:
    <p>Impurity F of Calcipotriol is a impurity of Calcipotriol. Calcipotriol (MC 903; Calcipotriene) is a ligand of VDR-like receptors.</p>
    Fórmula:C39H68O3Si2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:641.13
  • hCYP3A4-IN-1


    <p>hCYP3A4-IN-1 (compound C6) is a potent, orally active inhibitor of hCYP3A4, exhibiting IC50 values of 43.93 nM in human liver microsomes (HLMs) and 153.00 nM in</p>
    Cor e Forma:Odour Solid
  • α-Glucosidase-IN-60


    <p>α-Glucosidase-IN-60 (Compound 5k) acts as a competitive inhibitor of α-Glucosidase, with an IC50 of 10.8 μM.</p>
    Fórmula:C23H14N2O5
    Peso molecular:398.09027
  • α-Amylase/α-Glucosidase-IN-16


    <p>α-Amylase/α-Glucosidase-IN-16 (compound 15) is a potent dual inhibitor of α-amylase and α-glucosidase, with IC50 values of 0.8 μM and 1.2 μM, respectively. It is applicable for research in diabetes (DM).</p>
    Fórmula:C16H9Cl2F3N4S
    Peso molecular:415.98771
  • LYP-8


    <p>LYP-8 is a potent NAMPT degrader that achieves a maximum degradation rate of 97% in NAMPT within SKOV-3 cells at a concentration of 0.5 μM. LYP-8 also demonstrates anticancer activity both in vitro and in vivo.</p>
    Fórmula:C56H74N8O10S
    Peso molecular:1050.52486
  • α-Glucosidase-IN-46


    <p>α-Glucosidase-IN-46 is a potent inhibitor of α-glucosidase, with an IC50 of 26.0 μM. This compound is applicable in the research of Type 2 diabetes.</p>
    Fórmula:C35H32N4O5
    Peso molecular:588.23727
  • hCAIX/XII-IN-11


    <p>hCAIX/XII-IN-11 (Compound 6c) is an inhibitor of hCA IX and hCA XII, exhibiting Ki values of 0.7 μM for both isoforms. This compound is applicable in cancer research.</p>
    Fórmula:C13H10FN3O4
    Peso molecular:291.06553
  • MTHFD2-IN-3


    <p>MTHFD2-IN-3 (compound 10), a potent inhibitor of methylenetetrahydrofolate dehydrogenase (MTHFD2), demonstrates significant efficacy in obstructing the activity</p>
    Fórmula:C22H19NO7S
    Cor e Forma:Solid
    Peso molecular:441.45
  • DSPE-PEG5000-VIP


    <p>DSPE-PEG5000-PP1 is a PEG compound composed of DSPE and the cell-penetrating peptide (TAT) peptide. DSPE-PEG2000-TAT is applicable for drug delivery.</p>
    Cor e Forma:Odour Solid
  • Poststatin

    CAS:
    <p>Poststatin is a prolyl endopeptidase inhibitor produced by Streptomyces viridochromogenes MH534-30F3.</p>
    Fórmula:C26H47N5O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:541.69
  • α-Glucosidase-IN-49


    <p>α-Glucosidase-IN-49 (compound C23) is a potent inhibitor of α-Glucosidase, with an IC50 of 0.52 μM. This compound exhibits oral bioactivity, effectively lowering blood glucose levels and enhancing glucose tolerance in mice.</p>
    Fórmula:C21H13F3N4O3S3
    Peso molecular:522.01019
  • α-Amylase/α-Glucosidase-IN-13


    <p>α-Amylase/α-Glucosidase-IN-13 (Compound 5d) is a dual inhibitor of α-amylase and α-glucosidase, and is useful in diabetes research.</p>
    Fórmula:C22H16N2O5
    Peso molecular:388.10592
  • Pantothenoylcysteine

    CAS:
    <p>Pantothenoylcysteine is a bioactive chemical.</p>
    Fórmula:C12H22N2O6S
    Cor e Forma:Solid
    Peso molecular:322.38
  • LTA4H-IN-4


    <p>LTA4H-IN-4 (compound 3) is an orally active inhibitor of LTA4H. It exhibits an IC50 value of 156 μM against hERG and is applicable for inflammation-related research.</p>
  • Abiraterone N-oxide

    CAS:
    <p>Abiraterone N-oxide is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .</p>
    Fórmula:C24H31NO2
    Cor e Forma:Solid
    Peso molecular:365.51
  • Hydroxy desmethyl Bosentan

    CAS:
    <p>Hydroxy desmethyl Bosentan (Ro 64-105) is a Bosentan metabolism produced by the cytochrome P450 enzymes CYP2C9 and CYP3A4 in the liver.</p>
    Fórmula:C26H27N5O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:553.59
  • Retinyl glucoside

    CAS:
    <p>Retinyl-β-D-glucoside, a biologically active metabolite of vitamin A, naturally occurs in fish and mammals.</p>
    Fórmula:C26H40O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:448.59
  • DSPE-PEG-Maleimide (MW 3400) ammonium


    <p>DSPE-PEG-Maleimide (MW 3400) ammonium combines DSPE phospholipids with maleimide for the preparation of nanostructured lipid carriers. It is applicable in drug delivery research.</p>
    Cor e Forma:Odour Solid
  • Antibacterial agent 218


    <p>Antibacterialagent 218 (compound d28) is an orally active inhibitor of sterol 24-C-methyltransferase with an IC50 value of 0.273 μM. It also displays antifungal activity against Candida albicans SC5314, with an IC50 of 0.25 μg/mL.</p>
    Fórmula:C30H24N4OS
    Peso molecular:488.16708
  • IDO1-IN-24


    <p>IDO1-IN-24 (compound 2c) inhibits the production of IDO1 during cell assays, with an IC50 value of 17 μM.</p>
    Fórmula:C18H22N2O4
    Peso molecular:330.15796
  • Triethyl phosphate

    CAS:
    <p>Triethyl phosphate is a chemical compound. It can be called "phosphoric acid, triethyl ester".</p>
    Fórmula:C6H15O4P
    Pureza:98%
    Cor e Forma:Clear Liquid
    Peso molecular:182.16
  • MAGL-IN-5

    CAS:
    <p>MAGL-IN-5 is a non-selective lipase inhibitor.</p>
    Fórmula:C18H17N3O5
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:355.34
  • Boc-Ile-Glu-Gly-Arg-AMC

    CAS:
    <p>Boc-IEGR-AMC: fluorogenic substrate for factor Xa and Halocynthia roretzi acrosin.</p>
    Fórmula:C34H50N8O10
    Pureza:98%
    Cor e Forma:White Powder
    Peso molecular:730.81
  • N-Nitrosoglyphosate sodium

    CAS:
    <p>N-Nitrosoglyphosate sodium, a nitrosamine degradation product and synthetic impurity of glyphosate herbicide [1], is a chemical compound resulting from the</p>
    Fórmula:C3H6N2NaO6P
    Cor e Forma:Solid
    Peso molecular:220.05
  • Beauveriolide I

    CAS:
    <p>Beauveriolide I, a cyclodepsipeptide from Beauveria, inhibits lipid droplet and cholesterol synthesis in mouse macrophages; IC50=0.78 μM.</p>
    Fórmula:C27H41N3O5
    Cor e Forma:Solid
    Peso molecular:487.63
  • Metabolism Compound Library


    <p>A unique collection of xnum metabolic pathway-related bioactive small molecule compounds for high-throughput, high-content screening.</p>
    Cor e Forma:Liquid
  • Biotin sodium

    CAS:
    <p>Biotin (Vitamin B7) sodium aids in metabolism, cell growth, fatty acid synthesis, and gluconeogenesis.</p>
    Fórmula:C10H15N2NaO3S
    Cor e Forma:Solid
    Peso molecular:266.29
  • Hepaxanthin

    CAS:
    <p>Hepaxanthin is a carotenoid.</p>
    Fórmula:C20H30O2
    Cor e Forma:Solid
    Peso molecular:302.45
  • (±)9-HODE cholesteryl ester

    CAS:
    <p>(±)9-HODE cholesteryl ester was originally extracted from atherosclerotic lesions and shown to be produced by Cu2+-catalyzed oxidation of LDL.</p>
    Fórmula:C45H76O3
    Cor e Forma:Solid
    Peso molecular:665.1
  • Hexokinase II VDAC binding domain peptide, cell-permeable


    <p>HexokinaseIIVDACbinding domain peptide (Hxk2VBD peptide) is a cell-permeable peptide derived from the hexokinase II VDAC binding domain. This peptide inhibits the mitochondrial localization of hexokinase 2 (HXK2) and also suppresses neurotrophic factor-induced axon growth.</p>
    Fórmula:C188H291N53O40S2
    Peso molecular:3995.18073
  • Lurasidone Metabolite 14283 hydrochloride

    CAS:
    <p>Lurasidone Metabolite 14283 hydrochloride is a major active metabolite of Lurasidone.</p>
    Fórmula:C28H37ClN4O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:545.14
  • Tuftsin diacetate

    CAS:
    <p>Tuftsin diacetate, Thr-Lys-Pro-Arg, activates macrophages/microglia; it's in immunoglobulin G's Fc and boosts immunity.</p>
    Fórmula:C25H48N8O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:620.7
  • DSPE-PEG1000-APRPG


    <p>DSPE-PEG1000-APRPG is a PEG compound composed of DSPE and the APRPG peptide. It is applicable for drug delivery.</p>
    Cor e Forma:Odour Solid
  • (S,R,S)-AHPC-C2-amide-benzofuranylmethyl-pyridine

    CAS:
    <p>(S,R,S)-AHPC-C2-amide targets Smad3 degradation and boosts HIF-α; it has anti-fibrotic and renal protective roles.</p>
    Fórmula:C41H46N6O6S
    Cor e Forma:Solid
    Peso molecular:750.91
  • Tetomilast

    CAS:
    <p>Tetomilast (OPC-6535) is a phosphodiesterase-4 (PDE4) inhibitor, potentially effective in treating inflammatory bowel disease (IBD) and chronic obstructive</p>
    Fórmula:C19H18N2O4S
    Cor e Forma:Solid
    Peso molecular:370.42
  • Zymostenol

    CAS:
    <p>Zymostenol (5a-Cholest-8-en-3b-ol) is a RORγ agonist with an EC50 of 1 μM.Zymostenol is a late stage precursor of cholesterol biosynthesis.</p>
    Fórmula:C27H46O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.65
  • Ascorbate oxidase

    CAS:
    <p>Ascorbate oxidase, a REDOX enzyme, catalyzes ascorbic acid and oxygen to dehydroascorbic acid, regulating the extracellular matrix.</p>
    Cor e Forma:Solid
  • Asundexian

    CAS:
    <p>Asundexian (BAY-2433334) is a potent and orally active inhibitor of the coagulation factor FXIa that directly and reversibly binds to the active site of FXIa,</p>
    Fórmula:C26H21ClF4N6O4
    Pureza:99.89% - 99.90%
    Cor e Forma:Solid
    Peso molecular:592.93
  • Impurity C of Alfacalcidol

    CAS:
    <p>Impurity of Alfacalcidol is an impurity of Alfacalcidol. Alfacalcidol is a non-selective VDR activator medication.</p>
    Fórmula:C35H49N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:575.78
  • Bacterial α-Amylase

    CAS:
    <p>Bacterial α-Amylase is an enzyme that catalyzes the hydrolysis reaction of starch into smaller sugar molecules such as maltose and glucose.</p>
    Cor e Forma:Solid
  • LDHA-IN-3

    CAS:
    <p>LDHA-IN-3 is a potent selenobenzene-based LDHA inhibitor with a 145.2 nM IC50, useful in cancer research.</p>
    Fórmula:C13H9F3Se
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:301.17
  • N-acetyl Leukotriene E4

    CAS:
    <p>N-acetyl Leukotriene E4 is an endogenous metabolite of Leukotriene E4, less active than Leukotriene E4, causing constriction of the airways.</p>
    Fórmula:C25H39NO6S
    Cor e Forma:Solid
    Peso molecular:481.65
  • RXP-407

    CAS:
    <p>RXP 407 selectively inhibits ACE N-domain, preserving acetyl-Ser-Asp-Lys-Pro and not affecting angiotensin I in vivo.</p>
    Fórmula:C21H31N4O8P
    Cor e Forma:Solid
    Peso molecular:498.47
  • TEI-9647

    CAS:
    <p>TEI-9647 is a vitamin D3 analog and VDR/DRE genomic antagonist.</p>
    Fórmula:C27H38O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:426.59
  • Sulotroban potassium


    <p>Sulotroban potassium is a small molecule thromboxane A2 receptor (TXA2R) antagonist that can be used to study myocardial infarction and thrombosis.</p>
    Fórmula:C16H16KNO5S
    Pureza:98.02%
    Cor e Forma:Soild
    Peso molecular:373.46
  • Ser-Ala-alloresact acetate


    <p>Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.</p>
    Fórmula:C44H75N13O16S2
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:1106.28
  • Axl-IN-16


    <p>Axl-IN-16, a dual Axl/HIF inhibitor, promotes Flammulina velutipes fruiting body formation and suppresses hypoxia-inducible factor activity along with receptor</p>
    Fórmula:C14H19ClO8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:350.75
  • α-Amylase/α-Glucosidase-IN-14


    <p>α-Amylase/α-Glucosidase-IN-14 is an orally bioactive inhibitor of α-amylase and α-glucosidase, with IC50 values of 45.53 μM and 27.73 μM, respectively.</p>
    Fórmula:C24H19FN4O2S
    Peso molecular:446.12128
  • Pestalotin

    CAS:
    <p>Pestalotin, a fungal derivative, promotes rice seedling growth and sugar release, has antifungal properties, and is cytotoxic to certain cells.</p>
    Fórmula:C11H18O4
    Cor e Forma:Solid
    Peso molecular:214.26
  • SGK1-IN-4

    CAS:
    <p>SGK1-IN-4 is a selective inhibitor of SGK1 and can be used in studies about osteoarthritis.</p>
    Fórmula:C23H21ClFN5O4S
    Pureza:97.03%
    Cor e Forma:Solid
    Peso molecular:517.96
  • Galactose 1-phosphate

    CAS:
    <p>Galactose 1-phosphate, an intermediate substance in both galactose metabolism and nucleotide sugar processes, plays a crucial role in the biochemical pathways</p>
    Fórmula:C6H13O9P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:260.14
  • AP-III-a4 hydrochloride

    CAS:
    <p>AP-III-a4 hydrochloride (ENOblock hydrochloride) is a direct enolase (enolase) inhibitor that inhibit metastasis and affect glucose homeostasis.</p>
    Fórmula:C31H44ClFN8O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:631.18
  • Aldosterone-d8

    CAS:
    <p>Aldosterone D8, a deuterium-labeled variant of Aldosterone produced in the adrenal zona glomerulosa, regulates blood pressure.</p>
    Fórmula:C21H28O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:368.49
  • DSPE-PEG1000-LyP-1


    <p>DSPE-PEG1000-LyP-1 is a PEG compound composed of DSPE and a nine-residue peptide (LyP-1). LyP-1 specifically targets tumor-associated lymphatic vessels and macrophages.</p>
    Cor e Forma:Odour Solid
  • (S)-3-Thienylglycine

    CAS:
    <p>(S)-3-Thienylglycine is a thiophene derivative and can be used to investigate the genotoxicity of the similar structures with thiophene derivatives.</p>
    Fórmula:C6H7NO2S
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:157.19
  • tetranor-PGAM

    CAS:
    <p>PGE2 is a biomarker for inflammation and disease; its unstable urinary metabolite, tetranor-PGEM, and its byproduct, tetranor-PGAM, indicate biosynthesis.</p>
    Fórmula:C16H22O6
    Cor e Forma:Solid
    Peso molecular:310.346
  • 3-HIB

    CAS:
    <p>3-HIB is a paracrine regulator of transendothelial fatty acid transport.</p>
    Fórmula:C4H7NaO3
    Cor e Forma:Solid
    Peso molecular:126.09
  • Avenacin A 1

    CAS:
    <p>Avenacin A 1 is a biochemical.</p>
    Fórmula:C55H83NO21
    Cor e Forma:Solid
    Peso molecular:1094.255
  • α-Glucosidase-IN-58


    <p>α-Glucosidase-IN-58 (Compound 6d) is an α-glucosidase inhibitor with an IC50 of 1.47 μM.</p>
    Fórmula:C22H13F3N2OS
    Peso molecular:410.07007
  • ALR2-IN-1

    CAS:
    <p>ALR2-IN-1: potent, selective inhibitor of ALR2 (IC50=1.42 μM), antiglycemic, antioxidant; for diabetes research.</p>
    Fórmula:C16H17N3O2S
    Pureza:98.79%
    Cor e Forma:Soild
    Peso molecular:315.39
  • (Rac)-5-Keto Fluvastatin

    CAS:
    <p>(Rac)-5-Keto Fluvastatin (rac 5-Keto Fluvastatin) is an impurity of Fluvastatin which is an inhibitor of HMG-CoA reductase.</p>
    Fórmula:C24H24FNO4
    Pureza:95.04%
    Cor e Forma:Solid
    Peso molecular:409.45
  • 3-O-(2-Aminoethyl)-25-hydroxyvitamin D3

    CAS:
    <p>3-O-(2-Aminoethyl)-25-hydroxyvitamin D3 is a Vitamin D3 derivative.</p>
    Fórmula:C30H51NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:457.743
  • BSO-07


    <p>BSO-07 is a ROS/JNK activator that exhibits potent anti-cancer properties, demonstrated by an IC50 of 24.81 μM in human breast cancer (BC) cells. The mechanism of action for BSO-07 involves JNK activation and the promotion of increased ROS levels, which lead to the induction of apoptosis (Apoptosis) and tumorigenic apoptosis. This includes enhanced expression of apoptosis-related proteins such as PARP, Bax, phosphorylated p53, ATF4, and CHOP, along with a reduction in the levels of anti-apoptotic proteins (e.g., Bcl-2, Bcl-xL, and Survivin). BSO-07 holds promise for research in the field of breast cancer.</p>
    Cor e Forma:Odour Solid
  • hBChE-IN-3


    <p>hBChE-IN-3 (compound 30) serves as both an activator of carbonic anhydrase (CA) and an inhibitor of cholinesterase (ChE), exhibiting IC50 values of 7.4 nM for AchE and 1.9 nM for BchE. This compound is utilized in the research of neurodegenerative and psychiatric disorders.</p>
    Cor e Forma:Odour Solid
  • CAIX/CAXII-IN-3


    <p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>
    Cor e Forma:Odour Solid
  • β-Glucosidase

    CAS:
    <p>β-Glucosidase is a glucoside bond hydrolase involved in glucose metabolism and can be used to study diseases caused by abnormal glucose metabolism.</p>
    Fórmula:C24H44O12
    Cor e Forma:Solid
    Peso molecular:524.6
  • SAICAR

    CAS:
    <p>SAICAR is an intermediate of de novo purine nucleotide biosynthesis, activates pyruvate kinase isoform M2 (PKM2) in an isozyme-selective manner (EC50: 0.3 mM).</p>
    Fórmula:C13H19N4O12P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:454.28
  • NLG802

    CAS:
    <p>NLG802 is a prodrug of indoximod, an orally active indoleamine 2,3-dioxygenase (IDO) inhibitor.</p>
    Fórmula:C20H30ClN3O3
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:395.92
  • NF-κB/HIF-1α-IN-1


    <p>NF-κB/HIF-1α-IN-1 (compound 9c) effectively inhibits the NF-κB activation pathway and demonstrates selective antifibrotic activity. This compound exhibits no significant cytotoxicity in NCI tumor cell lines. In rat models, NF-κB/HIF-1α-IN-1 successfully ameliorates liver fibrosis, suppresses the expression levels of NF-κB and HIF-1α, and induces Nrf2.</p>
    Fórmula:C24H27N7O4
    Cor e Forma:Solid
    Peso molecular:477.21245
  • Saccharopine

    CAS:
    <p>L-Saccharopine is a product of the breakdown of essential amino acid Lysine.</p>
    Fórmula:C11H20N2O6
    Cor e Forma:Solid
    Peso molecular:276.29
  • Hydroxy bosentan

    CAS:
    <p>Hydroxy bosentan (Ro 48-5033), a Bosentan metabolite, is liver-processed with 10-20% of its activity.</p>
    Fórmula:C27H29N5O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:567.61
  • Xanthine oxidase-IN-16


    <p>Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.</p>
    Cor e Forma:Odour Solid
  • Isodihydroauroglaucin

    CAS:
    <p>Isodihydroauroglaucin is a useful organic compound for research related to life sciences. The catalog number is T124274 and the CAS number is 74886-31-0.</p>
    Fórmula:C19H24O3
    Cor e Forma:Solid
    Peso molecular:300.398
  • WXC-25


    <p>WXC-25 is an α-glucosidase inhibitor with an IC50 value of 2.02 μM.</p>
    Cor e Forma:Odour Solid
  • 10(S),17(S)-DiHDHA

    CAS:
    <p>Protectin D1, or neuroprotectin D1 in neurons, is anti-inflammatory. 10(S),17(S)-DiHDHA, also PDX, differs in structure and inhibits neutrophils and platelets.</p>
    Fórmula:C22H32O4
    Cor e Forma:Solid
    Peso molecular:360.494
  • α-Amylase/α-Glucosidase-IN-9


    <p>α-Amylase/α-Glucosidase-IN-9 (compound 5h) is a dual inhibitor of α-amylase (IC50= 16.4 μM) and α-glucosidase (IC50= 31.6 μM).</p>
    Fórmula:C20H16ClN5O4
    Peso molecular:425.08908
  • Resveratrol-3-O-sulfate sodium

    CAS:
    <p>Resveratrol-3-O-sulfate reduces IL-1α/β, IL-6, TNF-α in LPS-stimulated U-937 cells, inhibits Caco-2 cell growth, induces apoptosis, and binds mitoNEET.</p>
    Fórmula:C14H11NaO6S
    Cor e Forma:Solid
    Peso molecular:330.29
  • α-Amylase/α-Glucosidase-IN-15


    <p>α-Amylase/α-Glucosidase-IN-15 (compound 6C) is an orally active inhibitor of α-glucosidase (α-Glucosidase) and α-amylase (α-amylase), with IC50 values of 21 μM and 61 μM, respectively.</p>
    Fórmula:C26H24N4O3S
    Peso molecular:472.15691
  • 1-Naphthyl 3,5-dinitrobenzoate

    CAS:
    <p>1-Naphthyl 3,5-dinitrobenzoate (JMC-4) is an inhibitor of 5-LOX can be used in studies about inflammatory therapy.</p>
    Fórmula:C17H10N2O6
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:338.27
  • hCAIX/XII-IN-14


    <p>hCAIX/XII-IN-14 (Compound 1i) is an inhibitor of hCAIX and hCAXII, with Ki values of 9.4 nM for hCAII, 5.6 nM for hCAIX, and 6.3 nM for hCAXII.</p>
    Fórmula:C16H14F3N3O4S
    Cor e Forma:Solid
    Peso molecular:401.36
  • Mevinolinic acid

    CAS:
    <p>Mevinolinic acid is an active metabolite of Lovastatin. Lovastatin is an HMG-CoA reductase inhibitor.</p>
    Fórmula:C24H38O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:422.562
  • SX29


    <p>SX29 is a non-competitive α-glucosidase inhibitor with oral activity, exhibiting an IC50 of 2.12 μM. It possesses hypoglycemic properties; oral administration of SX29 reduces blood glucose levels and enhances glucose tolerance in diabetic mice.</p>
    Cor e Forma:Odour Solid
  • α-Glucosidase-IN-74


    <p>α-Glucosidase-IN-74, a nicotinamide-thiazole derivative, functions as an α-glucosidase (α-glucosidase) inhibitor. It demonstrates antidiabetic activity by reducing blood glucose and triglyceride levels in Streptozotocin-induced diabetic animals.</p>
    Cor e Forma:Odour Solid
  • WVSAV


    <p>WVSAV is a ligand for the PDZ2 domain (tyrosine phosphatase) with a dissociation constant (Kd) of 111 μM. It is utilized in studies of protein-ligand interactions.</p>
    Fórmula:C27H40N6O7
    Cor e Forma:Solid
    Peso molecular:560.64
  • Seco Rapamycin ethyl ester


    <p>Seco Rapamycin ethyl ester, an open-ring metabolite of the Rapamycin derivative, reportedly does not impact mTOR function [1].</p>
    Fórmula:C53H83NO13
    Cor e Forma:Solid
    Peso molecular:942.23
  • (Rac)-Azide-phenylalanine

    CAS:
    <p>(Rac)-Azide-phenylalanine: racemate, non-natural amino acid derivative for protein labeling.</p>
    Fórmula:C9H10N4O2
    Cor e Forma:Solid
    Peso molecular:206.20
  • NIM811

    CAS:
    <p>NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.</p>
    Fórmula:C62H111N11O12
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1202.635
  • DSPE-PEG5000-NGR


    <p>DSPE-PEG5000-NGR is a PEG compound composed of DSPE and the Asn-Gly-Arg (NGR) peptide. The NGR peptide has the capability to target tumor vasculature antigen CD13. DSPE-PEG5000-NGR is applicable in drug delivery.</p>
    Cor e Forma:Odour Solid
  • Phenacaine

    CAS:
    <p>Phenacaine, also known as Holocaine, is a local anesthetic that blocks certain Ca 2+ enzymes in red blood cells, brain, and heart.</p>
    Fórmula:C18H22N2O2
    Cor e Forma:Solid
    Peso molecular:298.38
  • DSPE-PEG2000-CSTSMLKAC


    <p>DSPE-PEG2000-CSTSMLKAC is a PEG compound composed of DSPE and CSTSMLKAC. CSTSMLKAC can mediate phage selective homing to ischemic heart tissue. DSPE-PEG2000-CSTSMLKAC is suitable for drug delivery.</p>
    Cor e Forma:Odour Solid
  • Methyl 3,4,5-trimethoxy-2-(2-(nicotinamido)benzamido)benzoate

    CAS:
    <p>Preterramide C is a fungal metabolite that has been found inA.</p>
    Fórmula:C24H23N3O7
    Cor e Forma:Solid
    Peso molecular:465.46
  • Lysinoalanine

    CAS:
    <p>Lysinoalanine is an unusual amino acid, not a dipeptide, which exists in proteins of cooked foods. It is formed in food that is heated or treated with alkali.</p>
    Fórmula:C9H19N3O4
    Cor e Forma:Solid
    Peso molecular:233.26
  • Leucylproline

    CAS:
    <p>Leucylproline is a peptide that proteolytic breakdown product by larger proteins.</p>
    Fórmula:C11H20N2O3
    Cor e Forma:Solid
    Peso molecular:228.29
  • 8-Demethyl Ivabradine

    CAS:
    <p>8-Demethyl Ivabradine, a metabolite of Ivabradine, is an oral HCN channel blocker.</p>
    Fórmula:C26H34N2O5
    Cor e Forma:Solid
    Peso molecular:454.567
  • MC 1046

    CAS:
    <p>MC 1046 is an impurity of Calcipotriol. Calcipotriol is a ligand of VDR-like receptors.</p>
    Fórmula:C27H38O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:410.59
  • Anti-Cancer Metabolism Compound Library


    <p>A unique collection of 1268 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS</p>
    Cor e Forma:Odour Solid
  • Tacalcitol monohydrate

    CAS:
    <p>Tacalcitol monohydrate(Curatoderm monohydrate), a vitamin D3 analog that promotes bone development by regulating calcium ions, can be used to study psoriasis.</p>
    Fórmula:C27H46O4
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:434.65
  • DF-461

    CAS:
    <p>DF-461 is an inhibitor of squalene synthase.</p>
    Fórmula:C20H14Cl2F3N3O4
    Cor e Forma:Solid
    Peso molecular:488.24
  • 8′-Hydroxy ABA

    CAS:
    <p>8′-Hydroxy ABA (8'-OH-ABA), a key metabolite of abscisic acid (ABA), exhibits hormonal activity by promoting enhanced oil synthesis.</p>
    Fórmula:C15H20O5
    Cor e Forma:Solid
    Peso molecular:280.32
  • 23,25-Dihydroxy-24-oxovitamin D3

    CAS:
    <p>23,25-Dihydroxy-24-oxovitamin D3, a prominent metabolite of 24(R),25-Dihydroxyvitamin D3, holds significant potential for studying metabolic disorders[1].</p>
    Fórmula:C27H42O4
    Cor e Forma:Solid
    Peso molecular:430.629
  • CYP1B1-IN-7

    CAS:
    <p>CYP1B1-IN-7 is a CYP1B1 inhibitor that can be used in synergy with anticancer compounds for the treatment of cancers.</p>
    Fórmula:C19H13ClO
    Pureza:99.49%
    Cor e Forma:Soild
    Peso molecular:292.76
  • DSPE-PEG1000-pPB


    <p>DSPE-PEG1000-pPB is a PEG compound consisting of DSPE and a cyclic oligopeptide (pPB). The pPB component exhibits a strong binding affinity to PDGFRβ, which is overexpressed in activated hepatic stellate cells (HSC). DSPE-PEG1000-pPB is applicable for drug delivery.</p>
    Cor e Forma:Odour Solid
  • Glycerol-3-phosphate oxidase

    CAS:
    <p>Glycerol-3-phosphate oxidase, from E. coli, is crucial in glycerol metabolism and phospholipid formation, producing electrons via oxidation.</p>
    Cor e Forma:Solid
  • DSPE-PEG1000-CREKA


    <p>DSPE-PEG1000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide has the capability to target tumor cells and tumor vasculature, exhibiting anti-tumor activity. Additionally, DSPE-PEG1000-CREKA can be utilized for drug delivery.</p>
    Cor e Forma:Odour Solid
  • PKM2-IN-3

    CAS:
    <p>PKM2-IN-3 inhibits PKM2 kinase with 4.1 μM IC50, curbing glycolysis and NLRP3, reducing neuroinflammation.</p>
    Fórmula:C21H22O4
    Cor e Forma:Solid
    Peso molecular:338.403
  • 1-Methylhistamine

    CAS:
    <p>2-(1-Methyl-1H-imidazol-4-yl)ethan-1-amine is a histamine metabolite.</p>
    Fórmula:C6H11N3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:125.1716
  • S32826

    CAS:
    <p>S32826, a potent autotaxin inhibitor with an IC50 of 8.8 nM, blocks LPA release and targets α, β, γ isoforms.</p>
    Fórmula:C21H36NO4P
    Cor e Forma:Solid
    Peso molecular:397.496
  • TPH1-IN-1


    <p>TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.</p>
    Fórmula:C21H18N6O4S
    Cor e Forma:Solid
    Peso molecular:450.47
  • Ciwujianoside D2

    CAS:
    <p>Ciwujianoside D2 is a useful organic compound for research related to life sciences. The catalog number is T126336 and the CAS number is 114892-57-8.</p>
    Fórmula:C54H84O22
    Cor e Forma:Solid
    Peso molecular:1085.24
  • GLUT1-IN-1


    <p>GLUT1-IN-1 inhibits GLUT1; cytotoxic to HeLa, A549, HepG2 (IC50: 5.49, 11.14, 8.73 μM); potential in PDT and cancer research.</p>
    Fórmula:C25H31BF2I2N6O7
    Cor e Forma:Solid
    Peso molecular:830.17
  • Mevalonic acid 5-pyrophosphate tetralithium

    CAS:
    <p>Mevalonic acid 5-pyrophosphate (also known as 5-Diphosphomevalonic acid) tetralithium is an endogenous metabolite involved in the mevalonate pathway.</p>
    Fórmula:C6H10Li4O10P2
    Cor e Forma:Solid
    Peso molecular:331.85
  • PDE1-IN-5


    <p>PDE1-IN-5 (Compound 10c) is a selective PDE1C inhibitor with an IC50 of 15 nM, exhibiting anti-inflammatory properties through the inhibition of iNOS, TNF-α, IL</p>
    Fórmula:C27H29FN4O
    Cor e Forma:Solid
    Peso molecular:444.54
  • (±)14(15)-EpEDE

    CAS:
    <p>8,11,14-Eicosatrienoic acid, also known as dihomo-γ-linolenic acid , is a polyunsaturated fatty acid (PUFA) produced from γ-linolenic acid by the action of</p>
    Fórmula:C20H34O3
    Cor e Forma:Solid
    Peso molecular:322.489
  • Carbonic anhydrase inhibitor 31


    <p>Carbonic anhydrase inhibitor31 is an mtCA2 inhibitor (Ki: 5.2 nM) that can be used in antituberculosis research.</p>
    Fórmula:C24H20N6O5S
    Cor e Forma:Solid
    Peso molecular:504.12159
  • Ophiobolin A

    CAS:
    <p>Ophiobolin A: Fungal metabolite, phytotoxin, inhibits calmodulin-activated phosphodiesterase (IC50: 9μM), with antimicrobial and anticancer properties.</p>
    Fórmula:C25H36O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:400.559
  • Thymidine 5′-diphosphate

    CAS:
    <p>Thymidine 5′-diphosphate (dTDP), a crucial product of pyrimidine synthesis in organisms, is synthesized through the thymidylate kinase (TMPK)-catalyzed</p>
    Fórmula:C10H16N2O11P2
    Cor e Forma:Solid
    Peso molecular:402.19
  • ONO-8430506

    CAS:
    <p>ONO-8430506 is an orally available, potent autotaxin (ATX)/ENPP2 inhibitor (IC90: 100 nM) that inhibits ATX activity in mouse plasma.</p>
    Fórmula:C27H28FN3O3
    Pureza:98.34%
    Cor e Forma:Solid
    Peso molecular:461.53
  • Cholesterol glucuronide

    CAS:
    <p>Cholesterol glucuronide is an endogenous metabolite of lipid generated by UDP glucuonyltransferase in the liver.</p>
    Fórmula:C33H54O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:562.78
  • hCAII-IN-8

    CAS:
    <p>Compound CDy9 is a highly selective inhibitor of carbonic anhydrase (CA) with an IC50 value of 0.18 μM for hCA II.</p>
    Fórmula:C15H16N2O5S
    Pureza:99.73%
    Cor e Forma:Soild
    Peso molecular:336.36
  • 2-Nitrophenyl a-D-glucopyranoside

    CAS:
    <p>2-Nitrophenyl a-D-glucopyranoside is a substrate of β-glucosidase [1] .</p>
    Fórmula:C12H15NO8
    Cor e Forma:Solid
    Peso molecular:301.25
  • Netupitant metabolite Netupitant N-oxide

    CAS:
    <p>Netupitant N-oxide is a highly selective antagonist of NK1 receptor, is Netupitant metabolite.</p>
    Fórmula:C30H32F6N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:594.59
  • α-Glycerophosphate Dehydrogenase-Triosephosphate


    <p>α-Glycerophosphate Dehydrogenase-Triosephosphate (GDH-TIM) is an enzyme mixture composed of glycerophosphate dehydrogenase (GDH) and triosephosphate isomerase (TIM). This compound is employed to measure transketolase (TK) activity in erythrocyte hemolysates, which helps in assessing vitamin B deficiency.</p>
  • 1,2-Dihexadecyl-sn-glycero-3-PC

    CAS:
    <p>1,2-Dihexadecyl-sn-glycero-3-PC can be used in related research in the field of life sciences. Its product number is T37043 and CAS number is 36314-47-3.</p>
    Fórmula:C40H84NO6P
    Cor e Forma:Solid
    Peso molecular:706.07
  • CETP-IN-4

    CAS:
    <p>CETP-IN-4 is a cholesteryl ester transfer protein (CETP) inhibitor.</p>
    Fórmula:C36H28F9N3O4
    Cor e Forma:Solid
    Peso molecular:737.623
  • Desoxycarbadox

    CAS:
    <p>Desoxycarbadox, derived from Carbadox, is a quinoxaline-di-N-oxide antibiotic compound.</p>
    Fórmula:C11H10N4O2
    Cor e Forma:Solid
    Peso molecular:230.227
  • ML171

    CAS:
    <p>Compound PDK0326, with CAS No. 6631-94-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0326 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Fórmula:C14H11NOS
    Cor e Forma:Mustard-Colored Powder
    Peso molecular:241.3
  • VDR agonist 2


    <p>VDR agonist 2 (compound 16i), a vitamin D receptor (VDR) agonist, effectively inhibits TGF-β1-induced hepatic stellate cell (HSC) activation, demonstrating</p>
    Fórmula:C20H21F3O3
    Cor e Forma:Solid
    Peso molecular:366.37
  • Carbonic anhydrase inhibitor 18


    <p>Carbonic anhydrase inhibitor18 (Compound 9) is an inhibitor of human carbonic anhydrase (hCA) isozymes, with Ki values of 604.8 nM for hCA I, 333.6 nM for hCA II, 1.9 nM for hCA IX, and 6.7 nM for hCA XII. Carbonic anhydrase inhibitor18 is applicable in cancer research.</p>
    Fórmula:C26H28N4O6S2
    Peso molecular:556.14503