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Neurociência

Neurociência

Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.

Subcategorias de "Neurociência"

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Foram encontrados 5400 produtos de "Neurociência"

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  • MPEP

    CAS:
    <p>MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.</p>
    Fórmula:C14H11N
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:193.24
  • VU0152100

    CAS:
    <p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>
    Fórmula:C18H19N3O2S
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:341.43
  • Tiaprofenic acid

    CAS:
    <p>Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.</p>
    Fórmula:C14H12O3S
    Pureza:99.51%
    Cor e Forma:Solid
    Peso molecular:260.31
  • Rebamipide mofetil

    CAS:
    <p>Rebamipide mofetil is an orally active prodrug of Rebamipide which is a mucoprotective agent.</p>
    Fórmula:C25H26ClN3O5
    Pureza:98.17%
    Cor e Forma:Solid
    Peso molecular:483.94
  • Homocarnosine acetate


    <p>Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.</p>
    Fórmula:C12H20N4O5
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:300.31
  • Losartan Carboxaldehyde

    CAS:
    <p>Losartan Carboxaldehyde is an endothelial cyclooxygenase (COX)-2 inhibitor.</p>
    Fórmula:C22H21ClN6O
    Pureza:99.1%
    Cor e Forma:Solid
    Peso molecular:420.89
  • Nitrocaramiphen hydrochloride

    CAS:
    <p>Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.</p>
    Fórmula:C18H27ClN2O4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:370.87
  • AVN-101

    CAS:
    <p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C21H25ClN2
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:340.89
  • α-Asarone

    CAS:
    <p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>
    Fórmula:C12H16O3
    Pureza:99.64% - 99.64%
    Cor e Forma:Monoclinic Needles From Water Monoclinic Needles From Water
    Peso molecular:208.25
  • LY2119620

    CAS:
    <p>LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.</p>
    Fórmula:C19H24ClN5O3S
    Pureza:99.7%
    Cor e Forma:Solid
    Peso molecular:437.94
  • MK-0752

    CAS:
    <p>MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).</p>
    Fórmula:C21H21ClF2O4S
    Pureza:98% - 99.55%
    Cor e Forma:Solid
    Peso molecular:442.9
  • LRRK2-IN-1

    CAS:
    <p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>
    Fórmula:C31H38N8O3
    Pureza:98% - 98.82%
    Cor e Forma:Solid
    Peso molecular:570.69
  • JHU37160

    CAS:
    <p>JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.</p>
    Fórmula:C19H20ClFN4
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:358.84
  • RU 24969 free base

    CAS:
    <p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>
    Fórmula:C14H16N2O
    Pureza:97.38%
    Cor e Forma:Solid
    Peso molecular:228.29
  • HM-30181 mesylate monohydrate

    CAS:
    <p>HM-30181 mesylate monohydrate is an oral P-glycoprotein (P-gp) inhibitor, used to enhance the oral bioavailability of P-gp substrate drugs.</p>
    Fórmula:C39H42N6O11S
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:802.85
  • ONO-8590580

    CAS:
    <p>ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.</p>
    Fórmula:C21H21FN6
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:376.43
  • LY334370

    CAS:
    <p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>
    Fórmula:C21H22FN3O
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:351.42
  • PNU-282987 S enantiomer free base

    CAS:
    <p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>
    Fórmula:C14H17ClN2O
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:264.75
  • 4i

    CAS:
    <p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>
    Fórmula:C16H12ClN3O
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:297.74
  • Edrophonium chloride

    CAS:
    <p>Edrophonium chloride is an acetylcholinesterase (AChE) inhibitor that is known to prevent the breakdown of the neurotransmitter acetylcholine by binding</p>
    Fórmula:C10H16ClNO
    Pureza:97.41%
    Cor e Forma:Liquid
    Peso molecular:201.69
  • Kavain

    CAS:
    <p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>
    Fórmula:C14H14O3
    Pureza:99.93% - ≥95%
    Cor e Forma:Solid
    Peso molecular:230.26
  • Prucalopride Succinate

    CAS:
    <p>Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).</p>
    Fórmula:C18H26ClN3O3·C4H6O4
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:485.96
  • α-Conotoxin PIA acetate


    <p>α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.</p>
    Pureza:98%
    Cor e Forma:Liquid
    Peso molecular:N/A
  • Flibanserin

    CAS:
    <p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>
    Fórmula:C20H21F3N4O
    Pureza:99.37% - 99.93%
    Cor e Forma:White Powder
    Peso molecular:390.4
  • CCMI

    CAS:
    <p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>
    Fórmula:C19H15Cl2N3O2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:388.25
  • AF-353

    CAS:
    <p>AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).</p>
    Fórmula:C14H17IN4O2
    Pureza:92.98% - 99.356%
    Cor e Forma:Solid
    Peso molecular:400.21
  • L-701324

    CAS:
    <p>L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.</p>
    Fórmula:C21H14ClNO3
    Pureza:98.63% - >99.99%
    Cor e Forma:Solid
    Peso molecular:363.79
  • Melitracen

    CAS:
    <p>Melitracen is a tricyclic antidepressant.</p>
    Fórmula:C21H25N
    Cor e Forma:Solid
    Peso molecular:291.43
  • Metergoline

    CAS:
    <p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>
    Fórmula:C25H29N3O2
    Pureza:99.83% - 99.97%
    Cor e Forma:Solid
    Peso molecular:403.52
  • Vortioxetine hydrobromide

    CAS:
    <p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>
    Fórmula:C18H22N2S·HBr
    Pureza:98.85% - 99.98%
    Cor e Forma:Solid
    Peso molecular:379.36
  • Opiranserin hydrochloride

    CAS:
    <p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>
    Fórmula:C21H35ClN2O5
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:430.97
  • Cerlapirdine

    CAS:
    <p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>
    Fórmula:C22H23N3O3S
    Pureza:98.77%
    Cor e Forma:Solid
    Peso molecular:409.5
  • MK-1064

    CAS:
    <p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>
    Fórmula:C24H20ClN5O3
    Pureza:99.19% - 99.82%
    Cor e Forma:Solid
    Peso molecular:461.9
  • Lurasidone

    CAS:
    <p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>
    Fórmula:C28H36N4O2S
    Pureza:99.78% - 99.91%
    Cor e Forma:Solid
    Peso molecular:492.68
  • Suritozole

    CAS:
    <p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>
    Fórmula:C10H10FN3S
    Pureza:99.25%
    Cor e Forma:Solid
    Peso molecular:223.27
  • NMDAR antagonist 1

    CAS:
    <p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>
    Fórmula:C20H20BrN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:414.3
  • γ-Mangostin

    CAS:
    <p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>
    Fórmula:C23H24O6
    Pureza:98.55% - 99.08%
    Cor e Forma:Solid
    Peso molecular:396.43
  • NS9283

    CAS:
    <p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>
    Fórmula:C14H8N4O
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:248.24
  • Pozanicline dihydrochloride

    CAS:
    <p>Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)</p>
    Fórmula:C11H18Cl2N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:265.18
  • Gadoteridol

    CAS:
    <p>Gadoteridol (Gd-HP-DO3A) is a gadolinium-based MRI contrast agent that can be used for central nervous system imaging.</p>
    Fórmula:C17H29GdN4O7
    Pureza:99.77% - 99.91%
    Cor e Forma:Solid
    Peso molecular:558.69
  • A-484954

    CAS:
    <p>A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.</p>
    Fórmula:C13H15N5O3
    Pureza:97.47% - 99.86%
    Cor e Forma:Solid
    Peso molecular:289.29
  • Venlafaxine

    CAS:
    <p>Venlafaxine (Wy 45030), an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI), is used to treat major generalised anxiety disorder (GAD),</p>
    Fórmula:C17H27NO2
    Pureza:99.2%
    Cor e Forma:White Solid Crystalline
    Peso molecular:277.4
  • Fluralaner

    CAS:
    <p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>
    Fórmula:C22H17Cl2F6N3O3
    Pureza:99.72% - 99.90%
    Cor e Forma:Solid Powder
    Peso molecular:556.29
  • N-Desmethylclozapine

    CAS:
    <p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>
    Fórmula:C17H17ClN4
    Pureza:97.25% - 99.83%
    Cor e Forma:Yellow Crystalline Solid
    Peso molecular:312.8
  • Tinoridine hydrochloride

    CAS:
    <p>Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.</p>
    Fórmula:C17H21ClN2O2S
    Pureza:97.49%
    Cor e Forma:Solid
    Peso molecular:352.88
  • OXA (17-33) acetate


    <p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>
    Fórmula:C79H125N23O22
    Pureza:98.52%
    Cor e Forma:Solid
    Peso molecular:1748.98
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Cor e Forma:Solid
    Peso molecular:538.64
  • Melatonin

    CAS:
    <p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>
    Fórmula:C13H16N2O2
    Pureza:98% - 99.89%
    Cor e Forma:Pale Yellow Leaflets From Benzene Solid
    Peso molecular:232.28
  • Radiprodil

    CAS:
    <p>Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.</p>
    Fórmula:C21H20FN3O4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:397.4
  • Mofezolac

    CAS:
    <p>Mofezolac (formerly known as Disopain or N-22) is a highly selective COX-1 (cyclooxygenase-1) inhibitor with COXs selectivity index &gt; 6000</p>
    Fórmula:C19H17NO5
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:339.34
  • RS-67333

    CAS:
    <p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>
    Fórmula:C19H29ClN2O2
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:352.9
  • Harmine

    CAS:
    <p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>
    Fórmula:C13H12N2O
    Pureza:98.29% - 99.92%
    Cor e Forma:Off-White Solid
    Peso molecular:212.25
  • Metoclopramide

    CAS:
    <p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>
    Fórmula:C14H22ClN3O2
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:299.80
  • Afloqualone

    CAS:
    <p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>
    Fórmula:C16H14FN3O
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:283.3
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Cor e Forma:Solid
    Peso molecular:417.97
  • Nelotanserin

    CAS:
    <p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>
    Fórmula:C18H15BrF2N4O2
    Pureza:98.42% - 99.88%
    Cor e Forma:Solid
    Peso molecular:437.24
  • Cholesterol myristate

    CAS:
    <p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>
    Fórmula:C41H72O2
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:597.01
  • Idalopirdine Hydrochloride

    CAS:
    <p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>
    Fórmula:C20H20ClF5N2O
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:434.83
  • p-Hydroxybenzaldehyde

    CAS:
    <p>1.</p>
    Fórmula:C7H6O2
    Pureza:99.05% - 99.86%
    Cor e Forma:Solid
    Peso molecular:122.12
  • Isocarboxazid

    CAS:
    <p>Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.</p>
    Fórmula:C12H13N3O2
    Pureza:98.32% - 99.94%
    Cor e Forma:Solid
    Peso molecular:231.25
  • AMN082 free base

    CAS:
    <p>AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.</p>
    Fórmula:C28H28N2
    Pureza:97.75% - 97.79%
    Cor e Forma:Solid
    Peso molecular:392.54
  • XAP044

    CAS:
    <p>XAP044 blocks mGlu7, inhibiting long-term potentiation in mouse brain with a half-maximal effect at 88nm.</p>
    Fórmula:C15H9IO4
    Pureza:97.41%
    Cor e Forma:Solid
    Peso molecular:380.13
  • PHCCC

    CAS:
    <p>PHCCC is a Group I mGluR antagonist and enhances mGluR4 function; also blocks mGluR2/8.</p>
    Fórmula:C17H14N2O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:294.3
  • Perospirone

    CAS:
    <p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>
    Fórmula:C23H30N4O2S
    Pureza:99.23%
    Cor e Forma:White Powder
    Peso molecular:426.57
  • Ipsapirone hydrochloride

    CAS:
    <p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>
    Fórmula:C19H24ClN5O3S
    Cor e Forma:Solid
    Peso molecular:437.94
  • Piboserod

    CAS:
    <p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>
    Fórmula:C22H31N3O2
    Pureza:97.21% - 99.49%
    Cor e Forma:Solid
    Peso molecular:369.5
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Fórmula:C19H21ClF2N4O
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:394.85
  • IGS-1.76

    CAS:
    <p>IGS-1.76 binds strongly to hNCS-1, modulates its Ric8a interaction, and inhibits the hNCS-1/Ric8a complex.</p>
    Fórmula:C22H18N2OS
    Pureza:98.18% - 98.56%
    Cor e Forma:Solid
    Peso molecular:358.46
  • SKF-83566

    CAS:
    <p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>
    Fórmula:C17H18BrNO
    Pureza:95.00% - 99.82%
    Cor e Forma:Solid
    Peso molecular:332.23
  • Zosuquidar

    CAS:
    <p>Zosuquidar (RS 33295-198) is a potent P-glycoprotein inhibitor with antitumor activity that inhibits tumor growth.</p>
    Fórmula:C32H31F2N3O2
    Cor e Forma:Solid
    Peso molecular:527.6
  • IKK 16

    CAS:
    <p>IKK 16 (IKK Inhibitor VII) is a selective IκB kinase (IKK) inhibitor for IKK-2, IKK complex and IKK-1 with IC50 of 40 nM, 70 nM and 200 nM, respectively.</p>
    Fórmula:C28H29N5OS
    Pureza:98.76% - 99.61%
    Cor e Forma:Solid
    Peso molecular:483.63
  • VU0155094

    CAS:
    <p>VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.</p>
    Fórmula:C24H24N2O4S
    Pureza:97.21%
    Cor e Forma:Solid
    Peso molecular:436.52
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Fórmula:C18H21ClF3N3O
    Pureza:99.03% - 99.95%
    Cor e Forma:Solid
    Peso molecular:387.83
  • PNU-120596

    CAS:
    <p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>
    Fórmula:C13H14ClN3O4
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:311.72
  • CZC-25146

    CAS:
    <p>CZC-25146, a stable LRRK2 inhibitor, IC50: 4.76 nM (wild-type), 6.87 nM (G2019S).</p>
    Fórmula:C22H25FN6O4S
    Pureza:97.68%
    Cor e Forma:Solid
    Peso molecular:488.54
  • Cyclopentolate Hydrochloride

    CAS:
    <p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>
    Fórmula:C17H26ClNO3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:327.85
  • (+)-Kavain

    CAS:
    <p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>
    Fórmula:C14H14O3
    Pureza:97% - ≥95%
    Cor e Forma:White Fine Powder
    Peso molecular:230.26
  • KN-62

    CAS:
    <p>KN-62 is a potent and specific Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor with Ki of 0.9 μM.</p>
    Fórmula:C38H35N5O6S2
    Pureza:99.80% - >99.99%
    Cor e Forma:White Solid
    Peso molecular:721.84
  • Semagacestat

    CAS:
    <p>Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).</p>
    Fórmula:C19H27N3O4
    Pureza:97.1% - 99.9%
    Cor e Forma:Solid
    Peso molecular:361.44
  • Ondansetron

    CAS:
    <p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>
    Fórmula:C18H19N3O
    Pureza:99.92%
    Cor e Forma:White To Yellow Crystals
    Peso molecular:293.36
  • VU0361737

    CAS:
    <p>VU0361737 (ML-128) is a mGlu4 PAM; EC50 is 240 nM (human) and 110 nM (rat), weak at mGlu5/8, inactive at mGlu1/2/3/6/7, CNS-penetrant.</p>
    Fórmula:C13H11ClN2O2
    Pureza:99.60% - 99.85%
    Cor e Forma:Solid
    Peso molecular:262.69
  • Glypromate acetate(32302-76-4 free base)


    <p>Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.</p>
    Fórmula:C14H23N3O8
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:361.35
  • Buclizine dihydrochloride

    CAS:
    <p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>
    Fórmula:C28H33ClN2·2HCl
    Pureza:98.05%
    Cor e Forma:Off-White Powder
    Peso molecular:505.95
  • Ocinaplon

    CAS:
    <p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>
    Fórmula:C17H11N5O
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:301.3
  • Norfluoxetine Hydrochloride

    CAS:
    <p>Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.</p>
    Fórmula:C16H17ClF3NO
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:331.76
  • Ipratropium Bromide

    CAS:
    <p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>
    Fórmula:C20H30BrNO3
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:412.37
  • SB-200646

    CAS:
    <p>SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor</p>
    Fórmula:C15H14N4O
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:266.3
  • Bicuculline

    CAS:
    <p>Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.</p>
    Fórmula:C20H17NO6
    Pureza:98% - 99.99%
    Cor e Forma:Light Yellow Powder
    Peso molecular:367.35
  • Mosapride

    CAS:
    <p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>
    Fórmula:C21H25ClFN3O3
    Pureza:99.56%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:421.89
  • TCN 201

    CAS:
    <p>TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.</p>
    Fórmula:C21H17ClFN3O4S
    Pureza:98.5%
    Cor e Forma:Solid
    Peso molecular:461.89
  • Revefenacin

    CAS:
    <p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>
    Fórmula:C35H43N5O4
    Pureza:98.12%
    Cor e Forma:Solid
    Peso molecular:597.75
  • RO4929097

    CAS:
    <p>RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).</p>
    Fórmula:C22H20F5N3O3
    Pureza:98.5% - 99.51%
    Cor e Forma:Solid
    Peso molecular:469.4
  • Miltirone

    CAS:
    <p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>
    Fórmula:C19H22O2
    Pureza:99.22% - 99.66%
    Cor e Forma:Solid
    Peso molecular:282.38
  • Pimavanserin tartrate

    CAS:
    <p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>
    Fórmula:C50H68F2N6O4·C4H6O6
    Pureza:99.24% - 99.98%
    Cor e Forma:Solid
    Peso molecular:1005.2
  • JHU37152

    CAS:
    <p>JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.</p>
    Fórmula:C19H20ClFN4
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:358.84
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    <p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>
    Fórmula:C2H5NO3·5HCl
    Pureza:98.03%
    Cor e Forma:Light Beige Crystalline Powder
    Peso molecular:109.3
  • Encenicline hydrochloride

    CAS:
    <p>Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).</p>
    Fórmula:C16H17ClN2OS·HCl
    Pureza:98.34% - 99.85%
    Cor e Forma:Solid
    Peso molecular:357.3
  • Acetoxyvalerensre

    CAS:
    <p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>
    Fórmula:C17H24O4
    Pureza:98.22%
    Cor e Forma:Solid
    Peso molecular:292.37
  • Amentoflavone

    CAS:
    <p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>
    Fórmula:C30H18O10
    Pureza:98.21% - 99.22%
    Cor e Forma:Odourless Whitish Solid
    Peso molecular:538.46
  • 5-HT1A modulator 2 hydrochloride

    CAS:
    <p>5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.</p>
    Fórmula:C11H16ClNO
    Pureza:98.5%
    Cor e Forma:Solid
    Peso molecular:213.7
  • pep2-SVKI acetate


    <p>Pep2-SVKI acetate(pep2-SVKI acetate (328944-75-8 free base)) is a synthetic peptide salt that prevents internalization of AMPA-type glutamate receptor.</p>
    Fórmula:C62H97N13O20
    Pureza:97.14%
    Cor e Forma:Solid
    Peso molecular:1344.51
  • Piperazine citrate

    CAS:
    <p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>
    Fórmula:C24H46N6O14
    Pureza:99.8%
    Cor e Forma:Crystals Indication
    Peso molecular:642.65
  • EUK-134

    CAS:
    <p>EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.</p>
    Fórmula:C18H18ClMnN2O4
    Pureza:98.39%
    Cor e Forma:Solid
    Peso molecular:416.74
  • LY310762

    CAS:
    <p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>
    Fórmula:C24H27FN2O2·HCl
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:430.94
  • MK-3697

    CAS:
    <p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>
    Fórmula:C23H21N5O3S
    Pureza:97.69% - 98.15%
    Cor e Forma:Solid
    Peso molecular:447.51
  • Metadoxine

    CAS:
    <p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>
    Fórmula:C8H11NO3·C5H7NO3
    Pureza:99.19%
    Cor e Forma:Off-White Powder
    Peso molecular:298.29
  • Tiagabine

    CAS:
    <p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>
    Fórmula:C20H25NO2S2
    Pureza:99.25%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:375.55
  • Clomipramine

    CAS:
    <p>Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by hindering serotonin reuptake.</p>
    Fórmula:C19H23ClN2
    Pureza:99.31% - 99.71%
    Cor e Forma:Solid
    Peso molecular:314.85
  • DNQX

    CAS:
    <p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C8H4N4O6
    Pureza:97.27% - 99.1%
    Cor e Forma:Off-White Powder With A Yellow Tinge
    Peso molecular:252.14
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:354.38
  • ADX88178

    CAS:
    <p>ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 of 4 nM for human mGluR4.</p>
    Fórmula:C12H12N6S
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:272.33
  • ZL006

    CAS:
    <p>ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.</p>
    Fórmula:C14H11Cl2NO4
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:328.15
  • Acamprosate

    CAS:
    <p>Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust</p>
    Fórmula:C5H11NO4S
    Pureza:98.30%
    Cor e Forma:Solid
    Peso molecular:181.21
  • Verubecestat

    CAS:
    <p>Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor.</p>
    Fórmula:C17H17F2N5O3S
    Pureza:92.24% - 99.55%
    Cor e Forma:Solid
    Peso molecular:409.41
  • VU0364770

    CAS:
    <p>VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu</p>
    Fórmula:C12H9ClN2O
    Pureza:99.65% - >99.99%
    Cor e Forma:Solid
    Peso molecular:232.67
  • GW791343 dihydrochloride

    CAS:
    <p>GW791343 dihydrochloride (GW791343 (HCl)) is a P2X7 allosteric modulator.</p>
    Fórmula:C20H26Cl2F2N4O
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:447.35
  • pyridostigmine

    CAS:
    <p>Pyridostigmine(Regonol) is an acetylcholinesterase inhibitor that can treat myasthenia gravis by increasing acetylcholine at the postsynaptic motor endplate.</p>
    Fórmula:C9H13N2O2
    Pureza:98.10%
    Cor e Forma:Solid
    Peso molecular:181.21
  • Lu AF21934

    CAS:
    <p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>
    Fórmula:C14H16Cl2N2O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:315.2
  • GALANTHAMINONE

    CAS:
    <p>Galanthaminone ((-)-Narwedine) is a cholinesterase (AChE) inhibitor, used for the treatment of mild to moderate Alzheimer's disease and other memory impairments</p>
    Fórmula:C17H19NO3
    Pureza:99.93%
    Cor e Forma:White To Off-White Chemical
    Peso molecular:285.34
  • A-867744

    CAS:
    <p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>
    Fórmula:C20H19ClN2O3S
    Pureza:95.66%
    Cor e Forma:Solid
    Peso molecular:402.89
  • NS-398

    CAS:
    <p>NS-398 (N-(2-cyclohexyloxy-4-nitrophenyl)methane sulfonamide) is a COX-2 inhibitor wih anti-inflammatory activity.</p>
    Fórmula:C13H18N2O5S
    Pureza:99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:314.36
  • PNU 22394 hydrochloride

    CAS:
    <p>PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist</p>
    Fórmula:C13H17ClN2
    Pureza:97.83%
    Cor e Forma:Solid
    Peso molecular:236.74
  • N-ACETYLTRYPTAMINE

    CAS:
    <p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>
    Fórmula:C12H14N2O
    Pureza:98.79%
    Cor e Forma:Powder
    Peso molecular:202.25
  • GR 125743

    CAS:
    <p>GR 125743 is a novel antagonist of 5-HT1B/1D receptor.</p>
    Fórmula:C25H28N4O2
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:416.52
  • Intepirdine

    CAS:
    <p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>
    Fórmula:C19H19N3O2S
    Pureza:98% - 98.63%
    Cor e Forma:Solid
    Peso molecular:353.44
  • JNJ-40411813

    CAS:
    <p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>
    Fórmula:C20H25ClN2O
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:344.88
  • Acotiamide monohydrochloride trihydrate

    CAS:
    <p>Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.</p>
    Fórmula:C21H37ClN4O8S
    Pureza:98% - 99.54%
    Cor e Forma:Solid
    Peso molecular:541.06
  • Mosapride Citrate

    CAS:
    <p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>
    Fórmula:C21H25ClFN3O3·C6H8O7
    Pureza:99.70%
    Cor e Forma:White Powder
    Peso molecular:614.02
  • 1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide

    CAS:
    <p>1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide is the inhibitor of human erythrocyte AChE.</p>
    Fórmula:C20H30Br2N2
    Pureza:98.17%
    Cor e Forma:Solid
    Peso molecular:458.27
  • 5-BDBD

    CAS:
    <p>5-BDBD is a potent and selective P2X4 receptor antagonist.</p>
    Fórmula:C17H11BrN2O2
    Pureza:97.78%
    Cor e Forma:Solid
    Peso molecular:355.19
  • Gabazine

    CAS:
    <p>Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)</p>
    Fórmula:C15H18BrN3O3
    Pureza:98.51% - 99.24%
    Cor e Forma:Solid
    Peso molecular:368.23
  • Guvacine hydrochloride

    CAS:
    <p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>
    Fórmula:C6H10ClNO2
    Pureza:98.42%
    Cor e Forma:Solid
    Peso molecular:163.602
  • Edonerpic maleate

    CAS:
    <p>Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).</p>
    Fórmula:C20H25NO6S
    Pureza:98.24%
    Cor e Forma:Solid
    Peso molecular:407.48
  • NPS ALX Compound 4a

    CAS:
    <p>NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>
    Fórmula:C25H25N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:431.55
  • Tianeptine

    CAS:
    <p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Fórmula:C21H25ClN2O4S
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:436.95
  • Volinanserin

    CAS:
    <p>Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.</p>
    Fórmula:C22H28FNO3
    Pureza:98.94% - 99.95%
    Cor e Forma:Solid
    Peso molecular:373.46
  • Niaprazine

    CAS:
    <p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>
    Fórmula:C20H25FN4O
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:356.44
  • Ginkgolide A

    CAS:
    <p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>
    Fórmula:C20H24O9
    Pureza:98.76% - 99.81%
    Cor e Forma:White Powder
    Peso molecular:408.4
  • Rapastinel Trifluoroacetate

    CAS:
    <p>Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.</p>
    Fórmula:C20H32F3N5O8
    Pureza:99.01% - 99.77%
    Cor e Forma:Solid
    Peso molecular:527.49
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Cor e Forma:Off-White To Pale Yellow Solid
    Peso molecular:440.94
  • NS 1738

    CAS:
    <p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>
    Fórmula:C14H9Cl2F3N2O2
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:365.13
  • A-582941 dihydrochloride

    CAS:
    <p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:353.29
  • Dolasetron Mesylate hydrate

    CAS:
    <p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>
    Fórmula:C20H26N2O7S
    Pureza:99.86% - 99.9%
    Cor e Forma:Solid
    Peso molecular:438.49
  • m-Chlorophenylbiguanide hydrochloride

    CAS:
    <p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>
    Fórmula:C8H11Cl2N5
    Pureza:99.43% - 99.87%
    Cor e Forma:Solid
    Peso molecular:248.11
  • Donepezil

    CAS:
    <p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>
    Fórmula:C24H29NO3
    Pureza:99.69%
    Cor e Forma:White Or Almost White Crystal Powder
    Peso molecular:379.49
  • CNQX disodium

    CAS:
    <p>CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.</p>
    Fórmula:C9H2N4Na2O4
    Pureza:97.77%
    Cor e Forma:Solid
    Peso molecular:276.12
  • Ritanserin

    CAS:
    <p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C27H25F2N3OS
    Pureza:99.77% - 99.89%
    Cor e Forma:Solid
    Peso molecular:477.57
  • Frentizole

    CAS:
    <p>Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interaction</p>
    Fórmula:C15H13N3O2S
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:299.35
  • α-Conotoxin MII acetate


    <p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>
    Fórmula:C69H107N23O24S4
    Pureza:94.82% - 97.79%
    Cor e Forma:Solid
    Peso molecular:1770.99
  • TAE-1

    CAS:
    <p>TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. It inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively.</p>
    Fórmula:C39H51I3N6O9
    Pureza:94.58%
    Cor e Forma:Solid
    Peso molecular:1128.57
  • CALP2 acetate(261969-04-4 free base)


    <p>CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.</p>
    Fórmula:C68H104N14O13S
    Pureza:97.43%
    Cor e Forma:Solid
    Peso molecular:1357.7
  • Nefazodone hydrochloride

    CAS:
    <p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>
    Fórmula:C25H33Cl2N5O2
    Pureza:99% - 99.86%
    Cor e Forma:White Solid
    Peso molecular:506.47
  • Pitofenone hydrochloride

    CAS:
    <p>Pitofenone hydrochloride (Pitophenone hydrochloride), a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and</p>
    Fórmula:C22H26ClNO4
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:403.9
  • Naratriptan hydrochloride

    CAS:
    <p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>
    Fórmula:C17H25N3O2S·HCl
    Pureza:99.17% - 99.93%
    Cor e Forma:Beige Solid
    Peso molecular:371.93
  • 4BP-TQS

    CAS:
    <p>4BP-TQS is an allosteric agonist of α7 nAChRs.</p>
    Fórmula:C18H17BrN2O2S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:405.31
  • Cyclodrine hydrochloride

    CAS:
    <p>Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of</p>
    Fórmula:C19H30ClNO3
    Pureza:98.59%
    Cor e Forma:Solid
    Peso molecular:355.9
  • LX2343

    CAS:
    <p>LX2343 inhibits BACE1 (IC50: 11.43 μM) and PI3K non-competitively (IC50: 15.99 μM), and enhances autophagy for Aβ removal.</p>
    Fórmula:C22H19ClN2O6S
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:474.91
  • Syntide 2 acetate(108334-68-5 free base)


    <p>Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).</p>
    Fórmula:C70H126N20O20
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:1567.85
  • Aftin-4

    CAS:
    <p>Aftin-4, an amyloid forty-two inducer, activates γ-secretase, promoting the generation of amyloid-β-1-42 (Aβ1-42) from amyloid-β protein precursor.</p>
    Fórmula:C20H28N6O
    Pureza:98.51%
    Cor e Forma:Solid
    Peso molecular:368.48
  • PF-06454589

    CAS:
    <p>PF-06454589 is a potent inhibitor of LRRK2.</p>
    Fórmula:C14H16N6O
    Pureza:99.06%
    Cor e Forma:Solid
    Peso molecular:284.32
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Fórmula:C11H11N3O
    Pureza:99.03%
    Cor e Forma:Solid
    Peso molecular:201.22
  • Cannabigerol

    CAS:
    <p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>
    Fórmula:C21H32O2
    Pureza:99.59% - 99.92%
    Cor e Forma:Solid
    Peso molecular:316.48
  • Ursulcholic acid

    CAS:
    <p>Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.</p>
    Fórmula:C24H40O10S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:552.7
  • Temanogrel

    CAS:
    <p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>
    Fórmula:C24H28N4O4
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:436.5
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Fórmula:C16H14O4
    Pureza:98.75%
    Cor e Forma:Solid
    Peso molecular:270.28
  • Fesoterodine

    CAS:
    <p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>
    Fórmula:C26H37NO3
    Pureza:97.1%
    Cor e Forma:Solid
    Peso molecular:411.58
  • DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Fórmula:C19H23Cl2N3
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:364.31
  • Baclofen hydrochloride

    CAS:
    <p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:250.122
  • A-740003

    CAS:
    <p>A-740003 is a potent P2X7 receptor blocker, inhibiting rat/human receptors (IC50: 18/40 nM), lessens pain in animals, and shrinks mouse neuroblastoma.</p>
    Fórmula:C26H30N6O3
    Pureza:96.53% - 99.68%
    Cor e Forma:Solid
    Peso molecular:474.55
  • Melitracen hydrochloride

    CAS:
    <p>Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.</p>
    Fórmula:C21H26ClN
    Pureza:99.99%
    Cor e Forma:Crystalline Solid
    Peso molecular:327.90
  • Darifenacin

    CAS:
    <p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>
    Fórmula:C28H30N2O2
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:426.55
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Fórmula:C22H21O2P
    Pureza:97.985%
    Cor e Forma:White Or Slight Yellow Powder
    Peso molecular:348.37
  • Nuciferine

    CAS:
    <p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>
    Fórmula:C19H21NO2
    Pureza:98.76% - 99.79%
    Cor e Forma:Solid
    Peso molecular:295.38
  • Ro0711401

    CAS:
    <p>Ro0711401 is an agonist of mGlu1 receptor.</p>
    Fórmula:C18H11F3N2O3
    Pureza:97.57%
    Cor e Forma:Solid
    Peso molecular:360.29
  • Traxoprodil

    CAS:
    <p>Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).</p>
    Fórmula:C20H25NO3
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:327.42
  • 6-Methylflavone

    CAS:
    <p>6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.</p>
    Fórmula:C16H12O2
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:236.27
  • Dolasetron

    CAS:
    <p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>
    Fórmula:C19H20N2O3
    Pureza:99.84% - 99.86%
    Cor e Forma:White Powder
    Peso molecular:324.37
  • Ampiroxicam

    CAS:
    <p>Ampiroxicam (Flucam) is a nonselective cyclooxygenase inhibitor uesd as anti-inflammatory drug.</p>
    Fórmula:C20H21N3O7S
    Pureza:97.27% - 99.2%
    Cor e Forma:Powder
    Peso molecular:447.46
  • YM90K

    CAS:
    <p>YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.</p>
    Fórmula:C11H8ClN5O4
    Pureza:98.23%
    Cor e Forma:Solid
    Peso molecular:309.66
  • TCS-OX2-29

    CAS:
    <p>TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays &gt;250-fold selectivity for OX2 over OX1.</p>
    Fórmula:C23H31N3O3
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:397.51
  • Xanthotoxol

    CAS:
    <p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>
    Fórmula:C11H6O4
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:202.16
  • A-804598

    CAS:
    <p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>
    Fórmula:C19H17N5
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:315.37
  • SB 242084

    CAS:
    <p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>
    Fórmula:C21H19ClN4O2
    Pureza:99.75% - ≥98%
    Cor e Forma:Solid
    Peso molecular:394.85
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Fórmula:C17H16FN3
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:281.33
  • Ocaperidone

    CAS:
    <p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>
    Fórmula:C24H25FN4O2
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:420.48
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Fórmula:C21H32Cl2N4O
    Pureza:99.68% - 99.87%
    Cor e Forma:Solid
    Peso molecular:427.41
  • Demecarium bromide

    CAS:
    <p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>
    Fórmula:C32H52Br2N4O4
    Pureza:98%
    Cor e Forma:White Powder Solid
    Peso molecular:716.59
  • 3-MATIDA

    CAS:
    <p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>
    Fórmula:C8H9NO4S
    Pureza:99.75% - 99.96%
    Cor e Forma:Solid
    Peso molecular:215.23
  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Fórmula:C17H25N3O2S·C4H6O5
    Pureza:99.95%
    Cor e Forma:Pale Yellow Solid
    Peso molecular:469.55
  • A 438079 hydrochloride

    CAS:
    <p>A 438079 hydrochloride (A-438079 HCl) is a potent and selective P2X7 receptor antagonist with pIC50 of 6.9.</p>
    Fórmula:C13H10Cl3N5
    Pureza:99.74% - >99.99%
    Cor e Forma:Solid
    Peso molecular:342.61
  • Desvenlafaxine succinate hydrate

    CAS:
    <p>Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).</p>
    Fórmula:C20H33NO7
    Pureza:99.26%
    Cor e Forma:White Crystalline Powde
    Peso molecular:399.48
  • suvn-911

    CAS:
    <p>suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.</p>
    Fórmula:C11H14Cl2N2O
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:261.15
  • Encequidar

    CAS:
    <p>Encequidar (HM30181A) is a potent and selective P-glycoprotein inhibitor.</p>
    Fórmula:C38H36N6O7
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:688.73
  • Serotonin hydrochloride

    CAS:
    <p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>
    Fórmula:C10H13ClN2O
    Pureza:98.05% - 99.93%
    Cor e Forma:White To Cream Powder
    Peso molecular:212.676
  • DL-Menthol

    CAS:
    <p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>
    Fórmula:C10H20O
    Pureza:99.74%
    Cor e Forma:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)
    Peso molecular:156.27
  • LY2811376

    CAS:
    <p>LY2811376, an orally available non-peptidic β-secretase(BACE1) inhibitor (IC50: 239-249 nM), can decrease Aβ secretion (EC50: 300 nM).</p>
    Fórmula:C15H14F2N4S
    Pureza:99% - 99.01%
    Cor e Forma:Solid
    Peso molecular:320.36
  • Azaphen

    CAS:
    <p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>
    Fórmula:C16H21Cl2N5O
    Pureza:97.62%
    Cor e Forma:Solid
    Peso molecular:370.28
  • HG-10-102-01

    CAS:
    <p>HG-10-102-01 is an inhibitor of leucine-rich repeat kinase 2 (LRRK2, IC50 of 20.3 nM).</p>
    Fórmula:C17H20ClN5O3
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:377.83
  • Harmine hydrochloride

    CAS:
    <p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>
    Fórmula:C13H13ClN2O
    Pureza:99.61% - >99.99%
    Cor e Forma:Yellow To Slightly Green Crystalline Powder
    Peso molecular:248.71
  • Anle138b

    CAS:
    <p>Anle138b: a novel oligomer modulator for disease-modifying therapy of neurodegenerative diseases such as prion and Parkinson's disease</p>
    Fórmula:C16H11BrN2O2
    Pureza:98.88% - 99.82%
    Cor e Forma:Solid
    Peso molecular:343.17