
Neurociência
Os inibidores de neurociência são compostos projetados para modular a atividade de proteínas, enzimas ou receptores específicos no sistema nervoso. Esses inibidores são cruciais para estudar os mecanismos moleculares subjacentes à função neural, transmissão sináptica e doenças neurodegenerativas. Ao direcionar receptores de neurotransmissores, canais iônicos e vias de sinalização, os inibidores de neurociência ajudam na exploração da função cerebral e no desenvolvimento de estratégias terapêuticas para distúrbios neurológicos como Alzheimer, Parkinson e epilepsia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de neurociência de alta qualidade para apoiar sua pesquisa em neurobiologia, neurofarmacologia e ciências cognitivas.
Subcategorias de "Neurociência"
- Receptor 5-HT(940 produtos)
- ACK(1 produtos)
- AChR(574 produtos)
- ATP Citrato Liase(16 produtos)
- Receptor adrenérgico(2.942 produtos)
- BACE(36 produtos)
- Beta Amilóide(204 produtos)
- CaMK(68 produtos)
- COX(562 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor GABA(336 produtos)
- Gama-secretase(59 produtos)
- GluR(255 produtos)
- GlyT(24 produtos)
- Receptor de Histamina(358 produtos)
- LRRK2(33 produtos)
- Receptor de Melatonina(24 produtos)
- NMDAR(28 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(296 produtos)
Exibir 12 mais subcategorias
Foram encontrados 5400 produtos de "Neurociência"
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FG8119
CAS:<p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>Fórmula:C17H15N5O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:321.33SB-737050A
CAS:<p>SB-737050A, a 5-HT antagonist, is used potentially for the treatment of schizophrenia.</p>Fórmula:C22H23ClN2O3S2Cor e Forma:SolidPeso molecular:463.01Chlorpyrifos-oxon
CAS:<p>Chlorpyrifos-oxon, an active metabolite of Chlorpyrifos, is a potent phosphorylating agent that significantly inhibits AChE activity and induces cross-linking between tubulin subunits, thereby disrupting microtubule function [4].</p>Fórmula:C9H11Cl3NO4PCor e Forma:SolidPeso molecular:334.52Ro 04-6790
CAS:<p>Ro 04-6790 is a 5-HT6 receptor antagonist.</p>Fórmula:C12H16N6O2SPureza:98%Cor e Forma:SolidPeso molecular:308.36(S)-3,5-DHPG
CAS:<p>group I mGlu receptor agonist</p>Fórmula:C8H9NO4Pureza:98%Cor e Forma:SolidPeso molecular:183.16S 16924
CAS:<p>S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.</p>Fórmula:C22H24FNO4Pureza:99.35% - 99.6%Cor e Forma:SolidPeso molecular:385.43L-CCG-l
CAS:<p>group II metabotropic glutamate receptor agonist</p>Fórmula:C6H9NO4Pureza:98%Cor e Forma:SolidPeso molecular:159.14DS2
CAS:<p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>Fórmula:C18H12ClN3OSPureza:98%Cor e Forma:SolidPeso molecular:353.83RS 39604
CAS:<p>potent and selective 5-HT4 antagonist</p>Fórmula:C26H37Cl2N3O6SPureza:98%Cor e Forma:SolidPeso molecular:590.56(1S,3R)-ACPD
CAS:<p>(1S,3R)-ACPD is a group I and II mGlu receptor agonist.</p>Fórmula:C7H11NO4Pureza:98%Cor e Forma:SolidPeso molecular:173.17Anti-inflammatory agent 56
CAS:<p>Anti-inflammatory agent 56 (Compound 9), a selective COX-2 inhibitor with an IC50 of 0.54 μM, exhibits anti-oxidant and anti-inflammatory properties by</p>Fórmula:C21H15F3N4O4SPureza:98%Cor e Forma:SolidPeso molecular:476.43MAO-B-IN-21
CAS:<p>MAO-B-IN-21: MAO-B inhibitor with antioxidant, anti-amyloid aggregation, neuroprotective properties, BBB permeable, improves memory in Alzheimer's mice.</p>Fórmula:C24H25ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:440.92SB357134
CAS:<p>SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.</p>Fórmula:C17H18Br2FN3O3SPureza:98%Cor e Forma:SolidPeso molecular:523.21BChE-IN-13
CAS:<p>BChE-IN-13 (17c): Oral, potent, selective BChE inhibitor; IC50: eqBChE 0.22μM, hBChE 0.016μM; aids memory, Alzheimer's research.</p>Fórmula:C24H28N2OCor e Forma:SolidPeso molecular:360.49Depramine
CAS:<p>Depramine (GP 31406), a tricyclic antidepressant, exhibits pharmacological activity by inhibiting acetylcholinesterase, Mg^2+-ATPase, and Na^+/K^+ ATPase</p>Fórmula:C19H22N2Cor e Forma:SolidPeso molecular:278.39Alniditan dihydrochloride
CAS:<p>Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.</p>Fórmula:C17H28Cl2N4OCor e Forma:SolidPeso molecular:375.34TC 1698 dihydrochloride
CAS:<p>nicotinic α7 receptor agonist</p>Fórmula:C13H18N2Pureza:98%Cor e Forma:SolidPeso molecular:202.3ZAPA sulfate
CAS:<p>GABAA receptors agonist</p>Fórmula:C4H8N2O6S2Pureza:98%Cor e Forma:SolidPeso molecular:244.25TASP0433864
CAS:<p>TASP0433864 enhances mGlu2 activity; EC50: 199 nM (human), 206 nM (rat); not an agonist.</p>Fórmula:C18H23N3O3Pureza:98%Cor e Forma:SolidPeso molecular:329.39GABAA receptor agent 8
CAS:<p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>Fórmula:C19H16N4OCor e Forma:SolidPeso molecular:316.36Tacitin
CAS:<p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>Fórmula:C18H20ClNPureza:98%Cor e Forma:SolidPeso molecular:285.81Piperilate
CAS:<p>Piperilate (Pipethanate), a hetrazepine PAF antagonist and anticholinergic used in asthma studies, counters organophosphate toxicity.</p>Fórmula:C21H25NO3Cor e Forma:SolidPeso molecular:339.43JNJ-40068782
CAS:<p>JNJ-40068782 is a potent, selective and systemically active positive allosteric modulator of the mGlu2 receptor.</p>Fórmula:C21H23N3OPureza:98%Cor e Forma:SolidPeso molecular:333.43Distigmine Bromide
CAS:<p>Distigmine Bromide is an acetylcholinesterase inhibitor. It is used for the treatment of underactive neurogenic bladder and myasthenia gravis.</p>Fórmula:C22H32BrN4O4Pureza:98%Cor e Forma:SolidPeso molecular:496.42ASP2535
CAS:<p>ASP2535 is a potent, selective, orally bioavailable, brain permeable and centrally-active glycine transporter-1 (GlyT1) inhibitor.ASP2535 can improve cognitive</p>Fórmula:C22H18N6OPureza:98%Cor e Forma:SolidPeso molecular:382.42PF-4479745
CAS:<p>PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.</p>Fórmula:C17H22N4Pureza:98%Cor e Forma:SolidPeso molecular:282.38HZ166
CAS:<p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>Fórmula:C21H16N4O2Pureza:98%Cor e Forma:SolidPeso molecular:356.38LY 2087101
CAS:<p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>Fórmula:C15H11FN2OS2Pureza:98%Cor e Forma:SolidPeso molecular:318.39Pruvanserin hydrochloride
CAS:<p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>Fórmula:C22H22ClFN4OPureza:99.6%Cor e Forma:SolidPeso molecular:412.89VU0404251
CAS:<p>VU0404251 is a positive allosteric modulator of mGlu5.</p>Fórmula:C19H23FN2O2Cor e Forma:SolidPeso molecular:330.45-Iodo-A-85380 dihydrochloride
CAS:<p>α4β2 and α6β2 nicotinic acetylcholine receptors agonist</p>Fórmula:C9H13Cl2IN2OPureza:98%Cor e Forma:SolidPeso molecular:363.02BChE-IN-4
CAS:<p>BChE-IN-4, a potent butyrylcholinesterase inhibitor, crosses blood-brain barrier, improves memory in mice; promising for Alzheimer's research.</p>Fórmula:C24H37N3OCor e Forma:SolidPeso molecular:383.57Thiobencarb
CAS:<p>Thiobencarb (Siacarb), a thiocarbamate herbicide, is a cholinesterase inhibitor.</p>Fórmula:C12H16ClNOSPureza:99.63%Cor e Forma:Clear Colorless Liquid Thiobencarb Is A Pale Yellow To Brownish Yellow Liquid Non Corrosive Used As An HerbicidePeso molecular:257.78Irindalone
CAS:<p>IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.</p>Fórmula:C24H29FN4OPureza:98%Cor e Forma:SolidPeso molecular:408.51LY-411575 isomer 1
CAS:<p>LY-411575 isomer 1 is a potent γ-secretase inhibitor. LY-411575 isomer 1 is an isomer of LY411575.</p>Fórmula:C26H23F2N3O4Pureza:98%Cor e Forma:SolidPeso molecular:479.48LY456066
CAS:<p>LY456066 is a mGluR1 receptor-selective, negative allosteric modulator.</p>Fórmula:C19H23N3OSPureza:98%Cor e Forma:SolidPeso molecular:341.47Muscarine iodide
CAS:<p>Muscarinic acetylcholine receptor agonist</p>Fórmula:C9H20INO2Pureza:98%Cor e Forma:SolidPeso molecular:301.17Tedatioxetine hydrobromide
CAS:<p>Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.</p>Fórmula:C18H22BrNSPureza:99.65%Cor e Forma:SolidPeso molecular:364.34BuChE-IN-4
CAS:<p>BuChE-IN-4 is a potent inhibitor of BuChE (IC50: 7.7 nM) and exhibits mild antioxidant capacity, non-toxicity, lipophilicity and neuroprotective effects.</p>Fórmula:C21H21BrFN3O4SCor e Forma:SolidPeso molecular:510.38VU0410425
CAS:<p>VU0410425 is a metabotropic glutamate receptor subtype 1 negative allosteric modulator.</p>Fórmula:C19H16ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:369.8Z-Cyclopentyl-AP4
CAS:<p>Group III mGlu receptor agonist</p>Fórmula:C6H12NO5PPureza:98%Cor e Forma:SolidPeso molecular:209.14ML289
CAS:<p>ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, >15-fold selectivity over mGlu2, and inactive against mGlu5.</p>Fórmula:C22H23NO3Pureza:99.54%Cor e Forma:SolidPeso molecular:349.42Mavoglurant racemate
CAS:<p>Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant.</p>Fórmula:C19H23NO3Pureza:98%Cor e Forma:SolidPeso molecular:313.39Alniditan
CAS:<p>Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.</p>Fórmula:C17H26N4OPureza:98%Cor e Forma:SolidPeso molecular:302.41PNU-282987 S enantiomer hydrochloride
CAS:<p>(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.</p>Fórmula:C14H18Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:301.21Indisetron Dihydrochloride
CAS:<p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>Fórmula:C17H24ClN5OCor e Forma:SolidPeso molecular:349.86hMAO-B-IN-2
CAS:<p>hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.</p>Fórmula:C18H23NO3Cor e Forma:SolidPeso molecular:301.38T 82
CAS:<p>T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.</p>Fórmula:C56H62N6O8Pureza:98%Cor e Forma:SolidPeso molecular:947.146OPC-14523 hydrochloride
CAS:<p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>Fórmula:C23H29Cl2N3O2Pureza:99.60%Cor e Forma:SolidPeso molecular:450.4CGP 36216 hydrochloride
CAS:<p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>Fórmula:C5H14NO2PPureza:98%Cor e Forma:SolidPeso molecular:151.14Piclozotan
CAS:<p>Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)</p>Fórmula:C23H24ClN3O2Pureza:98.59%Cor e Forma:SolidPeso molecular:409.91RR-11a
CAS:<p>RR-11a is a synthetic enzyme Legumain inhibitor.</p>Fórmula:C24H28N6O10Pureza:98%Cor e Forma:SolidPeso molecular:560.51SIB 1508Y maleate
CAS:<p>neuronal nicotinic ACh receptor agonist</p>Fórmula:C16H18N2O4Pureza:98%Cor e Forma:SolidPeso molecular:302.33ML337
CAS:<p>ML337 is a negative allosteric modulator of mGlu3 with an IC50 of 593 nM.</p>Fórmula:C21H20FNO3Pureza:99.83%Cor e Forma:SolidPeso molecular:353.39LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Fórmula:C19H23FN4Pureza:98%Cor e Forma:SolidPeso molecular:326.41AY1511
CAS:<p>AY1511 is a low cytotoxic inhibitor of amyloid β (Aβ) aggregation [1].</p>Fórmula:C17H14O6Cor e Forma:SolidPeso molecular:314.29VU0400195
CAS:<p>VU0400195 is a oral effective, positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu(4)).</p>Fórmula:C21H16ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:393.82LY487379 hydrochloride
CAS:<p>Positive allosteric modulator of mGlu2 receptors</p>Fórmula:C21H20ClF3N2O4SPureza:98%Cor e Forma:SolidPeso molecular:488.91SLV-310
CAS:<p>SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.</p>Fórmula:C25H24FN3O2Pureza:99.39%Cor e Forma:SolidPeso molecular:417.48WAY-361789
CAS:<p>WAY-361789 is an agonist of alpha7 nicotinic acetylcholine receptor.</p>Fórmula:C22H31N5O3Cor e Forma:SolidPeso molecular:413.51PXS-4787
CAS:<p>PXS-4787 selectively inhibits LOX with IC50 values: 2 μM (Bovine), 3.2 μM (LOXL1), 0.6 μM (LOXL2), 1.4 μM (LOXL3), 0.2 μM (LOXL4).</p>Fórmula:C10H12FNO2SCor e Forma:SolidPeso molecular:229.275-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Fórmula:C21H23N7Cor e Forma:SolidPeso molecular:373.45ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Fórmula:C25H29BrF3N5OCor e Forma:SolidPeso molecular:552.43Deramciclane fumarate
CAS:<p>Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.</p>Fórmula:C24H35NO5Cor e Forma:SolidPeso molecular:417.54Talsaclidine
CAS:<p>Talsaclidine: full M1 agonist, partial M2/M3 agonist with neuron-stimulating effects.</p>Fórmula:C10H15NOPureza:98%Cor e Forma:SolidPeso molecular:165.23A-85380 HCl
CAS:<p>A-85380 is an agonist of nicotinic acetylcholine receptor.</p>Fórmula:C9H14Cl2N2OCor e Forma:SolidPeso molecular:237.13Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Fórmula:C23H31N5O6Cor e Forma:SolidPeso molecular:473.53Radequinil
CAS:<p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>Fórmula:C18H14N4O3Pureza:98%Cor e Forma:SolidPeso molecular:334.33MAO-B-IN-11
CAS:<p>MAO-B-IN-11 (Compound 8c) is a strong MAO-B blocker with a 1.3 μM IC50 and neuroprotective effects.</p>Fórmula:C22H32O3Cor e Forma:SolidPeso molecular:344.49SEN-1269
CAS:<p>SEN-1269 prevents amyloid-β aggregation, shields neurons, and improves memory by hindering Aβ(1-42)-induced issues.</p>Fórmula:C18H18N4O2Pureza:98%Cor e Forma:SolidPeso molecular:322.36NRA-0160
CAS:<p>NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)</p>Fórmula:C24H23F2N3OSPureza:98%Cor e Forma:SolidPeso molecular:439.52Carburazepam
CAS:<p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>Fórmula:C17H16ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:329.78LRRK2-IN-10
CAS:<p>LRRK2-IN-10 (compound 34) is a potent, mutation-selective, brain-penetrant inhibitor targeting G2019S-LRRK2 kinase with IC50 values of 11 nM for G2019S-LRRK2</p>Fórmula:C20H15N5OPureza:98%Cor e Forma:SolidPeso molecular:341.37MAO-B ligand-1
CAS:<p>MAO-B ligand-1 is a selective MAO-B inhibitor.</p>Fórmula:C19H19N5O4SCor e Forma:SolidPeso molecular:413.45AR-R 17779 hydrochloride
CAS:<p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>Fórmula:C9H15ClN2O2Cor e Forma:SolidPeso molecular:218.68LRE1
CAS:<p>LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.</p>Fórmula:C12H13ClN4SPureza:>99.99%Cor e Forma:SolidPeso molecular:280.78DFMTI
CAS:<p>DFMTI can completely block the rmGlu1 L757V glutamate response.</p>Fórmula:C20H18F2N4OCor e Forma:SolidPeso molecular:368.38GRN-529
CAS:<p>GRN-529 is a selective negative allosteric modulator of the mGluR5 receptor.</p>Fórmula:C22H15F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:391.37Ro4491533
CAS:<p>Ro4491533 is a potent and selective negative allosteric modulator for group II of the metabotropic glutamate receptors (mGluR2/3).</p>Fórmula:C24H20F3N3OCor e Forma:SolidPeso molecular:423.43Dizocilpine
CAS:<p>MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.</p>Fórmula:C16H15NPureza:99.85% - 99.97%Cor e Forma:SolidPeso molecular:221.3γ-secretase modulator 2
CAS:<p>Gamma-secretase modulator 2 selectively targets Alzheimer's by reducing Aβ(1-42), aiding in prevention and treatment.</p>Fórmula:C25H22F4N6O2Pureza:98%Cor e Forma:SolidPeso molecular:514.47BuChE-IN-3
CAS:<p>BuChE-IN-3 (Compound C4) is a potent inhibitor of BuChE (IC50: 8.3 nM). buChE-IN-3 is a mild antioxidant, non-toxic, lipophilic and neuroprotective agent.</p>Fórmula:C21H21F2N3O4SCor e Forma:SolidPeso molecular:449.47AChE/BChE-IN-2
CAS:<p>AChE/BChE-IN-2 (Compound 13b) is a potent inhibitor of AChE/BChE with IC50 values of 0.96 ± 0.14 μM and 1.23 ± 0.23 μM for AChE and BChE, respectively.</p>Fórmula:C23H25N3O5Cor e Forma:SolidPeso molecular:423.46(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:<p>5-HT1A serotonin receptor agonist</p>Fórmula:C16H26BrNOPureza:98%Cor e Forma:SolidPeso molecular:328.29VMY-2-95
CAS:<p>VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.</p>Fórmula:C17H16N2OCor e Forma:SolidPeso molecular:264.32Pozanicline
CAS:<p>Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.</p>Fórmula:C11H16N2OPureza:98%Cor e Forma:SolidPeso molecular:192.26Arecaidine propargyl ester tosylate
CAS:<p>Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.</p>Fórmula:C17H21NO5SPureza:98%Cor e Forma:SolidPeso molecular:351.42MAP4
CAS:<p>metabotropic glutamate receptor modulator</p>Fórmula:C5H12NO5PPureza:98%Cor e Forma:White SolidPeso molecular:197.13mGlu4 receptor agonist 1
CAS:<p>Compound 62, an mGlu4 agonist, has a 308 nM EC50 with anxiolytic and antipsychotic effects.</p>Fórmula:C21H15ClN4O2Cor e Forma:SolidPeso molecular:390.82S-14671
CAS:<p>S-14671: 5-HT1A agonist (pKi 9.3), potent in vivo; 5-HT2A/2C antagonist (pKi 7.8).</p>Fórmula:C22H25N3O2SCor e Forma:SolidPeso molecular:395.52ADX71743
CAS:<p>ADX71743 is a potent and selective negative allosteric modulator of metabotropic glutamate receptor 7.</p>Fórmula:C17H19NO2Cor e Forma:SolidPeso molecular:269.34FTEAA
<p>FTEAA is a dual MAO-A and MAO-B inhibitor with IC50 of 0.52 μM and 1.02 μM, used in cardiovascular and neurological research.</p>Fórmula:C34H26F8N2O2Cor e Forma:SolidPeso molecular:646.57SKF-83566 hydrobromide
CAS:<p>D1-like dopamine receptor antagonist</p>Fórmula:C17H19BrClNOPureza:98%Cor e Forma:SolidPeso molecular:368.7GABA-AT-IN-1
CAS:<p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>Fórmula:C23H18N2O6Cor e Forma:SolidPeso molecular:418.4SB-221284
CAS:<p>5-HT2C/2B receptor antagonist</p>Fórmula:C16H14F3N3OSPureza:98%Cor e Forma:SolidPeso molecular:353.36ETAP
CAS:<p>ETAP, a dual inhibitor of both monoamine oxidase A (MAO-A) and monoamine oxidase B (MAO-B), exhibits antidepressant-like effects and is utilized in the research</p>Fórmula:C18H17N3OPureza:98%Cor e Forma:SolidPeso molecular:291.35(Rac)-WAY-161503
CAS:<p>(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.</p>Fórmula:C11H11Cl2N3OPureza:99.51%Cor e Forma:SolidPeso molecular:272.13Org-25935
CAS:<p>Org-25935, a GlyT-1 inhibitor, is used potentially for the treatment of schizophrenia and alcohol dependence.</p>Fórmula:C21H26ClNO3Cor e Forma:SolidPeso molecular:375.89Phenoxyacetone
CAS:<p>Phenoxyacetone (NSC-1876) is an inhibitor of acetylcholinesterase.</p>Fórmula:C9H10O2Pureza:98.21%Cor e Forma:Clear Light Yellow LiquidPeso molecular:150.17Elucaine
CAS:<p>Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.</p>Fórmula:C19H23NO2Pureza:98%Cor e Forma:SolidPeso molecular:297.39MS 245 oxalate
CAS:<p>MS 245 oxalate is a 5-HT6 antagonist.</p>Fórmula:C21H24N2O7SPureza:98%Cor e Forma:SolidPeso molecular:448.49JNJ1930942
CAS:<p>JNJ1930942 is a novel positive allosteric modulator of the α7 nicotinic acetylcholine receptor.</p>Fórmula:C16H11F4N3OSCor e Forma:SolidPeso molecular:369.34(+/-)-Marmesin
CAS:<p>Marmesin is a novel angiogenesis inhibitor.</p>Fórmula:C14H14O4Pureza:98.00% - 98.00%Cor e Forma:SolidPeso molecular:246.26BMT-145027
CAS:<p>BMT-145027 is a positive allosteric modulator of mGluR5 without inherent agonist activity (EC50 = 47 nM).</p>Fórmula:C23H14ClF3N4Pureza:99.62%Cor e Forma:SolidPeso molecular:438.83A-7 hydrochloride
CAS:<p>A-7 hydrochloride is a calmodulin antagonist and causes alterations in the subpopulation of CD44+CD24- in MDA-MB-231 cells.</p>Fórmula:C20H30Cl2N2O2SPureza:99.38%Cor e Forma:SolidPeso molecular:433.44BPN-15606
CAS:<p>BPN-15606, an oral γ-secretase modulator, reduces Aβ42/Aβ40 with IC50 of 7/17 nM; promising PK/PD, lowers Aβ in rodent CNS.</p>Fórmula:C23H23FN6OCor e Forma:SolidPeso molecular:418.47(±)-Homoproline Hydrochloride
CAS:<p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>Fórmula:C6H12ClNO2Pureza:99.69%Cor e Forma:SolidPeso molecular:165.62S 14063
CAS:<p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>Fórmula:C22H29Cl2N3O2SCor e Forma:SolidPeso molecular:470.45ZLWH-23
CAS:<p>ZLWH-23: AChE inhibitor (IC50: 0.27μM), GSK-3β (6.78μM), BChE (20.82μM), potential in Alzheimer's research.</p>Fórmula:C30H32FN5O2Cor e Forma:SolidPeso molecular:513.61NO 711
CAS:<p>NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>Fórmula:C21H22N2O3Pureza:99.70%Cor e Forma:SolidPeso molecular:350.41CCD-3693
CAS:<p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>Fórmula:C21H31F3O2Pureza:98%Cor e Forma:SolidPeso molecular:372.46SIB-1553A hydrochloride
CAS:<p>SIB-1553A hydrochloride is a nicotinic acetylcholine receptor agonist and a selective neuronal nAChR ligand</p>Fórmula:C13H20ClNOSPureza:99.56% - 99.73%Cor e Forma:SolidPeso molecular:273.82Fonazine
CAS:<p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>Fórmula:C19H25N3O2S2Cor e Forma:SolidPeso molecular:391.55mHTT-IN-2
CAS:<p>mHTT-IN-2 (compound 27) is a potent inhibitor of mutant huntingtin protein (mHTT), with an EC50 value of 0.066 μM.</p>Fórmula:C20H22FN7OPureza:98%Cor e Forma:SolidPeso molecular:395.43Org-13011 fumarate
CAS:<p>Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.</p>Fórmula:C22H29F3N4O5Pureza:98.92%Cor e Forma:SolidPeso molecular:486.48LY 125180
CAS:<p>LY 125180 is a serotonin antagonist.</p>Fórmula:C18H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:305.84ENS-163 phosphate
CAS:<p>Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.</p>Fórmula:C11H19N2O5PSPureza:98%Cor e Forma:SolidPeso molecular:322.32Rivanicline oxalate
CAS:<p>Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).</p>Fórmula:C12H16N2O4Pureza:98%Cor e Forma:SolidPeso molecular:252.27Hexafluronium Bromide
CAS:<p>Hexafluronium bromide enhances muscle relaxation in surgery by blocking acetylcholine receptors.</p>Fórmula:C36H42BrN2Cor e Forma:SolidPeso molecular:582.649ML375
CAS:<p>ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).</p>Fórmula:C23H15ClF2N2O2Cor e Forma:SolidPeso molecular:424.83Rapacuronium bromide
CAS:<p>Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.</p>Fórmula:C37H61BrN2O4Pureza:98%Cor e Forma:SolidPeso molecular:677.8LY 334370 hydrochloride
CAS:<p>5-HT1F receptor agonist</p>Fórmula:C21H23ClFN3OPureza:98%Cor e Forma:SolidPeso molecular:387.88FK960
CAS:<p>FK962 boosts somatostatin, enhances cognition, and raises synaptic density in rat hippocampus.</p>Fórmula:C13H16FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:265.28Bemesetron
CAS:<p>Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.</p>Fórmula:C15H17Cl2NO2Pureza:99.77%Cor e Forma:SolidPeso molecular:314.21Dimethyl-W84 (dibromide)
CAS:<p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>Fórmula:C34H48Br2N4O4Cor e Forma:SolidPeso molecular:736.59Pivalylbenzhydrazine
CAS:<p>Pivhydrazine: strong MAO inhibitor, stunts rat cartilage growth, used in depression research.</p>Fórmula:C12H18N2OCor e Forma:SolidPeso molecular:206.28MAO-IN-M30 dihydrochloride
CAS:<p>MAO-IN-M30 dihydrochloride: potent, brain-specific MAO-A/B inhibitor, iron chelator with antioxidant effects, counters Parkinson's in mice.</p>Fórmula:C14H16Cl2N2OPureza:99.83%Cor e Forma:SolidPeso molecular:299.2Aβ42-IN-1 free base
CAS:<p>Aβ42-IN-1 free base (compound 1v), an orally active γ-secretase modulator with high brain exposure, effectively lowers Aβ42 levels, exhibiting an IC 50 of 0.091</p>Fórmula:C29H26N4O2Pureza:98%Cor e Forma:SolidPeso molecular:462.54VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Fórmula:C24H17ClF2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:438.85PNU-96391
CAS:<p>PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.</p>Fórmula:C15H23NO2SPureza:99.53%Cor e Forma:SolidPeso molecular:281.41Penehyclidine hydrochloride
CAS:<p>Penehyclidine hydrochloride: M1/M3 antagonist, activates NF-κB, anti-inflammatory, anticholinergic.</p>Fórmula:C20H30ClNO2Pureza:99.79%Cor e Forma:SolidPeso molecular:351.91Neuroinflammatory-IN-2
CAS:<p>Neuroinflammatory-IN-2: anti-neuroinflammatory, inhibits MAO-B (IC50: 10.30µM), 96.33% Aβ1-42 aggregation reduction, neuroprotective in PC-12 cells.</p>Fórmula:C25H27FN2O3Cor e Forma:SolidPeso molecular:422.49PAT-1251 Hydrochloride
CAS:<p>PAT-1251 Hydrochloride: Potent, selective, oral LOXL2 inhibitor; IC50s - 0.71 μM (hLOXL2), 1.17 μM (hLOXL3).</p>Fórmula:C18H18ClF4N3O3Pureza:98%Cor e Forma:SolidPeso molecular:435.8WAY 629 hydrochloride
CAS:<p>5-HT2C agonist</p>Fórmula:C15H19ClN2Pureza:98%Cor e Forma:SolidPeso molecular:262.78TMPH hydrochloride
CAS:<p>neuronal nicotinic ACh receptors (nAChRs) antagonist</p>Fórmula:C16H32ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:305.88Alosetron ((Z)-2-butenedioate)
CAS:<p>Alosetron (GR 68755) (Z)-2-butenedioate is a Serotonin 5HT3-receptor antagonist that is used in the treatment of irritable bowel syndrome.</p>Fórmula:C21H22N4O5Pureza:98%Cor e Forma:SolidPeso molecular:410.42LP44 hydrochloride
CAS:<p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>Fórmula:C27H38ClN3OSPureza:98.06%Cor e Forma:SolidPeso molecular:488.13VU 0360223
CAS:<p>VU 0360223 is a negative allosteric modulator of mGlu5.</p>Fórmula:C15H9FN2SPureza:98%Cor e Forma:SolidPeso molecular:268.31Enciprazine
CAS:<p>Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.</p>Fórmula:C23H32N2O6Pureza:98.63%Cor e Forma:SolidPeso molecular:432.51BACE1/2-IN-1
CAS:<p>BACE1/2-IN-1 inhibits BACE1/2 with IC50s of 0.01μM/0.0053μM, has better permeability and lower Pgp efflux but reduced metabolic stability.</p>Fórmula:C21H31N5OSCor e Forma:SolidPeso molecular:401.57UMB68 sodium
CAS:<p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.</p>Fórmula:C6H12NaO3Cor e Forma:SolidPeso molecular:155.149AC260584
CAS:<p>AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).</p>Fórmula:C20H29FN2O2Cor e Forma:SolidPeso molecular:348.45Oxetorone fumarate
CAS:<p>Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.</p>Fórmula:C25H25NO6Pureza:99.809%Cor e Forma:SolidPeso molecular:435.48Bibn 99
CAS:<p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>Fórmula:C31H42ClN5O3Cor e Forma:SolidPeso molecular:568.15MAO-B-IN-16
CAS:<p>MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.</p>Fórmula:C18H19NO3Cor e Forma:SolidPeso molecular:297.35Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Fórmula:C26H31FN2O4Pureza:98%Cor e Forma:SolidPeso molecular:454.53FR-188582
CAS:<p>FR-188582 is a highly selective cyclooxygenase (COX)-2 inhibitor (IC50: 17 nM).</p>Fórmula:C16H13ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:332.8β-CCB
CAS:<p>benzodiazepine receptor ligand</p>Fórmula:C16H16N2O2Pureza:98%Cor e Forma:SolidPeso molecular:268.31Trimedoxime bromide
CAS:<p>Trimedoxime bromide is a cholinesterase reactivator used as an antidote in alkyl phosphate poisoning.</p>Fórmula:C15H18Br2N4O2Cor e Forma:SolidPeso molecular:446.14Nerispirdine HCl
CAS:<p>Nerispirdine enhances acetylcholine, blocks Na+ channels (IC50 11.9µM) and K(v) 1.1/1.2 channels (IC50 3.6/3.7µM).</p>Fórmula:C17H19ClFN3Pureza:98%Cor e Forma:SolidPeso molecular:319.8Tracazolate hydrochloride
CAS:<p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>Fórmula:C16H25ClN4O2Pureza:99.52%Cor e Forma:SolidPeso molecular:340.85LY 2365109 hydrochloride
CAS:<p>glycine transporter 1 (GlyT1) inhibitor</p>Fórmula:C22H27NO5Pureza:98%Cor e Forma:SolidPeso molecular:385.45AChE/BuChE-IN-2
CAS:<p>Compound 5f, an oral AChE/BuChE inhibitor, crosses BBB; IC50: 0.72 μM (AChE), 0.16 μM (BuChE), 62.52 μM (Aβ aggregation).</p>Fórmula:C20H18N2O2Cor e Forma:SolidPeso molecular:318.37DH97
CAS:<p>MT2 melatonin receptor antagonist</p>Fórmula:C22H26N2OPureza:98%Cor e Forma:SolidPeso molecular:334.45CP-457920
CAS:<p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>Fórmula:C18H17N3O3Pureza:99.06% - 99.74%Cor e Forma:SolidPeso molecular:323.35AChE-IN-21
CAS:<p>AChE-IN-21 (I-8), potent, selective AChE inhibitor, IC50: 2.66 nM, good BBB permeability.</p>Fórmula:C24H29NO4Cor e Forma:SolidPeso molecular:395.49FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Fórmula:C27H29F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:465.53RU-505
CAS:<p>RU-505 is an interaction inhibitor of Aβ-fibrinogen that acts by rescuing altered thrombosis and cognitive decline in Alzheimer's disease mice.</p>Fórmula:C28H32FN5OPureza:98%Cor e Forma:SolidPeso molecular:473.58CB-7921220
CAS:<p>CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.</p>Fórmula:C14H12N2O2Pureza:99.59%Cor e Forma:SolidPeso molecular:240.26L-AP4 monohydrate
CAS:<p>L-AP4 (L-APB) is a group III mGluR agonist with EC50s: 0.13μM (mGlu4), 0.29μM (mGlu8), 1.0μM (mGlu6), 249μM (mGlu7).</p>Fórmula:C4H12NO6PCor e Forma:SolidPeso molecular:201.115NAP-1
CAS:<p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>Fórmula:C20H18ClNO2Cor e Forma:SolidPeso molecular:339.82TIK-301
CAS:<p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>Fórmula:C14H17ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:280.75RJR 2429 dihydrochloride
CAS:<p>nAChR agonist that displays selectivity for α4β2</p>Fórmula:C12H18Cl2N2Pureza:98%Cor e Forma:SolidPeso molecular:261.19SERT-IN-2
<p>SERT-IN-2, a potent SERT inhibitor (IC 50 = 0.58 nM), exhibits promising efficacy as an anti-depressant.</p>Cor e Forma:SolidTG41
CAS:<p>TG41 is a GABAA receptors positive modulator.</p>Fórmula:C18H13BrCl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:440.12Dihydro Donepezil
CAS:<p>Dihydro Donepezil (Dihydro E2020), a Donepezil metabolite, is a potent AChE inhibitor (IC50: hAChE 11.6 nM, bAChE 8.12 nM).</p>Fórmula:C24H31NO3Cor e Forma:SolidPeso molecular:381.51LY314228
CAS:<p>LY314228 is an antagonist of 5-HT2A receptor.</p>Fórmula:C20H24N4O3Cor e Forma:SolidPeso molecular:368.43LY 344864 hydrochloride
CAS:<p>LY 344864 hydrochloride is a selective receptor agonist with an affinity of 6 nM (Ki) at the 5-HT1F receptor.</p>Fórmula:C21H23ClFN3OCor e Forma:SolidPeso molecular:387.88Ro 60-0175 fumarate
CAS:<p>5-HT2 receptor agonist</p>Fórmula:C15H16ClFN2O4Pureza:98%Cor e Forma:SolidPeso molecular:342.75VU0455691
CAS:<p>VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.</p>Fórmula:C24H25N5O3SPureza:98%Cor e Forma:SolidPeso molecular:463.55CP-601927
CAS:<p>CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.</p>Fórmula:C12H12F3NCor e Forma:SolidPeso molecular:227.23Antioxidant agent-2
CAS:<p>Antioxidant agent-2 (3c), BBB-permeable, selectively chelates metals; shows neuroprotection, fights liver damage in Alzheimer's research.</p>Fórmula:C23H26N2O7Cor e Forma:SolidPeso molecular:442.46BChE-IN-15
<p>BChE-IN-15 is a compound characterized as a pseudo-irreversible, covalent inhibitor of butyrylcholinesterase (BChE), demonstrating potent activity with an</p>Fórmula:C22H33N3O2Cor e Forma:SolidPeso molecular:371.52MAO-B-IN-12
CAS:<p>MAO-B-IN-12 (16c) is a potent MAO-B inhibitor with an IC50 of 1.3 μM and has neuroprotective properties.</p>Fórmula:C22H30O4Cor e Forma:SolidPeso molecular:358.47PF-0713
CAS:<p>PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.</p>Fórmula:C14H22OPureza:98%Cor e Forma:SolidPeso molecular:206.32(R)-Oxybutynin
CAS:<p>(R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.</p>Fórmula:C22H31NO3Cor e Forma:SolidPeso molecular:357.49Caroxazone
CAS:<p>Caroxazone is an antidepressant drug, monoamine oxidase inhibitor (MAOI) that is irreversible and nonselective meanwhile.</p>Fórmula:C10H10N2O3Cor e Forma:SolidPeso molecular:206.2SB 207710
CAS:<p>SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.</p>Fórmula:C19H27IN2O4Cor e Forma:SolidPeso molecular:474.33Ambutonium bromide
CAS:<p>Ambutonium bromide is an antagonist of acetylcholine.</p>Fórmula:C20H27BrN2OPureza:98%Cor e Forma:SolidPeso molecular:391.35BChE-IN-7
CAS:<p>BChE-IN-7 inhibits AChE/BChE selectively and reversibly; IC50 for BChE: 0.06 μM; crosses blood-brain barrier, protects neurons from Aβ toxicity.</p>Fórmula:C21H24N2O2Cor e Forma:SolidPeso molecular:336.43P-gp inhibitor 1
CAS:<p>P-gp inhibitor 1 inhibits reversing P-glycoprotein-mediated multidrug resistance with an EC50 of 57.9 nM (K562/A02 cells).</p>Fórmula:C32H31N5O2Pureza:98.65%Cor e Forma:SolidPeso molecular:517.62IEM 1925 dihydrobromide
CAS:<p>AMPA receptor antagonist</p>Fórmula:C17H30Br2N2Pureza:98%Cor e Forma:SolidPeso molecular:422.24Rivanicline
CAS:<p>Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.</p>Fórmula:C10H14N2Pureza:98%Cor e Forma:SolidPeso molecular:162.23ONT-093
CAS:<p>ONT-093 (OC-144-093) is an oral P-glycoprotein (P-gp) inhibitor with potential anti-cancer activity, used in the study of myelodysplastic syndromes.</p>Fórmula:C32H38N4OPureza:98.86%Cor e Forma:SolidPeso molecular:494.67RR-11a analog
CAS:<p>RR-11a (aza-peptide) inhibits asparaginyl endopeptidase: IC50 - 4.5 nM (T. Vaginalis, I. ricinus), 31 nM (S. mansoni).</p>Fórmula:C22H29N5O8Pureza:98.80%Cor e Forma:SolidPeso molecular:491.49BisQ
CAS:<p>BisQ is an agonist of photochromic. It used for the muscle-type nAChR.</p>Fórmula:C20H30IN4Pureza:98%Cor e Forma:SolidPeso molecular:453.392PHCCC(4Me)
CAS:<p>THCCC, a PHCCC analog, is a dual metabotropic glutamate receptor 2/3 negative/positive allosteric modulator.</p>Fórmula:C18H16N2O3Cor e Forma:SolidPeso molecular:308.33GABAA receptor agent 7
CAS:<p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>Fórmula:C18H13ClN4OCor e Forma:SolidPeso molecular:336.77Yhhu-3792
CAS:<p>Yhhu-3792 activates Notch, boosts Hes3/Hes5, enhances NSC renewal, expands NSC pool, and may improve memory.</p>Fórmula:C24H24N4O2Cor e Forma:SolidPeso molecular:400.47EMD 386088 hydrochloride
CAS:<p>EMD 386088 hydrochloride is a 5-HT6 receptor agonist.</p>Fórmula:C14H16Cl2N2Pureza:98%Cor e Forma:SolidPeso molecular:283.2sEH inhibitor-5
CAS:<p>sEH inhibitor-5 is a potent inhibitor of sEH (soluble epoxide hydrolase) (IC50: 0.1 nM).</p>Fórmula:C27H26Cl2N6O3SCor e Forma:SolidPeso molecular:585.5Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Fórmula:C22H27ClN2Cor e Forma:SolidPeso molecular:354.92D-NMAPPD
CAS:<p>Litifilimab (BIIB059) is a humanized antibody targeting BDCA2 and CLEC4C for the study of cutaneous lupus erythematosus.</p>Fórmula:C23H38N2O5Cor e Forma:SolidPeso molecular:422.56CGS-12066 maleate salt
CAS:<p>CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.</p>Fórmula:C21H21F3N4O4Cor e Forma:SolidPeso molecular:450.41Ethybenztropine
CAS:<p>Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.</p>Fórmula:C22H27NOPureza:98%Cor e Forma:SolidPeso molecular:321.46Adatanserin
CAS:<p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>Fórmula:C21H31N5OPureza:99.33%Cor e Forma:SolidPeso molecular:369.5Ro 41-3290
CAS:<p>Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.</p>Fórmula:C24H21ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:420.89Alaproclate (hydrochloride)
CAS:<p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>Fórmula:C13H19Cl2NO2Cor e Forma:SolidPeso molecular:292.2Pheniprazine
CAS:<p>Pheniprazine, a potent and long-acting monoamine oxidase inhibitor, shows promise for depression research.</p>Fórmula:C9H14N2Cor e Forma:SolidPeso molecular:150.22

