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Receptor adrenérgico

Receptor adrenérgico

Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.

Subcategorias de "Receptor adrenérgico"

Foram encontrados 645 produtos de "Receptor adrenérgico"

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  • Oxaprotiline hydrochloride

    CAS:
    <p>Oxaprotiline hydrochloride is an antidepressant.</p>
    Fórmula:C20H24ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.86
  • AG-825

    CAS:
    <p>AG-825(Tyrphostin C15) is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (Tyrphostin</p>
    Fórmula:C19H15N3O3S2
    Pureza:98.43%
    Cor e Forma:Yellow Solid
    Peso molecular:397.47
  • O-Desmethyl Mebeverine alcohol

    CAS:
    <p>Mebeverine metabolite O-desmethyl alcohol inhibits α1 receptors, relaxing the gut.</p>
    Fórmula:C15H25NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:251.36
  • Propranolol hydrochloride

    CAS:
    <p>Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse</p>
    Fórmula:C16H22ClNO2
    Pureza:99.94% - >99.99%
    Cor e Forma:White Or Almost White Powder White Powder
    Peso molecular:295.80
  • Nolomirole

    CAS:
    <p>Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.</p>
    Fórmula:C19H27NO4
    Cor e Forma:Solid
    Peso molecular:333.42
  • Terazosin dimer impurity dihydrochloride

    CAS:
    <p>Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.</p>
    Fórmula:C24H30Cl2N8O4
    Cor e Forma:Solid
    Peso molecular:565.46
  • Carvedilol

    CAS:
    <p>Carvedilol (SKF 105517) Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity. The S enantiomer of carvedilol nonselectively binds to and blocks beta-adrenergic receptors, thereby exerting negative inotropic and chronotropic effects, and leading to a reduction in cardiac output. In addition, both enantiomers of carvedilol bind to and block alpha 1-adrenergic receptors, thereby causing vasodilation and reducing peripheral vascular resistance.</p>
    Fórmula:C24H26N2O4
    Pureza:99.73% - 99.97%
    Cor e Forma:Colourless Crystalline Powder
    Peso molecular:406.47
  • L-770644 dihydrochloride

    CAS:
    <p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>
    Fórmula:C30H38ClN7O4S
    Cor e Forma:Solid
    Peso molecular:628.19
  • Ethylnorepinephrine hydrochloride

    CAS:
    <p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>
    Fórmula:C10H16ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:233.69
  • Bromchlorbuterol hydrochloride

    CAS:
    <p>Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.</p>
    Fórmula:C12H19BrCl2N2O
    Cor e Forma:Solid
    Peso molecular:358.1
  • Mabuterol free base

    CAS:
    <p>Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.</p>
    Fórmula:C13H18ClF3N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:310.74
  • Ivabradine-d3 hydrochloride

    CAS:
    <p>Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.</p>
    Fórmula:C27H37ClN2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:508.07
  • Tienoxolol FA


    <p>Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.</p>
    Fórmula:C22H30N2O7S
    Pureza:97.05% - 98.85%
    Cor e Forma:Soild
    Peso molecular:466.55
  • Meluadrine tartrate

    CAS:
    <p>Meluadrine tartrate is an endogenous metabolite.</p>
    Fórmula:C16H24ClNO8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:393.82
  • Benzquinamide

    CAS:
    <p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>
    Fórmula:C22H32N2O5
    Pureza:94.86%
    Cor e Forma:Solid
    Peso molecular:404.5
  • Corynanthine

    CAS:
    <p>Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.</p>
    Fórmula:C21H26N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:354.44
  • SB-206606

    CAS:
    <p>SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.</p>
    Fórmula:C19H22ClNO4
    Cor e Forma:Solid
    Peso molecular:363.83
  • Abediterol napadisylate

    CAS:
    <p>Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.</p>
    Fórmula:C60H68F4N4O14S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1209.32
  • Metaraminol

    CAS:
    <p>Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>
    Fórmula:C9H13NO2
    Cor e Forma:Solid
    Peso molecular:167.21
  • AdTx1


    <p>Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.</p>
    Fórmula:C310H481N87O100S8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:7283.22