
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(940 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.943 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(196 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(69 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(164 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5338 produtos de "GPCR/Proteína-G"
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Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Fórmula:C21H24N4O2SPureza:99.64%Cor e Forma:Light Yellow To Yellow SolidPeso molecular:396.51Monatepil 2maleate
<p>Monatepil 2maleate is an orally active Ca2+-channel antagonist and ACAT inhibitor with alpha(1)-adrenergic receptor blocking activity and antiarrhythmic properties that inhibit vasoconstriction.Monatepil 2maleate may be used to study atherosclerosis.</p>Fórmula:C32H34FN3O5SPureza:98%Cor e Forma:SolidPeso molecular:591.69Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Fórmula:C21H28N2O5Pureza:99.61%Cor e Forma:5 1 (Ntp 1992)Peso molecular:388.46Prostaglandin E1
CAS:<p>Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.</p>Fórmula:C20H34O5Pureza:99.78% - >99.99%Cor e Forma:SolidPeso molecular:354.48Abarelix
CAS:<p>Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.</p>Fórmula:C72H95ClN14O14Pureza:>99.99%Cor e Forma:SolidPeso molecular:1416.06Nortriptyline hydrochloride
CAS:<p>Nortriptyline HCl, a metabolite of amitriptyline, treats major and atypical depression, dysthymia.</p>Fórmula:C19H22ClNPureza:99.85% - ≥95%Cor e Forma:SolidPeso molecular:299.84Volagidemab
CAS:<p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>Pureza:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)Cor e Forma:LiquidMizolastine
CAS:<p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>Fórmula:C24H25FN6OPureza:98% - 99.75%Cor e Forma:SolidPeso molecular:432.49Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Fórmula:C15H24N2O4S·HClPureza:99.4% - 99.77%Cor e Forma:SolidPeso molecular:364.89[Leu15]-Gastrin I, human
CAS:<p>[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.</p>Fórmula:C98H126N20O31Pureza:98.02% - 98.84%Cor e Forma:SolidPeso molecular:2080.16NS-2028
CAS:<p>NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.</p>Fórmula:C9H5BrN2O3Pureza:99.44%Cor e Forma:A Crystalline SolidPeso molecular:269.05Dexchlorpheniramine Maleate
CAS:<p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>Fórmula:C20H23ClN2O4Pureza:99.58%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:390.86Procaine hydrochloride
CAS:<p>Procaine HCl is a benzoic acid derivative used as a local anesthetic, blocking nerve impulses and sensation.</p>Fórmula:C13H20N2O2·HClPureza:99.1% - 99.22%Cor e Forma:White Crystalline PowderPeso molecular:272.77AZ084
CAS:<p>AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.</p>Fórmula:C26H34N4O2Pureza:97.12%Cor e Forma:SolidPeso molecular:434.57Terazosin hydrochloride
CAS:<p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>Fórmula:C19H26ClN5O4Pureza:99.69% - 99.91%Cor e Forma:SolidPeso molecular:423.89Agomelatine
CAS:<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Fórmula:C15H17NO2Pureza:99.92%Cor e Forma:White SolidPeso molecular:243.3Bufotenidine hydrochloride(487-91-2 Free base)
CAS:<p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>Fórmula:C13H19ClN2OPureza:99.88%Cor e Forma:SolidPeso molecular:254.76Carteolol hydrochloride
CAS:<p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>Fórmula:C16H24N2O3·HClPureza:99.84% - 99.91%Cor e Forma:SolidPeso molecular:328.83SR59230A
CAS:<p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>Fórmula:C23H29NO6Pureza:98.84%Cor e Forma:SolidPeso molecular:415.48Frovatriptan succinate hydrate
CAS:<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Fórmula:C18H25N3O6Pureza:99.66%Cor e Forma:SolidPeso molecular:379.41Heptaminol hydrochloride
CAS:<p>Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.</p>Fórmula:C8H20ClNOPureza:98.61%Cor e Forma:White Crystalline PowderPeso molecular:181.71Imidazolidinyl urea
CAS:<p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>Fórmula:C11H16N8O8Pureza:98.6%Cor e Forma:White Fluid Powder With Slight Characteristic OdorPeso molecular:388.29Benserazide hydrochloride
CAS:<p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>Fórmula:C10H15N3O5·HClPureza:98.63% - 99.74%Cor e Forma:White Crystalline SolidPeso molecular:293.7Pheniramine maleate
CAS:<p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>Fórmula:C16H20N2·C4H4O4Pureza:99.85%Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecular:356.42Clomipramine hydrochloride
CAS:<p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>Fórmula:C19H23ClN2·HClPureza:99.04% - 99.47%Cor e Forma:White To Slightly Yellow Crystalline PowderPeso molecular:351.31Isoxsuprine hydrochloride
CAS:<p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>Fórmula:C18H24ClNO3Pureza:99.38%Cor e Forma:Crystals From Water SolidPeso molecular:337.84Naftidrofuryl oxalate
CAS:<p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>Fórmula:C26H35NO7Pureza:97.12% - 98.38%Cor e Forma:SolidPeso molecular:473.56CGS 15943
CAS:<p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>Fórmula:C13H8ClN5OPureza:97.4%Cor e Forma:SolidPeso molecular:285.69Astemizole
CAS:<p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>Fórmula:C28H31FN4OPureza:98.24% - 99.67%Cor e Forma:White Crystals SolidPeso molecular:458.57Orphenadrine hydrochloride
CAS:<p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>Fórmula:C18H23NO·HClPureza:99.88%Cor e Forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Peso molecular:305.85Cefaclor monohydrate
CAS:<p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>Fórmula:C15H16ClN3O5SPureza:97.36% - 99.9%Cor e Forma:White Crystaling PowderPeso molecular:385.82Triflupromazine hydrochloride
CAS:<p>Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.</p>Fórmula:C18H20ClF3N2SPureza:99.76% - 99.82%Cor e Forma:CrystalsPeso molecular:388.88Alosetron hydrochloride
CAS:<p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>Fórmula:C17H19ClN4OPureza:99.90%Cor e Forma:Off-White PowderPeso molecular:330.81Bromopride
CAS:<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Fórmula:C14H22BrN3O2Pureza:99.95%Cor e Forma:SolidPeso molecular:344.252-(1-Piperazinyl)pyrimidine
CAS:<p>2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.</p>Fórmula:C8H12N4Pureza:98.46%Cor e Forma:Liquid - Crystal - LumpPeso molecular:164.21Propafenone
CAS:<p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>Fórmula:C21H27NO3Pureza:99.02%Cor e Forma:SolidPeso molecular:341.44Cericlamine
CAS:<p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>Fórmula:C12H17Cl2NOPureza:99.38%Cor e Forma:SolidPeso molecular:262.18Mebhydrolin napadisylate
CAS:<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Fórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.96%Cor e Forma:White Or Almost White CrystallinePeso molecular:420.52Flopropione
CAS:<p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>Fórmula:C9H10O4Pureza:99.93%Cor e Forma:SolidPeso molecular:182.17Atomoxetine hydrochloride
CAS:<p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>Fórmula:C17H22ClNOPureza:99.86%Cor e Forma:White SolidPeso molecular:291.82RS102895 hydrochloride
CAS:<p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>Fórmula:C21H22ClF3N2O2Pureza:98.95%Cor e Forma:SolidPeso molecular:426.86Azasetron hydrochloride
CAS:<p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>Fórmula:C17H20ClN3O3·HClPureza:99.50%Cor e Forma:SolidPeso molecular:386.27Degarelix acetate(214766-78-6 free base)
CAS:<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Fórmula:C84H107ClN18O18Pureza:98.66%Cor e Forma:SolidPeso molecular:1692.34Pamabrom
CAS:<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Fórmula:C11H18BrN5O3Pureza:99.84% - >99.99%Cor e Forma:CoaPeso molecular:348.2DSP-4 hydrochloride
CAS:<p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>Fórmula:C11H16BrCl2NPureza:99.9%Cor e Forma:SolidPeso molecular:313.06Mefexamide hydrochloride
CAS:<p>Mefexamide hydrochloride is a central stimulant.</p>Fórmula:C15H25ClN2O3Pureza:99.95%Cor e Forma:SolidPeso molecular:316.83Fezolinetant
CAS:<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Fórmula:C16H15FN6OSPureza:98.62% - 99.7%Cor e Forma:SolidPeso molecular:358.39Mepyramine maleate
CAS:<p>Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.</p>Fórmula:C21H27N3O5Pureza:99.51% - 99.7%Cor e Forma:White Crystalline PowderPeso molecular:401.47Glycerol phenylbutyrate
CAS:<p>Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).</p>Fórmula:C33H38O6Pureza:98.54% - 99.74%Cor e Forma:SolidPeso molecular:530.65EMPA
CAS:<p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>Fórmula:C23H26N4O4SPureza:99.11%Cor e Forma:SolidPeso molecular:454.54JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Fórmula:C11H19N5Pureza:98.33% - 99.62%Cor e Forma:SolidPeso molecular:221.3Ogerin
CAS:<p>Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).</p>Fórmula:C17H17N5OPureza:99.5% - 99.75%Cor e Forma:SolidPeso molecular:307.35Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Fórmula:C20H23ClN2O5Pureza:99.97%Cor e Forma:Off-White SolidPeso molecular:406.86Nicergoline
CAS:<p>Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.</p>Fórmula:C24H26BrN3O3Pureza:98% - 99.80%Cor e Forma:SolidPeso molecular:484.39DPTN dihydrochloride
CAS:<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Fórmula:C22H20Cl2N4OSPureza:99.95%Cor e Forma:SoildPeso molecular:459.39Vabicaserin hydrochloride
CAS:<p>Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).</p>Fórmula:C15H21ClN2Pureza:98.32%Cor e Forma:SolidPeso molecular:264.79Isoprenaline hydrochloride
CAS:<p>Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.</p>Fórmula:C11H18ClNO3Pureza:98% - 99.65%Cor e Forma:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)Peso molecular:247.719GANT 58
CAS:<p>GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).</p>Fórmula:C24H16N4SPureza:99.53%Cor e Forma:SolidPeso molecular:392.48Terbutaline Sulfate
CAS:Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.Fórmula:C12H19NO3H2SO4Pureza:99.47% - 99.94%Cor e Forma:Crystalline PowderPeso molecular:274.32Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Fórmula:C21H26ClN3OSPureza:99.3% - 99.99%Cor e Forma:SolidPeso molecular:403.97Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Fórmula:C34H36Cl2N6O5S·2ClHPureza:99.17% - 99.58%Cor e Forma:SoildPeso molecular:784.58Gevotroline
CAS:<p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>Fórmula:C19H20FN3Pureza:98.65%Cor e Forma:SolidPeso molecular:309.38Senktide acetate
<p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>Fórmula:C42H59N7O13SPureza:98.26%Cor e Forma:SolidPeso molecular:902.02Terfenadine
CAS:<p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>Fórmula:C32H41NO2Pureza:98.76% - 99.75%Cor e Forma:SolidPeso molecular:471.67hGPR91 antagonist 1
CAS:<p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>Fórmula:C31H23F4N3OPureza:98.89%Cor e Forma:SolidPeso molecular:529.53Alfuzosin hydrochloride
CAS:<p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>Fórmula:C19H27N5O4·HClPureza:99.78%Cor e Forma:White To Off-White SolidPeso molecular:425.91Naluzotan hydrochloride
CAS:<p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>Fórmula:C23H39ClN4O3SPureza:99.96%Cor e Forma:SolidPeso molecular:487.1Proglumide
CAS:<p>Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.</p>Fórmula:C18H26N2O4Pureza:99.4% - 99.45%Cor e Forma:White Crystalline PowderPeso molecular:334.41TSHR antagonist S37
CAS:<p>TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).</p>Fórmula:C25H20N2O3S2Pureza:98.35%Cor e Forma:SolidPeso molecular:460.57Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Fórmula:C10H7KN6OPureza:98.91% - 99.63%Cor e Forma:Crystals From Dimethylformamide Crystalline SolidPeso molecular:266.31Mifentidine
CAS:<p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>Fórmula:C13H16N4Pureza:98.34% - 99.73%Cor e Forma:SolidPeso molecular:228.29Oxeladin citrate
CAS:<p>Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.</p>Fórmula:C26H41NO10Pureza:97.23%Cor e Forma:SolidPeso molecular:527.6Salmeterol
CAS:<p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>Fórmula:C25H37NO4Pureza:99.2% - 99.9%Cor e Forma:SolidPeso molecular:415.57Carbetapentane citrate
CAS:<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Cor e Forma:White To Off-White SolidPeso molecular:525.59(Rac)-MGV354
CAS:<p>(Rac)-MGV354: a racemic sGC activator; EC50s <0.5 nM (CHO cells), 5 nM (GTM-3 E cells).</p>Fórmula:C35H37N5O3Pureza:99.26%Cor e Forma:SolidPeso molecular:575.7Phentolamine mesylate
CAS:<p>Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.</p>Fórmula:C17H19N3O·CH4O3SPureza:99.77% - >99.99%Cor e Forma:By The Metabolic Processes Of Bacillus Subtilis And LicheniformisPeso molecular:377.46Cloroperone
CAS:<p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>Fórmula:C22H23ClFNO2Pureza:98.40%Cor e Forma:SoildPeso molecular:387.88Apelin-13
CAS:<p>Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor</p>Fórmula:C69H111N23O16SPureza:96.81%Cor e Forma:SolidPeso molecular:1550.83Ondansetron hydrochloride dihydrate
CAS:<p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>Fórmula:C18H19N3O·HCl·2H2OPureza:99.92%Cor e Forma:White Crystal PowderPeso molecular:365.86Bambuterol hydrochloride
CAS:<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Fórmula:C18H30ClN3O5Pureza:99.53% - 99.61%Cor e Forma:White SolidPeso molecular:403.91(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:<p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>Fórmula:C20H29N3O8Pureza:99.72%Cor e Forma:SoildPeso molecular:439.46Tropanserin
CAS:<p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>Fórmula:C17H23NO2Pureza:99.74%Cor e Forma:SolidPeso molecular:273.37Amiselimod hydrochloride
CAS:<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Fórmula:C19H31ClF3NO3Pureza:99.55%Cor e Forma:SolidPeso molecular:413.9Tetrahydrozoline
CAS:<p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>Fórmula:C13H16N2Pureza:97.85% - 99.77%Cor e Forma:SolidPeso molecular:200.28Metoclopramide hydrochloride
CAS:<p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>Fórmula:C14H22ClN3O2·HClPureza:99.99%Cor e Forma:White To Off-White PowderPeso molecular:336.26SEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Fórmula:C9H14ClNOSPureza:99.86% - 99.99%Cor e Forma:SolidPeso molecular:219.73JP1302 dihydrochloride
CAS:<p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>Fórmula:C24H26Cl2N4Pureza:99.61%Cor e Forma:SolidPeso molecular:441.4Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Fórmula:C21H23N3OSPureza:99.61%Cor e Forma:SolidPeso molecular:365.49Nepafenac
CAS:<p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>Fórmula:C15H14N2O2Pureza:98.94% - 99.43%Cor e Forma:SolidPeso molecular:254.28Latanoprostene bunod
CAS:<p>LBN is a NO-donating prostaglandin analog for reducing IOP in glaucoma or OHT patients.</p>Fórmula:C27H41NO8Pureza:99.33% - 99.69%Cor e Forma:SolidPeso molecular:507.62Fexofenadine hydrochloride
CAS:<p>Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with</p>Fórmula:C32H40ClNO4Pureza:>99.99%Cor e Forma:White Crystalline PowderPeso molecular:538.12Dexpramipexole dihydrochloride
CAS:<p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>Fórmula:C10H19Cl2N3SPureza:99.75% - 99.88%Cor e Forma:SolidPeso molecular:284.25Ifenprodil Tartrate
CAS:<p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>Fórmula:C21H27NO2C4H6O6Pureza:99.02% - 99.55%Cor e Forma:SolidPeso molecular:400.49Evatanepag
CAS:<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Fórmula:C25H28N2O5SPureza:97.09%Cor e Forma:SolidPeso molecular:468.57Prochlorperazine Maleate
CAS:<p>Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.</p>Fórmula:C28H32ClN3O8SPureza:99.78%Cor e Forma:Off-White PowderPeso molecular:606.09PF-610355 HCl
<p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>Fórmula:C19H22ClN7O6Pureza:97.97%Cor e Forma:SolidPeso molecular:479.87Luzindole
CAS:<p>Luzindole (N-0774) is a selective melatonin receptor antagonist.</p>Fórmula:C19H20N2OPureza:98.53%Cor e Forma:Off-White Amorphous SolidPeso molecular:292.37Ziprasidone hydrochloride monohydrate
CAS:<p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>Fórmula:C21H21ClN4OS·HCl·H2OPureza:98% - 99.83%Cor e Forma:Off-White PowderPeso molecular:467.12NEO 376
CAS:<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Fórmula:C20H24ClN3OPureza:99.56%Cor e Forma:SolidPeso molecular:357.88Rimonabant hydrochloride
CAS:<p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>Fórmula:C22H22Cl4N4OPureza:98.24% - 99.5%Cor e Forma:Off-White To White Crystalline PowderPeso molecular:500.25Citalopram hydrobromide
CAS:<p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>Fórmula:C20H22BrFN2OPureza:99.81%Cor e Forma:White Crystalline PowderPeso molecular:405.304L-741626
CAS:<p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>Fórmula:C20H21ClN2OPureza:98.57%Cor e Forma:SolidPeso molecular:340.85Ketanserin
CAS:<p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Cor e Forma:SolidPeso molecular:395.43Indusatumab
CAS:<p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>Pureza:> 95% - > 95%Cor e Forma:LiquidPeso molecular:145.18 kDaAnamorelin
CAS:<p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>Fórmula:C31H42N6O3Pureza:99.35% - 99.94%Cor e Forma:SolidPeso molecular:546.7Tripelennamine hydrochloride
CAS:<p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>Fórmula:C16H21N3·HClPureza:99.54% - 99.81%Cor e Forma:White SolidPeso molecular:291.82PF-06882961
CAS:<p>PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Fórmula:C31H30FN5O4Pureza:98.06% - 99.54%Cor e Forma:SolidPeso molecular:555.62-Bromo-6-methoxynaphthalene
CAS:<p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>Fórmula:C11H9BrOPureza:98.51%Cor e Forma:White To Off-White PowderPeso molecular:237.09Cisapride
CAS:<p>Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.</p>Fórmula:C23H29ClFN3O4Pureza:99.77%Cor e Forma:White To Slightly Biege Powder SolidPeso molecular:465.95Protriptyline hydrochloride
CAS:<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Fórmula:C19H21N·HClPureza:98.54% - 99.98%Cor e Forma:SolidPeso molecular:299.84Urocortin (rat) acetate
<p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>Pureza:97.76%Cor e Forma:SoildNylidrin hydrochloride
CAS:<p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.</p>Fórmula:C19H26ClNO2Pureza:99.35%Cor e Forma:SolidPeso molecular:335.87Terlipressin Acetate
CAS:<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Cor e Forma:SolidPeso molecular:1347.5Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Pureza:SDS-PAGE:95% SEC-HPLC:98.90%Cor e Forma:LiquidPeso molecular:146.43 kDaLafutidine
CAS:<p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>Fórmula:C22H29N3O4SPureza:98.55%Cor e Forma:Yellowish White Crystalline PowderPeso molecular:431.55Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Fórmula:C18H26ClN3O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:367.87Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Cor e Forma:White Crystalline PowderPeso molecular:313.86Erenumab
CAS:<p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>Pureza:99.43% (SEC-HPLC) - > 95%Cor e Forma:LiquidPeso molecular:146.2 kDaTalastine
CAS:<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Fórmula:C19H21N3OPureza:98.50% - 99.44%Cor e Forma:SolidPeso molecular:307.39Methyldopa
CAS:<p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>Fórmula:C10H13NO4Pureza:98.95% - 99.86%Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21Desipramine hydrochloride
CAS:<p>Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.</p>Fórmula:C18H23ClN2Pureza:99.58% - 99.94%Cor e Forma:White To Off-White PowderPeso molecular:302.842Naftifine hydrochloride
CAS:<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Fórmula:C21H22ClNPureza:98.75% - 99.84%Cor e Forma:SolidPeso molecular:323.86Fluoxetine hydrochloride
CAS:<p>Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.</p>Fórmula:C17H19ClF3NOPureza:99.6% - 99.98%Cor e Forma:White To Off-White Crystalline Solid White To Off-White PowderPeso molecular:345.787Clonidine hydrochloride
CAS:<p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Cor e Forma:SolidPeso molecular:266.55Sergliflozin A
CAS:<p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>Fórmula:C20H24O7Pureza:99.43%Cor e Forma:SolidPeso molecular:376.4Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:463.79Indacaterol maleate
CAS:<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Fórmula:C28H32N2O7Pureza:99.03% - 99.67%Cor e Forma:SolidPeso molecular:508.56ML-180
CAS:<p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>Fórmula:C20H25ClN4O2Pureza:99.74%Cor e Forma:SolidPeso molecular:388.89CD80-IN-3
CAS:<p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>Fórmula:C17H10FN3O3Pureza:98.08%Cor e Forma:SolidPeso molecular:323.28CYM 50769
CAS:<p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>Fórmula:C24H17ClN2O3Pureza:98% - 99.08%Cor e Forma:SolidPeso molecular:416.86Fluvoxamine maleate
CAS:<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Fórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Cor e Forma:White Crystalline PowderPeso molecular:434.41Silodosin
CAS:<p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Cor e Forma:Colorless To Pink SolidPeso molecular:495.53Metaproterenol hemisulfate
CAS:<p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>Fórmula:C11H17NO3·5H2O4SPureza:98.53% - 99.74%Cor e Forma:SolidPeso molecular:260.3Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Fórmula:C21H24ClNOPureza:99.77% - >99.99%Cor e Forma:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Urapidil hydrochloride
CAS:<p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>Fórmula:C20H29N5O3·HClPureza:99.58%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:423.94Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:383.51JNJ-18038683
CAS:<p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>Fórmula:C26H28ClN3O7Pureza:97.29%Cor e Forma:SolidPeso molecular:529.97PF429242 dihydrochloride
CAS:<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Fórmula:C25H37Cl2N3O2Pureza:99.68%Cor e Forma:SolidPeso molecular:482.49Acetophenazine dimaleate
CAS:<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Fórmula:C31H37N3O10SPureza:99.39% - 99.48%Cor e Forma:SolidPeso molecular:643.71Naftopidil
CAS:<p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>Fórmula:C24H28N2O3Pureza:99.60% - 99.97%Cor e Forma:White Crystalline PowderPeso molecular:392.49Ifenprodil
CAS:<p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>Fórmula:C21H27NO2Pureza:99.58%Cor e Forma:White Crystalline PowderPeso molecular:325.44Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Fórmula:C18H25ClN4OPureza:99.88% - 99.93%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:348.87Fluparoxan hydrochloride
CAS:<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Fórmula:C10H11ClFNO2Pureza:99.98%Cor e Forma:SoildPeso molecular:231.65Blonanserin
CAS:<p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>Fórmula:C23H30FN3Pureza:99.85%Cor e Forma:SolidPeso molecular:367.5Fosopamine(HCl)
CAS:<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Fórmula:C9H15ClNO5PPureza:99.84%Cor e Forma:SolidPeso molecular:283.65NF-56-EJ40 hydrochloride
CAS:<p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>Fórmula:C27H31Cl2N3O3Pureza:99.33%Cor e Forma:SoildPeso molecular:516.46Levosulpiride
CAS:<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Cor e Forma:White Crystalline PowderPeso molecular:341.43Fluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Fórmula:C17H18F3NOPureza:99.07% - 99.28%Cor e Forma:SolidPeso molecular:309.33Astressin acetate
<p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>Fórmula:C163H273N49O44Pureza:96.87%Cor e Forma:SolidPeso molecular:3623.21Diphenylpyraline hydrochloride
CAS:<p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>Fórmula:C19H23NO·HClPureza:98.72%Cor e Forma:SolidPeso molecular:317.85Chlorprothixene hydrochloride
CAS:<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Fórmula:C18H18ClNS·HClPureza:99.76%Cor e Forma:White PowderPeso molecular:352.32Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:PowderPeso molecular:522.55Olanzapine
CAS:<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Fórmula:C17H20N4SPureza:99.86% - ≥95%Cor e Forma:Yellowish Crystalline PowderPeso molecular:312.43CP-809101 hydrochloride
CAS:<p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Fórmula:C15H18Cl2N4OPureza:99.5%Cor e Forma:SolidPeso molecular:341.24Trazodone hydrochloride
CAS:<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Fórmula:C19H23Cl2N5OPureza:99.5% - 99.52%Cor e Forma:SolidPeso molecular:408.33MK-0249 FA
<p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>Fórmula:C24H26F3N3O4Pureza:99.98%Cor e Forma:SolidPeso molecular:477.48Antazoline hydrochloride
CAS:<p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>Fórmula:C17H19N3·HClPureza:98% - 99.53%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:301.82Brefonalol HCl
<p>Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.</p>Fórmula:C22H29ClN2O2Pureza:99.45%Cor e Forma:SolidPeso molecular:388.93Aripiprazole
CAS:<p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Cor e Forma:Colourless Flake Crystalline SolidPeso molecular:448.39YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Fórmula:C33H37N5O5SPureza:99.67%Cor e Forma:SolidPeso molecular:615.74Alverine citrate
CAS:<p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>Fórmula:C26H35NO7Pureza:98.53% - 99.43%Cor e Forma:CoaPeso molecular:473.57KGA-2727
CAS:<p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>Fórmula:C26H40N4O8Pureza:98.46%Cor e Forma:SolidPeso molecular:536.62(3aR,9aR)-Fluparoxan
CAS:<p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Fórmula:C10H10FNO2Pureza:97.82%Cor e Forma:SoildPeso molecular:195.19Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Fórmula:C14H15Cl2NSPureza:99.85% - >99.99%Cor e Forma:White PowderPeso molecular:300.25Zolmitriptan
CAS:<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Cor e Forma:White Or Kind Of White PowderPeso molecular:287.36Timonacic
CAS:<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Fórmula:C4H7NO2SPureza:99.99%Cor e Forma:SolidPeso molecular:133.17AH 6809
CAS:<p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>Fórmula:C17H14O5Pureza:97.59%Cor e Forma:SolidPeso molecular:298.29Phenothiazine
CAS:<p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>Fórmula:C12H9NSPureza:99.95%Cor e Forma:Yellow Solid PelletsPeso molecular:199.27Noradrenaline bitartrate
CAS:<p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>Fórmula:C12H19NO10Pureza:99.53% - >99.99%Cor e Forma:SolidPeso molecular:337.28ESI-05
CAS:<p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>Fórmula:C16H18O2SPureza:97.22%Cor e Forma:SolidPeso molecular:274.38AB928
CAS:<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Fórmula:C23H22N8OPureza:98.09% - >99.99%Cor e Forma:SolidPeso molecular:426.47Asenapine Maleate
CAS:<p>Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.</p>Fórmula:C21H20ClNO5Pureza:99.28%Cor e Forma:SolidPeso molecular:401.84DREADD agonist 21
CAS:<p>DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).</p>Fórmula:C17H18N4Pureza:99.94%Cor e Forma:SolidPeso molecular:278.35LCKLSL hydrochloride
<p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>Fórmula:C30H58ClN7O8SPureza:98.02% - 99.31%Cor e Forma:SolidPeso molecular:712.34(R)-Elagolix
CAS:<p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>Fórmula:C32H30F5N3O5Pureza:99.08%Cor e Forma:SolidPeso molecular:631.59Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Fórmula:C31H38N2OPureza:97.49%Cor e Forma:SolidPeso molecular:454.65Hydroxyzine Pamoate
CAS:<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Fórmula:C44H43ClN2O8Pureza:99.49%Cor e Forma:SolidPeso molecular:763.27Leronlimab
CAS:<p>Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.</p>Pureza:SDS-PAGE:95.0%;SEC-HPLC:99.6%Cor e Forma:LiquidPeso molecular:146.66 kDaFilorexant
CAS:<p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).</p>Fórmula:C24H25FN4O2Pureza:98.88%Cor e Forma:SolidPeso molecular:420.48Levodropropizine
CAS:<p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>Fórmula:C13H20N2O2Pureza:99.87% - 99.93%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.31Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Fórmula:C19H24N2O·HClPureza:99.84% - 99.92%Cor e Forma:White SolidPeso molecular:332.87Ro 10-5824 dihydrochloride
CAS:<p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>Fórmula:C17H22Cl2N4Pureza:99.79%Cor e Forma:SolidPeso molecular:353.29Moxisylyte hydrochloride
CAS:<p>Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.</p>Fórmula:C16H26ClNO3Pureza:99.93% - ≥95%Cor e Forma:SolidPeso molecular:315.84Ziprasidone hydrochloride
CAS:<p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>Fórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Cor e Forma:SolidPeso molecular:449.4Vilazodone
CAS:<p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>Fórmula:C26H27N5O2Pureza:99.61%Cor e Forma:Light Yellow SolidPeso molecular:441.52Dopexamine hydrochloride
CAS:<p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>Fórmula:C22H34Cl2N2O2Pureza:98.55%Cor e Forma:SolidPeso molecular:429.42Dimenhydrinate
CAS:<p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96Adrenalone hydrochloride
CAS:<p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>Fórmula:C9H11NO3·HClPureza:99.94%Cor e Forma:SolidPeso molecular:217.65Carvedilol EP IMpurity E
CAS:<p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>Fórmula:C9H14ClNO2Pureza:99.53%Cor e Forma:White To Almost White Solid CrystallinePeso molecular:203.666Promazine hydrochloride
CAS:<p>Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.</p>Fórmula:C17H21ClN2SPureza:99.90%Cor e Forma:SolidPeso molecular:320.88Acebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Fórmula:C18H29ClN2O4Pureza:99.92% - >99.99%Cor e Forma:White Or Slightly Off-White Crystalline Powder SolidPeso molecular:372.89Pizotifen
CAS:<p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>Fórmula:C19H21NSPureza:99.93%Cor e Forma:SolidPeso molecular:295.44Linaclotide
CAS:<p>Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.</p>Fórmula:C59H79N15O21S6Pureza:97.93% - 98.71%Cor e Forma:SolidPeso molecular:1526.74MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Fórmula:C27H25N3O4S2Pureza:97.44%Cor e Forma:SolidPeso molecular:519.64Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Fórmula:C15H20N2O2·HClPureza:99.64% - 99.92%Cor e Forma:SolidPeso molecular:296.79Desvenlafaxine
CAS:<p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>Fórmula:C16H25NO2Pureza:99.46% - 99.81%Cor e Forma:White Crystalline PowderPeso molecular:263.38Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Fórmula:C21H27Cl3N2O3Pureza:99.4% - 99.97%Cor e Forma:SolidPeso molecular:461.81Olinciguat
CAS:<p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>Fórmula:C21H16F5N7O3Pureza:99.33% - 99.71%Cor e Forma:SolidPeso molecular:509.39Roxatidine Acetate hydrochloride
CAS:<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Fórmula:C19H29ClN2O4Pureza:99.49%Cor e Forma:SolidPeso molecular:384.9Tolnaftate
CAS:<p>Tolnaftate (NP-27) is a synthetic antifungal agent.</p>Fórmula:C19H17NOSPureza:98.85%Cor e Forma:White PowderPeso molecular:307.41

