CymitQuimica logo
GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

Exibir 18 mais subcategorias

Foram encontrados 5338 produtos de "GPCR/Proteína-G"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
produtos por página.
  • Mirabegron

    CAS:
    <p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>
    Fórmula:C21H24N4O2S
    Pureza:99.64%
    Cor e Forma:Light Yellow To Yellow Solid
    Peso molecular:396.51
  • Monatepil 2maleate


    <p>Monatepil 2maleate is an orally active Ca2+-channel antagonist and ACAT inhibitor with alpha(1)-adrenergic receptor blocking activity and antiarrhythmic properties that inhibit vasoconstriction.Monatepil 2maleate may be used to study atherosclerosis.</p>
    Fórmula:C32H34FN3O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:591.69
  • Doxylamine succinate

    CAS:
    <p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>
    Fórmula:C21H28N2O5
    Pureza:99.61%
    Cor e Forma:5 1 (Ntp 1992)
    Peso molecular:388.46
  • Prostaglandin E1

    CAS:
    <p>Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.</p>
    Fórmula:C20H34O5
    Pureza:99.78% - >99.99%
    Cor e Forma:Solid
    Peso molecular:354.48
  • Abarelix

    CAS:
    <p>Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.</p>
    Fórmula:C72H95ClN14O14
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1416.06
  • Nortriptyline hydrochloride

    CAS:
    <p>Nortriptyline HCl, a metabolite of amitriptyline, treats major and atypical depression, dysthymia.</p>
    Fórmula:C19H22ClN
    Pureza:99.85% - ≥95%
    Cor e Forma:Solid
    Peso molecular:299.84
  • Volagidemab

    CAS:
    <p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>
    Pureza:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)
    Cor e Forma:Liquid
  • Mizolastine

    CAS:
    <p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>
    Fórmula:C24H25FN6O
    Pureza:98% - 99.75%
    Cor e Forma:Solid
    Peso molecular:432.49
  • Tiapride hydrochloride

    CAS:
    <p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>
    Fórmula:C15H24N2O4S·HCl
    Pureza:99.4% - 99.77%
    Cor e Forma:Solid
    Peso molecular:364.89
  • [Leu15]-Gastrin I, human

    CAS:
    <p>[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.</p>
    Fórmula:C98H126N20O31
    Pureza:98.02% - 98.84%
    Cor e Forma:Solid
    Peso molecular:2080.16
  • NS-2028

    CAS:
    <p>NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.</p>
    Fórmula:C9H5BrN2O3
    Pureza:99.44%
    Cor e Forma:A Crystalline Solid
    Peso molecular:269.05
  • Dexchlorpheniramine Maleate

    CAS:
    <p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>
    Fórmula:C20H23ClN2O4
    Pureza:99.58%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:390.86
  • Procaine hydrochloride

    CAS:
    <p>Procaine HCl is a benzoic acid derivative used as a local anesthetic, blocking nerve impulses and sensation.</p>
    Fórmula:C13H20N2O2·HCl
    Pureza:99.1% - 99.22%
    Cor e Forma:White Crystalline Powder
    Peso molecular:272.77
  • AZ084

    CAS:
    <p>AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.</p>
    Fórmula:C26H34N4O2
    Pureza:97.12%
    Cor e Forma:Solid
    Peso molecular:434.57
  • Terazosin hydrochloride

    CAS:
    <p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>
    Fórmula:C19H26ClN5O4
    Pureza:99.69% - 99.91%
    Cor e Forma:Solid
    Peso molecular:423.89
  • Agomelatine

    CAS:
    <p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>
    Fórmula:C15H17NO2
    Pureza:99.92%
    Cor e Forma:White Solid
    Peso molecular:243.3
  • Bufotenidine hydrochloride(487-91-2 Free base)

    CAS:
    <p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>
    Fórmula:C13H19ClN2O
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:254.76
  • Carteolol hydrochloride

    CAS:
    <p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>
    Fórmula:C16H24N2O3·HCl
    Pureza:99.84% - 99.91%
    Cor e Forma:Solid
    Peso molecular:328.83
  • SR59230A

    CAS:
    <p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>
    Fórmula:C23H29NO6
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:415.48
  • Frovatriptan succinate hydrate

    CAS:
    <p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>
    Fórmula:C18H25N3O6
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:379.41
  • Heptaminol hydrochloride

    CAS:
    <p>Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.</p>
    Fórmula:C8H20ClNO
    Pureza:98.61%
    Cor e Forma:White Crystalline Powder
    Peso molecular:181.71
  • Imidazolidinyl urea

    CAS:
    <p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>
    Fórmula:C11H16N8O8
    Pureza:98.6%
    Cor e Forma:White Fluid Powder With Slight Characteristic Odor
    Peso molecular:388.29
  • Benserazide hydrochloride

    CAS:
    <p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>
    Fórmula:C10H15N3O5·HCl
    Pureza:98.63% - 99.74%
    Cor e Forma:White Crystalline Solid
    Peso molecular:293.7
  • Pheniramine maleate

    CAS:
    <p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>
    Fórmula:C16H20N2·C4H4O4
    Pureza:99.85%
    Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
    Peso molecular:356.42
  • Clomipramine hydrochloride

    CAS:
    <p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>
    Fórmula:C19H23ClN2·HCl
    Pureza:99.04% - 99.47%
    Cor e Forma:White To Slightly Yellow Crystalline Powder
    Peso molecular:351.31
  • Isoxsuprine hydrochloride

    CAS:
    <p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>
    Fórmula:C18H24ClNO3
    Pureza:99.38%
    Cor e Forma:Crystals From Water Solid
    Peso molecular:337.84
  • Naftidrofuryl oxalate

    CAS:
    <p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>
    Fórmula:C26H35NO7
    Pureza:97.12% - 98.38%
    Cor e Forma:Solid
    Peso molecular:473.56
  • CGS 15943

    CAS:
    <p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>
    Fórmula:C13H8ClN5O
    Pureza:97.4%
    Cor e Forma:Solid
    Peso molecular:285.69
  • Astemizole

    CAS:
    <p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>
    Fórmula:C28H31FN4O
    Pureza:98.24% - 99.67%
    Cor e Forma:White Crystals Solid
    Peso molecular:458.57
  • Orphenadrine hydrochloride

    CAS:
    <p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>
    Fórmula:C18H23NO·HCl
    Pureza:99.88%
    Cor e Forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)
    Peso molecular:305.85
  • Cefaclor monohydrate

    CAS:
    <p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>
    Fórmula:C15H16ClN3O5S
    Pureza:97.36% - 99.9%
    Cor e Forma:White Crystaling Powder
    Peso molecular:385.82
  • Triflupromazine hydrochloride

    CAS:
    <p>Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.</p>
    Fórmula:C18H20ClF3N2S
    Pureza:99.76% - 99.82%
    Cor e Forma:Crystals
    Peso molecular:388.88
  • Alosetron hydrochloride

    CAS:
    <p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>
    Fórmula:C17H19ClN4O
    Pureza:99.90%
    Cor e Forma:Off-White Powder
    Peso molecular:330.81
  • Bromopride

    CAS:
    <p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>
    Fórmula:C14H22BrN3O2
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:344.25
  • 2-(1-Piperazinyl)pyrimidine

    CAS:
    <p>2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.</p>
    Fórmula:C8H12N4
    Pureza:98.46%
    Cor e Forma:Liquid - Crystal - Lump
    Peso molecular:164.21
  • Propafenone

    CAS:
    <p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>
    Fórmula:C21H27NO3
    Pureza:99.02%
    Cor e Forma:Solid
    Peso molecular:341.44
  • Cericlamine

    CAS:
    <p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>
    Fórmula:C12H17Cl2NO
    Pureza:99.38%
    Cor e Forma:Solid
    Peso molecular:262.18
  • Mebhydrolin napadisylate

    CAS:
    <p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>
    Fórmula:C19H20N2C10H8O6S2
    Pureza:99.35% - 99.96%
    Cor e Forma:White Or Almost White Crystalline
    Peso molecular:420.52
  • Flopropione

    CAS:
    <p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>
    Fórmula:C9H10O4
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:182.17
  • Atomoxetine hydrochloride

    CAS:
    <p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>
    Fórmula:C17H22ClNO
    Pureza:99.86%
    Cor e Forma:White Solid
    Peso molecular:291.82
  • RS102895 hydrochloride

    CAS:
    <p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>
    Fórmula:C21H22ClF3N2O2
    Pureza:98.95%
    Cor e Forma:Solid
    Peso molecular:426.86
  • Azasetron hydrochloride

    CAS:
    <p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>
    Fórmula:C17H20ClN3O3·HCl
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:386.27
  • Degarelix acetate(214766-78-6 free base)

    CAS:
    <p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>
    Fórmula:C84H107ClN18O18
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:1692.34
  • Pamabrom

    CAS:
    <p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>
    Fórmula:C11H18BrN5O3
    Pureza:99.84% - >99.99%
    Cor e Forma:Coa
    Peso molecular:348.2
  • DSP-4 hydrochloride

    CAS:
    <p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>
    Fórmula:C11H16BrCl2N
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:313.06
  • Mefexamide hydrochloride

    CAS:
    <p>Mefexamide hydrochloride is a central stimulant.</p>
    Fórmula:C15H25ClN2O3
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:316.83
  • Fezolinetant

    CAS:
    <p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>
    Fórmula:C16H15FN6OS
    Pureza:98.62% - 99.7%
    Cor e Forma:Solid
    Peso molecular:358.39
  • Mepyramine maleate

    CAS:
    <p>Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.</p>
    Fórmula:C21H27N3O5
    Pureza:99.51% - 99.7%
    Cor e Forma:White Crystalline Powder
    Peso molecular:401.47
  • Glycerol phenylbutyrate

    CAS:
    <p>Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).</p>
    Fórmula:C33H38O6
    Pureza:98.54% - 99.74%
    Cor e Forma:Solid
    Peso molecular:530.65
  • EMPA

    CAS:
    <p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>
    Fórmula:C23H26N4O4S
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:454.54
  • JNJ-39758979

    CAS:
    <p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>
    Fórmula:C11H19N5
    Pureza:98.33% - 99.62%
    Cor e Forma:Solid
    Peso molecular:221.3
  • Ogerin

    CAS:
    <p>Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).</p>
    Fórmula:C17H17N5O
    Pureza:99.5% - 99.75%
    Cor e Forma:Solid
    Peso molecular:307.35
  • Carbinoxamine Maleate Salt

    CAS:
    <p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>
    Fórmula:C20H23ClN2O5
    Pureza:99.97%
    Cor e Forma:Off-White Solid
    Peso molecular:406.86
  • Nicergoline

    CAS:
    <p>Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.</p>
    Fórmula:C24H26BrN3O3
    Pureza:98% - 99.80%
    Cor e Forma:Solid
    Peso molecular:484.39
  • DPTN dihydrochloride

    CAS:
    <p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>
    Fórmula:C22H20Cl2N4OS
    Pureza:99.95%
    Cor e Forma:Soild
    Peso molecular:459.39
  • Vabicaserin hydrochloride

    CAS:
    <p>Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).</p>
    Fórmula:C15H21ClN2
    Pureza:98.32%
    Cor e Forma:Solid
    Peso molecular:264.79
  • Isoprenaline hydrochloride

    CAS:
    <p>Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.</p>
    Fórmula:C11H18ClNO3
    Pureza:98% - 99.65%
    Cor e Forma:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
    Peso molecular:247.719
  • GANT 58

    CAS:
    <p>GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).</p>
    Fórmula:C24H16N4S
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:392.48
  • Terbutaline Sulfate

    CAS:
    Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
    Fórmula:C12H19NO3H2SO4
    Pureza:99.47% - 99.94%
    Cor e Forma:Crystalline Powder
    Peso molecular:274.32
  • Perphenazine

    CAS:
    <p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>
    Fórmula:C21H26ClN3OS
    Pureza:99.3% - 99.99%
    Cor e Forma:Solid
    Peso molecular:403.97
  • Anatibant 2HCl

    CAS:
    <p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>
    Fórmula:C34H36Cl2N6O5S·2ClH
    Pureza:99.17% - 99.58%
    Cor e Forma:Soild
    Peso molecular:784.58
  • Gevotroline

    CAS:
    <p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>
    Fórmula:C19H20FN3
    Pureza:98.65%
    Cor e Forma:Solid
    Peso molecular:309.38
  • Senktide acetate


    <p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>
    Fórmula:C42H59N7O13S
    Pureza:98.26%
    Cor e Forma:Solid
    Peso molecular:902.02
  • Terfenadine

    CAS:
    <p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>
    Fórmula:C32H41NO2
    Pureza:98.76% - 99.75%
    Cor e Forma:Solid
    Peso molecular:471.67
  • hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Fórmula:C31H23F4N3O
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:529.53
  • Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Fórmula:C19H27N5O4·HCl
    Pureza:99.78%
    Cor e Forma:White To Off-White Solid
    Peso molecular:425.91
  • Naluzotan hydrochloride

    CAS:
    <p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>
    Fórmula:C23H39ClN4O3S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:487.1
  • Proglumide

    CAS:
    <p>Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.</p>
    Fórmula:C18H26N2O4
    Pureza:99.4% - 99.45%
    Cor e Forma:White Crystalline Powder
    Peso molecular:334.41
  • TSHR antagonist S37

    CAS:
    <p>TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).</p>
    Fórmula:C25H20N2O3S2
    Pureza:98.35%
    Cor e Forma:Solid
    Peso molecular:460.57
  • Pemirolast potassium

    CAS:
    <p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>
    Fórmula:C10H7KN6O
    Pureza:98.91% - 99.63%
    Cor e Forma:Crystals From Dimethylformamide Crystalline Solid
    Peso molecular:266.31
  • Mifentidine

    CAS:
    <p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>
    Fórmula:C13H16N4
    Pureza:98.34% - 99.73%
    Cor e Forma:Solid
    Peso molecular:228.29
  • Oxeladin citrate

    CAS:
    <p>Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.</p>
    Fórmula:C26H41NO10
    Pureza:97.23%
    Cor e Forma:Solid
    Peso molecular:527.6
  • Salmeterol

    CAS:
    <p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>
    Fórmula:C25H37NO4
    Pureza:99.2% - 99.9%
    Cor e Forma:Solid
    Peso molecular:415.57
  • Carbetapentane citrate

    CAS:
    <p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>
    Fórmula:C20H31NO3·C6H8O7
    Pureza:99.46%
    Cor e Forma:White To Off-White Solid
    Peso molecular:525.59
  • (Rac)-MGV354

    CAS:
    <p>(Rac)-MGV354: a racemic sGC activator; EC50s &lt;0.5 nM (CHO cells), 5 nM (GTM-3 E cells).</p>
    Fórmula:C35H37N5O3
    Pureza:99.26%
    Cor e Forma:Solid
    Peso molecular:575.7
  • Phentolamine mesylate

    CAS:
    <p>Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.</p>
    Fórmula:C17H19N3O·CH4O3S
    Pureza:99.77% - >99.99%
    Cor e Forma:By The Metabolic Processes Of Bacillus Subtilis And Licheniformis
    Peso molecular:377.46
  • Cloroperone

    CAS:
    <p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>
    Fórmula:C22H23ClFNO2
    Pureza:98.40%
    Cor e Forma:Soild
    Peso molecular:387.88
  • Apelin-13

    CAS:
    <p>Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor</p>
    Fórmula:C69H111N23O16S
    Pureza:96.81%
    Cor e Forma:Solid
    Peso molecular:1550.83
  • Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Fórmula:C18H19N3O·HCl·2H2O
    Pureza:99.92%
    Cor e Forma:White Crystal Powder
    Peso molecular:365.86
  • Bambuterol hydrochloride

    CAS:
    <p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>
    Fórmula:C18H30ClN3O5
    Pureza:99.53% - 99.61%
    Cor e Forma:White Solid
    Peso molecular:403.91
  • (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid

    CAS:
    <p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>
    Fórmula:C20H29N3O8
    Pureza:99.72%
    Cor e Forma:Soild
    Peso molecular:439.46
  • Tropanserin

    CAS:
    <p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>
    Fórmula:C17H23NO2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:273.37
  • Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Fórmula:C19H31ClF3NO3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:413.9
  • Tetrahydrozoline

    CAS:
    <p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>
    Fórmula:C13H16N2
    Pureza:97.85% - 99.77%
    Cor e Forma:Solid
    Peso molecular:200.28
  • Metoclopramide hydrochloride

    CAS:
    <p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>
    Fórmula:C14H22ClN3O2·HCl
    Pureza:99.99%
    Cor e Forma:White To Off-White Powder
    Peso molecular:336.26
  • SEP-363856 hydrochloride

    CAS:
    <p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>
    Fórmula:C9H14ClNOS
    Pureza:99.86% - 99.99%
    Cor e Forma:Solid
    Peso molecular:219.73
  • JP1302 dihydrochloride

    CAS:
    <p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>
    Fórmula:C24H26Cl2N4
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:441.4
  • Pericyazine

    CAS:
    <p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>
    Fórmula:C21H23N3OS
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:365.49
  • Nepafenac

    CAS:
    <p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>
    Fórmula:C15H14N2O2
    Pureza:98.94% - 99.43%
    Cor e Forma:Solid
    Peso molecular:254.28
  • Latanoprostene bunod

    CAS:
    <p>LBN is a NO-donating prostaglandin analog for reducing IOP in glaucoma or OHT patients.</p>
    Fórmula:C27H41NO8
    Pureza:99.33% - 99.69%
    Cor e Forma:Solid
    Peso molecular:507.62
  • Fexofenadine hydrochloride

    CAS:
    <p>Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with</p>
    Fórmula:C32H40ClNO4
    Pureza:>99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:538.12
  • Dexpramipexole dihydrochloride

    CAS:
    <p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>
    Fórmula:C10H19Cl2N3S
    Pureza:99.75% - 99.88%
    Cor e Forma:Solid
    Peso molecular:284.25
  • Ifenprodil Tartrate

    CAS:
    <p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>
    Fórmula:C21H27NO2C4H6O6
    Pureza:99.02% - 99.55%
    Cor e Forma:Solid
    Peso molecular:400.49
  • Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Fórmula:C25H28N2O5S
    Pureza:97.09%
    Cor e Forma:Solid
    Peso molecular:468.57
  • Prochlorperazine Maleate

    CAS:
    <p>Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.</p>
    Fórmula:C28H32ClN3O8S
    Pureza:99.78%
    Cor e Forma:Off-White Powder
    Peso molecular:606.09
  • PF-610355 HCl


    <p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>
    Fórmula:C19H22ClN7O6
    Pureza:97.97%
    Cor e Forma:Solid
    Peso molecular:479.87
  • Luzindole

    CAS:
    <p>Luzindole (N-0774) is a selective melatonin receptor antagonist.</p>
    Fórmula:C19H20N2O
    Pureza:98.53%
    Cor e Forma:Off-White Amorphous Solid
    Peso molecular:292.37
  • Ziprasidone hydrochloride monohydrate

    CAS:
    <p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>
    Fórmula:C21H21ClN4OS·HCl·H2O
    Pureza:98% - 99.83%
    Cor e Forma:Off-White Powder
    Peso molecular:467.12
  • NEO 376

    CAS:
    <p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>
    Fórmula:C20H24ClN3O
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:357.88
  • Rimonabant hydrochloride

    CAS:
    <p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>
    Fórmula:C22H22Cl4N4O
    Pureza:98.24% - 99.5%
    Cor e Forma:Off-White To White Crystalline Powder
    Peso molecular:500.25
  • Citalopram hydrobromide

    CAS:
    <p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>
    Fórmula:C20H22BrFN2O
    Pureza:99.81%
    Cor e Forma:White Crystalline Powder
    Peso molecular:405.304
  • L-741626

    CAS:
    <p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>
    Fórmula:C20H21ClN2O
    Pureza:98.57%
    Cor e Forma:Solid
    Peso molecular:340.85
  • Ketanserin

    CAS:
    <p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>
    Fórmula:C22H22FN3O3
    Pureza:99.19% - 99.73%
    Cor e Forma:Solid
    Peso molecular:395.43
  • Indusatumab

    CAS:
    <p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>
    Pureza:> 95% - > 95%
    Cor e Forma:Liquid
    Peso molecular:145.18 kDa
  • Anamorelin

    CAS:
    <p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>
    Fórmula:C31H42N6O3
    Pureza:99.35% - 99.94%
    Cor e Forma:Solid
    Peso molecular:546.7
  • Tripelennamine hydrochloride

    CAS:
    <p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>
    Fórmula:C16H21N3·HCl
    Pureza:99.54% - 99.81%
    Cor e Forma:White Solid
    Peso molecular:291.82
  • PF-06882961

    CAS:
    <p>PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>
    Fórmula:C31H30FN5O4
    Pureza:98.06% - 99.54%
    Cor e Forma:Solid
    Peso molecular:555.6
  • 2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Fórmula:C11H9BrO
    Pureza:98.51%
    Cor e Forma:White To Off-White Powder
    Peso molecular:237.09
  • Cisapride

    CAS:
    <p>Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.</p>
    Fórmula:C23H29ClFN3O4
    Pureza:99.77%
    Cor e Forma:White To Slightly Biege Powder Solid
    Peso molecular:465.95
  • Protriptyline hydrochloride

    CAS:
    <p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>
    Fórmula:C19H21N·HCl
    Pureza:98.54% - 99.98%
    Cor e Forma:Solid
    Peso molecular:299.84
  • Urocortin (rat) acetate


    <p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>
    Pureza:97.76%
    Cor e Forma:Soild
  • Nylidrin hydrochloride

    CAS:
    <p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells &amp; human basophils.</p>
    Fórmula:C19H26ClNO2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:335.87
  • Terlipressin Acetate

    CAS:
    <p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>
    Fórmula:C56H82N16O19S2
    Pureza:98.50% - 99.69%
    Cor e Forma:Solid
    Peso molecular:1347.5
  • Sonepcizumab

    CAS:
    <p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>
    Pureza:SDS-PAGE:95% SEC-HPLC:98.90%
    Cor e Forma:Liquid
    Peso molecular:146.43 kDa
  • Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Fórmula:C22H29N3O4S
    Pureza:98.55%
    Cor e Forma:Yellowish White Crystalline Powder
    Peso molecular:431.55
  • Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Fórmula:C18H26ClN3O3
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:367.87
  • Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Fórmula:C17H28ClNO2
    Pureza:97.32% - 99.86%
    Cor e Forma:White Crystalline Powder
    Peso molecular:313.86
  • Erenumab

    CAS:
    <p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>
    Pureza:99.43% (SEC-HPLC) - > 95%
    Cor e Forma:Liquid
    Peso molecular:146.2 kDa
  • Talastine

    CAS:
    <p>Talastine is an antihistamine compound that can induce an allergic rash.</p>
    Fórmula:C19H21N3O
    Pureza:98.50% - 99.44%
    Cor e Forma:Solid
    Peso molecular:307.39
  • Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21
  • Desipramine hydrochloride

    CAS:
    <p>Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.</p>
    Fórmula:C18H23ClN2
    Pureza:99.58% - 99.94%
    Cor e Forma:White To Off-White Powder
    Peso molecular:302.842
  • Naftifine hydrochloride

    CAS:
    <p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>
    Fórmula:C21H22ClN
    Pureza:98.75% - 99.84%
    Cor e Forma:Solid
    Peso molecular:323.86
  • Fluoxetine hydrochloride

    CAS:
    <p>Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.</p>
    Fórmula:C17H19ClF3NO
    Pureza:99.6% - 99.98%
    Cor e Forma:White To Off-White Crystalline Solid White To Off-White Powder
    Peso molecular:345.787
  • Clonidine hydrochloride

    CAS:
    <p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>
    Fórmula:C9H10Cl3N3
    Pureza:99.16% - 99.86%
    Cor e Forma:Solid
    Peso molecular:266.55
  • Sergliflozin A

    CAS:
    <p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>
    Fórmula:C20H24O7
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:376.4
  • Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:463.79
  • Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Fórmula:C28H32N2O7
    Pureza:99.03% - 99.67%
    Cor e Forma:Solid
    Peso molecular:508.56
  • ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Fórmula:C20H25ClN4O2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:388.89
  • CD80-IN-3

    CAS:
    <p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>
    Fórmula:C17H10FN3O3
    Pureza:98.08%
    Cor e Forma:Solid
    Peso molecular:323.28
  • CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Fórmula:C24H17ClN2O3
    Pureza:98% - 99.08%
    Cor e Forma:Solid
    Peso molecular:416.86
  • Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Fórmula:C19H25F3N2O6
    Pureza:99.92% - 99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:434.41
  • Silodosin

    CAS:
    <p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>
    Fórmula:C25H32F3N3O4
    Pureza:99.282% - 99.76%
    Cor e Forma:Colorless To Pink Solid
    Peso molecular:495.53
  • Metaproterenol hemisulfate

    CAS:
    <p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>
    Fórmula:C11H17NO3·5H2O4S
    Pureza:98.53% - 99.74%
    Cor e Forma:Solid
    Peso molecular:260.3
  • Cyproheptadine hydrochloride sesquihydrate

    CAS:
    <p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>
    Fórmula:C21H24ClNO
    Pureza:99.77% - >99.99%
    Cor e Forma:White To Slightly Yellowish Crystalline Solid
    Peso molecular:341.88
  • Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3·HCl
    Pureza:99.58%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:423.94
  • Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:383.51
  • JNJ-18038683

    CAS:
    <p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>
    Fórmula:C26H28ClN3O7
    Pureza:97.29%
    Cor e Forma:Solid
    Peso molecular:529.97
  • PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Fórmula:C25H37Cl2N3O2
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:482.49
  • Acetophenazine dimaleate

    CAS:
    <p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>
    Fórmula:C31H37N3O10S
    Pureza:99.39% - 99.48%
    Cor e Forma:Solid
    Peso molecular:643.71
  • Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Fórmula:C24H28N2O3
    Pureza:99.60% - 99.97%
    Cor e Forma:White Crystalline Powder
    Peso molecular:392.49
  • Ifenprodil

    CAS:
    <p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 &amp; GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>
    Fórmula:C21H27NO2
    Pureza:99.58%
    Cor e Forma:White Crystalline Powder
    Peso molecular:325.44
  • Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Fórmula:C18H25ClN4O
    Pureza:99.88% - 99.93%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:348.87
  • Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H11ClFNO2
    Pureza:99.98%
    Cor e Forma:Soild
    Peso molecular:231.65
  • Blonanserin

    CAS:
    <p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>
    Fórmula:C23H30FN3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:367.5
  • Fosopamine(HCl)

    CAS:
    <p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>
    Fórmula:C9H15ClNO5P
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:283.65
  • NF-56-EJ40 hydrochloride

    CAS:
    <p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>
    Fórmula:C27H31Cl2N3O3
    Pureza:99.33%
    Cor e Forma:Soild
    Peso molecular:516.46
  • Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43
  • Fluoxetine

    CAS:
    <p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>
    Fórmula:C17H18F3NO
    Pureza:99.07% - 99.28%
    Cor e Forma:Solid
    Peso molecular:309.33
  • Astressin acetate


    <p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>
    Fórmula:C163H273N49O44
    Pureza:96.87%
    Cor e Forma:Solid
    Peso molecular:3623.21
  • Diphenylpyraline hydrochloride

    CAS:
    <p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>
    Fórmula:C19H23NO·HCl
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:317.85
  • Chlorprothixene hydrochloride

    CAS:
    <p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>
    Fórmula:C18H18ClNS·HCl
    Pureza:99.76%
    Cor e Forma:White Powder
    Peso molecular:352.32
  • Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>
    Fórmula:C28H30N2O8
    Pureza:99.7% - >99.99%
    Cor e Forma:Powder
    Peso molecular:522.55
  • Olanzapine

    CAS:
    <p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>
    Fórmula:C17H20N4S
    Pureza:99.86% - ≥95%
    Cor e Forma:Yellowish Crystalline Powder
    Peso molecular:312.43
  • CP-809101 hydrochloride

    CAS:
    <p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>
    Fórmula:C15H18Cl2N4O
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:341.24
  • Trazodone hydrochloride

    CAS:
    <p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>
    Fórmula:C19H23Cl2N5O
    Pureza:99.5% - 99.52%
    Cor e Forma:Solid
    Peso molecular:408.33
  • MK-0249 FA


    <p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>
    Fórmula:C24H26F3N3O4
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:477.48
  • Antazoline hydrochloride

    CAS:
    <p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>
    Fórmula:C17H19N3·HCl
    Pureza:98% - 99.53%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:301.82
  • Brefonalol HCl


    <p>Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.</p>
    Fórmula:C22H29ClN2O2
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:388.93
  • Aripiprazole

    CAS:
    <p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>
    Fórmula:C23H27Cl2N3O2
    Pureza:99.43% - 99.62%
    Cor e Forma:Colourless Flake Crystalline Solid
    Peso molecular:448.39
  • YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Fórmula:C33H37N5O5S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:615.74
  • Alverine citrate

    CAS:
    <p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>
    Fórmula:C26H35NO7
    Pureza:98.53% - 99.43%
    Cor e Forma:Coa
    Peso molecular:473.57
  • KGA-2727

    CAS:
    <p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>
    Fórmula:C26H40N4O8
    Pureza:98.46%
    Cor e Forma:Solid
    Peso molecular:536.62
  • (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H10FNO2
    Pureza:97.82%
    Cor e Forma:Soild
    Peso molecular:195.19
  • Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Fórmula:C14H15Cl2NS
    Pureza:99.85% - >99.99%
    Cor e Forma:White Powder
    Peso molecular:300.25
  • Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Fórmula:C16H21N3O2
    Pureza:99.69% - 99.91%
    Cor e Forma:White Or Kind Of White Powder
    Peso molecular:287.36
  • Timonacic

    CAS:
    <p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>
    Fórmula:C4H7NO2S
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:133.17
  • AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Fórmula:C17H14O5
    Pureza:97.59%
    Cor e Forma:Solid
    Peso molecular:298.29
  • Phenothiazine

    CAS:
    <p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>
    Fórmula:C12H9NS
    Pureza:99.95%
    Cor e Forma:Yellow Solid Pellets
    Peso molecular:199.27
  • Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Fórmula:C12H19NO10
    Pureza:99.53% - >99.99%
    Cor e Forma:Solid
    Peso molecular:337.28
  • ESI-05

    CAS:
    <p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>
    Fórmula:C16H18O2S
    Pureza:97.22%
    Cor e Forma:Solid
    Peso molecular:274.38
  • AB928

    CAS:
    <p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>
    Fórmula:C23H22N8O
    Pureza:98.09% - >99.99%
    Cor e Forma:Solid
    Peso molecular:426.47
  • Asenapine Maleate

    CAS:
    <p>Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.</p>
    Fórmula:C21H20ClNO5
    Pureza:99.28%
    Cor e Forma:Solid
    Peso molecular:401.84
  • DREADD agonist 21

    CAS:
    <p>DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).</p>
    Fórmula:C17H18N4
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:278.35
  • LCKLSL hydrochloride


    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Fórmula:C30H58ClN7O8S
    Pureza:98.02% - 99.31%
    Cor e Forma:Solid
    Peso molecular:712.34
  • (R)-Elagolix

    CAS:
    <p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>
    Fórmula:C32H30F5N3O5
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:631.59
  • Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Fórmula:C31H38N2O
    Pureza:97.49%
    Cor e Forma:Solid
    Peso molecular:454.65
  • Hydroxyzine Pamoate

    CAS:
    <p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>
    Fórmula:C44H43ClN2O8
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:763.27
  • Leronlimab

    CAS:
    <p>Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.</p>
    Pureza:SDS-PAGE:95.0%;SEC-HPLC:99.6%
    Cor e Forma:Liquid
    Peso molecular:146.66 kDa
  • Filorexant

    CAS:
    <p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki &lt;3 nM).</p>
    Fórmula:C24H25FN4O2
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:420.48
  • Levodropropizine

    CAS:
    <p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>
    Fórmula:C13H20N2O2
    Pureza:99.87% - 99.93%
    Cor e Forma:White Or Off White Crystalline Powder
    Peso molecular:236.31
  • Palonosetron hydrochloride

    CAS:
    <p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>
    Fórmula:C19H24N2O·HCl
    Pureza:99.84% - 99.92%
    Cor e Forma:White Solid
    Peso molecular:332.87
  • Ro 10-5824 dihydrochloride

    CAS:
    <p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:353.29
  • Moxisylyte hydrochloride

    CAS:
    <p>Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.</p>
    Fórmula:C16H26ClNO3
    Pureza:99.93% - ≥95%
    Cor e Forma:Solid
    Peso molecular:315.84
  • Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Fórmula:C21H22CL2N4OS
    Pureza:97.97% - 99.82%
    Cor e Forma:Solid
    Peso molecular:449.4
  • Vilazodone

    CAS:
    <p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>
    Fórmula:C26H27N5O2
    Pureza:99.61%
    Cor e Forma:Light Yellow Solid
    Peso molecular:441.52
  • Dopexamine hydrochloride

    CAS:
    <p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>
    Fórmula:C22H34Cl2N2O2
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:429.42
  • Dimenhydrinate

    CAS:
    <p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>
    Fórmula:C24H28ClN5O3
    Pureza:99.57% - 99.77%
    Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Peso molecular:469.96
  • Adrenalone hydrochloride

    CAS:
    <p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>
    Fórmula:C9H11NO3·HCl
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:217.65
  • Carvedilol EP IMpurity E

    CAS:
    <p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>
    Fórmula:C9H14ClNO2
    Pureza:99.53%
    Cor e Forma:White To Almost White Solid Crystalline
    Peso molecular:203.666
  • Promazine hydrochloride

    CAS:
    <p>Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.</p>
    Fórmula:C17H21ClN2S
    Pureza:99.90%
    Cor e Forma:Solid
    Peso molecular:320.88
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Fórmula:C18H29ClN2O4
    Pureza:99.92% - >99.99%
    Cor e Forma:White Or Slightly Off-White Crystalline Powder Solid
    Peso molecular:372.89
  • Pizotifen

    CAS:
    <p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>
    Fórmula:C19H21NS
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:295.44
  • Linaclotide

    CAS:
    <p>Linaclotide treats IBS-C &amp; chronic constipation; it's a selective guanylate cyclase C agonist.</p>
    Fórmula:C59H79N15O21S6
    Pureza:97.93% - 98.71%
    Cor e Forma:Solid
    Peso molecular:1526.74
  • MP-A08

    CAS:
    <p>MP-A08 selectively inhibits SPHK1; targets SphK1 &amp; SphK2 with Ki of 6.9 μM &amp; 27 μM, respectively.</p>
    Fórmula:C27H25N3O4S2
    Pureza:97.44%
    Cor e Forma:Solid
    Peso molecular:519.64
  • Fenspiride hydrochloride

    CAS:
    <p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>
    Fórmula:C15H20N2O2·HCl
    Pureza:99.64% - 99.92%
    Cor e Forma:Solid
    Peso molecular:296.79
  • Desvenlafaxine

    CAS:
    <p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>
    Fórmula:C16H25NO2
    Pureza:99.46% - 99.81%
    Cor e Forma:White Crystalline Powder
    Peso molecular:263.38
  • Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Fórmula:C21H27Cl3N2O3
    Pureza:99.4% - 99.97%
    Cor e Forma:Solid
    Peso molecular:461.81
  • Olinciguat

    CAS:
    <p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>
    Fórmula:C21H16F5N7O3
    Pureza:99.33% - 99.71%
    Cor e Forma:Solid
    Peso molecular:509.39
  • Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Fórmula:C19H29ClN2O4
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:384.9
  • Tolnaftate

    CAS:
    <p>Tolnaftate (NP-27) is a synthetic antifungal agent.</p>
    Fórmula:C19H17NOS
    Pureza:98.85%
    Cor e Forma:White Powder
    Peso molecular:307.41