
Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 358 produtos de "Receptor de Histamina"
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Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Fórmula:C19H23NOCor e Forma:SolidPeso molecular:281.39Cetirizine D8
CAS:<p>Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:396.94Cetirizine D4
CAS:<p>Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:392.91Acrivastine D7
CAS:<p>Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.</p>Fórmula:C22H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:355.48Doxepin D3 Hydrochloride
CAS:<p>Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and</p>Fórmula:C19H22ClNOPureza:98%Cor e Forma:SolidPeso molecular:318.86Fexofenadine-d6
CAS:<p>Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.</p>Fórmula:C32H39NO4Pureza:98%Cor e Forma:SolidPeso molecular:507.69Emedastine Difumarate
CAS:<p>Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.</p>Fórmula:C25H34N4O9Cor e Forma:SolidPeso molecular:534.56Gizzerosine
CAS:<p>Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.</p>Fórmula:C11H20N4O2Cor e Forma:SolidPeso molecular:240.3Emedastine
CAS:<p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>Fórmula:C17H26N4OPureza:97.1% - 97.76%Cor e Forma:OilPeso molecular:302.41Fexofenadine hydrochloride
CAS:<p>Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,</p>Fórmula:C32H39NO4·HClPureza:99.39% - ≥95%Cor e Forma:SolidPeso molecular:538.13Chlorpheniramine
CAS:<p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>Fórmula:C16H19ClN2Cor e Forma:SolidPeso molecular:274.79Hydroxyzine
CAS:<p>Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.</p>Fórmula:C21H27ClN2O2Pureza:99.54% - ≥95%Cor e Forma:Oil SolidPeso molecular:374.9VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Fórmula:C15H19N5Pureza:99.44% - 99.57%Cor e Forma:SolidPeso molecular:269.34SCH-37370
CAS:<p>SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.</p>Fórmula:C21H21ClN2OPureza:99.07%Cor e Forma:SolidPeso molecular:352.86H4 Receptor antagonist 1
CAS:<p>H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.</p>Fórmula:C16H17ClN4OPureza:98.81%Cor e Forma:SolidPeso molecular:316.79Metiamide
CAS:<p>Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .</p>Fórmula:C9H16N4S2Pureza:97.41%Cor e Forma:SolidPeso molecular:244.38Dimaprit dihydrochloride
CAS:<p>Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.</p>Fórmula:C6H15N3S·2HClPureza:99.79%Cor e Forma:SolidPeso molecular:234.19Conessine
CAS:<p>Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.</p>Fórmula:C24H40N2Pureza:99.65%Cor e Forma:SolidPeso molecular:356.59Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Fórmula:C28H37N3O3Pureza:99.86% - >99.99%Cor e Forma:SolidPeso molecular:463.61JNJ-7777120
CAS:<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Fórmula:C14H16ClN3OPureza:99.83% - 99.96%Cor e Forma:SolidPeso molecular:277.75
