
Antibiótico
Os inibidores de antibióticos são substâncias que interferem na atividade dos antibióticos, frequentemente utilizados para estudar os mecanismos de resistência a antibióticos ou para aumentar a eficácia dos antibióticos existentes. Esses inibidores desempenham um papel crítico na compreensão de como as bactérias evitam o tratamento com antibióticos e no desenvolvimento de estratégias para superar a resistência. Na CymitQuimica, oferecemos uma variedade de inibidores de antibióticos para apoiar sua pesquisa em resistência antimicrobiana, farmacologia e inovação terapêutica.
Foram encontrados 919 produtos de "Antibiótico"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Gatifloxacin hydrochloride
CAS:<p>Gatifloxacin hydrochloride, a fourth-gen fluoroquinolone antibiotic, blocks bacterial DNA rotase and topoisomerase IV.</p>Fórmula:C19H23ClFN3O4Pureza:99.85% - 99.89%Cor e Forma:SolidPeso molecular:411.86Avibactam sodium
CAS:<p>Avibactam sodium (NXL-104) is a β-lactamase inhibitor that inhibits TEM-1, P99, and KPC-2. Avibactam sodium has antimicrobial activity. Cost-effective and quality-assured.</p>Fórmula:C7H10N3NaO6SPureza:99.16% - >99.99%Cor e Forma:SolidPeso molecular:287.22Bedaquiline
CAS:<p>Bedaquiline, an anti-TB drug, blocks mycobacterial ATP synthesis, effective against all Mycobacterium tuberculosis states.</p>Fórmula:C32H31BrN2O2Pureza:98% - 99.8%Cor e Forma:SolidPeso molecular:555.5Doripenem
CAS:<p>Doripenem is a new parenteral carbapenem antibiotic with broad-spectrum activity against gram-negative and gram-positive pathogens.</p>Fórmula:C15H24N4O6S2Pureza:99.65% - 99.79%Cor e Forma:White To Off-White PowderPeso molecular:420.5Sulfamethoxazole sodium
CAS:<p>Sulfamethoxazole sodium (Ro 4-2130 sodium) is a sulfonamide bacteriostatic antibiotic</p>Fórmula:C10H10N3NaO3SPureza:99.13% - 99.43%Cor e Forma:SolidPeso molecular:275.26Ertapenem sodium
CAS:<p>Ertapenem sodium (MK-826) is a long-acting carbapenem antibiotic effective against a wide range of bacteria, including ESBL producers.</p>Fórmula:C22H24N3O7S·NaPureza:96.05% - 99.92%Cor e Forma:White Or Off-White PowderPeso molecular:497.5Tosufloxacin tosylate hydrate
CAS:<p>Tosufloxacin tosylate hydrate (A-61827 tosylate hydrate) is a fluoroquinolone antibacterial agent that is used to treat susceptible infections.</p>Fórmula:C26H25F3N4O7SPureza:99.21% - 99.25%Cor e Forma:SolidPeso molecular:594.60Luliconazole
CAS:<p>Luliconazole (NND 502) is an Azole Antifungal. The mechanism of action of luliconazole is as a Cytochrome P450 2C19 Inhibitor.</p>Fórmula:C14H9Cl2N3S2Pureza:98.27% - 99.83%Cor e Forma:SolidPeso molecular:354.28Sulfisomidin
CAS:<p>Sulfisomidin (Sulfaisodimidine) (Sulfaisodimidine) is a short-acting antibacterial agent.</p>Fórmula:C12H14N4O2SPureza:95% - 99.95%Cor e Forma:SolidPeso molecular:278.33Emodinanthrone
CAS:<p>Emodinanthrone is a natural product belongs to the class of organic compounds known as anthracenes.</p>Fórmula:C15H12O4Pureza:95% - 99.1%Cor e Forma:SolidPeso molecular:256.25Pretomanid
CAS:<p>Pretomanid ((S)-PA 824) , a nitroimidazole, is used as an anti-tuberculosis drug for tuberculosis with MIC less than 2.8 μM.</p>Fórmula:C14H12F3N3O5Pureza:98.75% - 99.96%Cor e Forma:SolidPeso molecular:359.26Aprepitant
CAS:<p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>Fórmula:C23H21F7N4O3Pureza:98% - 99.68%Cor e Forma:Off-White To Light Yellow Cyrstalline SolidPeso molecular:534.43Tacrolimus monohydrate
CAS:<p>Tacrolimus monohydrate (LCP-Tacro) is a macrolide from the culture broth of a strain of Streptomyces tsukubaensis, binds to FKBP to form a complex.</p>Fórmula:C44H71NO13Pureza:97.07% - 98.05%Cor e Forma:SolidPeso molecular:822.05Ceftaroline fosamil
CAS:<p>Ceftaroline fosamil (TAK-599) is a cephalosporin, with activity against Gram-positive pathogens.</p>Fórmula:C24H25N8O10PS4Pureza:97.09% - ≥98%Cor e Forma:SolidPeso molecular:744.74Micafungin sodium
CAS:<p>Micafungin sodium (FK 463) is the sodium salt form of micafungin, a semi-synthetic echinocandin derived from a natural product of the fungus Coleophoma empetri</p>Fórmula:C56H70N9NaO23SPureza:98% - 99.41%Cor e Forma:SolidPeso molecular:1292.26Sitafloxacin Hydrate
CAS:<p>Sitafloxacin Hydrate (DU-6859a) is a fluoroquinolone antibiotic that shows promise in the treatment of Buruli ulcer.</p>Fórmula:C19H18ClF2N3O3H2OPureza:99.73% - 99.77%Cor e Forma:SolidPeso molecular:436.84Isavuconazole
CAS:<p>Isavuconazole (RO-0094815) is an azole antifungal with MICs 0.002-0.5 mg/liter against C. albicans to C. glabrata.</p>Fórmula:C22H17F2N5OSPureza:99.74% - >99.99%Cor e Forma:SolidPeso molecular:437.47Clindamycin hydrochloride
CAS:<p>Clindamycin hydrochloride (Clinimycin HCl) inhibits protein synthesis by acting on the 50S ribosomal. Clindamycin is a chlorinated broad-spectrum antibiotic.</p>Fórmula:C18H33ClN2O5S·HClPureza:99.80%Cor e Forma:White Crystalline PowderPeso molecular:461.44Amoxicillin Sodium
CAS:<p>Amoxicillin Sodium (Clavulanate) is a moderate- spectrum, bacteriolytic, β-lactam antibiotic.</p>Fórmula:C16H18N3O5S·NaPureza:98.45% - 99.2%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:387.39Puromycin aminonucleoside
CAS:<p>Puromycin aminonucleoside (NSC-3056) increases podocyte permeability by modulating ZO-1 in an oxidative stress-dependent manner.</p>Fórmula:C12H18N6O3Pureza:99.85% - 99.9%Cor e Forma:SolidPeso molecular:294.31Tylvalosin tartrate
CAS:<p>Tylvalosin tartrate (Acetylisovaleryltylosin Tartrate) is a macrolide antibiotic that can against Gram-positive bacteria.</p>Fórmula:C57H93NO25Pureza:99.25%Cor e Forma:SolidPeso molecular:1192.34ML318
CAS:<p>ML318, a biaryl nitrile, inhibits PvdQ acylase (IC50=20nM) and P. aeruginosa growth (IC50=19µM), blocking pyoverdine production under low iron.</p>Fórmula:C14H8F4N2Pureza:98.93%Cor e Forma:SolidPeso molecular:280.22Epothilone B
CAS:<p>Epothilone B (EPO 906) is a compound isolated from the myxobacterium Sorangium cellulosum.</p>Fórmula:C27H41NO6SPureza:99.79% - 99.84%Cor e Forma:White PowderPeso molecular:507.68Benznidazol
CAS:<p>Benznidazol (Benznidazole)e has an antiprotozoal activity by interfering with parasite protein biosynthesis, influencing cytokines production and stimulating</p>Fórmula:C12H12N4O3Pureza:99.53% - >99.99%Cor e Forma:SolidPeso molecular:260.25Gastric mucin
CAS:Gastric mucin, a large glycoprotein, protects the gut from acid, enzymes, microbes, and physical damage.Pureza:98%Cor e Forma:SolidOmadacycline
CAS:<p>Omadacycline (Amadacycline), a new tetracycline antibiotic, can inhibit the 30s subunit of bacterial ribosome.</p>Fórmula:C29H40N4O7Pureza:98.33% - 99.76%Cor e Forma:SolidPeso molecular:556.65Sulfacetamide
CAS:<p>Sulfacetamide treats blepharitis, conjunctivitis, mild hidradenitis suppurativa, and acne by inhibiting bacterial folic acid.</p>Fórmula:C8H10N2O3SPureza:99.87%Cor e Forma:White To Yellowish Crystalline PowderPeso molecular:214.24Tebipenem Pivoxil
CAS:<p>Tebipenem Pivoxil (Orapenem) , an orally activity carbapenem antibiotic, is utilized in treating otolaryngologic and respiratory infections.</p>Fórmula:C22H31N3O6S2Pureza:97.96%Cor e Forma:SolidPeso molecular:497.63Quinocetone
CAS:<p>Quinocetone is an animal growth promoter and potential anti-tumor activity.</p>Fórmula:C18H14N2O3Pureza:98.06%Cor e Forma:SolidPeso molecular:306.32Wortmannin
CAS:<p>Wortmannin (SL-2052) is a PI3K inhibitor (IC50=3 nM) that is covalent and irreversible.</p>Fórmula:C23H24O8Pureza:95.84% - 99.76%Cor e Forma:White SolidPeso molecular:428.43Corylin
CAS:<p>Corylin is a major bioactive compound isolated from Psoralea corylifolia L; it has the activity of antibiotic or anticancer.</p>Fórmula:C20H16O4Pureza:98.44% - >99.99%Cor e Forma:SolidPeso molecular:320.34Benzyl isothiocyanate
CAS:<p>BITC, found in cruciferous veggies, exhibits anticancer, antimicrobial, and immunomodulatory effects.</p>Fórmula:C8H7NSPureza:99.25% - 99.83%Cor e Forma:Clear Yellow LiquidPeso molecular:149.21Tedizolid Phosphate
CAS:<p>Tedizolid Phosphate (TR-701FA) is an oxazolidinone-class antibiotic. Tedizolid phosphate is a phosphate ester prodrug of the active compound tedizolid.</p>Fórmula:C17H16FN6O6PPureza:97.96%Cor e Forma:SolidPeso molecular:450.32Chloramphenicol succinate sodium
CAS:<p>Chloramphenicol succinate sodium is broad-spectrum antibiotic with antibacterial activity.</p>Fórmula:C15H15Cl2N2NaO8Pureza:95.58%Cor e Forma:White PowderPeso molecular:445.2Tildipirosin
CAS:<p>Tildipirosin, a veterinary antibiotic, is a 16-membered macrolide that blocks bacterial protein synthesis and biofilm formation.</p>Fórmula:C41H71N3O8Pureza:98.47%Cor e Forma:SolidPeso molecular:734.02Geldanamycin
CAS:<p>Geldanamycin, an HSP90 inhibitor (Kd: 1.2 μM), specifically disrupts glucocorticoid receptor (GR)/HSP association.</p>Fórmula:C29H40N2O9Pureza:97.59% - 99.27%Cor e Forma:Yellow To Orange PowderPeso molecular:560.64Sulfadiazine sodium
CAS:<p>Sulfadiazine sodium (Sulfadiazin-natrium) is a sodium salt form of sulfadiazine, an intermediate-acting bacteriostatic, synthetic sulfanilamide derivative.</p>Fórmula:C10H10N4O2S·NaPureza:99.75%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:272.26Ceftiofur
CAS:<p>Ceftiofur is a semisynthetic antibiotic, with activity against various gram-positive/negative, anaerobic and aerobic bacteria encountered by domestic animals.</p>Fórmula:C19H17N5O7S3Pureza:98.26%Cor e Forma:SolidPeso molecular:523.56Danofloxacin
CAS:<p>Danofloxacin (Danofloxacin free base) is a fluoroquinolone antibiotic used in veterinary medicine.</p>Fórmula:C19H20FN3O3Pureza:99.77% - 99.8%Cor e Forma:SolidPeso molecular:357.38Dihydrostreptomycin sulfate
CAS:<p>Dihydrostreptomycin sulfate (Dihydrostreptomycin sesquisulfate) inhibits protein synthesis by binding to the 30S ribosomal subunit.</p>Fórmula:C21H41N7O12·5H2SO4Pureza:97.38% - 99.9%Cor e Forma:SolidPeso molecular:730.71Cecropin A
CAS:<p>Cecropin A, a linear 37-residue antimicrobial polypeptide produced by the cecropia moth, has exhibited cytotoxicity in various human cancer cell lines and</p>Fórmula:C184H313N53O46Pureza:96.78%Cor e Forma:SolidPeso molecular:4003.78Cephalosporin C zinc salt
CAS:<p>Cephalosporin C zinc salt was a potent inhibitor of SAMHD1 (IC50 : 1.1 ± 0.1 μM), and this inhibition was largely attributable to the presence of zinc.</p>Fórmula:C16H19N3O8SZnPureza:99.14%Cor e Forma:SolidPeso molecular:478.78(6R,7S)-Cefminox sodium heptahydrate
CAS:<p>(6R,7S)-Cefminox sodium heptahydrate (Meicelin) is a broad-spectrum, bactericidal cephalosporin antibiotic.</p>Fórmula:C16H34N7NaO14S3Pureza:99.65%Cor e Forma:SolidPeso molecular:667.65Maduramicin ammonium
CAS:<p>Maduramicin ammonium (Maduramycin Ammonium) is an anticoccidial agent for the the treatment of Eimeria spp., E.</p>Fórmula:C47H83NO17Pureza:99.83%Cor e Forma:White Crystalline PowderPeso molecular:934.20Mezlocillin Sodium
CAS:<p>Mezlocillin Sodium (Baycipen) is a penicillin beta-lactam antibiotic used in the treatment of bacterial infections caused by susceptible, usually gram-positive</p>Fórmula:C21H25N5O8S2·NaPureza:99.44%Cor e Forma:SolidPeso molecular:561.56Gamithromycin
CAS:<p>Gamithromycin (ML-1709460) is a macrolide compound with antibacterial activity.</p>Fórmula:C40H76N2O12Pureza:99.38%Cor e Forma:SolidPeso molecular:777.04Dalfopristin
CAS:<p>Dalfopristin (RP54476), a semi-synthetic streptogramin, treats multi-resistant Enterococcus faecium.</p>Fórmula:C34H50N4O9SPureza:98.07%Cor e Forma:SolidPeso molecular:690.85Cefquinome sulfate
CAS:<p>Cefquinome Sulfate is a semisynthetic, broad-spectrum, fourth-generation aminothiazolyl cephalosporin with antibacterial activity.</p>Fórmula:C23H26N6O9S3Pureza:97.83%Cor e Forma:White Or Almost White PowderPeso molecular:626.67Oxytetracycline Dihydrate
CAS:<p>Oxytetracycline Dihydrate (Terramycin Dihydrate) is a prescription antibiotic, interfering with the ability of bacteria to produce essential proteins.</p>Fórmula:C22H24N2O9·2H2OPureza:99.80%Cor e Forma:CrystallinePeso molecular:496.46Oxiconazole
CAS:<p>Oxiconazole is a broad-spectrum imidazole antifungal, inhibiting ergosterol biosynthesi by disrupting cytochrome P450 enzymes (lanosterol 14- α demethylase).</p>Fórmula:C18H13Cl4N3OPureza:99.99%Cor e Forma:SolidPeso molecular:429.13
