CAS 2768029-03-2

TRPM5 agonist-1

CAS: 2768029-03-2

TRPM5 agonist-1 is an orally active TRPM5 agonist with a pEC50 value of 8.1. It displays excellent selectivity for related cation channels (TRPM8, TRPV1, TRPV4, TRPA1, TRPM4) with selectivity greater than 100-fold. TRPM5 agonist-1 induces local stimulation of gastrointestinal transit in mice and is useful for studying the promotion of gastric motility.

Formel: C₁₁H₇Cl₂N₃S₂

Molekulargewicht: 316.22

Ref: TM-T213675