CAS 896584-55-7

Formel: C16H14N2O5

InChl: InChI=1S/C16H14N2O5/c19-16(18-11-2-4-13-15(8-11)23-9-22-13)17-10-1-3-12-14(7-10)21-6-5-20-12/h1-4,7-8H,5-6,9H2,(H2,17,18,19)

InChI Key: XEOBUSLELWJDNO-UHFFFAOYSA-N

SMILES: C1COC2=C(O1)C=CC(=C2)NC(=O)NC3=CC4=C(C=C3)OCO4

TRPV1 antagonist 10

CAS: 896584-55-7

TRPV1 antagonist 10 is a potent, orally active TRPV1 antagonist with an IC50 of 33.06 nM and serves as a moderate to weak inhibitor of URAT1 (IC50 = 22.51 μM) and GLUT9 (inhibition of 60.25% at 50 μM). It exhibits analgesic and urate-lowering properties and is applicable for research in hyperuricemia and inflammatory pain.

Formel: C₁₆H₁₄N₂O₅

Farbe und Form: Solid

Molekulargewicht: 314.293

Ref: TM-T207037