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EGFR
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PF-6274484
CAS:1035638-91-5
PF-6274484, a high affinity, irreversible covalent inhibitor of EGFR kinase with Ki of 0.14 nM, …
Formel:
C18H14ClFN4O2
Reinheit:
99.12%
Farbe und Form:
Solid
Molekulargewicht:
372.78
Ref: TM-T22396
2mg | 40,00 € | ||
5mg | 60,00 € | ||
10mg | 90,00 € | ||
25mg | 184,00 € | ||
50mg | 343,00 € | ||
100mg | 510,00 € | ||
500mg | 1.112,00 € | ||
1ml*10 (DMSO) | 66,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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CP-724714
CAS:383432-38-0
CP-724714 (CP724714) is an effective and selective HER2/ErbB2 inhibitor (IC50: 10 nM), >640-fold selectivity against …
Formel:
C27H27N5O3
Reinheit:
99.1%
Farbe und Form:
Solid
Molekulargewicht:
469.54
Ref: TM-T4014
1mg | 43,00 € | ||
2mg | 57,00 € | ||
5mg | 94,00 € | ||
10mg | 153,00 € | ||
25mg | 267,00 € | ||
50mg | 445,00 € | ||
100mg | 646,00 € | ||
1ml*10 (DMSO) | 88,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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AZD8931 diFuMaric acid
CAS:1196531-39-1
AZD8931 is a reversible and ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 (IC50 of …
Formel:
C31H33ClFN5O11
Reinheit:
99%
Farbe und Form:
Solid
Molekulargewicht:
706.1
Ref: TM-T8751
1mg | 128,00 € | ||
5mg | 282,00 € | ||
10mg | 421,00 € | ||
25mg | 694,00 € | ||
50mg | 975,00 € | ||
100mg | 1.319,00 € | ||
1ml*10 (DMSO) | 418,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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SYR127063
CAS:871026-18-5
SYR127063 (BDBM-92454) (BDBM92454) is a potent and selective HER2 inhibitor, binds to HER2 in a …
Formel:
C23H20ClF3N4O3
Reinheit:
98.57%
Farbe und Form:
Solid
Molekulargewicht:
492.88
Ref: TM-T34760
1mg | 128,00 € | ||
5mg | 281,00 € | ||
10mg | 423,00 € | ||
25mg | 694,00 € | ||
50mg | 978,00 € | ||
1ml*10 (DMSO) | 348,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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AG490
CAS:133550-30-8
AG490 (Tyrphostin B42) is an inhibitor of EGFR (IC50: 0.1 μM). It is 135-fold more …
Formel:
C17H14N2O3
Reinheit:
99.7%
Farbe und Form:
Yellow Solid
Molekulargewicht:
294.3
Ref: TM-T2600
10mg | 55,00 € | ||
25mg | 74,00 € | ||
50mg | 90,00 € | ||
100mg | 100,00 € | ||
200mg | 162,00 € | ||
500mg | 278,00 € | ||
1ml*10 (DMSO) | 57,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Chrysophanol
CAS:481-74-3
Chrysophanol (Turkey Rhubarb) is an EGFR/mTOR pathway inhibitor, which can be found in rhubarb, and …
Formel:
C15H10O4
Reinheit:
99.7%
Farbe und Form:
Physical Description Golden Yellow Plates Or Brown Powder Melting Point 196°C
Molekulargewicht:
254.24
Ref: TM-T2995
50mg | 43,00 € | ||
100mg | 57,00 € | ||
1ml*10 (DMSO) | 59,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Canertinib dihydrochloride
CAS:289499-45-2
Canertinib dihydrochloride (PD-183805 dihydrochloride) is the hydrochloride salt of an orally bio-available quinazoline with potential …
Formel:
C24H27Cl3FN5O3
Reinheit:
99.23%
Farbe und Form:
Solid
Molekulargewicht:
558.86
Ref: TM-T2501
5mg | 38,00 € | ||
10mg | 52,00 € | ||
50mg | 74,00 € | ||
1ml*10 (DMSO) | 51,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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SU5214
CAS:186611-04-1
SU5214 is a modulator of tyrosine kinase signal transduction.
Formel:
C16H13NO2
Reinheit:
99.55%
Farbe und Form:
Solid
Molekulargewicht:
251.28
Ref: TM-T3569
5mg | 60,00 € | ||
10mg | 90,00 € | ||
25mg | 177,00 € | ||
50mg | 276,00 € | ||
100mg | 454,00 € | ||
1ml*10 (DMSO) | 66,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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ZM39923 hydrochloride
CAS:1021868-92-7
ZM39923 hydrochloride (JAK3 Inhibitor IV) is an JAK1/3 inhibitor with pIC50 of 4.4/7.1, almost no …
Formel:
C23H25NO·HCl
Reinheit:
98.05%
Farbe und Form:
Solid
Molekulargewicht:
367.91
Ref: TM-T6145
5mg | 58,00 € | ||
10mg | 93,00 € | ||
25mg | 168,00 € | ||
50mg | 304,00 € | ||
100mg | 455,00 € | ||
1ml*10 (DMSO) | 94,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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WZ8040
CAS:1214265-57-2
WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).
Formel:
C24H25ClN6OS
Reinheit:
98%
Farbe und Form:
Solid
Molekulargewicht:
481.01
Ref: TM-T6734
1mg | 47,00 € | ||
5mg | 92,00 € | ||
10mg | 147,00 € | ||
25mg | 241,00 € | ||
50mg | 358,00 € | ||
100mg | 527,00 € | ||
1ml*10 (DMSO) | 94,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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FIIN-3
CAS:1637735-84-2
FIIN-3 is an irreversible inhibitor of FGFR.
Formel:
C34H36Cl2N8O4
Reinheit:
97.7%
Farbe und Form:
Solid
Molekulargewicht:
691.61
Ref: TM-T3466
1mg | 60,00 € | ||
2mg | 82,00 € | ||
5mg | 118,00 € | ||
10mg | 185,00 € | ||
25mg | 412,00 € | ||
50mg | 612,00 € | ||
100mg | 867,00 € | ||
1ml*10 (DMSO) | 175,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Vandetanib
CAS:443913-73-3
Vandetanib (ZD6474) is a potent inhibitor of VEGFR2 (IC50: 40 nM). It also inhibits VEGFR3 …
Formel:
C22H24BrFN4O2
Reinheit:
100%
Farbe und Form:
White Solid
Molekulargewicht:
475.35
Ref: TM-T1656
10mg | 49,00 € | ||
25mg | 68,00 € | ||
50mg | 95,00 € | ||
100mg | 171,00 € | ||
200mg | 231,00 € | ||
500mg | 370,00 € | ||
1ml*10 (DMSO) | 54,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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KI8751
CAS:228559-41-9
KI8751 is a potent and selective inhibitor of VEGFR2 with IC50 of 0.9 nM.
Formel:
C24H18F3N3O4
Reinheit:
99.9%
Farbe und Form:
Solid
Molekulargewicht:
469.41
Ref: TM-T2446
2mg | 36,00 € | ||
5mg | 52,00 € | ||
10mg | 84,00 € | ||
25mg | 153,00 € | ||
50mg | 289,00 € | ||
100mg | 508,00 € | ||
200mg | 660,00 € | ||
500mg | 1.003,00 € | ||
1ml*10 (DMSO) | 55,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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PP1
CAS:172889-26-8
PP1 (AGL 1872), a specific and effective Src inhibitor, is with IC50 for Lck/Fyn is …
Formel:
C16H19N5
Reinheit:
99.97%
Farbe und Form:
Off-White To Grey Solid
Molekulargewicht:
281.36
Ref: TM-T6196
1mg | 40,00 € | ||
2mg | 57,00 € | ||
5mg | 92,00 € | ||
10mg | 122,00 € | ||
25mg | 202,00 € | ||
50mg | 283,00 € | ||
100mg | 440,00 € | ||
500mg | 979,00 € | ||
1ml*10 (DMSO) | 98,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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AZD3759 hydrochloride
CAS:1626387-81-2
AZD3759 (hydrochloride) is an effective, orally active and central nervous system-penetrant EGFR inhibitor. At Km …
Formel:
C22H24Cl2FN5O3
Reinheit:
99.41%
Farbe und Form:
Solid
Molekulargewicht:
496.36
Ref: TM-T4249
1mg | 43,00 € | ||
2mg | 54,00 € | ||
5mg | 74,00 € | ||
10mg | 95,00 € | ||
25mg | 163,00 € | ||
50mg | 277,00 € | ||
100mg | 456,00 € | ||
500mg | 1.044,00 € | ||
1ml*10 (DMSO) | 84,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Olafertinib
CAS:1660963-42-7
Olafertinib (RX-518) is a novel mutant-selective, irreversible, orally available EGFR inhibitor. It can overcome T790M-mediated …
Formel:
C29H28F2N6O2
Reinheit:
98.43%
Farbe und Form:
Solid
Molekulargewicht:
530.57
Ref: TM-TQ0255
1mg | 48,00 € | ||
5mg | 94,00 € | ||
10mg | 150,00 € | ||
25mg | 299,00 € | ||
50mg | 441,00 € | ||
100mg | 644,00 € | ||
1ml*10 (DMSO) | 109,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Naquotinib
CAS:1448232-80-1
Naquotinib (ASP8273) (ASP8273) is an orally available, mutant-selective and irreversible EGFR inhibitor; (IC50s: 8-33 nM …
Formel:
C30H42N8O3
Reinheit:
97.49%
Farbe und Form:
Solid
Molekulargewicht:
562.71
Ref: TM-TQ0092
1mg | 51,00 € | ||
2mg | 66,00 € | ||
5mg | 95,00 € | ||
50mg | Nachfragen | ||
1ml*10 (DMSO) | 131,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Tuxobertinib
CAS:2414572-47-5
Tuxobertinib (BDTX-189) is a potent and selective inhibitor of allosteric EGFR and HER2 oncogenic mutations(KDs …
Formel:
C29H29ClN6O4
Reinheit:
98.86%
Farbe und Form:
Solid
Molekulargewicht:
561.03
Ref: TM-T9072
2mg | 40,00 € | ||
5mg | 59,00 € | ||
10mg | 94,00 € | ||
25mg | 185,00 € | ||
50mg | 346,00 € | ||
100mg | 514,00 € | ||
200mg | 735,00 € | ||
1ml*10 (DMSO) | 73,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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WS6
CAS:1421227-53-3
WS6, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase …
Formel:
C29H31F3N6O3
Reinheit:
99.83%
Farbe und Form:
Solid
Molekulargewicht:
568.59
Ref: TM-T2106
1mg | 35,00 € | ||
2mg | 51,00 € | ||
5mg | 71,00 € | ||
10mg | 106,00 € | ||
25mg | 206,00 € | ||
50mg | 379,00 € | ||
100mg | 475,00 € | ||
1ml*10 (DMSO) | 90,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Saracatinib
CAS:379231-04-6
Saracatinib (AZD0530) (AZD0530) is an effective Src inhibitor (IC50: 2.7 nM), and effective to Lck, …
Formel:
C27H32ClN5O5
Reinheit:
99.63%
Farbe und Form:
Solid
Molekulargewicht:
542.03
Ref: TM-T6078
10mg | 64,00 € | ||
25mg | 94,00 € | ||
50mg | 143,00 € | ||
100mg | 224,00 € | ||
1ml*10 (DMSO) | 70,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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(±)-Norcantharidin
CAS:29745-04-8
(±)-Norcantharidin (Endothall anhydride) is a synthetic anticancer compound which is a dual inhibitor for c-Met …
Formel:
C8H8O4
Reinheit:
99.43%
Farbe und Form:
Solid
Molekulargewicht:
168.15
Ref: TM-T5656
1g | 530,00 € | ||
5mg | 44,00 € | ||
10mg | 54,00 € | ||
25mg | 77,00 € | ||
50mg | 103,00 € | ||
100mg | 151,00 € | ||
500mg | 357,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Alflutinib
CAS:1869057-83-9
Alflutinib (ASK120067) is an inhibitor of EGFR, and its targets including EGFR activating mutations and …
Formel:
C28H31F3N8O2
Reinheit:
99.61%
Farbe und Form:
Solid
Molekulargewicht:
568.59
Ref: TM-T22254
1mg | 210,00 € | ||
5mg | 428,00 € | ||
10mg | 610,00 € | ||
25mg | 920,00 € | ||
50mg | 1.295,00 € | ||
100mg | 1.755,00 € | ||
1ml*10 (DMSO) | 550,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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HKI-357
CAS:848133-17-5
HKI-357 is an irreversible dual inhibitor of EGFR and ERBB2 (IC50s: 34 nM and 33 …
Formel:
C31H29ClFN5O3
Reinheit:
98.31%
Farbe und Form:
Solid
Molekulargewicht:
574.05
Ref: TM-T11569
1mg | 78,00 € | ||
5mg | 149,00 € | ||
10mg | 222,00 € | ||
25mg | 452,00 € | ||
50mg | 647,00 € | ||
100mg | 920,00 € | ||
1ml*10 (DMSO) | 185,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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TX1-85-1
CAS:1603845-32-4
TX1-85-1 induces partial degradation of Her3 protein and attenuates Her3-dependent signaling. TX1-85-1 is an irreversible …
Formel:
C32H36N8O3
Reinheit:
98.12%
Farbe und Form:
Solid
Molekulargewicht:
580.68
Ref: TM-T17182
1mg | 69,00 € | ||
5mg | 125,00 € | ||
10mg | 212,00 € | ||
25mg | 362,00 € | ||
50mg | 532,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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PD168393
CAS:194423-15-9
PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, …
Formel:
C17H13BrN4O
Reinheit:
99.7%
Farbe und Form:
Solid
Molekulargewicht:
369.22
Ref: TM-T6932
1mg | 39,00 € | ||
2mg | 49,00 € | ||
5mg | 66,00 € | ||
10mg | 88,00 € | ||
25mg | 151,00 € | ||
50mg | 219,00 € | ||
100mg | 304,00 € | ||
1ml*10 (DMSO) | 55,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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HG-14-10-04
CAS:1356962-34-9
HG-14-10-04 is a potent and specific ALK inhibitor.
Formel:
C29H34ClN7O
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
532.08
Ref: TM-T4015
1mg | 59,00 € | ||
2mg | 87,00 € | ||
5mg | 121,00 € | ||
10mg | 194,00 € | ||
25mg | 274,00 € | ||
50mg | 343,00 € | ||
100mg | 493,00 € | ||
1ml*10 (DMSO) | 141,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Mutant EGFR inhibitor
CAS:1421373-62-7
Mutant EGFR inhibitor is a selective and potent Mutated EGFR inhibitor, inhibits L858R activating mutant, …
Formel:
C27H30ClN7O2
Reinheit:
98%
Farbe und Form:
Solid
Molekulargewicht:
520.03
Ref: TM-T2705
1mg | 36,00 € | ||
2mg | 52,00 € | ||
5mg | 79,00 € | ||
10mg | 95,00 € | ||
25mg | 170,00 € | ||
50mg | 258,00 € | ||
100mg | 371,00 € | ||
500mg | Nachfragen | ||
1ml*10 (DMSO) | 102,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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ZD-4190
CAS:413599-62-9
ZD-4190 is a compound that inhibits both the vascular endothelial growth factor receptor 2 (VEGFR2) …
Formel:
C19H16BrFN6O2
Reinheit:
99.42%
Farbe und Form:
Solid
Molekulargewicht:
459.27
Ref: TM-T5475
1mg | 123,00 € | ||
2mg | 179,00 € | ||
5mg | 299,00 € | ||
10mg | 449,00 € | ||
25mg | 714,00 € | ||
50mg | 981,00 € | ||
100mg | 1.318,00 € | ||
1ml*10 (DMSO) | 302,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Methyl 2,5-dihydroxycinnamate
CAS:63177-57-1
Methyl 2,5-dihydroxycinnamate is an EGF receptor-associated tyrosine kinases inhibitor.
Formel:
C10H10O4
Reinheit:
98.98%
Farbe und Form:
Crystalline
Molekulargewicht:
194.18
Ref: TM-T22974
5mg | 64,00 € | ||
10mg | 99,00 € | ||
25mg | 189,00 € | ||
50mg | 351,00 € | ||
100mg | 522,00 € | ||
1ml*10 (DMSO) | 59,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Tucatinib
CAS:937263-43-9
Tucatinib (ONT-380) is a potent and selective HER2 inhibitor (IC50: 8 nM).
Formel:
C26H24N8O2
Reinheit:
99.96%
Farbe und Form:
Solid
Molekulargewicht:
480.52
Ref: TM-T2364
1g | 1.110,00 € | ||
2mg | 40,00 € | ||
5mg | 54,00 € | ||
10mg | 83,00 € | ||
25mg | 127,00 € | ||
50mg | 189,00 € | ||
100mg | 343,00 € | ||
500mg | 812,00 € | ||
1ml*10 (DMSO) | 85,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Butein
CAS:487-52-5
Butein (2’,3,4,4’-tetrahydroxy Chalcone), a plant polyphenol, is isolated from Rhus verniciflua. It can inhibit the …
Formel:
C15H12O5
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
272.25
Ref: TM-T6427
1mg | 42,00 € | ||
2mg | 55,00 € | ||
5mg | 86,00 € | ||
10mg | 104,00 € | ||
25mg | 210,00 € | ||
50mg | 337,00 € | ||
100mg | 540,00 € | ||
1ml*10 (DMSO) | 86,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Osimertinib
CAS:1421373-65-0
Osimertinib (AZD-9291) is an EGFR third-generation inhibitor that inhibits the T790M resistance mutation produced by …
Formel:
C28H33N7O2
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
499.61
Ref: TM-T2490
1g | 121,00 € | ||
2mg | 30,00 € | ||
5mg | 45,00 € | ||
10mg | 49,00 € | ||
25mg | 59,00 € | ||
50mg | 70,00 € | ||
100mg | 91,00 € | ||
200mg | 91,00 € | ||
500mg | 100,00 € | ||
1ml*10 (DMSO) | 45,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Beta-Hydroxyisovalerylshikonin
CAS:7415-78-3
Beta-Hydroxyisovalerylshikonin is an inhibitor of protein-tyrosine kinases such as v-Src and EGFR, and has been …
Formel:
C21H24O7
Reinheit:
98.16%
Farbe und Form:
Solid
Molekulargewicht:
388.41
Ref: TM-TN1440
1mg | 134,00 € | ||
5mg | 395,00 € | ||
10mg | 575,00 € | ||
25mg | 894,00 € | ||
50mg | 1.199,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EGFR-IN-8
CAS:2407957-87-1
EGFR-IN-8, a dual inhibitor targeting both EGFR and c-Met, shows potential as a promising candidate …
Formel:
C32H23ClF3N7O4
Reinheit:
98%
Farbe und Form:
Solid
Molekulargewicht:
662.02
Ref: TM-T11162
1mg | 74,00 € | ||
5mg | 166,00 € | ||
10mg | 266,00 € | ||
25mg | 440,00 € | ||
50mg | 602,00 € | ||
100mg | 825,00 € | ||
1ml*10 (DMSO) | 235,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PD153035 hydrochloride
CAS:183322-45-4
PD153035 hydrochloride (ZM 252868) is a effective and selective inhibitor of EGFR (Ki: 5.2 pM, …
Formel:
C16H15BrClN3O2
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
396.67
Ref: TM-T1761
5mg | 35,00 € | ||
10mg | 44,00 € | ||
25mg | 81,00 € | ||
50mg | 142,00 € | ||
100mg | 233,00 € | ||
500mg | 530,00 € | ||
1ml*10 (DMSO) | 35,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PP 3
CAS:5334-30-5
PP 3 is a Negative control for the Src kinase inhibitor PP 2
Formel:
C11H9N5
Reinheit:
98.92%
Farbe und Form:
Whit To Off-White Solid
Molekulargewicht:
211.22
Ref: TM-T23176
5mg | 56,00 € | ||
10mg | 83,00 € | ||
25mg | 143,00 € | ||
50mg | 203,00 € | ||
100mg | 306,00 € | ||
500mg | 719,00 € | ||
1ml*10 (DMSO) | 54,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Poziotinib
CAS:1092364-38-9
Poziotinib (NOV120101)(NOV120101; HM781-36B) is an irreversible HER1/2/4 inhibitor (IC50s: 3/5/23 nM).
Formel:
C23H21Cl2FN4O3
Reinheit:
99.78%
Farbe und Form:
Solid
Molekulargewicht:
491.34
Ref: TM-T2630
1mg | 35,00 € | ||
5mg | 69,00 € | ||
10mg | 95,00 € | ||
25mg | 183,00 € | ||
50mg | 323,00 € | ||
100mg | 508,00 € | ||
1ml*10 (DMSO) | 73,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EAI045
CAS:1942114-09-1
EAI045, an allosteric inhibitor, targets towards drug-resistant EGFR mutants but avoids the wild-type receptor.
Formel:
C19H14FN3O3S
Reinheit:
99.73%
Farbe und Form:
Solid
Molekulargewicht:
383.4
Ref: TM-T6824
5mg | 43,00 € | ||
10mg | 58,00 € | ||
25mg | 90,00 € | ||
50mg | 121,00 € | ||
100mg | 193,00 € | ||
1ml*10 (DMSO) | 54,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
ONO-7475
CAS:1646839-59-9
ONO-7475 is an inhibitor with high specificity for anexelekto and MER tyrosine kinase
Formel:
C32H26N4O6
Reinheit:
98.33%
Farbe und Form:
Solid
Molekulargewicht:
562.57
Ref: TM-T8327
1mg | 62,00 € | ||
5mg | 134,00 € | ||
10mg | 206,00 € | ||
25mg | 352,00 € | ||
50mg | 520,00 € | ||
100mg | 733,00 € | ||
1ml*10 (DMSO) | 166,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Poziotinib hydrochloride
CAS:1429757-68-5
Poziotinib hydrochloride irreversibly inhibits EGFR (HER1 or ErbB1), including EGFR mutants, HER2, and HER4, thereby …
Formel:
C23H22Cl3FN4O3
Reinheit:
99.69%
Farbe und Form:
Solid
Molekulargewicht:
527.8
Ref: TM-T8758
5mg | 54,00 € | ||
10mg | 81,00 € | ||
25mg | 124,00 € | ||
50mg | 179,00 € | ||
100mg | 267,00 € | ||
200mg | 401,00 € | ||
500mg | 666,00 € | ||
1ml*10 (DMSO) | 87,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AZ7550
CAS:1421373-99-0
AZ7550, an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).
Formel:
C27H31N7O2
Reinheit:
97.07%
Farbe und Form:
Solid
Molekulargewicht:
485.58
Ref: TM-T13564
1mg | 129,00 € | ||
5mg | 282,00 € | ||
10mg | 417,00 € | ||
25mg | 689,00 € | ||
50mg | 920,00 € | ||
100mg | 1.287,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tyrphostin A9
CAS:10537-47-0
Tyrphostin A9 (SF 6847) is an Agricultural acaricide, now superseded. Tyrphostin A9 is firstly designed …
Formel:
C18H22N2O
Reinheit:
99.36%
Farbe und Form:
Yellow Solid
Molekulargewicht:
282.38
Ref: TM-T2479
25mg | 54,00 € | ||
50mg | 63,00 € | ||
100mg | 95,00 € | ||
200mg | 169,00 € | ||
500mg | 374,00 € | ||
1ml*10 (DMSO) | 40,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Dacomitinib
CAS:1110813-31-4
Dacomitinib (PF299)(PF299804; PF-00299804) is a highly selective, orally bioavailable small-molecule inhibitor of the HER family …
Formel:
C24H25ClFN5O2
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
469.94
Ref: TM-T2483
1mg | 38,00 € | ||
2mg | 49,00 € | ||
5mg | 78,00 € | ||
10mg | 124,00 € | ||
25mg | 170,00 € | ||
50mg | 222,00 € | ||
100mg | 348,00 € | ||
200mg | 435,00 € | ||
500mg | 717,00 € | ||
1ml*10 (DMSO) | 78,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AZ-5104
CAS:1421373-98-9
AZ5104 is a potent EGFR inhibitor.
Formel:
C27H31N7O2
Reinheit:
99.9%
Farbe und Form:
Solid Powder
Molekulargewicht:
485.58
Ref: TM-T2491
5mg | 57,00 € | ||
10mg | 79,00 € | ||
25mg | 126,00 € | ||
50mg | 188,00 € | ||
100mg | 251,00 € | ||
200mg | 314,00 € | ||
1ml*10 (DMSO) | 57,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Afatinib Dimaleate
CAS:850140-73-7
Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the receptor …
Formel:
C32H33ClFN5O11
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
718.08
Ref: TM-T1773
1g | 460,00 € | ||
5mg | 40,00 € | ||
10mg | 58,00 € | ||
25mg | 85,00 € | ||
50mg | 105,00 € | ||
100mg | 138,00 € | ||
200mg | 184,00 € | ||
500mg | 308,00 € | ||
1ml*10 (DMSO) | 65,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Epidermal Growth Factor
CAS:62253-63-8
Epidermal Growth Factor binds to epidermal growth factor receptor (EGFR) and stimulates cell growth and …
Formel:
C270H401N73O83S7
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
6222
Ref: TM-T8679
1mg | 129,00 € | ||
2mg | 184,00 € | ||
5mg | 278,00 € | ||
10mg | 421,00 € | ||
25mg | 697,00 € | ||
50mg | 976,00 € | ||
100mg | 1.319,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
CP-380736
CAS:179688-29-0
CP-380736 (PF-00520893) is an epidermal growth factor receptor (EGFR) inhibitor. EGFR is a tyrosine kinase …
Formel:
C14H18N2O5
Reinheit:
99.91%
Farbe und Form:
White To Off-White Solid
Molekulargewicht:
294.3
Ref: TM-T19814
5mg | 54,00 € | ||
10mg | 81,00 € | ||
25mg | 123,00 € | ||
50mg | 180,00 € | ||
100mg | 267,00 € | ||
200mg | 402,00 € | ||
1ml*10 (DMSO) | 70,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
NSC 228155
CAS:113104-25-9
NSC 228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and …
Formel:
C11H6N4O4S
Reinheit:
99.84%
Farbe und Form:
Solid
Molekulargewicht:
290.25
Ref: TM-T6908
5mg | 50,00 € | ||
10mg | 66,00 € | ||
25mg | 123,00 € | ||
50mg | 215,00 € | ||
100mg | 373,00 € | ||
200mg | 484,00 € | ||
1ml*10 (DMSO) | 52,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
(E)-AG 556
CAS:133550-41-1
AG 556 is a selective inhibitor of EGFR and blocks LPS-induced TNF-α production.
Formel:
C20H20N2O3
Reinheit:
98%
Farbe und Form:
Light Yellow Powder
Molekulargewicht:
336.38
Ref: TM-T21853
5mg | 51,00 € | ||
10mg | 86,00 € | ||
25mg | 157,00 € | ||
50mg | 231,00 € | ||
100mg | 342,00 € | ||
200mg | 507,00 € | ||
500mg | 801,00 € | ||
1ml*10 (DMSO) | 56,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Alflutinib mesylate
CAS:2130958-55-1
Alflutinib mesylate (AST2818 mesylate) ,is an irreversible tyrosine kinase inhibitor that selectively inhibits EGFR mutations, …
Formel:
C29H35F3N8O5S
Reinheit:
99.81%
Farbe und Form:
Solid
Molekulargewicht:
664.7
Ref: TM-T7175
1mg | 77,00 € | ||
5mg | 160,00 € | ||
10mg | 230,00 € | ||
25mg | 388,00 € | ||
50mg | 576,00 € | ||
100mg | 816,00 € | ||
500mg | 1.662,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tyrphostin 23
CAS:118409-57-7
Tyrphostin 23 (AG18) inhibits EGFR with IC50 of 35 μM.
Formel:
C10H6N2O2
Reinheit:
99.19%
Farbe und Form:
Yellow-Tan Solid
Molekulargewicht:
186.17
Ref: TM-T2063
10mg | 59,00 € | ||
25mg | 120,00 € | ||
50mg | 221,00 € | ||
100mg | 332,00 € | ||
1ml*10 (DMSO) | 43,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EGFR-IN-12
CAS:879127-07-8
EGFR-IN-12 (EGFR Inhibitor) is a cell permeable and selective inhibitor of EGFR kinase (IC50: 21 …
Formel:
C21H18F3N5O
Reinheit:
99.15%
Farbe und Form:
Solid
Molekulargewicht:
413.4
Ref: TM-T5168
1mg | 81,00 € | ||
5mg | 156,00 € | ||
10mg | 255,00 € | ||
25mg | 511,00 € | ||
50mg | 727,00 € | ||
100mg | 985,00 € | ||
500mg | 1.977,00 € | ||
1ml*10 (DMSO) | 170,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WHI-P154
CAS:211555-04-3
WHI-P154 (Jak3 inhibitor ii) is a potent JAK3 inhibitor.
Formel:
C16H14BrN3O3
Reinheit:
99.6%
Farbe und Form:
Solid
Molekulargewicht:
376.2
Ref: TM-T1985
2mg | 46,00 € | ||
5mg | 65,00 € | ||
10mg | 100,00 € | ||
25mg | 178,00 € | ||
50mg | 331,00 € | ||
100mg | 534,00 € | ||
1ml*10 (DMSO) | 68,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Avitinib maleate
CAS:1557268-88-8
Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor.
Formel:
C30H30FN7O6
Reinheit:
99.77%
Farbe und Form:
Solid
Molekulargewicht:
603.61
Ref: TM-T3721
5mg | 72,00 € | ||
10mg | 113,00 € | ||
25mg | 205,00 € | ||
50mg | 346,00 € | ||
100mg | 557,00 € | ||
1ml*10 (DMSO) | 87,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Avitinib
CAS:1557267-42-1
Avitinib (AC0010), also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth …
Formel:
C26H26FN7O2
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
487.53
Ref: TM-T3024
2mg | 48,00 € | ||
5mg | 73,00 € | ||
10mg | 113,00 € | ||
25mg | 212,00 € | ||
50mg | 347,00 € | ||
100mg | 513,00 € | ||
1ml*10 (DMSO) | 85,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
BI-4020
CAS:2664214-60-0
BI-4020 is a fourth-generation, orally active, and non-covalent inhibitor of EGFR tyrosine kinase. BI-4020 exhibits …
Formel:
C30H38N8O2
Reinheit:
100.00%
Farbe und Form:
Solid
Molekulargewicht:
542.68
Ref: TM-T10534
1mg | 268,00 € | ||
5mg | 650,00 € | ||
10mg | 925,00 € | ||
25mg | 1.388,00 € | ||
50mg | 1.859,00 € | ||
1ml*10 (DMSO) | 790,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
(S)-Sunvozertinib
CAS:2370013-49-1
(S)-Sunvozertinib (DZD9008) is a rationally designed selective, irreversible EGFR/HER2 inhibitor.
Formel:
C29H35ClFN7O3
Reinheit:
99.69%
Farbe und Form:
Solid
Molekulargewicht:
584.08
Ref: TM-T9304
1mg | 62,00 € | ||
5mg | 134,00 € | ||
10mg | 207,00 € | ||
25mg | 415,00 € | ||
50mg | 612,00 € | ||
100mg | 878,00 € | ||
1ml*10 (DMSO) | 172,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
ALK-IN-1
CAS:1197958-12-5
ALK-IN-1 (AP26113) is a potent ALK inhibitor with IC50 of 0.62 nM in a cell-free …
Formel:
C26H34ClN6O2P
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
529.01
Ref: TM-T3059
5mg | 48,00 € | ||
10mg | 70,00 € | ||
25mg | 94,00 € | ||
50mg | 142,00 € | ||
100mg | 230,00 € | ||
200mg | 346,00 € | ||
500mg | 561,00 € | ||
1ml*10 (DMSO) | 51,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Zorifertinib
CAS:1626387-80-1
Zorifertinib (AZD3759) is an orally active, effective and central nervous system-penetrant EGFR inhibitor. The IC50 …
Formel:
C22H23ClFN5O3
Reinheit:
98.32%
Farbe und Form:
White To Off-White Solid
Molekulargewicht:
459.9
Ref: TM-T3659
10mg | 46,00 € | ||
25mg | 67,00 € | ||
50mg | 96,00 € | ||
100mg | 134,00 € | ||
1ml*10 (DMSO) | 50,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
MTX-211
CAS:1952236-05-3
MTX-211, an inhibitor of EGFR and PI3K, is used for the therapy of cancer and …
Formel:
C20H14Cl2FN5O2S
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
478.33
Ref: TM-T4296
1mg | 93,00 € | ||
2mg | 161,00 € | ||
5mg | 304,00 € | ||
10mg | 462,00 € | ||
25mg | 765,00 € | ||
50mg | 1.054,00 € | ||
100mg | 1.430,00 € | ||
500mg | 2.775,00 € | ||
1ml*10 (DMSO) | 310,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Desmethyl Erlotinib hydrochloride
CAS:183320-51-6
Desmethyl Erlotinib hydrochloride (OSI 420) is an active metabolite of erlotinib which is an orally …
Formel:
C21H21N3O4·HCl
Reinheit:
99.03%
Farbe und Form:
Solid
Molekulargewicht:
415.87
Ref: TM-T6619
1mg | 59,00 € | ||
2mg | 82,00 € | ||
5mg | 113,00 € | ||
10mg | 184,00 € | ||
25mg | 329,00 € | ||
50mg | 495,00 € | ||
100mg | 704,00 € | ||
1ml*10 (DMSO) | 124,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Allitinib tosylate
CAS:1050500-29-2
Allitinib tosylate (AST-1306) is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of …
Formel:
C31H26ClFN4O5S
Reinheit:
98.52%
Farbe und Form:
Solid
Molekulargewicht:
621.08
Ref: TM-T6331
1mg | 55,00 € | ||
5mg | 118,00 € | ||
10mg | 183,00 € | ||
25mg | 346,00 € | ||
50mg | 517,00 € | ||
100mg | 727,00 € | ||
500mg | 1.538,00 € | ||
1ml*10 (DMSO) | 162,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
RG14620
CAS:136831-49-7
RG14620 (Tyrphostin RG14620) is an epidermal growth factor receptor (EGFR) inhibitor.
Formel:
C14H8Cl2N2
Reinheit:
99.79%
Farbe und Form:
Solid
Molekulargewicht:
275.13
Ref: TM-T3554
2mg | 35,00 € | ||
5mg | 52,00 € | ||
10mg | 76,00 € | ||
25mg | 134,00 € | ||
50mg | 255,00 € | ||
100mg | 425,00 € | ||
500mg | 920,00 € | ||
1ml*10 (DMSO) | 58,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AG 555
CAS:133550-34-2
AG 555 (Tyrphostin B46) is an EGFR tyrosine kinase inhibitor.
Formel:
C19H18N2O3
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
322.36
Ref: TM-T4326
5mg | 46,00 € | ||
10mg | 69,00 € | ||
25mg | 109,00 € | ||
50mg | 166,00 € | ||
100mg | 241,00 € | ||
1ml*10 (DMSO) | 51,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WHI-P258
CAS:21561-09-1
WHI-P258 is a dimethoxyquinazoline inhibitor of JAK3. This compound binds JAK3 weakly and may be …
Formel:
C16H15N3O2
Reinheit:
99.95%
Farbe und Form:
Solid
Molekulargewicht:
281.31
Ref: TM-T2035
5mg | 55,00 € | ||
10mg | 86,00 € | ||
25mg | 150,00 € | ||
50mg | 233,00 € | ||
100mg | 391,00 € | ||
500mg | 893,00 € | ||
1ml*10 (DMSO) | 62,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
RG13022
CAS:136831-48-6
RG13022 (Tyrphostin RG13022) is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF …
Formel:
C16H14N2O2
Reinheit:
98.38%
Farbe und Form:
Solid
Molekulargewicht:
266.29
Ref: TM-T3545
2mg | 46,00 € | ||
5mg | 60,00 € | ||
10mg | 87,00 € | ||
25mg | 177,00 € | ||
50mg | 298,00 € | ||
100mg | 470,00 € | ||
1ml*10 (DMSO) | 63,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Osimertinib mesylate
CAS:1421373-66-1
Osimertinib mesylate (Mereletinib mesylate) is an irreversible and mutant selective EGFR inhibitor (IC50s: 12/1 nM …
Formel:
C29H37N7O5S
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
595.71
Ref: TM-T3634
1g | 149,00 € | ||
5mg | 49,00 € | ||
10mg | 60,00 € | ||
50mg | 86,00 € | ||
100mg | 94,00 € | ||
200mg | 111,00 € | ||
500mg | 129,00 € | ||
1ml*10 (DMSO) | 68,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AG-1478
CAS:153436-53-4
AG-1478 (NSC-693255) (Tyrphostin AG-1478) is a selective EGFR inhibitor.
Formel:
C16H14ClN3O2
Reinheit:
99.71%
Farbe und Form:
Solid
Molekulargewicht:
315.75
Ref: TM-T2047
5mg | 54,00 € | ||
10mg | 71,00 € | ||
25mg | 115,00 € | ||
50mg | 198,00 € | ||
100mg | 273,00 € | ||
200mg | 355,00 € | ||
1ml*10 (DMSO) | 59,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Neratinib
CAS:698387-09-6
Neratinib (HKI-272) (HKI-272) is an orally available, irreversible tyrosine kinase inhibitor for HER2 and EGFR …
Formel:
C30H29ClN6O3
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
557.04
Ref: TM-T2325
5mg | 35,00 € | ||
10mg | 51,00 € | ||
25mg | 69,00 € | ||
50mg | 92,00 € | ||
100mg | 122,00 € | ||
200mg | 184,00 € | ||
500mg | 307,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AG-494
CAS:133550-35-3
AG-494 (Tyrphostin B48) is an inhibitor of epidermal growth factor receptor kinase.
Formel:
C16H12N2O3
Reinheit:
98.9%
Farbe und Form:
Solid
Molekulargewicht:
280.28
Ref: TM-T4205
5mg | 65,00 € | ||
10mg | 93,00 € | ||
25mg | 162,00 € | ||
50mg | 244,00 € | ||
100mg | 387,00 € | ||
1ml*10 (DMSO) | 66,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Withanolide A
CAS:32911-62-9
Withanolide A extends the lifespan in human EGFR-driven cancerous Caenorhabditis elegans.
Formel:
C28H38O6
Reinheit:
98.49%
Farbe und Form:
Solid
Molekulargewicht:
470.6
Ref: TM-TN2309
1mg | 98,00 € | ||
5mg | 233,00 € | ||
10mg | 357,00 € | ||
25mg | 567,00 € | ||
50mg | 841,00 € | ||
1ml*10 (DMSO) | 366,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
G5-7
CAS:939681-36-4
JAK2 inhibitor G5-7 (JAK2 inhibitor G5-7) is an orally active JAK2 inhibitor, selectively inhibits JAK2-mediated …
Formel:
C22H19F2NO3
Reinheit:
99.37%
Farbe und Form:
Solid
Molekulargewicht:
383.39
Ref: TM-T8742
1mg | 82,00 € | ||
5mg | 158,00 € | ||
10mg | 230,00 € | ||
25mg | 424,00 € | ||
50mg | 613,00 € | ||
100mg | 856,00 € | ||
500mg | 1.700,00 € | ||
1ml*10 (DMSO) | 171,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Benidipine hydrochloride
CAS:91599-74-5
Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker …
Formel:
C28H32ClN3O6
Reinheit:
99.56%
Farbe und Form:
Solid
Molekulargewicht:
542.03
Ref: TM-T6227
1g | 130,00 € | ||
50mg | 36,00 € | ||
100mg | 48,00 € | ||
200mg | 61,00 € | ||
500mg | 90,00 € | ||
1ml*10 (DMSO) | 52,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Desmethyl Erlotinib
CAS:183321-86-0
Desmethyl Erlotinib (CP-473420) is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 …
Formel:
C21H21N3O4
Reinheit:
98.62%
Farbe und Form:
Solid
Molekulargewicht:
379.41
Ref: TM-T6328
1mg | 52,00 € | ||
2mg | 75,00 € | ||
5mg | 114,00 € | ||
10mg | 185,00 € | ||
25mg | 324,00 € | ||
50mg | 489,00 € | ||
100mg | 703,00 € | ||
1ml*10 (DMSO) | 125,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Almonertinib
CAS:1899921-05-1
Almonertinib (HS-10296) is an inhibitor of EGFR activation mutation and tolerant mutation of EGFR T790M, …
Formel:
C30H35N7O2
Reinheit:
99.85%
Farbe und Form:
Solid
Molekulargewicht:
525.64
Ref: TM-T5462
1mg | 88,00 € | ||
5mg | 193,00 € | ||
10mg | 305,00 € | ||
25mg | 514,00 € | ||
50mg | 739,00 € | ||
100mg | 1.016,00 € | ||
500mg | 2.070,00 € | ||
1ml*10 (DMSO) | 245,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Dacomitinib hydrate
CAS:1042385-75-0
Dacomitinib hydrate (PF 299804) is a highly selective and second-generation small-molecule inhibitor of the pan-epidermal …
Formel:
C24H27ClFN5O3
Reinheit:
98.05%
Farbe und Form:
Solid
Molekulargewicht:
487.96
Ref: TM-T19965
1mg | 37,00 € | ||
2mg | 52,00 € | ||
5mg | 78,00 € | ||
10mg | 118,00 € | ||
25mg | 167,00 € | ||
50mg | 223,00 € | ||
100mg | 346,00 € | ||
500mg | 810,00 € | ||
1ml*10 (DMSO) | 88,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tesevatinib
CAS:781613-23-8
Tesevatinib (XL-647) is an orally available, multi-target tyrosine kinase inhibitor (IC50s: 0.3, 16, 1.5, 8.7, …
Formel:
C24H25Cl2FN4O2
Reinheit:
97.89%
Farbe und Form:
Solid
Molekulargewicht:
491.39
Ref: TM-TQ0166
1mg | 106,00 € | ||
2mg | 152,00 € | ||
5mg | 232,00 € | ||
10mg | 450,00 € | ||
25mg | 737,00 € | ||
50mg | 1.003,00 € | ||
1ml*10 (DMSO) | 250,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EBE-A22
CAS:229476-53-3
EBE-A22 (PD153035 Analog 63) is a derivative of PD 153035 which can inhibit ErbB-1-phosphorylation, whereas …
Formel:
C17H16BrN3O2
Reinheit:
99.88%
Farbe und Form:
Solid
Molekulargewicht:
374.23
Ref: TM-T3558
1mg | 46,00 € | ||
2mg | 59,00 € | ||
5mg | 91,00 € | ||
10mg | 114,00 € | ||
25mg | 223,00 € | ||
50mg | 339,00 € | ||
100mg | 508,00 € | ||
500mg | 1.087,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Gefitinib-based PROTAC 3
CAS:2230821-27-7
Gefitinib-based PROTAC 3, conjugating an EGFR binding element to a VHL ligand via a linker, …
Formel:
C47H57ClFN7O8S
Reinheit:
98.25%
Farbe und Form:
Solid
Molekulargewicht:
934.51
Ref: TM-T5437
1mg | 49,00 € | ||
2mg | 69,00 € | ||
5mg | 94,00 € | ||
10mg | 171,00 € | ||
25mg | 278,00 € | ||
50mg | 424,00 € | ||
100mg | 611,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
MAZ51
CAS:163655-37-6
MAZ51 is a VEGFR-3 (Flt-4) tyrosine kinase inhibitor.
Formel:
C21H18N2O
Reinheit:
98.53%
Farbe und Form:
Solid
Molekulargewicht:
314.38
Ref: TM-T8496
1mg | 40,00 € | ||
2mg | 56,00 € | ||
5mg | 88,00 € | ||
10mg | 126,00 € | ||
25mg | 242,00 € | ||
50mg | 403,00 € | ||
100mg | 599,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Brigatinib
CAS:1197953-54-0
Brigatinib (AP-26113) is a highly potent and selective ALK inhibitor.
Formel:
C29H39ClN7O2P
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
584.09
Ref: TM-T3621
1ml | 65,00 € | ||
2mg | 36,00 € | ||
5mg | 50,00 € | ||
10mg | 66,00 € | ||
25mg | 87,00 € | ||
50mg | 112,00 € | ||
100mg | 163,00 € | ||
200mg | 235,00 € | ||
500mg | 400,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WZ4002
CAS:1213269-23-8
WZ4002 is a mutant-selective EGFR inhibitor for EGFR(L858R) and EGFR(T790M) with IC50 of 2 nM/8 …
Formel:
C25H27ClN6O3
Reinheit:
98.12%
Farbe und Form:
Solid
Molekulargewicht:
494.97
Ref: TM-T6238
2mg | 35,00 € | ||
5mg | 51,00 € | ||
10mg | 72,00 € | ||
25mg | 115,00 € | ||
50mg | 183,00 € | ||
100mg | 325,00 € | ||
200mg | 478,00 € | ||
1ml*10 (DMSO) | 52,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tyrphostin A1
CAS:2826-26-8
Tyrphostin A1 (Tyrphostin 1) is an inhibitor of EGFR tyrosine kinase .
Formel:
C11H8N2O
Reinheit:
99.13%
Farbe und Form:
Solid
Molekulargewicht:
184.19
Ref: TM-T7649
5mg | 35,00 € | ||
10mg | 51,00 € | ||
25mg | 96,00 € | ||
50mg | 121,00 € | ||
100mg | 158,00 € | ||
1ml*10 (DMSO) | 40,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Pelitinib
CAS:257933-82-7
Pelitinib (EKB-569) (EKB-569) is an effective irreversible EGFR inhibitor (IC50: 38.5 nM).
Formel:
C24H23ClFN5O2
Reinheit:
99.86%
Farbe und Form:
Off-White Solid
Molekulargewicht:
467.92
Ref: TM-T2327
5mg | 55,00 € | ||
10mg | 71,00 € | ||
25mg | 109,00 € | ||
50mg | 133,00 € | ||
100mg | 189,00 € | ||
500mg | 455,00 € | ||
1ml*10 (DMSO) | 57,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WZ-3146
CAS:1214265-56-1
WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and EGFR(E746_A750) with IC50 of 2 nM …
Formel:
C24H25ClN6O2
Reinheit:
98.95%
Farbe und Form:
Solid
Molekulargewicht:
464.95
Ref: TM-T6733
1mg | 52,00 € | ||
2mg | 73,00 € | ||
5mg | 95,00 € | ||
10mg | 176,00 € | ||
25mg | 312,00 € | ||
50mg | 499,00 € | ||
100mg | 713,00 € | ||
1ml*10 (DMSO) | 104,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
CZC-8004
CAS:916603-07-1
CZC-8004 (CZC-00008004) is a pan-kinase(ABL kinase) inhibitor and binds a range of tyrosine kinases.
Formel:
C17H16FN5
Reinheit:
98%
Farbe und Form:
Solid
Molekulargewicht:
309.34
Ref: TM-T7186
1mg | 47,00 € | ||
5mg | 96,00 € | ||
10mg | 142,00 € | ||
25mg | 291,00 € | ||
50mg | 435,00 € | ||
100mg | 625,00 € | ||
1ml*10 (DMSO) | 95,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Lazertinib
CAS:1903008-80-9
Lazertinib (GNS-1480) is an effective, highly mutant-selective and irreversible EGFR-TKI with IC50 values of 1.7 …
Formel:
C30H34N8O3
Reinheit:
99.96%
Farbe und Form:
Solid
Molekulargewicht:
554.64
Ref: TM-T4485
1mg | 48,00 € | ||
2mg | 64,00 € | ||
5mg | 90,00 € | ||
10mg | 147,00 € | ||
25mg | 253,00 € | ||
50mg | 319,00 € | ||
100mg | 462,00 € | ||
500mg | 1.072,00 € | ||
1ml*10 (DMSO) | 108,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
CNX-2006
CAS:1375465-09-0
CNX-2006 is a novel irreversible mutant-selective EGFR inhibitor with IC50 of < 20 nM, with very …
Formel:
C26H27F4N7O2
Reinheit:
99.16%
Farbe und Form:
Solid
Molekulargewicht:
545.53
Ref: TM-T6008
1mg | 40,00 € | ||
2mg | 52,00 € | ||
5mg | 82,00 € | ||
10mg | 123,00 € | ||
25mg | 219,00 € | ||
50mg | 397,00 € | ||
1ml*10 (DMSO) | 89,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Sapitinib
CAS:848942-61-0
Sapitinib (AZD-8931) , a reversible, ATP competitive inhibitor of EGFR(IC50=4 nM), ErbB2(IC50=3 nM) and ErbB3(IC50=4 …
Formel:
C23H25ClFN5O3
Reinheit:
99.83%
Farbe und Form:
Solid
Molekulargewicht:
473.93
Ref: TM-T6092
2mg | 38,00 € | ||
5mg | 56,00 € | ||
10mg | 85,00 € | ||
25mg | 109,00 € | ||
50mg | 163,00 € | ||
100mg | 235,00 € | ||
1ml*10 (DMSO) | 59,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Olmutinib
CAS:1353550-13-6
Olmutinib (HM61713, BI 1482694) is an orally available small molecule, a mutant-selective inhibitor of epidermal …
Formel:
C26H26N6O2S
Reinheit:
99.27%
Farbe und Form:
Solid
Molekulargewicht:
486.59
Ref: TM-T6918
2mg | 39,00 € | ||
5mg | 56,00 € | ||
10mg | 87,00 € | ||
25mg | 134,00 € | ||
50mg | 176,00 € | ||
100mg | 276,00 € | ||
200mg | 454,00 € | ||
1ml*10 (DMSO) | 58,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Cyasterone
CAS:17086-76-9
Cyasterone (Cyasteron), a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, …
Formel:
C29H44O8
Reinheit:
99.26%
Farbe und Form:
Solid
Molekulargewicht:
520.65
Ref: TM-T3870
1mg | 35,00 € | ||
5mg | 69,00 € | ||
10mg | 109,00 € | ||
25mg | 199,00 € | ||
50mg | 298,00 € | ||
100mg | 442,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Leptomycin B
CAS:87081-35-4
Leptomycin B (LMB) is a potent inhibitor of the nuclear export of proteins and is …
Formel:
C33H48O6
Reinheit:
99.71%
Farbe und Form:
White Crystalline Solid
Molekulargewicht:
540.73
Ref: TM-T15735
1mg | 203,00 € | ||
2mg | 335,00 € | ||
5mg | 611,00 € | ||
10mg | 867,00 € | ||
25mg | 1.296,00 € | ||
50mg | 1.747,00 € | ||
100mg | 2.349,00 € | ||
1ml*10 (DMSO) | 277,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PD-161570
CAS:192705-80-9
PD-161570 is a potent and ATP-competitive human FGF-1 receptor inhibitor with an IC50 of 39.9 …
Formel:
C26H35Cl2N7O
Reinheit:
99.23%
Farbe und Form:
Solid
Molekulargewicht:
532.51
Ref: TM-T23127
1mg | 95,00 € | ||
2mg | 133,00 € | ||
5mg | 207,00 € | ||
10mg | 306,00 € | ||
25mg | 516,00 € | ||
50mg | 735,00 € | ||
100mg | 997,00 € | ||
1ml*10 (DMSO) | 241,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Almonertinib hydrochloride
CAS:2134096-03-8
Almonertinib hydrochloride (HS-10296 hydrochloride) is a small molecule inhibitor of EGFR-activating mutations and T790M-resistant mutation …
Formel:
C30H36ClN7O2
Reinheit:
98.01%
Farbe und Form:
Solid
Molekulargewicht:
562.1
Ref: TM-T5675
1mg | 90,00 € | ||
5mg | 182,00 € | ||
10mg | 305,00 € | ||
25mg | 525,00 € | ||
50mg | 740,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Genistein
CAS:446-72-0
Genistein (NPI 031L) is an isoflavonoid derived from soy products. It inhibits protein-tyrosine kinase and …
Formel:
C15H10O5
Reinheit:
99.69%
Farbe und Form:
Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether Solid
Molekulargewicht:
270.24
Ref: TM-T1737
50mg | 45,00 € | ||
100mg | 58,00 € | ||
500mg | 93,00 € | ||
1ml*10 (DMSO) | 62,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Rostafuroxin
CAS:156722-18-8
Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.
Formel:
C23H34O4
Reinheit:
100%
Farbe und Form:
Solid
Molekulargewicht:
374.51
Ref: TM-T2621
2mg | 43,00 € | ||
5mg | 64,00 € | ||
10mg | 105,00 € | ||
25mg | 184,00 € | ||
50mg | 345,00 € | ||
100mg | 510,00 € | ||
1ml*10 (DMSO) | 71,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tyrphostin AG30
CAS:122520-79-0
Tyrphostin AG30 (AG30) (AG30) is a potent protein tyrosine kinases (PTK) inhibitor.
Formel:
C10H7NO4
Reinheit:
98%
Farbe und Form:
Solid
Molekulargewicht:
205.17
Ref: TM-T7101
2mg | 46,00 € | ||
5mg | 69,00 € | ||
10mg | 86,00 € | ||
25mg | 172,00 € | ||
50mg | 301,00 € | ||
100mg | 500,00 € | ||
1ml*10 (DMSO) | 52,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Almonertinib mesylate
CAS:2134096-06-1
Almonertinib mesylate is an irreversible inhibitor of EGFR tyrosine kinase with high selectivity for EGFR-sensitizing …
Formel:
C31H39N7O5S
Reinheit:
98.85%
Farbe und Form:
Solid
Molekulargewicht:
621.75
Ref: TM-T9865
1mg | 90,00 € | ||
5mg | 185,00 € | ||
10mg | 306,00 € | ||
25mg | 518,00 € | ||
50mg | 732,00 € | ||
100mg | 1.044,00 € | ||
500mg | 2.070,00 € | ||
1ml*10 (DMSO) | 270,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
(Rac)-JBJ-04-125-02
CAS:2140807-05-0
(Rac)-JBJ-04-125-02 (JBJ-04-125-02) is effective as a single agent in both in vitro and in vivo …
Formel:
C29H26FN5O3S
Reinheit:
95.85%
Farbe und Form:
Solid
Molekulargewicht:
543.61
Ref: TM-T8872
1mg | 103,00 € | ||
5mg | 212,00 € | ||
10mg | 346,00 € | ||
25mg | 585,00 € | ||
50mg | 832,00 € | ||
100mg | 1.133,00 € | ||
1ml*10 (DMSO) | 257,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024
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Mobocertinib
CAS:1847461-43-1
Mobocertinib (tak788) is a potent inhibitor of epidermal growth factor receptor (EGFR) and an antineoplastic …
Formel:
C32H39N7O4
Reinheit:
99.72%
Farbe und Form:
Solid
Molekulargewicht:
585.7
Ref: TM-T8151
5mg | 35,00 € | ||
10mg | 51,00 € | ||
25mg | 78,00 € | ||
50mg | 118,00 € | ||
100mg | 185,00 € | ||
500mg | 479,00 € | ||
1ml*10 (DMSO) | 52,00 € |
Voraussichtliche Lieferung in Vereinigte Staaten, am Montag 15. Juli 2024