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CAS 1000819-21-5

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  • GnRH-R antagonist-2

    CAS:
    GnRH-R antagonist-2 (Compound 44c) is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist, with IC50 values of 43 nM for rat and 88 nM for human GnRH-R. It is applicable in studies related to hormone-dependent diseases such as endometriosis, breast cancer, and prostate cancer[1].
    Fórmula:C37H50N4O3S
    Peso molecular:630.89

    Ref: TM-T213283

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