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Caspasa

Caspasa

Los inhibidores de caspasas son compuestos que bloquean la actividad de las caspasas, una familia de proteasas que son ejecutores centrales de la apoptosis. Las caspasas escinden sustratos específicos dentro de la célula para desencadenar el proceso apoptótico, lo que conduce a la muerte celular programada. Los inhibidores de caspasas se utilizan para estudiar los mecanismos de la apoptosis, así como para prevenir la muerte celular no deseada en varios modelos de investigación. Estos inhibidores también se exploran en contextos terapéuticos para proteger las células de la apoptosis en enfermedades como la neurodegeneración. En CymitQuimica, ofrecemos una amplia gama de inhibidores de caspasas de alta calidad para apoyar su investigación en apoptosis, muerte celular y campos relacionados.

Se han encontrado 125 productos de "Caspasa"

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  • Phenoxodiol

    CAS:
    <p>Phenoxodiol (Idronoxil) activates the mitochondrial caspase system, inhibits X-linked inhibitor of apoptosis(XIAP), disrupts FLICE inhibitory protein(FLIP)</p>
    Fórmula:C15H12O3
    Pureza:98.07%
    Forma y color:Solid
    Peso molecular:240.25
  • AVN-944

    CAS:
    <p>AVN-944 (VX-944)(VX-944) is a selective, noncompetitive inhibitor of human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.</p>
    Fórmula:C25H27N5O5
    Pureza:99.07% - ≥95%
    Forma y color:Solid
    Peso molecular:477.51
  • Taurodeoxycholic acid sodium hydrate

    CAS:
    <p>Taurodeoxycholic acid sodium hydrate (Sodium taurodeoxycholate monohydrate), a hydrophilic bile salt, on bile salt and biliary lipid secretion in the rat.</p>
    Fórmula:C26H46NNaO7S
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:539.70
  • 5,7-Dihydroxychromone

    CAS:
    <p>1.</p>
    Fórmula:C9H6O4
    Pureza:99.76% - ≥95%
    Forma y color:Solid
    Peso molecular:178.14
  • Boc-Asp(OMe)-fluoromethyl ketone

    CAS:
    <p>Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.</p>
    Fórmula:C11H18FNO5
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:263.26
  • Tauroursodeoxycholate sodium

    CAS:
    <p>Tauroursodeoxycholate sodium (TUDC) is an endoplasmic reticulum (ER) stress inhibitor, used for the treatment of gallstones and liver cirrhosis.</p>
    Fórmula:C26H44NNaO6S
    Pureza:97.90%
    Forma y color:Solid
    Peso molecular:521.69
  • Z-VAD-FMK

    CAS:
    <p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>
    Fórmula:C21H28FN3O7
    Pureza:98.24% - 99.79%
    Forma y color:Solid
    Peso molecular:453.46
  • (E/Z)-Necrosulfonamide

    CAS:
    <p>(E/Z)-Necrosulfonamide is a novel inhibitor of MLKL.</p>
    Fórmula:C18H15N5O6S2
    Pureza:97.62% - 98%
    Forma y color:Solid
    Peso molecular:461.47
  • Lobaplatin

    CAS:
    <p>Lobaplatin (D-19466) (D-19466) is a diastereometric mixture of platinum(II) complexe.</p>
    Fórmula:C9H18N2O3Pt
    Pureza:98.00%
    Forma y color:Solid
    Peso molecular:397.33
  • Z-DEVD-FMK

    CAS:
    <p>Z-DEVD-FMK (Caspase-3 Inhibitor) is a selective, irreversible Caspase-3 inhibitor, and also exhibits effective inhibition activity on caspase-6, caspase-7,</p>
    Fórmula:C30H41FN4O12
    Pureza:96.19% - 99.69%
    Forma y color:Solid
    Peso molecular:668.66
  • Arnicolide D

    CAS:
    <p>Arnicolide D is a sesquiterpene lactone.</p>
    Fórmula:C19H24O5
    Pureza:96.66%
    Forma y color:Solid
    Peso molecular:332.39
  • Dehydrocorydaline nitrate

    CAS:
    <p>DHC curbs antibody and cell-mediated allergies, inhibits mitochondrial potential in macrophages, and has antinociceptive, anti-inflammatory effects.</p>
    Fórmula:C22H24N2O7
    Pureza:99.79% - 99.92%
    Forma y color:Solid
    Peso molecular:428.44
  • Dehydrotrametenolic acid

    CAS:
    <p>Dehydrotrametenolic acid (Dehydroeburicoic acid) induces necrotic cell death that involves Ca(2+) overload, mitochondrial dysfunction, and calpain activation in</p>
    Fórmula:C31H48O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:468.71
  • Limonin glucoside

    CAS:
    <p>Limonin glucoside: a citrus compound, blocks HIV/HTLV-1, triggers cancer cell death, kills Aedes larvae.</p>
    Fórmula:C32H42O14
    Forma y color:Solid
    Peso molecular:650.674
  • Caspase-3-IN-1

    CAS:
    <p>Caspase-3-IN-1 is a potent inhibitor of Caspase-3 (IC50: 14.5 nM).</p>
    Fórmula:C26H25N3O6S
    Forma y color:Solid
    Peso molecular:507.56
  • Tigilanol tiglate

    CAS:
    <p>Tigilanol tiglate (EBC-46) is a PKC/C1 domain activator. Tigilanol tiglate induces immunogenic cell death and tumour regression.</p>
    Fórmula:C30H42O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:562.65
  • Anisperimus

    CAS:
    <p>Anisperimus (LF 15-0195) is an immunosuppressant that prevents CNS autoimmunity by promoting the development of regulatory CD4 T cells expressing Foxp3.</p>
    Fórmula:C18H39N7O3
    Pureza:98.10%
    Forma y color:Solid
    Peso molecular:401.55
  • AD-2646

    CAS:
    <p>AD-2646 has antidepressant activity and inhibits 2-deoxy-D-glucose (2-DG)-induced gastric acid secretion.</p>
    Fórmula:C23H40N2O4
    Forma y color:Solid
    Peso molecular:408.57
  • ZYZ-488

    CAS:
    <p>ZYZ-488 is an Apoptosis protease activating factor-1 (Apaf-1) inhibitor, which suppresses the activation of procaspase-9 and procaspase-3.</p>
    Fórmula:C20H29N3O11
    Pureza:99.04%
    Forma y color:Solid
    Peso molecular:487.46
  • Caspase-9 Inhibitor III

    CAS:
    <p>Caspase-9 Inhibitor III (Ac-LEHD-cmk) blocks caspase-9, protects against ischemic heart damage.</p>
    Fórmula:C24H35ClN6O9
    Forma y color:Solid
    Peso molecular:587.02