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Integrin

Integrin

Los inhibidores de integrinas se dirigen a las integrinas, una familia de receptores en la superficie celular que desempeñan un papel crucial en la adhesión celular, la migración y la transducción de señales. Las integrinas están involucradas en la regulación del ciclo celular, particularmente en procesos como la división y la diferenciación celular. Inhibir las integrinas puede interrumpir estos procesos, lo que lleva al arresto del ciclo celular y la apoptosis, lo que hace que estos inhibidores sean valiosos en la investigación del cáncer y el estudio de la metástasis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de integrinas de alta calidad para apoyar su investigación en la regulación del ciclo celular, la biología del cáncer y el desarrollo terapéutico.

Se han encontrado 224 productos de "Integrin"

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  • A-205804

    CAS:
    <p>A-205804 is a specific and effective inhibitor of E-selectin( IC50=20 nM ) and ICAM-1(IC50=25 nM) expression.</p>
    Fórmula:C15H12N2OS2
    Pureza:98.07% - 98.52%
    Forma y color:Solid
    Peso molecular:300.4
  • Cyclo(-RGDfK)

    CAS:
    <p>Cyclo(-RGDfK) is a selective and potent inhibitor of integrin αvβ3 with an IC50 value of 0.94 nM.Cost-effective and quality-assured.</p>
    Fórmula:C27H41N9O7
    Pureza:95.29% - >99.99%
    Forma y color:Solid
    Peso molecular:603.67
  • PND-1186

    CAS:
    <p>PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).</p>
    Fórmula:C25H26F3N5O3
    Pureza:99.14% - 99.75%
    Forma y color:Solid
    Peso molecular:501.5
  • GLPG0187

    CAS:
    <p>GLPG0187, a broad spectrum integrin receptor antagonist, inhibits αvβ1-integrin (IC50: 1.3 nM).</p>
    Fórmula:C29H37N7O5S
    Pureza:99.4% - 99.70%
    Forma y color:Solid
    Peso molecular:595.71
  • OSU-T315

    CAS:
    <p>OSU-T315 (OSU-T315 (1,5-regioisomer)) (1,5-regioisomer) is a ILK inhibitor.</p>
    Fórmula:C30H30F3N5O
    Pureza:98.69%
    Forma y color:Solid
    Peso molecular:533.59
  • Arginine-glycine-aspartic acid

    CAS:
    <p>RGD (RGD (Arg-Gly-Asp) Peptides) (Arg-Gly-Asp) Peptides is a cell adhesion motif which can mimic cell adhesion proteins and bind to integrins.</p>
    Fórmula:C12H22N6O6
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:346.34
  • Cyclo(RADfK)

    CAS:
    <p>Cyclo(RADfK) is a selective α(v)β(3) integrin ligand used in neoangiogenesis research, therapy, and diagnostics; it's a control for RGD peptides.</p>
    Fórmula:C28H43N9O7
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:617.7
  • Cyclo(-RGDfK) TFA

    CAS:
    <p>Cyclo(-RGDfK) is a selective αvβ3 integrin inhibitor(IC50 : 0.94 nM).</p>
    Fórmula:C29H42F3N9O9
    Pureza:98.99% - 99.54%
    Forma y color:Solid
    Peso molecular:717.69
  • CWHM-12

    CAS:
    <p>CWHM-12 is a potent inhibitor of αV integrins (IC50s of 0.2/0.8/1.5/1.8 nM for αvβ8/αvβ3/αvβ6/αvβ1).</p>
    Fórmula:C26H32BrN5O6
    Pureza:98.05% - 99.83%
    Forma y color:Solid
    Peso molecular:590.47
  • H-Gly-Arg-Gly-Asp-Asn-Pro-OH

    CAS:
    <p>RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.</p>
    Fórmula:C23H38N10O10
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:614.61
  • iRGD peptide

    CAS:
    <p>iRGD peptide: 9-amino acid cyclic compound (CRGDKGPDC), found through phage display in mice with tumors.</p>
    Fórmula:C35H57N13O14S2
    Pureza:98.77%
    Forma y color:Solid
    Peso molecular:948.04
  • Leukadherin-1

    CAS:
    <p>Leukadherin-1 boosts CD11b/CD18 adhesion, lowers leukocyte movement, cuts inflammation.</p>
    Fórmula:C22H15NO4S2
    Pureza:98.49% - 98.93%
    Forma y color:Solid
    Peso molecular:421.49
  • Pyrintegrin

    CAS:
    <p>Pyrintegrin: β1-integrin agonist, boosts embryonic stem cell survival, and podocyte protection, improves cell-matrix adhesion.</p>
    Fórmula:C23H25N5O3S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:451.54
  • Orbofiban

    CAS:
    <p>Orbofiban, an orally administered antagonist of the platelet GPIIb/IIIa receptor, effectively inhibits platelet aggregation.</p>
    Fórmula:C17H23N5O4
    Forma y color:Solid
    Peso molecular:361.4
  • Cucurbitacin B

    CAS:
    <p>Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells.</p>
    Fórmula:C32H46O8
    Pureza:97.1% - 99.33%
    Forma y color:Solid
    Peso molecular:558.7
  • ILK-IN-2

    CAS:
    <p>ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.</p>
    Fórmula:C30H30F3N5O
    Pureza:99.30%
    Forma y color:Solid
    Peso molecular:533.59
  • A-286982

    CAS:
    <p>A 286982 blocks the LFA-1 and ICAM-1 integrin-ligand interaction.</p>
    Fórmula:C24H27N3O4S
    Pureza:97.81%
    Forma y color:Solid
    Peso molecular:453.55
  • Arg-Gly-Asp TFA (99896-85-2(free base))


    <p>Arg-Gly-Asp TFA (RGD, 99896-85-2) is a tripeptide that promotes cell adhesion and integrin binding.</p>
    Fórmula:C14H23F3N6O8
    Pureza:99.2% - ≥98%
    Forma y color:Solid
    Peso molecular:460.36
  • roxifiban

    CAS:
    <p>Roxifiban, a prodrug of XV459, is an antiplatelet agent with high affinity and specificity for platelet glycoprotein IIb/IIIa complex(GPIIb/IIIa) receptors.</p>
    Fórmula:C21H29N5O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:447.48
  • LXW7

    CAS:
    <p>LXW7 is an octamer disulfide cyclic peptide and αvβ3 integrin ligand, acts as a potent and specific endothelial progenitor cells (EPCs) and endothelial cells (</p>
    Fórmula:C29H48N12O12S2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:820.89
  • Natalizumab

    CAS:
    <p>Natalizumab used for the treatment of relapsing remitting multiple sclerosis and Crohn's disease.</p>
    Pureza:98.00%
    Forma y color:Liquid
    Peso molecular:N/A
  • Lifitegrast

    CAS:
    <p>Lifitegrast (SAR 1118) is a lymphocyte, function-associated antigen-1 antagonist.</p>
    Fórmula:C29H24Cl2N2O7S
    Pureza:99.39% - 99.66%
    Forma y color:Solid
    Peso molecular:615.48
  • Irigenin

    CAS:
    <p>Irigenin mediates its antimetastatic effect by specifically and selectively blocking the α9β1 and α4β1 integrin binding sites on the C-C loop of the Extra</p>
    Fórmula:C18H16O8
    Pureza:99.50% - 99.85%
    Forma y color:Solid
    Peso molecular:360.31
  • Carotegrast methyl

    CAS:
    <p>Carotegrast methyl (AJM300), an orally-active small molecule, can antagonize the α4 integrin receptor. It is a specific and dual α4β1/α4β7 integrin antagonist.</p>
    Fórmula:C28H26Cl2N4O5
    Pureza:99.26% - 99.72%
    Forma y color:Solid
    Peso molecular:569.44
  • Tirofiban hydrochloride monohydrate

    CAS:
    <p>Tirofiban(MK383) hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>
    Fórmula:C22H39ClN2O6S
    Pureza:98.81% - >99.99%
    Forma y color:White Solid
    Peso molecular:495.07
  • E7820

    CAS:
    <p>E7820 (ER68203-00) is an angiogenesis inhibitor by suppressing integrin a2 (a cell adhesion molecule expressed on endothelial cells).</p>
    Fórmula:C17H12N4O2S
    Pureza:98.31% - 99.11%
    Forma y color:Solid
    Peso molecular:336.37
  • ILK-IN-3

    CAS:
    <p>ILK-IN-3 is an inhibitor of integrin linked kinase, and with antitumor activity.</p>
    Fórmula:C10H12N6O
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:232.24
  • Cyclo(RGDyK) trifluoroacetate

    CAS:
    <p>Cyclo(RGDyK) trifluoroacetate is a potent and selective αVβ3 integrin inhibitor with IC50 of 20 nM.</p>
    Fórmula:C31H43F6N9O12
    Pureza:95.28% - ≥95%
    Forma y color:Solid
    Peso molecular:847.72
  • TR-14035

    CAS:
    <p>TR-14035 (MDK-1191) is a dual antagonist of α4β7/α4β1 integrins (IC50s: 7/87nM).</p>
    Fórmula:C24H21Cl2NO5
    Pureza:98.98%
    Forma y color:Solid
    Peso molecular:474.33
  • BIO-1211

    CAS:
    <p>BIO-1211 is a more potent inhibitor of α4β1 (VLA-4, IC50 = 4 nM) over α4β7(IC50 = 2 μM).</p>
    Fórmula:C36H48N6O9
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:708.8
  • Eptifibatide acetate (148031-34-9 free base)

    CAS:
    <p>Eptifibatide acetate (148031-34-9), a cyclic heptapeptide GP IIb/IIIa inhibitor antiplatelet drug.</p>
    Fórmula:C35H49N11O9S2·xC2H4O2
    Pureza:99.7% - 99.87%
    Forma y color:Solid
    Peso molecular:831.96 (free base)
  • GPRP acetate (67869-62-9 free base)

    CAS:
    <p>GPRP acetate (Pefabloc FG) is fibrinogen-related peptides, which inhibit the interaction of fibrinogen with the platelet membrane glycoprotein IIbIIIa complex.</p>
    Fórmula:C20H35N7O7
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:485.53
  • Bexotegrast

    CAS:
    <p>Bexotegrast (PLN-74809) is an αvβ6 and αvβ1 integrin inhibitor with antifibrotic properties for the study of idiopathic pulmonary fibrosis (IPF).</p>
    Fórmula:C27H36N6O3
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:492.61
  • Etaracizumab

    CAS:
    <p>Etaracizumab (LM 609) is a humanized monoclonal antibody targeting integrin αvβ3, inhibiting angiogenesis and melanoma growth, used in the study of melanoma.</p>
    Pureza:96.77% (SEC-HPLC) - 99.32% (SEC-HPLC)
    Forma y color:Liquid
    Peso molecular:144.3 (kDa)
  • Muromonab

    CAS:
    <p>Muromonab (OKT3) is a mouse-derived antibody targeting the CD3 receptor, blocking all cytotoxic T cell functions.</p>
    Pureza:95% - 97.51% (SEC-HPLC)
    Forma y color:Liquid
  • RO0270608

    CAS:
    <p>RO0270608 is an α4β1/α4β7 integrin antagonist with anti-inflammatory activity for the study of allergic inflammatory responses.</p>
    Fórmula:C24H19Cl3N2O4
    Pureza:98.26%
    Forma y color:Solid
    Peso molecular:505.78
  • Voxalatamab

    CAS:
    <p>Voxalatamab (JNJ-63898081), an IgG4 bispecific antibody targeting PSMA and CD3, demonstrates anti-cancer efficacy in prostate cancer research [1].</p>
    Forma y color:Liquid
  • Rovelizumab

    CAS:
    <p>Rovelizumab: humanized anti-CD11/CD18 antibody for MS, hemorrhagic shock, MI, and stroke research.</p>
    Forma y color:Liquid
  • Vepsitamab

    CAS:
    <p>Vepsitamab (AMG 199), an anti-MUC17/CD3 BiTE, targets T cells and tumors for cell lysis and T cell activation.</p>
    Forma y color:Liquid
  • Cevostamab

    CAS:
    <p>Cevostamab (BFCR4350A, RG6160, RO7187797) is a humanized BsAb IgG1 targeting FcRH5 on MM cells and CD3 on T cells to enhance T-cell-mediated MM cell killing.</p>
    Forma y color:Liquid
  • Pavurutamab

    CAS:
    <p>Pavurutamab (AMG-701) is a bispecific T cell engager targeting CD3 and BCMA with extended half-life, designed to treat MM.</p>
    Forma y color:Liquid
  • Enlimomab

    CAS:
    <p>Enlimomab (BI-RR 0001), a mouse IgG2a antibody, blocks leukocyte binding to ICAM-1, reducing inflammation and used in stroke research.</p>
    Forma y color:Liquid
  • Anti-Mouse IL-1a Antibody (ALF-161)


    <p>Anti-Mouse IL-1a Antibody is an IgG1 subtype inhibitor specific to mouse IL-1a, derived from the Armenian Hamster.</p>
    Pureza:98%
    Forma y color:Odour Liquid
  • Pasotuxizumab

    CAS:
    <p>Pasotuxizumab (BAY 2010112) is a BiTE that targets PSMA &amp; CD3 with K D s 47.0 &amp; 9.4 nM, for mCRPC research.</p>
    Forma y color:Liquid
  • Ubamatamab

    CAS:
    <p>Ubamatamab (REGN4018), a human bispecific antibody targeting Mucin 16 (MUC16) and CD3, exhibits potent antitumor activity [1].</p>
    Forma y color:Liquid
  • Vatelizumab

    CAS:
    <p>Vatelizumab is a humanised monoclonal antibody targeting Integrin α2β1 ( VLA-2, CD49b), which enhances the frequency of regulatory T cells multiple sclerosis.</p>
    Pureza:95%
    Forma y color:Liquid
  • Tepoditamab

    CAS:
    <p>Tepoditamab (MCLA-117) is a bispecific antibody targeting CLEC12A and CD3, inducing T cell lysis of AML cells.</p>
    Forma y color:Liquid
  • Vonsetamig

    CAS:
    <p>Vonsetamig, a humanized immunoglobulin G4-kappa monoclonal antibody, targets both TNFRSF17 and CD3E. It serves as an antineoplastic agent.</p>
    Forma y color:Liquid
  • Flotetuzumab

    CAS:
    <p>Flotetuzumab (MGD006/S80880) is a CD123/CD3 bispecific DART antibody, reactivating T-cells for AML treatment.</p>
    Forma y color:Liquid
  • Linvoseltamab

    CAS:
    <p>Linvoseltamab, a bispecific antibody, targets both BCMA (TNFRSF17) and CD3 epsilon, demonstrating a favorable safety profile and promising efficacy in relapsed/</p>
    Forma y color:Liquid
  • Vibecotamab

    CAS:
    <p>Vibecotamab, a bispecific antibody, targets CD123/CD3 for T-cell killing of tumors, promising for acute myeloid leukemia.</p>
    Forma y color:Liquid
  • Obrindatamab

    CAS:
    <p>Obrindatamab: a humanized bispecific antibody targeting B7-H3/CD3, enhances CTL-mediated cancer cell killing.</p>
    Forma y color:Liquid
  • Pacanalotamab

    CAS:
    <p>Pacanalotamab (AMG 420/BI-836909), a BiTE, directs T-cells to BCMA+ MM cells, causing lysis.</p>
    Forma y color:Liquid
  • OS-2966


    <p>OS-2966 is a humanised de-immunised monoclonal antibody that target Integrin b1/ITGB1/CD29, malignant gliomas, glioblastomas, and astrocytomas.</p>
    Pureza:95%
    Forma y color:Odour Liquid
  • Anti-Mouse CD3ε Antibody (145-2C11)


    <p>Anti-Mouse CD3ε Antibody (145-2C11) is an antibody inhibitor targeting CD3ε in Armenian hamsters, in TCR formation and in T lymphocyte activation</p>
    Pureza:99%
    Forma y color:Odour Liquid
  • Gresonitamab

    CAS:
    <p>Gresonitamab (AMG 910) is an HLE BiTE antibody targeting CD3+ T cells and CLDN18.2+ tumors, for adenocarcinoma research.</p>
    Forma y color:Liquid
  • SB273005

    CAS:
    <p>SB273005 is a potent integrin inhibitor with Ki of 1.2 nM and 0.3 nM for αvβ3 receptor and αvβ5 receptor, respectively.</p>
    Fórmula:C22H24F3N3O4
    Pureza:99.58%
    Forma y color:Solid
    Peso molecular:451.44
  • Tirofiban

    CAS:
    <p>Tirofiban (L700462) (MK-383) is a selective palate GPIIb/IIIa antagonist which inhibits platelet aggregation with IC50 of 9 nM.</p>
    Fórmula:C22H36N2O5S
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:440.6
  • GR 144053 trihydrochloride

    CAS:
    <p>platelet fibrinogen receptor glycoprotein IIb/IIIa (GpIIb/IIIa) antagonist</p>
    Fórmula:C18H30Cl3N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:454.82
  • Sibrafiban

    CAS:
    <p>Sibrafiban (RO 48-3657), an oral, nonpeptide prodrug, inhibits platelet aggregation as a selective IIb/IIIa antagonist.</p>
    Fórmula:C20H28N4O6
    Forma y color:Solid
    Peso molecular:420.46
  • UR-3216

    CAS:
    <p>UR-3216 is a prodrug, selectively antagonizing GPIIb/IIIa receptors orally, with its active form, UR-2992, binding tightly to platelets.</p>
    Fórmula:C27H29N7O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:563.56
  • L 703014

    CAS:
    <p>L 703014 is an antagonist of the fibrinogen receptor.</p>
    Fórmula:C24H34N4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:442.55
  • Balamapimod

    CAS:
    <p>Balamapimod is a reversible inhibitor of Ras/Raf/MEK. It also has a potential anti-tumor activity.</p>
    Fórmula:C30H32ClN7OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:574.14
  • BMS-587101

    CAS:
    <p>BMS-587101 is a small molecule antagonist of LFA-1, which can reduce inflammation and joint destruction in the mouse model of arthritis.</p>
    Fórmula:C26H20Cl2N4O4S
    Forma y color:Solid
    Peso molecular:555.43
  • BMS-688521

    CAS:
    <p>BMS-688521 is an LFA-1/ICAM interaction inhibitor, a small molecule antagonist of LFA-1 with potential anti-inflammatory activity.</p>
    Fórmula:C26H19Cl2N5O4
    Pureza:98.87%
    Forma y color:Solid
    Peso molecular:536.37
  • MK-0668

    CAS:
    <p>MK-0668 is a very potent and orally active very late antigen-4 antagonist.</p>
    Fórmula:C31H30Cl2N6O6S
    Forma y color:Solid
    Peso molecular:685.58
  • NSC47924

    CAS:
    <p>NSC47924 is a laminin receptor (LR) inhibitor.</p>
    Fórmula:C18H17NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:279.33
  • Zalunfiban

    CAS:
    <p>RUC-4 is an aIIb 3 antagonist. It is also used for prehospital therapy of myocardial infarction.</p>
    Fórmula:C16H18N8O2S
    Forma y color:Solid
    Peso molecular:386.43
  • TCS 2314

    CAS:
    <p>TCS 2314 is an orally active and selective very late antigen-4 antagonist (IC50: 4.4 nM).</p>
    Fórmula:C28H34N4O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:522.59
  • Chrysotobibenzyl

    CAS:
    <p>Chrysotobibenzyl from Dendrobium pulchellum stems may trigger cell death in detached cells and hinder lung cancer growth.</p>
    Fórmula:C19H24O5
    Forma y color:Solid
    Peso molecular:332.39
  • αvβ1 integrin-IN-1 TFA (1689540-62-2 free base)


    <p>αvβ1 integrin-IN-1 TFA is an effective and selective αvβ1 integrin inhibitor (IC50: 0.63 nM).</p>
    Fórmula:C28H35F3N6O8S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:672.67
  • Zaurategrast ethyl ester sulfate

    CAS:
    <p>Zaurategrast ethyl ester sulfate is a α4β1/α4β7 integrin antagonist, and used for the treatment of inflammatory and autoimmune disorders.</p>
    Fórmula:C56H60Br2N8O10S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1197.01
  • RUC-1

    CAS:
    <p>RUC-1 is an αIIbβ3-selective ADP-induced platelet aggregation inhibitor.</p>
    Fórmula:C11H15N5OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:265.33
  • Zaurategrast ethyl ester

    CAS:
    <p>Zaurategrast ethyl ester, an α4β1/α4β7 integrin antagonist prodrug of CT7758, treats inflammatory/autoimmune conditions.</p>
    Fórmula:C28H29BrN4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:549.46
  • IMB-10

    CAS:
    <p>IMB-10 is an alphaMbeta2 integrin modulator, inhibiting leukocyte migration and recruitment in vitro and in vivo.</p>
    Fórmula:C19H15NOS2
    Forma y color:Solid
    Peso molecular:337.46
  • Ro 43-5054

    CAS:
    <p>Ro 43-5054 is a small molecular, noncyclic peptidomimetic inhibitor.</p>
    Fórmula:C24H27N5O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:497.5
  • BOP sodium

    CAS:
    <p>BOP sodium salt is an inhibitor of alpha9beta1 and alpha4beta1 integrin.</p>
    Fórmula:C25H29N3NaO7S
    Forma y color:Solid
    Peso molecular:538.57
  • GSK-3008348

    CAS:
    <p>GSK-3008348 is an antagonist of integrin alpha(v)beta6.</p>
    Fórmula:C29H37N5O2
    Pureza:99.547%
    Forma y color:Solid
    Peso molecular:487.64
  • Valategrast

    CAS:
    <p>Valategrast: potent, oral dual α4β1/α4β7 integrin antagonist, may treat COPD and asthma.</p>
    Fórmula:C30H32Cl3N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:604.95
  • Valategrast hydrochloride

    CAS:
    <p>Valategrast hydrochloride (R411), a dual antagonist of integrin α4β1 (VLA-4), is used for the potential treatment of asthma.</p>
    Fórmula:C30H33Cl4N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:641.41
  • CLT-28643

    CAS:
    <p>CLT-28643 is a specific α5β1-Integrin inhibitor that prevents fibrosis in GFS, inhibits tumor growth and angiogenesis, suppresses fibrosis and inflammation.</p>
    Fórmula:C19H17N3O4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:351.36
  • Integrin-IN-2

    CAS:
    <p>Integrin-IN-2, an oral αv integrin blocker, enhances αvβ6/3/5/8 affinities with pIC50s: 7.8/8.4/8.4/7.4.</p>
    Fórmula:C27H30N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:458.55
  • XVA143

    CAS:
    <p>XVA143, an α/β I-like allosteric antagonist, blocks LFA-1 adhesion and combats P. gingivalis in mice, preventing bone loss.</p>
    Fórmula:C25H21Cl2N3O8
    Forma y color:Solid
    Peso molecular:562.36
  • Integrin modulator 1

    CAS:
    <p>Integrin modulator 1 is a selective α4β1 integrin agonist (IC50 9.8 nM) that enhances adhesion with EC50 12.9 nM, aiding integrin-dependent studies.</p>
    Fórmula:C13H14N2O4
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:262.26
  • Firategrast

    CAS:
    <p>Firategrast (SB 683699) is an orally active and specific α4β1/α4β7 integrin antagonist.Firategrast reduces the transport of lymphocytes into the central nervous</p>
    Fórmula:C27H27F2NO6
    Pureza:99.16%
    Forma y color:Solid
    Peso molecular:499.5
  • Elarofiban

    CAS:
    <p>Elarofiban(RWJ-53308) is a novel and orally active GPIIb/IIIa antagonist.</p>
    Fórmula:C22H32N4O4
    Pureza:98.76%
    Forma y color:Solid
    Peso molecular:416.51
  • 3-Hydroxyxanthone

    CAS:
    <p>3-Hydroxyxanthone (3-Hydroxy-xanthen-9-one), a xanthone derivative, exhibits inhibitory effects on NADPH-catalyzed lipid peroxidation in human umbilical vein</p>
    Fórmula:C13H8O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:212.2
  • ICAM-1-IN-1

    CAS:
    <p>ICAM-1-IN-1 is a potent and selective E-selectin(IC50 = 7 nM) and ICAM-1(IC50 = 5 nM) inhibitor.</p>
    Fórmula:C15H11BrN2O2S
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:363.23
  • BI-1950

    CAS:
    <p>BI-1950: potent inhibitor of LFA-1, key in immune function and drug target.</p>
    Fórmula:C32H26Cl2FN7O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:646.5
  • Teclistamab

    CAS:
    <p>Teclistamab(JNJ-64007957) is a human bispecific monoclonal antibody targeting the CD3 receptor on t-cells and the BCMA for relapsed and refractory multiple myeloma.</p>
    Pureza:95%
    Forma y color:Liquid
  • Synstatin (92-119)

    CAS:
    <p>Synstatin (92-119) serves as an anti-tumor agent by suppressing angiogenesis and cancer cell invasion, chiefly through the down-regulation of integrin αvβ3 and</p>
    Fórmula:C133H207N35O46
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3032.27
  • TAK 029

    CAS:
    <p>TAK 029 is a local glycoprotein IIb/IIIa receptor inhibitor.</p>
    Fórmula:C19H23N5O7
    Forma y color:Solid
    Peso molecular:433.42
  • αvβ6 integrin inhibitor 2

    CAS:
    <p>αvβ6 Integrin Inhibitor 2 is a potent inhibitor of αvβ6 integrin, demonstrating an inhibition concentration (IC50) of 96.5 nM.</p>
    Fórmula:C21H30N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:386.49
  • Lotrafiban

    CAS:
    <p>Lotrafiban: Oral GP IIb/IIIa inhibitor for treating coronary and cerebrovascular disease.</p>
    Fórmula:C23H32N4O4
    Forma y color:Solid
    Peso molecular:428.52
  • JNJ-26076713

    CAS:
    <p>JNJ-26076713, an oral alpha V integrin blocker, may treat macular edema, AMD, and diabetic retinopathy.</p>
    Fórmula:C29H38N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:490.64
  • SB-267268

    CAS:
    <p>SB-267268: αvβ3 inhibitor (IC50: 0.68 nM human, 0.29 nM mouse), blocks αvβ3/αvβ5 integrins (Ki: 0.9 nM human, 0.5 nM monkey αvβ3, 0.7 nM human αvβ5).</p>
    Fórmula:C22H24F3N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:451.44
  • Zaurategrast

    CAS:
    <p>Zaurategrast is an effective and oral-effective inhibitor of the α4-integrin.</p>
    Fórmula:C26H25BrN4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:521.41
  • Solitomab

    CAS:
    <p>Solitomab (AMG 110) is a bispecific antibody targeting CD3 and EpCAM, used in uterine/ovarian carcinosarcoma research.</p>
    Forma y color:Liquid
  • Carotegrast

    CAS:
    <p>Carotegrast, an orally available α4 integrin receptor inhibitor, has anti-inflammatories activities.</p>
    Fórmula:C27H24Cl2N4O5
    Forma y color:Solid
    Peso molecular:555.41
  • Tirofiban HCl

    CAS:
    <p>Tirofiban HCl is an antagonist of platelet glycoprotein-IIb/IIIa receptor.</p>
    Fórmula:C22H37ClN2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:477.06