
c-Myc
Los inhibidores de c-Myc se dirigen a la proteína c-Myc, un factor de transcripción que juega un papel crucial en el crecimiento celular, la proliferación y la apoptosis. c-Myc regula la expresión de numerosos genes involucrados en el ciclo celular y a menudo está sobreexpresado en varios tipos de cáncer, lo que lleva a una proliferación celular descontrolada y al crecimiento tumoral. Inhibir c-Myc puede interrumpir estos procesos, induciendo el arresto del ciclo celular y la apoptosis en células cancerosas. Los inhibidores de c-Myc son herramientas importantes en la investigación del cáncer y el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de c-Myc de alta calidad para apoyar su investigación en oncología, regulación del ciclo celular y control transcripcional.
Se han encontrado 69 productos de "c-Myc"
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NNK
CAS:<p>NNK is a procarcinogen and a major tobacco-specific toxicant. It inhibits the expression of lysyl oxidase which is a tumor suppressor.Cost-effective and quality-assured.</p>Fórmula:C10H13N3O2Pureza:99.63% - 99.92%Forma y color:SolidPeso molecular:207.23Lusianthridin
CAS:<p>Lusianthridin is a natural product from Dendrobium venustum.</p>Fórmula:C15H14O3Pureza:98.49%Forma y color:SolidPeso molecular:242.27Agrimol B
CAS:<p>1. Agrimol B is a main active ingredient isolated from Agrimonia pilosa Ledeb.</p>Fórmula:C37H46O12Pureza:99.06% - ≥95%Forma y color:SolidPeso molecular:682.7510058-F4
CAS:<p>10058-F4 inhibits c-Myc-Max, blocking c-Myc target gene activation, causing cell-cycle arrest & apoptosis.</p>Fórmula:C12H11NOS2Pureza:98% - 99.87%Forma y color:SolidPeso molecular:249.35APTO-253 HCl
CAS:<p>APTO-253 (LOR-253/LT-253) is a small-molecule MTF-1 inhibitor with antitumor properties, reducing cyclin D1, hypoxia, and angiogenesis gene expression.</p>Fórmula:C22H15ClFN5Forma y color:SolidPeso molecular:403.8410074-A4
CAS:<p>10074-A4 is a c-Myc binding compound that associates with c-Myc370–409 and behaves like a “ligand cloud” around a “protein cloud”, with distinct features from</p>Fórmula:C18H14Cl2N2O3SPureza:99.06%Forma y color:SolidPeso molecular:409.29Artemisitene
CAS:<p>Artemisitene, an oxidized antimalarial derivative of Artemisinin, stems from precursors like Artemisinin B and Artemisinic acid.</p>Fórmula:C15H20O5Pureza:99.58%Forma y color:SolidPeso molecular:280.32NY2267
CAS:<p>NY2267 (Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl</p>Fórmula:C38H43N3O6Pureza:99.16% - 99.27%Forma y color:SolidPeso molecular:637.76Idarubicin hydrochloride
CAS:<p>Idarubicin hydrochloride (Zavedos), a hydrochloride salt form of Idarubicin, is a DNA topoisomerase II (topo II) inhibitor for MCF-7 cells ( IC50: 3.3 ng/mL).</p>Fórmula:C26H27NO9·HClPureza:98.91% - 99.96%Forma y color:SolidPeso molecular:533.95BTYNB
CAS:<p>BTYNB (MDK6620) is an inhibitor of the oncofetal mRNA-binding protein IMP1. MDK6620 downregulates β-TrCP1 mRNA and reduces activation of NF-κB.</p>Fórmula:C12H9BrN2OSPureza:≥95%Forma y color:SolidPeso molecular:309.18EN4
CAS:<p>EN4 (EN4 MYC inhibitor) MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC.</p>Fórmula:C25H24N2O4Pureza:98.51%Forma y color:SolidPeso molecular:416.47PARL Protein, Human, Recombinant (Myc)
<p>Required for the control of apoptosis during postnatal growth.</p>Forma y color:Lyophilized PowderPeso molecular:37.8 kDa (predicted)ACOX1 Protein, Mouse, Recombinant (Myc)
<p>Catalyzes the desaturation of acyl-CoAs to 2-trans-enoyl-CoAs.</p>Forma y color:Lyophilized PowderPeso molecular:76.2 kDa (predicted)2-5A-dependent Rnase Protein, Human, Recombinant (Myc)
<p>2-5A-dependent Rnase Protein, Human, Recombinant (Myc) is expressed in E.</p>Pureza:85% - 85%Forma y color:Lyophilized PowderPeso molecular:85.1 kDa (predicted)c-Myc inhibitor 9
CAS:<p>c-Myc inhibitor 9 (compound 332) with logEC50 ≥6, suppresses tumors in mice, useful for cancer research.</p>Fórmula:C27H31N5OSForma y color:SolidPeso molecular:473.63RK-9123016
CAS:<p>RK-9123016 is a SIRT2 inhibitor.</p>Fórmula:C16H18N6O3SPureza:99.65%Forma y color:SolidPeso molecular:374.42FUBP1-IN-2
CAS:<p>FUBP1-IN-2 hinders FUBP1, affects c-Myc and p21 expression, and depletes polyamines.</p>Fórmula:C26H26ClN3O4Forma y color:SolidPeso molecular:479.96KSI-3716
CAS:<p>KSI-3716 is a c-Myc inhibitor, a bladder chemotherapy agent that blocks the formation of complexes between c-MYC/MAX and target gene promoters.</p>Fórmula:C17H11BrCl2N2O2Pureza:98.94%Forma y color:SolidPeso molecular:426.09BI8622
CAS:<p>BI8622 is a HUWE1 antagonist that restores levels of RP2 mutants in retinal cell lines and inhibits cellular activation of NLRP3 and AIM2 inflammatory vesicles.</p>Fórmula:C25H26N6OPureza:98.28%Forma y color:SolidPeso molecular:426.51VPC-70619
CAS:<p>VPC-70619: Oral, selective N-Myc inhibitor; blocks cancer growth by hindering N-Myc-Max/DNA binding; well-absorbed.</p>Fórmula:C16H8ClF3N4OForma y color:SolidPeso molecular:364.71
