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Cromatina / Epigenética

Cromatina / Epigenética

Los inhibidores de cromatina/epigenética son compuestos que modulan la estructura y función de la cromatina o interfieren con modificaciones epigenéticas, como la metilación del ADN y la modificación de histonas. Estos inhibidores son herramientas esenciales para estudiar la regulación de la expresión génica y el papel de la epigenética en enfermedades como el cáncer, los trastornos neurológicos y las anomalías del desarrollo. Al dirigirse a los procesos epigenéticos, estos inhibidores pueden alterar los patrones de expresión génica y ofrecer nuevas vías terapéuticas. En CymitQuimica, ofrecemos una amplia selección de inhibidores de cromatina/epigenética de alta calidad para apoyar su investigación en biología molecular, genética y epigenética.

Subcategorías de "Cromatina / Epigenética"

Se han encontrado 2242 productos de "Cromatina / Epigenética"

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  • Anti-PARP1 Antibody (8I163)


    <p>Anti-PARP1 Antibody (8I163) is a Mouse antibody targeting PARP1. Anti-PARP1 Antibody (8I163) can be used in IHC-P.</p>
    Forma y color:Odour Liquid
  • Anti-PARP Antibody (1W26)


    <p>Anti-PARP Antibody (1W26) is a Mouse antibody targeting PARP. Anti-PARP Antibody (1W26) can be used in WB,IHC-P,IP.</p>
    Forma y color:Odour Liquid
  • Anti-PARP1 Antibody (6I459)


    <p>Anti-PARP1 Antibody (6I459) is an antibody targeting PARP1. Anti-PARP1 Antibody (6I459) can be used in ELISA, IHC.</p>
    Forma y color:Odour Liquid
  • Anti-PARP1 Antibody (7A800)


    <p>Anti-PARP1 Antibody (7A800) is an antibody targeting PARP1. Anti-PARP1 Antibody (7A800) can be used in ELISA, WB, IHC.</p>
    Forma y color:Odour Liquid
  • Anti-PARP1 Antibody (9E313)


    <p>Anti-PARP1 Antibody (9E313) is a Mouse antibody targeting PARP1. Anti-PARP1 Antibody (9E313) can be used in IHC-P.</p>
    Forma y color:Odour Liquid
  • Anti-PARP1 Antibody (8S756)


    <p>Anti-PARP1 Antibody (8S756) is an antibody targeting PARP1. Anti-PARP1 Antibody (8S756) can be used in ELISA, WB, IHC, IF, FCM.</p>
    Forma y color:Odour Liquid
  • Gintemetostat

    CAS:
    <p>Gintemetostat (KTX-1001) is a potent NSD2 inhibitor (IC50=0.001-0.01μM) for treating NSD2-dysregulated cancers.</p>
    Fórmula:C25H26F4N8O2
    Forma y color:Solid
    Peso molecular:546.52
  • PROTAC PARP1 degrader

    CAS:
    <p>PROTAC PARP1 degrader suppresses MDA-MB-231 cells at 10 μM, IC50: 6.12 μM in 24h.</p>
    Fórmula:C58H63Cl2N11O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1145.1
  • 7-Chloro-4-(piperazin-1-yl)quinoline

    CAS:
    <p>7-Cl-4-(piperazin-1-yl)quinolone: sirtuin inhibitor, serotonin uptake blocker, antimalarial (D10 IC50 1.18µM, K1 IC50 0.97µM).</p>
    Fórmula:C13H14ClN3
    Pureza:99.52%
    Forma y color:Light Yellow Solid
    Peso molecular:247.72
  • I-BET567

    CAS:
    <p>I-BET567: potent, oral pan-BET inhibitor; pIC50s: 6.9 (BRD4 BD1), 7.2 (BD2); effective in mouse cancer and inflammation models.</p>
    Fórmula:C17H18ClN5O2
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:359.81
  • AMI-1 free acid

    CAS:
    <p>AMI-1: Potent reversible PRMT inhibitor; IC50: 8.8 μM (hPRMT1), 3.0 μM (yeast-Hmt1p); blocks substrate binding.</p>
    Fórmula:C21H16N2O9S2
    Pureza:97.8%
    Forma y color:Solid
    Peso molecular:504.49
  • PR5-LL-CM01

    CAS:
    <p>PR5-LL-CM01 is a novel protein arginine methyltransferase 5 (PRMT5) inhibitor in colorectal and pancreatic cancers.</p>
    Fórmula:C23H27N7
    Forma y color:Solid
    Peso molecular:401.51
  • PCAF-IN-1

    CAS:
    <p>PCAF-IN-1 is a highly selective PCAF inhibitor with potential anti-tumor, anti-inflammatory, and anti-heart disease effects.</p>
    Fórmula:C15H11ClN6
    Forma y color:Solid
    Peso molecular:310.74
  • N-Descyclopropanecarbaldehyde Olaparib

    CAS:
    <p>N-Descyclopropanecarbaldehyde Olaparib is a CRBN ligand for dual EGFR/PARP PROTAC, suitable for F-18 radiolabeling and tumor imaging via PET.</p>
    Fórmula:C20H19FN4O2
    Forma y color:Solid
    Peso molecular:366.39
  • Ifidancitinib

    CAS:
    <p>Ifidancitinib (ATI-50002) is a JAK kinase 1/3 inhibitor used to study autoimmune diseases.</p>
    Fórmula:C20H18FN5O3
    Pureza:98.05%
    Forma y color:Solid
    Peso molecular:395.39
  • Eicosapentaenoic Acid (Standard)

    CAS:
    Eicosapentaenoic Acid (Standard) is the standard substance of Eicosapentaenoic Acid, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Eicosapentaenoic Acid is an ω-3 fatty acid and an inhibitor of fatty acid synthase (FASN). Eicosapentaenoic Acid promotes DNA demethylation in the reexpression of the tumor suppressor gene CCAAT/ enhancer-binding protein δ (C/EBPδ). Eicosapentaenoic Acid activates the RAS/ERK/C/EBPβ pathway in U937 leukemia cells through demethylation of the CpG island of H-RAS intron 1. Eicosapentaenoic Acid promotes the relaxation of vascular smooth muscle cells and vasodilation.
    Fórmula:C20H30O2
    Peso molecular:302.45
  • TCS PIM-1 1

    CAS:
    <p>TCS PIM-1 1 (SC 204330) is a potent ATP-competitive inhibitor of Pim-1 kinase with an IC50 of 50 nM, selective over MEK1/2 and Pim-2.</p>
    Fórmula:C18H11BrN2O2
    Pureza:97% - 97.98%
    Forma y color:Solid
    Peso molecular:367.2
  • Nudifloramide

    CAS:
    <p>Nudifloramide (1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide) is one of the end degradation products of nicotinamide-adenine dinucleotide (NAD).</p>
    Fórmula:C7H8N2O2
    Pureza:99.7% - ≥95%
    Forma y color:Solid
    Peso molecular:152.15
  • BI-7273

    CAS:
    <p>BI-7273 is an effective, specific, BRD9 BD Inhibitor, which can infiltrate cell.</p>
    Fórmula:C20H23N3O3
    Pureza:97.37% - 99.57%
    Forma y color:Solid
    Peso molecular:353.41
  • BIX-01294

    CAS:
    <p>BIX-01294 is an G9a Histone Methyltransferase inhibitor(IC50 : 1.9 μM).</p>
    Fórmula:C28H38N6O2
    Pureza:98.58% - 99.64%
    Forma y color:Solid
    Peso molecular:490.64