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Cromatina / Epigenética

Cromatina / Epigenética

Los inhibidores de cromatina/epigenética son compuestos que modulan la estructura y función de la cromatina o interfieren con modificaciones epigenéticas, como la metilación del ADN y la modificación de histonas. Estos inhibidores son herramientas esenciales para estudiar la regulación de la expresión génica y el papel de la epigenética en enfermedades como el cáncer, los trastornos neurológicos y las anomalías del desarrollo. Al dirigirse a los procesos epigenéticos, estos inhibidores pueden alterar los patrones de expresión génica y ofrecer nuevas vías terapéuticas. En CymitQuimica, ofrecemos una amplia selección de inhibidores de cromatina/epigenética de alta calidad para apoyar su investigación en biología molecular, genética y epigenética.

Subcategorías de "Cromatina / Epigenética"

Se han encontrado 2238 productos de "Cromatina / Epigenética"

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  • Ritlecitinib

    CAS:
    <p>Ritlecitinib (PF-06651600) is an orally available, selective JAK3 inhibitor and does not affect the activity of JAK1/2.Cost-effective and quality-assured.</p>
    Fórmula:C15H19N5O
    Pureza:98.82% - 99.92%
    Forma y color:Solid
    Peso molecular:285.34
  • GSK-J1 sodium salt

    CAS:
    <p>GSK-J1 sodium salt is a potent inhibitor of the H3K27 histone demethylases JMJD3 and UTX.</p>
    Fórmula:C22H22N5NaO2
    Forma y color:Solid
    Peso molecular:411.4408
  • Senaparib

    CAS:
    <p>Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor activity.</p>
    Fórmula:C24H20F2N6O3
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:478.45
  • Aurora kinase inhibitor-3

    CAS:
    <p>Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) is a potent inhibitor of Aurora A kinase (IC50 = 42 nM).1 It is selective for Aurora A over BMX, BTK,</p>
    Fórmula:C21H18F3N5O
    Pureza:98.91%
    Forma y color:Solid
    Peso molecular:413.4
  • NSC 228155

    CAS:
    <p>NSC 228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and modulate EGFR tyrosine phosphorylation.</p>
    Fórmula:C11H6N4O4S
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:290.25
  • PF-CBP1

    CAS:
    <p>PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).</p>
    Fórmula:C29H36N4O3
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:488.62
  • 653-47

    CAS:
    <p>653-47 enhances the effects of 666-15 on inhibiting CREB and is a mild CREB inhibitor itself (IC50: 26.3μM).</p>
    Fórmula:C20H19ClN2O3
    Forma y color:Solid
    Peso molecular:370.83
  • PF 477736

    CAS:
    <p>PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) and also inhibits FGFR3, Aurora-A, VEGFR2, Flt3, Fms (</p>
    Fórmula:C22H25N7O2
    Pureza:97.58% - 99.94%
    Forma y color:Solid
    Peso molecular:419.48
  • Paris saponin VII

    CAS:
    <p>Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.</p>
    Fórmula:C51H82O21
    Pureza:99.51% - 99.63%
    Forma y color:Solid
    Peso molecular:1031.18
  • CPI-637

    CAS:
    <p>CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibitor.</p>
    Fórmula:C22H22N6O
    Pureza:99.89% - 99.95%
    Forma y color:Solid
    Peso molecular:386.45
  • 6-Bromo-3-methyl-1,4-dihydroquinazolin-2-one

    CAS:
    <p>CHEMBRDG-BB 7118966 is an inhibitor of Bromodomain-containing protein 4 (human).</p>
    Fórmula:C9H9BrN2O
    Pureza:99.28%
    Forma y color:Solid
    Peso molecular:241.08
  • Cerdulatinib

    CAS:
    <p>Cerdulatinib (PRT2070) is an novel oral dual Syk/JAK inhibitor.</p>
    Fórmula:C20H27N7O3S
    Pureza:98.74% - 99.49%
    Forma y color:Solid
    Peso molecular:445.54
  • UNC1079

    CAS:
    <p>UNC1079 is an selective L3MBTL3 domain inhibitor</p>
    Fórmula:C28H42N4O2
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:466.66
  • EPZ015666

    CAS:
    <p>EPZ015666 (GSK3235025) is an orally available inhibitor of PRMT5 enzymatic activity.</p>
    Fórmula:C20H25N5O3
    Pureza:98% - 99.64%
    Forma y color:Solid
    Peso molecular:383.44
  • BI-9564

    CAS:
    <p>BI-9564, a specific cell-permeable BRD9 BD inhibitor. The Kd for BRD9 is 5.9 nM, and IC50 for BET family is &gt; 100 μM.</p>
    Fórmula:C20H23N3O3
    Pureza:99.38%
    Forma y color:Solid
    Peso molecular:353.41
  • PF-9363

    CAS:
    <p>PF-9363 (CTX-3648) is a potent and high selective KAT6A/KAT6B inhibitor. PF-9363 can be used for the research of cancer.</p>
    Fórmula:C20H20N4O6S
    Pureza:99.03% - 99.7%
    Forma y color:Solid
    Peso molecular:444.46
  • Anacardic Acid

    CAS:
    <p>Anacardic Acid (6-pentadecylsalicylic Acid) is an effective inhibitor of p300 and p300/CBP-associated factor histone acetyltranferases.</p>
    Fórmula:C22H36O3
    Pureza:97.47% - 99.87%
    Forma y color:Solid
    Peso molecular:348.52
  • 666-15

    CAS:
    <p>666-15 is a selective CREB inhibitor with an IC50 of 81 nM. 666-15 can effectively inhibit the growth of breast cancer.Cost-effective and quality-assured.</p>
    Fórmula:C33H31Cl2N3O5
    Pureza:99.41% - 99.88%
    Forma y color:Solid
    Peso molecular:620.52
  • KDM4D-IN-1

    CAS:
    <p>KDM4D-IN-1 is a KDM4D inhibitor (IC50: 0.41±0.03 μM).</p>
    Fórmula:C11H7N5O
    Pureza:99.51% - >99.99%
    Forma y color:Solid
    Peso molecular:225.21
  • Nicotinamide riboside chloride

    CAS:
    <p>NR, also SRT647, is a B3 vitamin form; precursor to NAD+.</p>
    Fórmula:C11H15ClN2O5
    Pureza:98.92% - 99.86%
    Forma y color:Solid
    Peso molecular:290.7