CymitQuimica logo
Cromatina / Epigenética

Cromatina / Epigenética

Los inhibidores de cromatina/epigenética son compuestos que modulan la estructura y función de la cromatina o interfieren con modificaciones epigenéticas, como la metilación del ADN y la modificación de histonas. Estos inhibidores son herramientas esenciales para estudiar la regulación de la expresión génica y el papel de la epigenética en enfermedades como el cáncer, los trastornos neurológicos y las anomalías del desarrollo. Al dirigirse a los procesos epigenéticos, estos inhibidores pueden alterar los patrones de expresión génica y ofrecer nuevas vías terapéuticas. En CymitQuimica, ofrecemos una amplia selección de inhibidores de cromatina/epigenética de alta calidad para apoyar su investigación en biología molecular, genética y epigenética.

Subcategorías de "Cromatina / Epigenética"

Se han encontrado 2238 productos de "Cromatina / Epigenética"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
productos por página.
  • Upadacitinib

    CAS:
    <p>Upadacitinib (ABT-494), a selective JAK1 inhibitor, is researched for autoimmune diseases; IC50: 43 nM.</p>
    Fórmula:C17H19F3N6O
    Pureza:98.96% - 99.94%
    Forma y color:Solid
    Peso molecular:380.37
  • 1,5-Isoquinolinediol

    CAS:
    <p>1,5-Isoquinolinediol, a PARP1 inhibitor (IC50: 0.39 μM), is used in DNA repair and cell death studies.</p>
    Fórmula:C9H7NO2
    Pureza:98.29% - 99.35%
    Forma y color:Of White To White Powder
    Peso molecular:161.16
  • AZ505

    CAS:
    <p>AZ505 is an effective and specific SMYD2 inhibitor (IC50: 0.12 μM).</p>
    Fórmula:C29H38Cl2N4O4
    Pureza:98.18%
    Forma y color:Solid
    Peso molecular:577.54
  • Reversine

    CAS:
    <p>Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).</p>
    Fórmula:C21H27N7O
    Pureza:98% - 98.42%
    Forma y color:Solid
    Peso molecular:393.49
  • MLN8054

    CAS:
    <p>MLN8054 is a potent and selective Aurora A kinase inhibitor with an IC50 of 4 nM.</p>
    Fórmula:C25H15ClF2N4O2
    Pureza:98.07% - 98.26%
    Forma y color:Solid
    Peso molecular:476.86
  • 666-15

    CAS:
    <p>666-15 is a selective CREB inhibitor with an IC50 of 81 nM. 666-15 can effectively inhibit the growth of breast cancer.Cost-effective and quality-assured.</p>
    Fórmula:C33H31Cl2N3O5
    Pureza:99.41% - 99.88%
    Forma y color:Solid
    Peso molecular:620.52
  • GSK1379725A

    CAS:
    <p>GSK1379725A is a selective BPTF ligand (Kd = 2.8 μM).</p>
    Fórmula:C23H23FN6O3
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:450.47
  • CPI-637

    CAS:
    <p>CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibitor.</p>
    Fórmula:C22H22N6O
    Pureza:99.89% - 99.95%
    Forma y color:Solid
    Peso molecular:386.45
  • Bromosporine

    CAS:
    <p>Bromosporine is a broad spectrum inhibitor for bromodomains for BRD2/4/9 and CECR2 (IC50: 0.41/0.29/0.122/0.017 μM), respectively.</p>
    Fórmula:C17H20N6O4S
    Pureza:99.65% - 99.79%
    Forma y color:Solid
    Peso molecular:404.44
  • Ruboxistaurin mesylate

    CAS:
    <p>Ruboxistaurin: PKC beta inhibitor, eases oxidative stress, heart issues &amp; nephropathy in diabetic rats, halts retinal neovascularization.</p>
    Fórmula:C29H32N4O6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:564.65
  • Cerdulatinib

    CAS:
    <p>Cerdulatinib (PRT2070) is an novel oral dual Syk/JAK inhibitor.</p>
    Fórmula:C20H27N7O3S
    Pureza:98.74% - 99.49%
    Forma y color:Solid
    Peso molecular:445.54
  • PF-9363

    CAS:
    <p>PF-9363 (CTX-3648) is a potent and high selective KAT6A/KAT6B inhibitor. PF-9363 can be used for the research of cancer.</p>
    Fórmula:C20H20N4O6S
    Pureza:99.03% - 99.7%
    Forma y color:Solid
    Peso molecular:444.46
  • UNC1999

    CAS:
    <p>UNC1999 is a orally bioavailable, effective and specific inhibitor of EZH2 (IC50=2 nM) and EZH1 (IC50=45).</p>
    Fórmula:C33H43N7O2
    Pureza:99.19% - >99.99%
    Forma y color:Solid
    Peso molecular:569.74
  • Anacardic Acid

    CAS:
    <p>Anacardic Acid (6-pentadecylsalicylic Acid) is an effective inhibitor of p300 and p300/CBP-associated factor histone acetyltranferases.</p>
    Fórmula:C22H36O3
    Pureza:97.47% - 99.87%
    Forma y color:Solid
    Peso molecular:348.52
  • Bobcat339

    CAS:
    <p>Bobcat339 is a novel cytosine-based TET enzyme inhibitor (IC50s: 33/73 uM for TET1/2), but not DNMT3a, does not inhibit the DNA methyltransferase DNMT3a.</p>
    Fórmula:C16H12ClN3O
    Pureza:97.79% - 99.24%
    Forma y color:Solid
    Peso molecular:297.74
  • Nicotinamide Hydrochloride

    CAS:
    <p>Nicotinamide Hydrochloride, a vitamin B3 form, inhibits SIRT2 and melanoma growth, enhancing NAD+, ATP, ROS, and survival in melanoma mice.</p>
    Fórmula:C6H7ClN2O
    Forma y color:Solid
    Peso molecular:158.59
  • Nicotinamide riboside chloride

    CAS:
    <p>NR, also SRT647, is a B3 vitamin form; precursor to NAD+.</p>
    Fórmula:C11H15ClN2O5
    Pureza:98.92% - 99.86%
    Forma y color:Solid
    Peso molecular:290.7
  • 8-CHLOROQUINAZOLIN-4(1H)-ONE

    CAS:
    <p>8-CHLOROQUINAZOLIN-4(1H)-ONE is inhibitor of Poly [ADP-ribose] polymerase 1 (human)</p>
    Fórmula:C8H5ClN2O
    Pureza:98.79%
    Forma y color:Solid
    Peso molecular:180.59
  • ICG001

    CAS:
    <p>ICG001 antagonizes Wnt signaling, binds CBP with 3 μM IC50, not p300.</p>
    Fórmula:C33H32N4O4
    Pureza:99.06% - 99.95%
    Forma y color:Solid
    Peso molecular:548.63
  • (R)-(-)-JQ1 Enantiomer

    CAS:
    <p>(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1. (+)-JQ1 is a BET bromodomain inhibitor, acting on BRD4(1/2)(IC50 of 77 nM/33 nM in a cell-free assay)</p>
    Fórmula:C23H25ClN4O2S
    Pureza:99.38%
    Forma y color:Solid
    Peso molecular:456.99