Somatostatina
La somatostatina es una hormona peptídica que inhibe la liberación de varias otras hormonas, incluyendo la hormona de crecimiento, insulina y glucagón. Actúa al unirse a los receptores de somatostatina, que son receptores acoplados a proteínas G expresados en varios tejidos. Los análogos de la somatostatina se utilizan en el tratamiento de la acromegalia, tumores neuroendocrinos y trastornos gastrointestinales. Estos análogos también son herramientas valiosas para estudiar la secreción y señalización hormonal. En CymitQuimica, ofrecemos una gama completa de análogos de somatostatina de alta calidad para apoyar su investigación en endocrinología, regulación hormonal y desarrollo terapéutico.
Se han encontrado 54 productos de "Somatostatina"
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DOTA-JR11
CAS:DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.Fórmula:C74H98ClN19O21S2Forma y color:SolidPeso molecular:1689.27Dotanoc
CAS:Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.Fórmula:C69H94N14O17S2Forma y color:SolidPeso molecular:1455.71Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Fórmula:C53H71N11O14S2Forma y color:SolidPeso molecular:1150.33Cyclosomatostatin TFA
Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.Fórmula:C46H58F3N7O8Forma y color:SolidPeso molecular:893.99L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Fórmula:C31H44N6O9Pureza:98%Forma y color:SoildPeso molecular:644.72Tau conotoxin CnVA
CAS:Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Fórmula:C72H116N24O17S4Forma y color:SolidPeso molecular:1718.1SSTR4 agonist-1
CAS:<p>SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.</p>Fórmula:C16H23N3O2Forma y color:SolidPeso molecular:289.37L-797,591 hydrochloride
L-797,591 HCl activates SSTR1, boosts p-ERK5 with AG1478, and enhances p38 phosphorylation, reversible by AG1478.Fórmula:C38H50ClN5O2Pureza:98.65% - >99.99%Forma y color:SoildPeso molecular:644.30Neuronostatin-13 (human)
CAS:Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.Fórmula:C64H110N20O16Pureza:98%Forma y color:SolidPeso molecular:1415.68[D-Trp8,Tyr11] Somatostatin
CAS:[D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,Fórmula:C76H104N18O20S2Peso molecular:1653.88[Tyr11]-Somatostatin
CAS:[Tyr11]-Somatostatin, a neuroactive peptide, aids proteomics research and modulates retinal function.Fórmula:C76H104N18O20S2Peso molecular:1653.89DOTA-EB-TATE
DOTA-EB-TATE is formed by combining the SST peptide derivative DOTA-octreotate with an Evans blue analog (EB). This peptide drug conjugate (PDC) enhances the pharmacokinetics of SSTR2 analogs and reduces PRRT toxicity. Additionally, DOTA-EB-TATE serves in the synthesis/research of radiopharmaceutical conjugates (RDC).Fórmula:C105H133N21O30S5Peso molecular:2329.63Cortistatin-14
CAS:Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.Fórmula:C81H114N20O18S2Pureza:98.06% - 98.23%Forma y color:SolidPeso molecular:1720.03Cyclosomatostatin Acetate
<p>Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell</p>Fórmula:C46H61N7O8Pureza:98.83%Forma y color:SolidPeso molecular:840.02L803
CAS:L803 is a selective somatostatin receptor type 4 (SST4) agonist that can inhibit L-type calcium channel currents (ICa). It holds potential for research into degenerative diseases of retinal ganglion cells (RGC), such as glaucoma.Fórmula:C50H80N13O19PForma y color:SolidPeso molecular:1198.22Somatostatin 1-28 acetate
Somatostatin 1-28 acetate circulates in human plasma.Pureza:99.22%Forma y color:Soild(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide
CAS:Somatostatin analog (Compound 4) with Kd: SSTR5-0.61nM, SSTR3-11.05nM, SSTR2-23.5nM, SSTR1-1.2µM, SSTR4->1µM.Fórmula:C50H67N11O10S2Peso molecular:1046.26[Tyr1]-Somatostatin-14
CAS:[Tyr1]-Somatostatin-14 could binds to SSTR2.Fórmula:C82H108N18O20S2Peso molecular:1729.99Anti-Somatostatin Antibody (9L93)
Anti-Somatostatin Antibody (9L93) is a Rabbit antibody targeting Somatostatin. Anti-Somatostatin Antibody (9L93) can be used in ELISA.Forma y color:Odour Liquid
